Compile Data Set for Download or QSAR
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TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human TAOK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 11.7nMAssay Description:Inhibition of human TAOK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50244953(CHEMBL4063500)
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TAO2 expressed in sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50429615(CHEMBL2334586)
Affinity DataIC50: 89nMAssay Description:Inhibition of human wild type partial length TAOK2 (M1 to A320 residues) expressed in mammalian expression system by Kinomescan assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536316(CHEMBL4537058)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536316(CHEMBL4537058)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50536679(CHEMBL4568087)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human GST-tagged TAOK2 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50235830(CHEMBL2006765)
Affinity DataIC50: 529nMAssay Description:Inhibition of TAOK2 (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536313(CHEMBL4529072)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536333(CHEMBL4550547)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50618084(CHEMBL5437375)
Affinity DataIC50: 689nMAssay Description:Inhibition of TAO2 (unknown origin) by Z'-Lyte kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536342(CHEMBL4548193)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536358(CHEMBL2164269)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536348(CHEMBL4545777)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50563891(CHEMBL4793380)
Affinity DataIC50: 903nMAssay Description:Inhibition of recombinant human TAO2 (1 to 320 residues) using myelin basic protein as substrate incubated for 40 mins in presence of [gamma33P]ATP b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536329(CHEMBL1995377)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536335(CHEMBL4563650)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536338(CHEMBL4542920)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536344(CHEMBL600947 | GNF-Pf-2911)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536340(CHEMBL4528019)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM42286(MLS000034309 | cid_654122 | N*2*-(2,5-Dimethoxy-ph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536320(CHEMBL4590509)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536325(CHEMBL4483432)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536321(CHEMBL1622765)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536319(CHEMBL4566039)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536311(CHEMBL4593946)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536322(CHEMBL604514 | GNF-Pf-4167)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536323(CHEMBL4080220)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536326(CHEMBL4534844)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM286984(8-(3-(4-acryloylpiperazin-1-yl)propyl)-6-(2,6-dich...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human TAOK2 preincubated for 15 mins followed by peptide substrate addition measured after 3 hrs by caliper capillary electrophoresis m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536324(CHEMBL4072223)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50402265(CHEMBL2164280 | US8802861, 1)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536334(CHEMBL3715362)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536334(CHEMBL3715362)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536354(CHEMBL1305300)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536312(CHEMBL1458296)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536352(CHEMBL4561613)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536359(CHEMBL4527282)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536361(CHEMBL1613587)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536314(CHEMBL4543595)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536356(CHEMBL4591485)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536345(CHEMBL4519027)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536343(CHEMBL4581349)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536341(CHEMBL4520393)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536336(CHEMBL4536891)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536318(CHEMBL373492)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536357(CHEMBL4553536)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536327(CHEMBL4526718)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536355(CHEMBL4569913)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TAO2(Rat)
University of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50536346(CHEMBL4544171)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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