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TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103834(SPI-09 | US9791447, Compound SPI-09 | US11041859, ...)
Affinity DataIC50: 1.90E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103832(SPI-07 | US11041859, Code SPI-07)
Affinity DataIC50: 1.90E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103834(SPI-09 | US9791447, Compound SPI-09 | US11041859, ...)
Affinity DataIC50: 1.90E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM348889(NSC58046 | US9791447, Compound SPI-07)
Affinity DataIC50: 1.90E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103835(SPI-10 | US9791447, Compound SPI-10 | US11041859, ...)
Affinity DataIC50: 2.00E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103835(SPI-10 | US9791447, Compound SPI-10 | US11041859, ...)
Affinity DataIC50: 2.00E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103827(SPI-02 | US9791447, Compound SPI-02 | US11041859, ...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of His-tagged human SENP7 expressed in Escherichia coli (DE3) using YFP-SUMO-ECFP as substrate incubated for 15 mins by Coomassie staining...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103827(SPI-02 | US9791447, Compound SPI-02 | US11041859, ...)
Affinity DataIC50: 2.70E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103827(SPI-02 | US9791447, Compound SPI-02 | US11041859, ...)
Affinity DataIC50: 2.70E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103833(SPI-08 | US9791447, Compound SPI-08 | US11041859, ...)
Affinity DataIC50: 2.80E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103833(SPI-08 | US9791447, Compound SPI-08 | US11041859, ...)
Affinity DataIC50: 2.80E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103829(SPI-04 | US9791447, Compound SPI-04 | US11041859, ...)
Affinity DataIC50: 3.40E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103829(SPI-04 | US9791447, Compound SPI-04 | US11041859, ...)
Affinity DataIC50: 3.40E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103826(SPI-01 | US9791447, Compound SPI-01 | US11041859, ...)
Affinity DataIC50: 3.50E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103826(SPI-01 | US9791447, Compound SPI-01 | US11041859, ...)
Affinity DataIC50: 3.50E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81517(VEA-561)
Affinity DataIC50: 4.30E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103830(SPI-05 | US9791447, Compound SPI-05 | US11041859, ...)
Affinity DataIC50: 4.60E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103830(SPI-05 | US9791447, Compound SPI-05 | US11041859, ...)
Affinity DataIC50: 4.60E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM348888(NSC70551 | US9791447, Compound SPI-06 | US11041859...)
Affinity DataIC50: 4.70E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM348888(NSC70551 | US9791447, Compound SPI-06 | US11041859...)
Affinity DataIC50: 4.70E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM348885(NSC8676 | US9791447, Compound SPI-03)
Affinity DataIC50: 4.80E+3nMAssay Description:The binding of SPI-01 to the enzyme-substrate complex was investigated. CSP analysis was carried out on the 40 kDa complex of 15N-labeled full length...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM103828(SPI-03 | US11041859, Code SPI-03)
Affinity DataIC50: 4.80E+3nMAssay Description:The inhibitors confer the non-competitive inhibitory mechanism, as shown by nuclear magnetic resonance (NMR) and quantitative enzyme kinetic analysis...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81514(VEA-401)
Affinity DataIC50: 2.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: 3.65E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81513(VEA-422)
Affinity DataIC50: 7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81512(VEA-417)
Affinity DataIC50: 7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81510(JCP-666)
Affinity DataIC50: 7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81515(VEA-499)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSentrin-specific protease 7(Human)
City of Hope

US Patent
LigandPNGBDBM81516(VEA-500)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed