Compile Data Set for Download or QSAR
Report error Found 350 of ic50 data for polymerid = 49000273
LigandPNGBDBM50282363(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50: 0.160nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
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LigandPNGBDBM50030727(L-159,913 | CHEMBL97539 | CHEMBL279629 | 4''-[3-Bu...)
Affinity DataIC50: 0.310nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat brain tissue preparationMore data for this Ligand-Target Pair
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LigandPNGBDBM50030727(L-159,913 | CHEMBL97539 | CHEMBL279629 | 4''-[3-Bu...)
Affinity DataIC50: 0.330nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat adrenal tissue preparationMore data for this Ligand-Target Pair
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LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50287290(KRH-594 | CHEMBL34866 | Potassium; 2-[5-ethyl-3-[2...)
Affinity DataIC50: 0.440nMAssay Description:In vitro ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
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LigandPNGBDBM50287294(2-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 0.440nMAssay Description:In vitro ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285171(2-{2,6-Dioxo-4-propyl-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 0.650nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
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LigandPNGBDBM50287291(N-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 0.660nMAssay Description:In vitro ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50009712(CHEMBL315104 | 5,7-Dimethyl-2-propyl-3-[2'-(2H-tet...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50009719(L-158338 | CHEMBL296725 | 7-Methyl-2-propyl-3-[2'-...)
Affinity DataIC50: 1nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50282260(7-Butyl-8-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of specific binding of [125I]AII to Angiotensin II receptor, type 1 from rat liver membraneMore data for this Ligand-Target Pair
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LigandPNGBDBM50011977((E)-3-[2-n-butyl-1-{(4-carboxyphenyl)methyl}-1H-im...)
Affinity DataIC50: 1nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
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LigandPNGBDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50: 1nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50041701(2-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 measured by ability to displace [125I]- A II from its specific binding site in rat liver membran...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50041688({2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4...)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against AT1 receptor of rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibition of specific binding of [125I]AII to Angiotensin II receptor, type 1 from rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285164(1-Cyclohexyl-3-(2-{2,6-dioxo-4-propyl-3-[2'-(1H-te...)
Affinity DataIC50: 1.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
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LigandPNGBDBM50406795(Cozaar | LOSARTAN POTASSIUM)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50011975(4-[2-Butyl-5-(2-carboxy-3-thiophen-2-yl-propenyl)-...)
Affinity DataIC50: 1.5nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
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LigandPNGBDBM50041689(5-Benzyl-2-butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity against AT1 receptor of rat adrenal cortical membranesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50049186(CHEMBL1069 | (S)-3-Methyl-2-{pentanoyl-[2'-(1H-tet...)
Affinity DataIC50: 1.90nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50282261(7-Butyl-10,10-dimethyl-8-[2'-(2H-tetrazol-5-yl)-bi...)
Affinity DataIC50: 2.20nMAssay Description:In vitro inhibition of specific binding of [125I]AII to Angiotensin II receptor, type 1 from rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285165(2-{2,6-Dioxo-4-propyl-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 2.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
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LigandPNGBDBM50009338(Sar-Arg-Val-Tyr-Val-His-Pro-Ala | (S)-2-((S)-1-((S...)
Affinity DataIC50: 2.40nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 measured by ability to displace [125I]- A II from its specific binding site in rat liver membran...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50285163(2-{4-Butyl-2,6-dioxo-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50: 2.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50041683(2-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 3nMAssay Description:Binding affinity against AT1 receptor in the presence of 0.01% BSAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043244(4'-(1-Methyl-2'-propyl-1H-[2,5']bibenzoimidazolyl-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043257(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl-1-[...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043260(2-Butyl-6-(1,1-dioxo-1lambda*6*-[1,2]thiazinan-2-y...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataIC50: 3nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50044356(5-Butyl-2-phenethyl-4-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of [125I]angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranesMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50282270(4'-(2-Butyl-4-cyclopentyl-4-methyl-5-oxo-4,5-dihyd...)
Affinity DataIC50: 3.30nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
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LigandPNGBDBM50285166(3-Allyl-6-propyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 3.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
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LigandPNGBDBM50285160(N-(2-{2,6-Dioxo-4-propyl-3-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataIC50: 3.40nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50044345(5-Butyl-2-(2-hydroxy-2-phenyl-ethyl)-4-[2'-(1H-tet...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of [125I]angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50287289(2-Chloro-N-[5-ethyl-3-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50: 3.60nMAssay Description:In vitro ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50043246(4'-(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl...)
Affinity DataIC50: 4nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043277(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 4nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50145961(7-Methyl-2-propyl-3-{4-[3-(2H-tetrazol-5-yl)-pyrid...)
Affinity DataIC50: 4nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50145972(2-Amino-4-[4-(5,7-dimethyl-2-propyl-imidazo[4,5-b]...)
Affinity DataIC50: 4.20nMAssay Description:Binding affinity for rat angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50285177(6-Propyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 4.30nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50044334(5-{3-Butyl-5-oxo-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of [125I]angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50285167(6-Butyl-3-methyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 4.5nMAssay Description:Tested for binding affinity against angiotensin II receptor in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50043247(4-Methyl-2-propyl-6-pyridin-2-yl-1-[2'-(1H-tetrazo...)
Affinity DataIC50: 5nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50043279(1-Methyl-2'-propyl-3'-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50: 5nMAssay Description:Inhibition of specific binding of [125I]angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50: 5nMAssay Description:Binding affinity against angiotensin II receptor type 1 (AT1) from rat liver.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50044355(2,5-Dibutyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50: 5nMAssay Description:Displacement of [125-I]-labeled angiotensin II from Angiotensin II receptor, type 1 of rat uterine membranesMore data for this Ligand-Target Pair
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LigandPNGBDBM50044355(2,5-Dibutyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of [125I]angiotensin-II binding to the angiotensin II receptor type 1 in rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50282264(2-Butyl-5-cyclohexyl-5-methyl-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50: 5.20nMAssay Description:In vitro binding affinity at Angiotensin II receptor, type 1 from rat liver membrane by [125I]- A II displacement.More data for this Ligand-Target Pair
In DepthDetails Article

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