Compile Data Set for Download or QSAR
Report error Found 64 of ic50 data for polymerid = 2742
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.134nMAssay Description:Inhibition of human RSK4 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.159nMAssay Description:Inhibition of human RSK4 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM286091(US10758530, Compound 18 | BDBM286094 | US10081632,...)
Affinity DataIC50: 0.300nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM286091(US10758530, Compound 18 | BDBM286094 | US10081632,...)
Affinity DataIC50: 0.300nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50468574(CHEMBL4116008 | US11414410, Example 100)
Affinity DataIC50: 4nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520159(CHEMBL4543618)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM458758((R)-1-benzyl-N-(9-methyl-6-oxo-6,7,8,9-tetrahydrop...)
Affinity DataIC50: 8nMAssay Description:Radioisotope assays were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radioactive workin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM342166(US9771366, Compound 15 | (R)-1-benzyl-N-(9-methyl-...)
Affinity DataIC50: 8nMAssay Description:Radioisotope assays (SignalChem) were performed for the evaluation of the kinase target profiling and all assays were performed in a designated radio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578032(CHEMBL4847762)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578033(CHEMBL4847469)
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578046(CHEMBL4846725)
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578034(CHEMBL4870231)
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin) using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK a substrate by [32P] gammaATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] labe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578027(CHEMBL4870807)
Affinity DataIC50: 16nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578040(CHEMBL4846978)
Affinity DataIC50: 18nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50389154(CHEMBL2064666)
Affinity DataIC50: 19nMAssay Description:Inhibition of human Rsk4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578031(CHEMBL4845942)
Affinity DataIC50: 25nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578035(CHEMBL4872665)
Affinity DataIC50: 29nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578043(CHEMBL4852908)
Affinity DataIC50: 33nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50585046(CHEMBL5086263)
Affinity DataIC50: 37nMAssay Description:Inhibition of RSK4 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578036(CHEMBL4850890)
Affinity DataIC50: 55nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578029(CHEMBL4856762)
Affinity DataIC50: 84nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578024(CHEMBL4869608)
Affinity DataIC50: 117nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520148(CHEMBL4538751 | US10894784, Example 30.03.01.A)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520152(CHEMBL4594167 | US10894784, Example 150.02)
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520150(CHEMBL4566796)
Affinity DataIC50: 192nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520151(CHEMBL4537673)
Affinity DataIC50: 276nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578038(CHEMBL4852557)
Affinity DataIC50: 301nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520157(CHEMBL4436188)
Affinity DataIC50: 325nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578028(CHEMBL4850184)
Affinity DataIC50: 395nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578039(CHEMBL4874868)
Affinity DataIC50: 410nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520155(CHEMBL4552254 | US10894784, Example 30.01.01)
Affinity DataIC50: 434nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520158(CHEMBL4453292 | US10894784, Example 143.02)
Affinity DataIC50: 528nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50462709(CHEMBL4245507)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520160(CHEMBL4515413 | US10894784, Example 01.03)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520165(CHEMBL4454902)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578025(CHEMBL4865220)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520174(CHEMBL4553949 | US10894784, Example 16.06.02.A)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520175(CHEMBL4451595 | US10894784, Example 135.02)
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520142(CHEMBL4435393)
Affinity DataIC50: 3.22E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578042(CHEMBL4846647)
Affinity DataIC50: 3.59E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520161(CHEMBL4468020 | US10894784, Example 39.01.02)
Affinity DataIC50: 4.12E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578030(CHEMBL4866663)
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50520173(CHEMBL4538591 | US10894784, Example 179.02)
Affinity DataIC50: 6.11E+3nMAssay Description:Inhibition of recombinant full length human His6-tagged RSK4 expressed in baculovirus infected sf21 cells using biotin labelled Ahx-KKLNRTLSFAEPG pep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50626656(CHEMBL5418355)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50578044(CHEMBL4868071)
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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