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TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50: 16nMAssay Description:50% inhibitory concentration of competitive binding against hCyp-18 PPIase activity using uncoupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388298(CHEMBL2058794)
Affinity DataIC50: 710nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388318(CHEMBL2057227)
Affinity DataIC50: 890nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388311(CHEMBL2059026)
Affinity DataIC50: 1.07E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388314(CHEMBL2059029)
Affinity DataIC50: 2.13E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388314(CHEMBL2059029)
Affinity DataIC50: 2.13E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388325(CHEMBL2059239)
Affinity DataIC50: 2.64E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388323(CHEMBL2059237)
Affinity DataIC50: 2.64E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388323(CHEMBL2059237)
Affinity DataIC50: 2.64E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388309(CHEMBL2059024)
Affinity DataIC50: 2.80E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388324(CHEMBL2059238)
Affinity DataIC50: 2.88E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50621735(CHEMBL5437245)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of FKBP52 (unknown origin) expressed in HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50621733(CHEMBL5420939)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of FKBP52 (unknown origin) expressed in HEK293T cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388300(CHEMBL2058796)
Affinity DataIC50: 3.41E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388320(CHEMBL2059034)
Affinity DataIC50: 3.50E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388321(CHEMBL2059035)
Affinity DataIC50: 3.72E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388310(CHEMBL2059025)
Affinity DataIC50: 5.55E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388322(CHEMBL2059036)
Affinity DataIC50: 6.20E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50109811((S)-1-[2-Oxo-2-(3,4,5-trimethoxy-phenyl)-acetyl]-p...)
Affinity DataIC50: 7.37E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50068939(CHEMBL8597 | 17-Ethyl-1,14-dihydroxy-12-[2-(4-hydr...)
Affinity DataIC50: 8.00E+3nMAssay Description:50% inhibitory concentration of competitive binding against hCyp-18 PPIase activity using uncoupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388267(CHEMBL2058797)
Affinity DataIC50: 8.30E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataIC50: 9.37E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388319(CHEMBL2059033)
Affinity DataIC50: 9.50E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388319(CHEMBL2059033)
Affinity DataIC50: 9.50E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388326(CHEMBL2059240)
Affinity DataIC50: 9.77E+3nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataIC50: 1.05E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388312(CHEMBL2059027)
Affinity DataIC50: 1.16E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388316(CHEMBL2059031)
Affinity DataIC50: 1.17E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388280(CHEMBL2058234)
Affinity DataIC50: 1.43E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50118067(N-{1-[(Ethoxy-{2-[1-(4-nitro-phenylcarbamoyl)-2-ph...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Human Cyclophilin hCyp-18 Peptidyl-prolyl isomerase by using the standard trypsin-coupled PPIase (peptidyl-prolyl isomera...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50118067(N-{1-[(Ethoxy-{2-[1-(4-nitro-phenylcarbamoyl)-2-ph...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Human Cyclophilin hCyp-18 Peptidyl-prolyl isomerase by using the standard trypsin-coupled PPIase (peptidyl-prolyl isomera...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388270(CHEMBL2058800)
Affinity DataIC50: 1.51E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388279(CHEMBL2058233)
Affinity DataIC50: 1.57E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388289(CHEMBL2058495)
Affinity DataIC50: 1.77E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388288(CHEMBL2058494)
Affinity DataIC50: 2.03E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388290(CHEMBL2058496)
Affinity DataIC50: 2.05E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388266(CHEMBL2058500)
Affinity DataIC50: 2.65E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50087860(1-(2-{2-[3-(3H-Imidazol-4-yl)-2-(3-methyl-butyryla...)
Affinity DataIC50: 2.80E+4nMAssay Description:50% inhibitory concentration of competitive binding against hCyp-18 PPIase activity using uncoupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388273(CHEMBL2058224)
Affinity DataIC50: 3.25E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388272(CHEMBL2058223)
Affinity DataIC50: 3.28E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388283(CHEMBL2058237)
Affinity DataIC50: 4.03E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388303(CHEMBL2058801)
Affinity DataIC50: 4.16E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388291(CHEMBL2058498)
Affinity DataIC50: 4.39E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388304(CHEMBL2058802)
Affinity DataIC50: 4.92E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388296(CHEMBL2058792)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388297(CHEMBL2058793)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388299(CHEMBL2058795)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388293(CHEMBL2058787)
Affinity DataIC50: 6.65E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388276(CHEMBL2058227)
Affinity DataIC50: 6.99E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
Departement D'Ingenierie Et D'Etudes Des Proteines

Curated by ChEMBL
LigandPNGBDBM50388278(CHEMBL2058232)
Affinity DataIC50: 8.45E+4nMAssay Description:Binding affinity to FKBP52 FK1 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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