Compile Data Set for Download or QSAR
Report error Found 376 of ic50 data for polymerid = 50000420
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111856({(R)-2-Amino-4-[benzo[1,3]dioxol-5-ylmethyl-(4-met...)
Affinity DataIC50: 0.0240nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111848((R)-2-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-benz...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111848((R)-2-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-benz...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458764(CHEMBL4209125)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458765(CHEMBL4205697)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458766(CHEMBL4212386)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458771(CHEMBL4214046)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458773(CHEMBL4204567)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458774(CHEMBL4202714)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458775(CHEMBL4218415)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458763(CHEMBL4202848)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216807((3R)-6-cyclohexyl-3-[3-({[(3,4-dimethoxyphenyl)sul...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216831((3R)-6-cyclohexyl-N-hydroxy-3-[3-(4-pyridinyl)-1,2...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216796((3R)-3-(3-{[acetyl(methyl)amino]methyl}-1,2,4-oxad...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216824((3R)-6-cyclohexyl-N-hydroxy-3-(3-{4-[(methylsulfon...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216838((3R)-6-cyclohexyl-N-hydroxy-3-{3-[1-(methylsulfony...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50102948({(R)-4-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-ben...)
Affinity DataIC50: 3.90nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50102948({(R)-4-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-ben...)
Affinity DataIC50: 3.90nMAssay Description:The compound was evaluated for its inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111808({(R)-2-Amino-4-[benzo[1,3]dioxol-5-ylmethyl-(4-met...)
Affinity DataIC50: 4.60nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216841((3R)-6-cyclohexyl-N-hydroxy-3-[3-(4-morpholinylmet...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111840((R)-N-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-(2-tr...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216823(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216833((3R)-6-cyclohexyl-3-{3-[(cyclopropylamino)methyl]-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216830((3R)-3-{3-[(cyclobutylamino)methyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216842((3R)-6-cyclohexyl-N-hydroxy-3-[3-(2-pyridinylmethy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216843(3-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216848((3R)-6-cyclohexyl-N-hydroxy-3-[3-(3-pyridinylmethy...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216817((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(phenylsulfonyl...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216813((3R)-6-cyclohexyl-N-hydroxy-3-{3-[6-(4-methyl-1-pi...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216829((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(2-hydroxy-1,1-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50458758(CHEMBL4207907)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human N-terminal 6His/flag-tagged BMP1 (121 to 721 residues) expressed in CHO cells using ((5-FAM)-ELIDQYDVQRDDSSDGSLED-K(5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50102988({(R)-4-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-ben...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50102988({(R)-4-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-ben...)
Affinity DataIC50: 9nMAssay Description:The compound was evaluated for its inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50241177(5-{(1R)-4-cyclohexyl-1-[2-(hydroxylamino)-2-oxoeth...)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of human procollagen C-proteinase assessed as [3H]procollagen turnover by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50241177(5-{(1R)-4-cyclohexyl-1-[2-(hydroxylamino)-2-oxoeth...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cells by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111842((R)-2-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-benz...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against procollagen C-proteinase (PCP).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216790((3R)-6-cyclohexyl-3-[3-(2,4-dioxo-1,2,3,4-tetrahyd...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216855((3R)-3-{3-[(tert-butylamino)methyl]-1,2,4-oxadiazo...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50402510(CHEMBL2204087)
Affinity DataIC50: 10nMAssay Description:Inhibition of PCP after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216802((3R)-6-cyclohexyl-N-hydroxy-3-(3-{[(methylsulfonyl...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216801((3R)-6-cyclohexyl-N-hydroxy-3-{3-[6-(methylamino)-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216836((3R)-6-cyclohexyl-N-hydroxy-3-{3-[(4-hydroxy-1-pip...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111854({(R)-2-Amino-4-[benzo[1,3]dioxol-5-ylmethyl-(4-met...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216812((3R)-6-cyclohexyl-N-hydroxy-3-[3-({[(4-methylpheny...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216808((3R)-6-cyclohexyl-N-hydroxy-3-[3-(2-pyrazinyl)-1,2...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216809((3R)-6-cyclohexyl-N-hydroxy-3-[3-(5-pyrimidinyl)-1...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216805((3R)-6-cyclohexyl-3-[3-(1,1-dioxido-2-isothiazolid...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50111861({(R)-5-[Benzo[1,3]dioxol-5-ylmethyl-(4-methoxy-ben...)
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216811((3R)-6-cyclohexyl-N-hydroxy-3-[3-({[(4-methoxyphen...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBone morphogenetic protein 1(Human)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50216834(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human procollagen C-proteinase expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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