Compile Data Set for Download or QSAR
Report error Found 22 of ic50 data for polymerid = 50002748
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123407(2-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-pheny...)
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123417(2-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-pheny...)
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123431(7-{7-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-oxo-2...)
Affinity DataIC50: 28nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123412(1-Ethyl-2-{7-[1-(1-imino-ethyl)-piperidin-4-yloxy]...)
Affinity DataIC50: 58nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123414(((5-Carbamimidoyl-benzo[b]thiophen-2-ylmethyl)-{4-...)
Affinity DataIC50: 63nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084617(YM-60828 | ((7-carbamimidoyl-naphthalen-2-ylmethyl...)
Affinity DataIC50: 63nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123426(2-{7-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-oxo-2...)
Affinity DataIC50: 76nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123422(((7-Carbamimidoyl-naphthalen-2-ylmethyl)-{4-[1-(1-...)
Affinity DataIC50: 83nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123416(((5-Carbamimidoyl-benzo[b]thiophen-2-ylmethyl)-{4-...)
Affinity DataIC50: 86nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123420(7-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-pheny...)
Affinity DataIC50: 94nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123427(3'-{7-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-oxo-...)
Affinity DataIC50: 143nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123413(2-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-pheny...)
Affinity DataIC50: 167nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123429(((3'-Carbamimidoyl-biphenyl-3-ylmethyl)-{4-[1-(1-i...)
Affinity DataIC50: 269nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123425(((3'-Carbamimidoyl-biphenyl-3-ylmethyl)-{4-[1-(1-i...)
Affinity DataIC50: 292nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123415(3'-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataIC50: 360nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123408(4'-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataIC50: 769nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123423(3-{3-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-ph...)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123421(3-{5-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-ph...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123409(2'-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123411(2'-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123410(3-{5-[({4-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-ph...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin-2(Rat)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123419(3-(5-{7-[1-(1-Imino-ethyl)-piperidin-4-yloxy]-3-ox...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory concentration against trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed