Report error Found 268 of ic50 data for polymerid = 49000636,49000641,50007810
Affinity DataIC50: 1.07nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 11.5nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 41.7nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced whole cell currents ...More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
Affinity DataIC50: 58.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 60.3nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
Affinity DataIC50: 70.8nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
Affinity DataIC50: 72.4nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 89.1nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the onset of compound app...More data for this Ligand-Target Pair
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response by fl...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response by fl...More data for this Ligand-Target Pair
Affinity DataIC50: 151nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
