Compile Data Set for Download or QSAR
Report error Found 1030 of ic50 data for polymerid = 49000307,49000311,50000702,50002642,50006869
LigandPNGBDBM50487585(CHEMBL2237954)
Affinity DataIC50: 0.0309nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487598(CHEMBL2237953)
Affinity DataIC50: 0.0437nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487582(CHEMBL2237955)
Affinity DataIC50: 0.0457nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487589(CHEMBL2261189)
Affinity DataIC50: 0.0668nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487592(CHEMBL2261183)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487590(CHEMBL2261188)
Affinity DataIC50: 0.132nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487588(CHEMBL2261191)
Affinity DataIC50: 0.146nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487593(CHEMBL2261182)
Affinity DataIC50: 0.158nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486421(CHEMBL2237950)
Affinity DataIC50: 0.182nMAssay Description:Inhibition of L-type calcium channel in Cavia porcellus (guinea pig) ileal SMC assessed as inhibition of 80 mM KCl-induced currentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487591(CHEMBL2261187)
Affinity DataIC50: 0.212nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487587(CHEMBL2261192)
Affinity DataIC50: 0.488nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487595(CHEMBL2261195)
Affinity DataIC50: 0.543nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487600(CHEMBL2261196)
Affinity DataIC50: 0.564nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487594(CHEMBL2261181)
Affinity DataIC50: 0.596nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487599(CHEMBL2261184)
Affinity DataIC50: 0.748nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487580(CHEMBL2237952)
Affinity DataIC50: 0.906nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in Rabbit cardiac muscle.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50227241(CHEMBL1202817)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in Rabbit cardiac muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50487601(CHEMBL2261198)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002644(CHEMBL78656 | 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-...)
Affinity DataIC50: 1.40nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50486778(CHEMBL2236229)
Affinity DataIC50: 1.49nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486800(CHEMBL2236232)
Affinity DataIC50: 1.66nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486789(CHEMBL2236225)
Affinity DataIC50: 1.69nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486433(CHEMBL2237951)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of L-type calcium channel in Cavia porcellus (guinea pig) ileal SMC assessed as inhibition of 80 mM KCl-induced currentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487586(CHEMBL2261194)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486798(CHEMBL2236212)
Affinity DataIC50: 1.86nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487581(CHEMBL2261190)
Affinity DataIC50: 2nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486803(CHEMBL2236227)
Affinity DataIC50: 2.16nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50436176(Dynacirc | Dynacirc Cr | Isrodipine | PN-200-110 |...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of L-type calcium channel measured using 2-electrode voltage-clamp in human embryonic kidney cells heterologically expressing alpha-1C sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50486799(CHEMBL2236236)
Affinity DataIC50: 2.21nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486801(CHEMBL2236226)
Affinity DataIC50: 2.29nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486786(CHEMBL2236233)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486781(CHEMBL2236213)
Affinity DataIC50: 2.54nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50487602(CHEMBL2261185)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
In DepthDetails Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50487583(CHEMBL2261199)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of calcium channel in Cavia porcellus (guinea pig) ileum assessed as inhibition of KCl-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486787(CHEMBL2236230)
Affinity DataIC50: 2.79nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002628(CHEMBL78651 | 4-(2,3-Dichloro-phenyl)-2,6-dimethyl...)
Affinity DataIC50: 2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50486782(CHEMBL2236211)
Affinity DataIC50: 2.91nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50101963(CHEBI:76917 | BAY-K-5552 | Nisoldipine | Sular)
Affinity DataIC50: 3nMAssay Description:Inhibition of L-type calcium channel measured using 2-electrode voltage-clamp in Chinese hamster ovary cells heterologically expressing alpha-1C subu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50486777(CHEMBL2236209)
Affinity DataIC50: 3.05nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486779(CHEMBL2236231)
Affinity DataIC50: 3.15nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50486783(CHEMBL2236210)
Affinity DataIC50: 3.22nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002603(CHEMBL81326 | 2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-...)
Affinity DataIC50: 3.30nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50486790(CHEMBL2236224)
Affinity DataIC50: 3.54nMAssay Description:Antagonist activity at Cavia porcellus albino (guinea pig) calcium channel assessed as inhibition of KCl-induced ileal longitudinal smooth muscle con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002613(CHEMBL312276 | 2,6-Dimethyl-4-(2-trifluoromethyl-p...)
Affinity DataIC50: 3.60nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002607(CHEMBL432933 | 4-(2,3-Dichloro-phenyl)-2,6-dimethy...)
Affinity DataIC50: 5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Ortho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002626(CHEMBL80771 | 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-...)
Affinity DataIC50: 5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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