Compile Data Set for Download or QSAR
Report error Found 168 of ic50 data for polymerid = 187,50006749
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50135483(1-(6-methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino...)
Affinity DataIC50: 3nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50135482(1-(5-Methoxy-2-thiophen-2-yl-quinazolin-4-ylamino)...)
Affinity DataIC50: 8nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092879(2-Chloro-4-methyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 20nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50090430(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092879(2-Chloro-4-methyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340608(8-(6-methylpyridin-3-yl)-N-(4-(3-morpholino-1H-1,2...)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50295171(CHEMBL487194 | AILANTHINONE)
Affinity DataIC50: 32nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044568(CHEMBL85822)
Affinity DataIC50: 35nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340606(N-(4-(3-(6-methylpyridin-3-yl)-1H-1,2,4-triazol-1-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340627(7,8-bis(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholi...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340628(7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50349194(NSC-14975 | GLAUCARUBINONE)
Affinity DataIC50: 40nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044567(CHEMBL86615)
Affinity DataIC50: 45nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50062648(2-Chloro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50062648(2-Chloro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 50nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340629(8-methoxy-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-mor...)
Affinity DataIC50: 50nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213931(tylophorinidine | CHEMBL250854)
Affinity DataIC50: 65nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213932([(R)-(+)-deoxytylophorinidine | CHEMBL250474)
Affinity DataIC50: 68nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50295170(6R-senecionylchaparrin | CHEMBL564009)
Affinity DataIC50: 71nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044564(CHEMBL315804)
Affinity DataIC50: 98nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092877(2-Fluoro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50090444(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044572(CHEMBL3341912)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092877(2-Fluoro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340622(8-chloro-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morp...)
Affinity DataIC50: 100nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213934(tylophorinine | CHEMBL398325)
Affinity DataIC50: 110nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340600(N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)-7...)
Affinity DataIC50: 120nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340626(8-cyclopropyl-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3...)
Affinity DataIC50: 130nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340624(8-methyl-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morp...)
Affinity DataIC50: 160nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092882(2,4-Dichloro-pyrimidine-5-carboxylic acid (3,5-bis...)
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092882(2,4-Dichloro-pyrimidine-5-carboxylic acid (3,5-bis...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340614(N-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl)-8-(th...)
Affinity DataIC50: 200nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044566(CHEMBL87274)
Affinity DataIC50: 210nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340610(8-(3-fluoro-4-methoxyphenyl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 250nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340607(7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-(pyridin-2-yl...)
Affinity DataIC50: 290nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092872(2-Chloro-4-ethyl-pyrimidine-5-carboxylic acid (3,5...)
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092890(2-Chloro-pyrimidine-5-carboxylic acid (3,5-bis-tri...)
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044570(CHEMBL87433)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213935((12aS,13R)-2,3,6,7-tetramethoxy-9,10,11,12,12a,13-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213936((S)-2,3,6,7-tetramethoxy-8b,9,10,11,12,12a-hexahyd...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340599(7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 310nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340609(8-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 330nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092883(2-Chloro-4-phenyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044569(CHEMBL83026)
Affinity DataIC50: 400nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092883(2-Chloro-4-phenyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 400nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092871(2-Chloro-4-propyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 500nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044552(CHEMBL3341901)
Affinity DataIC50: 500nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044553(CHEMBL3341956)
Affinity DataIC50: 500nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340613(8-(3-fluoro-4-methoxyphenyl)-N-(4-(3-methyl-1H-1,2...)
Affinity DataIC50: 500nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092880(2-Chloro-4-pentafluoroethyl-pyrimidine-5-carboxyli...)
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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