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Report error Found 6 of ic50 data for polymerid = 50000867
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM24777(5-hydroxy-1,4-dihydronaphthalene-1,4-dione | CHEMB...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant ERp57 assessed as inhibition of E-GSH formation using Di-E-GSSG as substrate measured for 60 mins in presence of DTT ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50633548(CHEMBL5418475)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of human recombinant ERp57 assessed as inhibition of E-GSH formation using Di-E-GSSG as substrate measured for 60 mins in presence of DTT ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50633544(CHEMBL5399770)
Affinity DataIC50: 6.98E+3nMAssay Description:Inhibition of human recombinant ERp57 assessed as inhibition of E-GSH formation using Di-E-GSSG as substrate measured for 60 mins in presence of DTT ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtein disulfide-isomerase A3(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed