Compile Data Set for Download or QSAR
Report error Found 7 of ic50 data for polymerid = 50001793
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 392nMAssay Description:Inhibition of human CTK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 492nMAssay Description:Inhibition of human CTK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CTK using poly[Glu:Tyr] (4:1) as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50429477(CHEMBL2332840)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50499634(CHEMBL3741589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MATK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50252338(CHEMBL4090364)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of CTK/MATK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMegakaryocyte-associated tyrosine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human His-tagged MATK expressed in Escherichia coli using tyr-01 peptide as substrate incubated for 60 mins in ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed