Report error Found 421 of ic50 data for polymerid = 50002453
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of 8His-tagged Pin1 PPIase domain (45-163)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human N-terminal His6-tagged Pin1 PPIase activity expressed in Escherichia coli BL21 using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as su...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human N-terminal His-tagged Pin1 expressed in Escherichia coli BL21 using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate i...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of N-terminal His tagged human Pin1 expressed in Escherichia coli BL21 (DE3) using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate preincu...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of 8His-tagged Pin1 PPIase domain (45-163)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of 8His-tagged Pin1 PPIase domain (45-163)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Reversible inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human Pin1 PPIase Activity by protease free PPIase assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of Gst-tagged human Pin1 by Western blot analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Inhibition of Pin1 (unknown origin) by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of 8His-tagged Pin1 PPIase domain (45-163)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Displacement of FITC-WFYpSPFLE from human Pin1 (45-163) catalytic domain by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of 8His-tagged Pin1 PPIase domain (45-163)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of Pin1 by PIn1 PPIase assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human Pin1 (Met1 to Glu163 residues) expressed in Escherichia coli using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrat...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-pNA as substrate by spectrofluorometry assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Pin1 using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human Pin1 (Met1 to Glu163 residues) expressed in Escherichia coli using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrat...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-AEPF-pNA and WFYpSPR-pNA as substrate after 5 minsMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Pin1 by PIn1 PPIase assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Pin1 using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-4-nitroanilide as substrate after 30 mins by protease-coupled assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of Gst-tagged human Pin1by FP assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human Pin1More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of human recombinant PIN1 assessed as inhibition of MCA release using Suc-AEPF-MCA peptide as substrate preincubated with enzyme for 3 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human Pin1 using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrate preincubated for 30 mins follow...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human Pin1 (Met1 to Glu163 residues) expressed in Escherichia coli using Suc-Ala-Glu-cis-Pro-Phe-4-nitroanilide as substrat...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Displacement of 5-FITC-(Acp)-Bth-D-pThr-Pip-2-NaI-Q from N-terminal-GST-fused human Pin1 expressed in Escherichia coli BL21(DE3) incubated for 12 hrs...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Horizon Discovery
Curated by ChEMBL
Horizon Discovery
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of Pin1 (unknown origin) using Suc-Ala-Glu-Pro-Phe-pNA as substrate by spectrofluorometry assayMore data for this Ligand-Target Pair
