Compile Data Set for Download or QSAR
Report error Found 9 of ic50 data for polymerid = 4532
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 21.7nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 30.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 30.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 36.4nMAssay Description:Inhibition of human TLK1 using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM311210(US10155760, Example 66 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50154291(CHEMBL3775181)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human N-terminal FLAG, C-terminal HIS8-tagged TLK1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TLK1 using histone H3 as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human TLK1 using casein as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintill...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase tousled-like 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM8226(3-[(3-chlorophenyl)amino]-4-(2-methoxyphenyl)-2,5-...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of NanoLuc-fused TLK1 (unknown origin) expressed in HEK293T cells after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed