Compile Data Set for Download or QSAR
Report error Found 21 of ic50 data for polymerid = 50003278
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM59100(Bi-ligand, 3)
Affinity DataIC50: 400nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044967(CHEMBL3309759)
Affinity DataIC50: 500nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044973(CHEMBL3309761)
Affinity DataIC50: 700nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50126829((E)-1-(6-(3-acetyl-2,4,6-trihydroxy-5-methylbenzyl...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044971(CHEMBL3309760)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044974(CHEMBL3309762)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044975(CHEMBL3309763)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044976(CHEMBL2316879)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in absence of 0.01% Triton X100 by U...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50044976(CHEMBL2316879)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Thermus flavus MDH pre-incubated for 4 mins before reaction initiation in presence of OAA and NAPH in presence of 0.01% Triton X100 by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50111591(4-[2-(2,4-Difluoro-phenylamino)-thiazol-4-yl]-benz...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50111589(2-[(3,5-diiodo-4-oxidophenyl)(3,5-diiodo-4-oxocycl...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50023867(Indirubin)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50111585(4-bromophenylazophenol | 4-(4-Bromo-phenylazo)-phe...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM3175(Bisindolylmaleimide 11b | Ro 31-8220 | CHEMBL6291 ...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50126827(4-(1-Hydroxy-naphthalen-2-ylazo)-naphthalene-1-sul...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50310357(indigo | CHEMBL599552)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50072147(CHEMBL100473 | 2,3-Bis-[1-amino-1-(2-amino-phenyls...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50111604(3-[1-(4-Phenoxy-phenylamino)-meth-(Z)-ylidene]-3H-...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMalate dehydrogenase(Thermus thermophilus)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM2681(3-{1-[3-(dimethylamino)propyl]-1H-indol-3-yl}-4-(1...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory activity against malate dehydrogenase (MDH) from Thermus flavusMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed