Compile Data Set for Download or QSAR
Report error Found 3 of ic50 data for polymerid = 50000734
TargetHistone-lysine N-methyltransferase ASH1L(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50631854(CHEMBL5410484)
Affinity DataIC50: 790nMAssay Description:Inhibition of N-terminal Mocr-tagged ASH1L (2069 to 2288 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHistone-lysine N-methyltransferase ASH1L(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50530712(CHEMBL4591248)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ASH1L expressed in Escherichia coli assessed as reduction in methylated polynucleosome level using polynucleosome as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMed
TargetHistone-lysine N-methyltransferase ASH1L(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50530712(CHEMBL4591248)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ASH1L expressed in Escherichia coli assessed as reduction in methylated polynucleosome level using polynucleosome as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMed