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TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | Rucaparib | RUCAPARIB CAMSY...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of DNA polymerase alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408427(CHEMBL483492)
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408426(CHEMBL2092833)
Affinity DataIC50: 480nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50443277(CHEMBL5281189)
Affinity DataIC50: 680nMAssay Description:Inhibition of DNA polymerase alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50205415(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-2,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50205415(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-2,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184755((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(methoxycar...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184758((3aS,4S,7R,7aR)-1,6-didodecyl-2,7-bis(methoxycarbo...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184757((3aR,4R,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5' end radiolabeled 24nt DNA/48nt DNA as primer/template after 5 mins by PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50335554(({[({[2-(2-amino-6-oxo-6,9-dihydro-3H-purin-9-yl)e...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human DNA polymerase alpha by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.60E+3nMpH: 7.5Assay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Human alpha polymeraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184752((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(isopropoxy...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human DNA polymerase-alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184756((3aR,4S,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184754((E)-methyl-3,6-dioxo-4-docosenoate | CHEMBL425779)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50143526(Untenone A | CHEMBL366792)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5-end radiolabeled 24nt to 48nt DNA as primer template after 5 mins in presence of dCTP/dGTP/dTTP/dATP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5-end radiolabeled 24nt to 48nt DNA as primer template after 5 mins in presence of dCTP/dGTP/dTTP/dATP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50313783(N-(4-chlorobenzyl)-1-methyl-9-(morpholinomethyl)-2...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant DNA polymerase alpha expressed in baculovirus infected SF9 cells after 12 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50313784((R)-9-(((2-(benzofuran-2-yl)-2-hydroxyethyl)(methy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant DNA polymerase alpha expressed in baculovirus infected SF9 cells after 12 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184761((3aR,4R,7S,7aS)-dimethyl 3,5-dihexadecyl-1-oxo-7-(...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184750((2R,3S,4R)-4-hydroxy-5-[2-oxo-nonadec-ylidene]-1-p...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50153113([(3S,10R,13R,17R)-17-((E)-(1R,4S)-4-Ethyl-1,5-dime...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory concentration against human DNA polymerase alpha incubated with 0.05 unitsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184748((2S,3S,4R)-methyl 2-ethyl-4-hydroxy-5-(2-oxononade...)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181926(2-{4-[Bis-(4-dimethylcarbamoyl-phenyl)-methoxy]-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181922(2-(4-(bis(3-fluorophenyl)methoxy)phenyl)-1-cyclohe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181927(2-(4-(bis(4-fluorophenyl)methoxy)-2-fluorophenyl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181929(1-cyclohexyl-2-(4-(dip-tolylmethoxy)phenyl)-1H-ben...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181923(2-(4-(benzhydryloxy)phenyl)-1-cyclohexyl-1H-benzo[...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181932(2-(4-(bis(4-chlorophenyl)methoxy)phenyl)-1-cyclohe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181938(1-Cyclohexyl-2-[2-fluoro-4-(phenyl-pyridin-3-yl-me...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181935(1-Cyclohexyl-2-[4-(di-pyridin-3-yl-methoxy)-2-fluo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181941(2-(4-(benzhydryloxy)-2-fluorophenyl)-1-cyclohexyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50181933(2-(4-(bis(4-fluorophenyl)methoxy)phenyl)-1-cyclohe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50191511(2-{4-[4'-chloro-4-(2-oxopyrrolidin-1-yl)biphenyl-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408425(CHEMBL2092835)
Affinity DataIC50: 1.04E+4nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408425(CHEMBL2092835)
Affinity DataIC50: 1.04E+4nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50370476(Combivir | ZIDOVUDINE TRIPHOSPHATE)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184753((1R,1bR,2R,5S,5aS)-1a,3-dihexadecyl-6-oxo-1a,1b,2,...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50370476(Combivir | ZIDOVUDINE TRIPHOSPHATE)
Affinity DataIC50: 1.34E+4nMpH: 7.5Assay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human DNA polymerase alpha assessed as incorporation of [alpha-32P]dCTP up to 1mM preincubated for 30 mins by whatman DE81 paper bindin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50091981(3,7-Dihydroxy-naphthalene-2-carboxylic acid 4-chlo...)
Affinity DataIC50: 1.80E+4nMAssay Description:Compound was evaluated for the inhibitory activity against Human alpha polymeraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184760((2S,3S,4S)-methyl 1-benzyl-2-ethyl-4-hydroxy-5-(2-...)
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184749((2S,3S,4R)-methyl 1-benzyl-2-ethyl-4-hydroxy-5-(2-...)
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50153111([(3S,5S,10S,13R,17R)-17-((R)-1,5-Dimethyl-hexyl)-1...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against human DNA polymerase alpha incubated with 0.05 unitsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50011181(CHEMBL666 | (PFA)dihydroxyphosphinecarboxylic acid...)
Affinity DataIC50: 2.00E+4nMpH: 7.5Assay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50300193(2-[3-(1-Benzyl-1H-pyrazol-3-yl)-benzenesulfonylami...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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