Compile Data Set for Download or QSAR
Report error Found 1537 of ic50 data for polymerid = 49000268,49000274,49000277,50004523
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030726(3-[4-(2'-Benzoylsulfamoyl-3-fluoro-biphenyl-4-ylme...)
Affinity DataIC50: 0.0530nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50282708(Thiophene-2-carboxylic acid benzyl-{2-ethyl-4-oxo-...)
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030685(Pentanoic acid {4-chloro-3-[3-ethyl-4-(3-fluoro-2'...)
Affinity DataIC50: 0.0700nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50155247(CHEMBL385433)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]CGP42112A from human recombinant AT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125I]CGP 42112A from human recombinant AT2 receptor expressed in HEK293 cells measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030721(4-Bromo-N-butyl-3-{4-[2'-(2,5-dichloro-benzoylsulf...)
Affinity DataIC50: 0.0920nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030693(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.100nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032358(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-phenyl(4-pyridy...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283765(N-{3-[3-Butyl-4-(3-fluoro-2'-(ethyloxtycarbonyl)su...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against AT2 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50011972(CHEMBL385189 | Sar-Arg-Val-Tyr-Ile-His-Pro-Thi-OH)
Affinity DataIC50: 0.110nMAssay Description:In vitro inhibition of [125I]-AII specific binding towards angiotensin II receptor in rat mesenteric membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283763(N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-3-...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against AT1 receptor from rat adrenal tissuesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030711(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.120nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50030711(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030700(N-{4-Bromo-3-[4-(3-fluoro-2'-(N-t-butyloxycarbonyl...)
Affinity DataIC50: 0.140nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030720(N-{3-[4-(3-Fluoro-2'-(N-t-butyloxycarbonyl)-Sulfan...)
Affinity DataIC50: 0.140nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030687(N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-3-...)
Affinity DataIC50: 0.150nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032368(butyloxy 2-[2-(4-{4-ethyl-5-[3-phenyl(butyl)carbox...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030691(Pentanoic acid (4-bromo-3-{4-[2'-(2,5-difluoro-ben...)
Affinity DataIC50: 0.150nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283766(N-(3-{3-Butyl-4-[3-fluoro-2'-(2-fluoro-benzoylsulf...)
Affinity DataIC50: 0.150nMAssay Description:Inhibitory concentration against AT2 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283763(N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Inhibitory concentration against AT2 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030730(Pentanoic acid {4-bromo-3-[4-(3-fluoro-2'-(N-t-but...)
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030707(Pentanoic acid (4-bromo-3-{3-ethyl-4-[3-fluoro-2'-...)
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032367(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-[2-pyridyl(4-py...)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(Pentanoic acid {3-[3-butyl-4-(3-fluoro-2'-(N-t-but...)
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030686(N-{3-[3-Butyl-4-(3-fluoro-2'-(N-t-butyloxycarbonyl...)
Affinity DataIC50: 0.170nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030730(Pentanoic acid {4-bromo-3-[4-(3-fluoro-2'-(N-t-but...)
Affinity DataIC50: 0.170nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030732(N-{3-[3-Butyl-4-(3-fluoro-2'(tert-butoxycarbonyl) ...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against AT1 receptor from rat adrenal tissues.More data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032352(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-biphenylcarboxa...)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030695(N-Butyl-3-[3-butyl-4-(3-fluoro-2'-(N-t-butyloxycar...)
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030694(N-{4-Bromo-3-[3-ethyl-4-(3-fluoro-2'-(N-t-butyloxy...)
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030693(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032352(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-biphenylcarboxa...)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030726(3-[4-(2'-Benzoylsulfamoyl-3-fluoro-biphenyl-4-ylme...)
Affinity DataIC50: 0.190nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030683(N-Butyl-3-[4-(3-fluoro-2'-(N-t-butyloxycarbonyl)-S...)
Affinity DataIC50: 0.190nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283302(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
Affinity DataIC50: 0.200nMAssay Description:In vivo inhibitory concentration against AT2 receptor of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030684(N-{3-[3-Butyl-4-(3-fluoro-2-(N-t-butyloxycarbonyl)...)
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030720(N-{3-[4-(3-Fluoro-2'-(N-t-butyloxycarbonyl)-Sulfan...)
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50009718(CHEMBL7550 | 2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetraz...)
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to angiotensin AT2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283307(4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-...)
Affinity DataIC50: 0.210nMAssay Description:In vivo inhibitory concentration against AT2 receptor of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030691(Pentanoic acid (4-bromo-3-{4-[2'-(2,5-difluoro-ben...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030692(N-(3-{3-Butyl-4-[2'-(2-chloro-benzoylsulfamoyl)-3-...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030717(N-{4-Bromo-3-[4-(3-fluoro-2-(N-t-butyloxycarbonyl)...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030715(N-{3-[3-Butyl-4-(3-fluoro-2-(N-t-butyloxycarbonyl)...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030702(3-[3-Butyl-4-(3-fluoro-2'-(N-t-butyloxycarbonyl)-S...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030711(Pentanoic acid {4-bromo-3-[3-ethyl-4-(3-fluoro-2'-...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030688(N-(3-{3-Butyl-4-[2'-(3,3-dimethyl-butyrylsulfamoyl...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283305(3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propy...)
Affinity DataIC50: 0.210nMAssay Description:In vivo inhibitory concentration against AT2 receptor of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50283300(2-Butyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonylam...)
Affinity DataIC50: 0.210nMAssay Description:In vivo inhibitory concentration against Angiotensin II, type 2 of rat midbrain membraneMore data for this Ligand-Target Pair
In DepthDetails Article

TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(Pentanoic acid {3-[3-butyl-4-(3-fluoro-2'-(N-t-but...)
Affinity DataIC50: 0.220nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetType-2 angiotensin II receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50032354(isopentyloxy 2-[2-(4-{4-ethyl-5-[3-[3-pyridyl(3-py...)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of [125I]-[Sar1,Ile8]Ang II binding at rat angiotensin II (type 2) receptor.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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