Compile Data Set for Download or QSAR
Report error Found 36 of ic50 data for polymerid = 50003062
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50604141(CHEMBL5188433)
Affinity DataIC50: 6nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50604138(CHEMBL5184381)
Affinity DataIC50: 10nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311261(US10155760, Example 117 | (S)-methyl (5-((2-amino-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311210(US10155760, Example 66 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 30nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50585189(CHEMBL5083125)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human BIKe using peptide as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50585191(CHEMBL5079149)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human BIKe using peptide as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311208(US10155760, Example 64 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 90nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50573682(CHEMBL4872886)
Affinity DataIC50: 120nMAssay Description:Inhibition of wild-type human partial length BIKE (S34 to N329 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50603678(CHEMBL5202351)
Affinity DataIC50: 161nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311266(US10155760, Example 122 | (S)-1-((4-(difluoromethy...)
Affinity DataIC50: 180nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311268(US10155760, Example 124 | (S)-1-((2′,4-bis(d...)
Affinity DataIC50: 180nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311291(US10155760, Example 147 | (S)-1-((2′-chloro-...)
Affinity DataIC50: 260nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311193(US10155760, Example 37 | (S)-1-(2-(difluoromethyl)...)
Affinity DataIC50: 280nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511400(CHEMBL4535040)
Affinity DataIC50: 707nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50585189(CHEMBL5083125)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of NanoLuc-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511375(CHEMBL4593649)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511376(CHEMBL4516665)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511373(CHEMBL4571548)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311381(US10155760, Example 238 | (S)-1-((4-chloro-2′...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511395(CHEMBL4473140)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511398(CHEMBL4582326)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511379(CHEMBL4447403)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511383(CHEMBL4531680)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM311267(US10155760, Example 123 | (S)-1-((2′,6-bis(d...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511394(CHEMBL4552310)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511399(CHEMBL4542463)
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511397(CHEMBL4452939)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511377(CHEMBL4534571)
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511378(CHEMBL4470026)
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50585191(CHEMBL5079149)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of NanoLuc-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511384(CHEMBL4561238)
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511396(CHEMBL4472438)
Affinity DataIC50: 3.83E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 6.55E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50606012(CHEMBL5087558)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of BIKE (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50401152(CHEMBL2205766)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BMP2KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBMP-2-inducible protein kinase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50273541(N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl...)
Affinity DataIC50: 1.01E+4nMAssay Description:Binding affinity to biotinylated BMP2K (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed