Compile Data Set for Download or QSAR
Report error Found 34 of ic50 data for polymerid = 4934,50001922
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataIC50: 6.30E+3nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM618482(US11759530, Compound Table1.5)
Affinity DataIC50: 1.02E+4nMAssay Description:No assay is defined.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82310(Purine, 5)
Affinity DataKi:  4.30E+3nM ΔG°:  -31.9kJ/mole IC50: 1.02E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82329(Purine, 24)
Affinity DataIC50: 1.27E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82307(Purine, 2)
Affinity DataIC50: 1.35E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82308(Purine, 3)
Affinity DataIC50: 1.37E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82322(Purine, 17)
Affinity DataIC50: 1.82E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82328(Purine, 23)
Affinity DataIC50: 2.00E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82324(Purine, 19)
Affinity DataIC50: 2.34E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50132162(Phosphoric acid mono-(2,3,4-trihydroxy-5,6-bis-pho...)
Affinity DataIC50: 2.74E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50075651(1D-myo-inositol 1,3,4,5-tetrakis(dihydrogen phosph...)
Affinity DataIC50: 2.78E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82327(Purine, 22)
Affinity DataIC50: 2.80E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82326(Purine, 21)
Affinity DataIC50: 2.88E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50221652(CHEMBL3349691)
Affinity DataIC50: 3.94E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82309(Purine, 4)
Affinity DataIC50: 4.34E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataIC50: 4.37E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataIC50: 4.37E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82325(Purine, 20)
Affinity DataIC50: 4.90E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82306(Purine, 1)
Affinity DataIC50: 5.71E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82318(Purine, 13)
Affinity DataIC50: 6.30E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82323(Purine, 18)
Affinity DataIC50: 6.76E+4nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50132165(Phosphoric acid mono-(2,4,6-trihydroxy-3,5-bis-pho...)
Affinity DataIC50: 9.00E+4nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50221513(CHEMBL3349690)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Rat)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50221514(CHEMBL3351092)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity against recombinant plasmid rat brain IP3K by overexpressing in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82313(Purine, 8)
Affinity DataIC50: 1.02E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82320(Purine, 15)
Affinity DataIC50: 1.17E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82312(Purine, 7)
Affinity DataIC50: 1.38E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82315(Purine, 10)
Affinity DataIC50: 1.50E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82311(Purine, 6)
Affinity DataIC50: 1.50E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82321(Purine, 16)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82319(Purine, 14)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82317(Purine, 12)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82316(Purine, 11)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetInositol-trisphosphate 3-kinase A(Human)
City of Hope

US Patent
LigandPNGBDBM82314(Purine, 9)
Affinity DataIC50: 2.20E+5nMpH: 8.0 T: 2°CAssay Description:IP3K reactions were carried out in a 100ul solution that contained Tris-Cl, EGTA, ATP, DTT, 2,3-diphosphoglycerate, D-l(1,4,5)P3, [3H]-l(1,4,5)P3 and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed