Compile Data Set for Download or QSAR
Report error Found 213 of ic50 data for polymerid = 395
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605525(CHEMBL5175191)
Affinity DataIC50: 5nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605526(CHEMBL5188920)
Affinity DataIC50: 5nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605527(CHEMBL5186248)
Affinity DataIC50: 6nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605523(CHEMBL5197199)
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605535(CHEMBL5198962)
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508013(CHEMBL4541479)
Affinity DataIC50: 8nMAssay Description:Inhibition of ERK5 in human HeLa cells by KiNativ profiling methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605522(CHEMBL5172952)
Affinity DataIC50: 8nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508013(CHEMBL4541479)
Affinity DataIC50: 8nMAssay Description:Inhibition of ERK5 (unknown origin) incubated for 1 hr by KiNativ profiling analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508013(CHEMBL4541479)
Affinity DataIC50: 8nMAssay Description:Inhibition of ERK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50337130(2-((2-methoxy-4-(piperazin-1-yl)phenyl)amino)-5,11...)
Affinity DataIC50: 10nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50559468(CHEMBL4757477)
Affinity DataIC50: 11nMAssay Description:Inhibition of ERK5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605519(CHEMBL5175007)
Affinity DataIC50: 13nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605520(CHEMBL5202924)
Affinity DataIC50: 13nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50434070(CHEMBL2381340)
Affinity DataIC50: 13nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605521(CHEMBL5173346)
Affinity DataIC50: 14nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605528(CHEMBL5175760)
Affinity DataIC50: 14nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605536(CHEMBL5208879)
Affinity DataIC50: 16nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508008(CHEMBL4438379)
Affinity DataIC50: 17nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605533(CHEMBL5180089)
Affinity DataIC50: 19nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508013(CHEMBL4541479)
Affinity DataIC50: 20nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605523(CHEMBL5197199)
Affinity DataIC50: 20nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605534(CHEMBL5208123)
Affinity DataIC50: 22nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605524(CHEMBL5193573)
Affinity DataIC50: 25nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50629292(CHEMBL5422839)
Affinity DataIC50: 27nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605527(CHEMBL5186248)
Affinity DataIC50: 31nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50507989(CHEMBL4445670)
Affinity DataIC50: 35nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50507989(CHEMBL4445670)
Affinity DataIC50: 35nMAssay Description:Activation of ERK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50507989(CHEMBL4445670)
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged ERK5 (1 to 398 residues) expressed in Escherichia coli using biotinylated peptide Ahx-PPGDYSTTP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605518(CHEMBL5179461)
Affinity DataIC50: 37nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605521(CHEMBL5173346)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50363196(CHEMBL1944698)
Affinity DataIC50: 43nMAssay Description:Inhibition of ERK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50507990(CHEMBL4469661)
Affinity DataIC50: 51nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50337134(US9266890, IV-6 | Scaffold, B46 | CHEMBL1673046 | ...)
Affinity DataIC50: 52nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508009(CHEMBL4550589)
Affinity DataIC50: 54nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605528(CHEMBL5175760)
Affinity DataIC50: 58nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50: 59nMAssay Description:Inhibition of ERK5 phosphorylation in sorbitol-stimulated human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50: 59nMAssay Description:Inhibition of GST-tagged ERK5 (unknown origin) expressed in baculovirus expression system incubated for 90 mins by HTS assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50: 59nMAssay Description:Inhibition of ERK5 (unknown origin) expressed in baculovirus expression system incubated for 90 mins in presence of ATP by PKlight ATP detection reag...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50434072(CHEMBL2381342)
Affinity DataIC50: 59nMAssay Description:Inhibition of ERK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605522(CHEMBL5172952)
Affinity DataIC50: 60nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50629290(CHEMBL5394239)
Affinity DataIC50: 62nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508007(CHEMBL4542723)
Affinity DataIC50: 64nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50337139(11-ethyl-2-((2-methoxy-4-(4-methylpiperazin-1-yl)p...)
Affinity DataIC50: 66nMAssay Description:Inhibition of ERK5 in human HeLa cells assessed as reduction in EGF-induced ERK5 autophosphorylation pretreated for 1 hr followed by EGF stimulation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50629291(CHEMBL5440819)
Affinity DataIC50: 67nMAssay Description:Inhibition of ERK5 (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50508012(CHEMBL4526317)
Affinity DataIC50: 68nMAssay Description:Inhibition of His-tagged MAP2K5 activated N-terminal GST-tagged recombinant human ERK5 (1 to 398 residues) expressed in Escherichia coli using biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605526(CHEMBL5188920)
Affinity DataIC50: 70nMAssay Description:Inhibition of ERK5 phosphorylation in human HeLa cells incubated for 1 hr by Western blot densitometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605517(CHEMBL5209433)
Affinity DataIC50: 72nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605511(CHEMBL5193786)
Affinity DataIC50: 77nMAssay Description:Inhibition of ERK5 (1 to 492 residues) in HEK293 cells assessed as paradoxical activation of ERK5 transcriptional activity incubated for 20 hrs by du...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50539940(CHEMBL4636072)
Affinity DataIC50: 79nMAssay Description:Inhibition of ERK5 in human HeLa cells assessed as reduction in EGF-induced ERK5 autophosphorylation pretreated for 1 hr followed by EGF stimulation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Newcastle University Centre For Cancer

Curated by ChEMBL
LigandPNGBDBM50605511(CHEMBL5193786)
Affinity DataIC50: 79nMAssay Description:Inhibition of ERK5 (unknown origin) using K-5FAM-LVEPLTPSGEAPNQ-COOH as substrate incubated for 2 hrs in presence of ATP by IMAP-FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
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