Compile Data Set for Download or QSAR
Report error Found 21 of ic50 data for polymerid = 50000307
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50631859(CHEMBL5409682)
Affinity DataIC50: 96nMAssay Description:Inhibition of human N-terminal GST tagged GAS41 (1 to 148 residues) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616142(CHEMBL5428051)
Affinity DataIC50: 170nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS4 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616151(CHEMBL5397585)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS4 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616146(CHEMBL5411016)
Affinity DataIC50: 290nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS4 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616152(CHEMBL5439842)
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS4 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50616147(CHEMBL5434894)
Affinity DataIC50: 730nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS4 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625616(CHEMBL5398308)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625617(CHEMBL5421606)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625620(CHEMBL4762606)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625618(CHEMBL5429859)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625615(CHEMBL5435042)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625614(CHEMBL5427853)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625613(CHEMBL5394670)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625612(CHEMBL5416331)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50625604(CHEMBL5439680)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS4 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50566867(CHEMBL4855926)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50566890(CHEMBL4865432)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50566877(CHEMBL4863719)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 4(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50631858(CHEMBL1573062)
Affinity DataIC50: 2.10E+5nMAssay Description:Inhibition of human N-terminal GST tagged GAS41 (1 to 148 residues) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed