Compile Data Set for Download or QSAR
Report error Found 14 of ic50 data for polymerid = 50000613
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054482((S)-4-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarbam...)
Affinity DataIC50: 1.20nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054483((S)-4-{(S)-2-[(S)-1-(1-Carbamimidoyl-piperidin-3-y...)
Affinity DataIC50: 113nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054483((S)-4-{(S)-2-[(S)-1-(1-Carbamimidoyl-piperidin-3-y...)
Affinity DataIC50: 113nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054499(N-((S)-3-Carbamimidoyl-2-hydroxy-cyclohexyl)-2-((S...)
Affinity DataIC50: 293nMAssay Description:compound was tested in vitro for inhibition of serine protease Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054484(CVS-1778 | N-((S)-1-Formyl-4-guanidino-butyl)-2-((...)
Affinity DataIC50: 329nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054505(N-(3-Carbamimidoyl-2-hydroxy-cyclohexyl)-2-((S)-2-...)
Affinity DataIC50: 538nMAssay Description:compound was tested in vitro for inhibition of serine protease Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054503(N-((1S,2R)-3-Carbamimidoyl-2-hydroxy-cyclohexyl)-2...)
Affinity DataIC50: 1.02E+3nMAssay Description:compound was tested in vitro for inhibition of serine protease Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054488(N-((S)-1-Formyl-4-guanidino-butyl)-2-((S)-2-oxo-3-...)
Affinity DataIC50: 1.55E+3nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054497(N-((S)-3-Carbamimidoyl-2-hydroxy-cyclohexyl)-2-((S...)
Affinity DataIC50: 2.50E+3nMAssay Description:compound was tested in vitro for inhibition of serine protease Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054501(2-[(S)-3-(Butane-1-sulfonylamino)-2-oxo-piperidin-...)
Affinity DataIC50: 2.50E+3nMAssay Description:compound was tested in vitro for inhibition of serine protease Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054487(N-[(S)-1-(1-Carbamimidoyl-piperidin-3-ylmethyl)-2-...)
Affinity DataIC50: 1.51E+4nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054487(N-[(S)-1-(1-Carbamimidoyl-piperidin-3-ylmethyl)-2-...)
Affinity DataIC50: 1.51E+4nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054485(N-[(S)-1-((R)-1-Carbamimidoyl-piperidin-3-ylmethyl...)
Affinity DataIC50: 6.07E+4nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAnionic trypsin(Bovine)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50054486(N-[(S)-1-((S)-1-Carbamimidoyl-piperidin-3-ylmethyl...)
Affinity DataIC50: 6.48E+4nMAssay Description:Compound was evaluated for inhibition of amidolytic activity for chromogenic substrate trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed