Compile Data Set for Download or QSAR
Report error Found 2242 of ic50 data for polymerid = 2125,49000355,50000021,50000659
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245192(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245186(3-((S)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataIC50: 0.0160nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245205(2-((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataIC50: 0.0180nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50263230(3-(4-(1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-(2...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50263229(CHEMBL505225 | CHEMBL505969 | 3-(4-(1-(2,3-dihydro...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50343722(3-(4-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-(2...)
Affinity DataIC50: 0.0340nMAssay Description:Displacement of [I125]-CCK8 from human CCK1 receptor expressed in CHO Flip cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245195(2-(((R)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazo...)
Affinity DataIC50: 0.0390nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245187(CHEMBL504861 | CHEMBL446789 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517344(CHEMBL4526455)
Affinity DataIC50: 0.0407nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245188(3-((S)-3-((carboxymethoxy)methyl)-4-(1-(3-ethoxyph...)
Affinity DataIC50: 0.0410nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517358(CHEMBL4585323)
Affinity DataIC50: 0.0427nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50061829((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[...)
Affinity DataIC50: 0.0447nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(CHEMBL411079 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-...)
Affinity DataIC50: 0.0500nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517353(CHEMBL4525615)
Affinity DataIC50: 0.0501nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245201(3-(((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazo...)
Affinity DataIC50: 0.0520nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517333(CHEMBL4440419)
Affinity DataIC50: 0.0525nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245189(3-((R)-3-(acetamidomethyl)-4-(1-(3-ethoxyphenyl)-2...)
Affinity DataIC50: 0.0580nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245187(CHEMBL504861 | CHEMBL446789 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517373(CHEMBL4514283)
Affinity DataIC50: 0.0603nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517378(CHEMBL4440303)
Affinity DataIC50: 0.0631nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517375(CHEMBL4483457)
Affinity DataIC50: 0.0646nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245190(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50263227(3-(4-(2-(2,4-difluorophenyl)-1-(3-ethoxyphenyl)-1H...)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517349(CHEMBL4583158)
Affinity DataIC50: 0.0741nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517368(CHEMBL4441596)
Affinity DataIC50: 0.0741nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517382(CHEMBL4563364)
Affinity DataIC50: 0.0759nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0794nMAssay Description:Binding affinity against cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517357(CHEMBL4568746)
Affinity DataIC50: 0.0794nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517361(CHEMBL4534977)
Affinity DataIC50: 0.0794nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of cholecystokinin A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50263226(CHEMBL506201 | CHEMBL498942 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245184(3-((S)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245182(3-((S)-3-(acetamidomethyl)-4-(1-(3-ethoxyphenyl)-2...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Ability to inhibit the binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of [125I]Cholecystokinin-8 (125I-CCK-8) binding to Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I] CCK-8 from Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Antagonistic activity against cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin A receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of binding of [125I]- CCK-33 to rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Half maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of Cholecystokinin type A receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517376(CHEMBL4473468)
Affinity DataIC50: 0.0832nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517339(CHEMBL4551834)
Affinity DataIC50: 0.0871nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50517363(CHEMBL4471871)
Affinity DataIC50: 0.0891nMAssay Description:Displacement of [125I]-CCK-8 from human CCK1R expressed in human 1321N1 cell membranes after 2 hrs by SPA assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50170765([(S)-1-((4aS,5R)-2-Benzyl-1-mercapto-3-oxo-octahyd...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50170765([(S)-1-((4aS,5R)-2-Benzyl-1-mercapto-3-oxo-octahyd...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50106593([1-(2-Benzyl-3-oxo-1-thioxo-octahydro-4a(S)-pyrido...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholecystokinin receptor type A(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50245191(3-((R)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of human CCK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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