Compile Data Set for Download or QSAR
Report error Found 36 of ic50 data for polymerid = 50002206
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380109(CHEMBL2013099)
Affinity DataIC50: 5.42nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380110(CHEMBL2013100)
Affinity DataIC50: 5.53nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380107(CHEMBL2013097)
Affinity DataIC50: 5.69nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380108(CHEMBL2013098)
Affinity DataIC50: 6.62nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380111(CHEMBL2013101)
Affinity DataIC50: 7.74nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380106(CHEMBL2013096)
Affinity DataIC50: 8.36nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380103(CHEMBL2013093)
Affinity DataIC50: 9.71nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380104(CHEMBL2013094)
Affinity DataIC50: 10.4nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380105(CHEMBL2013095)
Affinity DataIC50: 13.2nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380101(CHEMBL2013091)
Affinity DataIC50: 24.2nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380112(CHEMBL2013102)
Affinity DataIC50: 61.4nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380102(CHEMBL2013092)
Affinity DataIC50: 86.7nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404853(CHEMBL156313)
Affinity DataIC50: 5.00E+3nMAssay Description:Effect on Aryl hydrocarbon hydroxylase activity in 3-methylcolanthrene-induced rat liver microsomes at 2.6x10E-4MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404855(CHEMBL158007)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404855(CHEMBL158007)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50017716(CHEMBL282567 | 2-Benzhydryl-pentanoic acid 2-dieth...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404852(CHEMBL345675)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404852(CHEMBL345675)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM24656(CHEMBL14145 | 4-phenyl-1H-imidazole | 4-Phenylimid...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404854(CHEMBL155867)
Affinity DataIC50: 8.13E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404854(CHEMBL155867)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404853(CHEMBL156313)
Affinity DataIC50: 8.40E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50208872(5,6-dimethyl-1H-benzimidazole | 5,6-dimethylbenzim...)
Affinity DataIC50: 9.70E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50208872(5,6-dimethyl-1H-benzimidazole | 5,6-dimethylbenzim...)
Affinity DataIC50: 9.77E+4nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404851(CHEMBL156439)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404851(CHEMBL156439)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404856(CHEMBL156134)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404856(CHEMBL156134)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404849(CHEMBL348508)
Affinity DataIC50: 4.79E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404849(CHEMBL348508)
Affinity DataIC50: 4.80E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404858(CHEMBL351569)
Affinity DataIC50: 6.30E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404858(CHEMBL351569)
Affinity DataIC50: 6.31E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404850(CHEMBL309135)
Affinity DataIC50: 6.70E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50404850(CHEMBL309135)
Affinity DataIC50: 6.76E+5nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM7939(1H-1,3-benzodiazole | Benzimidazole | Benzimidazol...)
Affinity DataIC50: 1.10E+6nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 1A1(Rat)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM7939(1H-1,3-benzodiazole | Benzimidazole | Benzimidazol...)
Affinity DataIC50: 1.10E+6nMAssay Description:Inhibition of Aryl hydrocarbon hydroxylase in phenobarbitone-treated ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed