Compile Data Set for Download or QSAR
Report error Found 477 of ic50 data for complexid = 50006035
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230790(CHEMBL292892)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230779(CHEMBL294686)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230811(CHEMBL293091)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230778(CHEMBL56211)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230771(CHEMBL55510)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230806(CHEMBL294415)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50212829(CHEMBL170944)
Affinity DataIC50: 1.20nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
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LigandPNGBDBM50228195(CHEBI:2719 | Angiotensin Ii)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50011975(4-[2-Butyl-5-(2-carboxy-3-thiophen-2-yl-propenyl)-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50236697(L-alpha-aspartyl-L-arginyl-L-valyl-L-tyrosyl-L-iso...)
Affinity DataIC50: 2nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50281848(L-158827 | 2-Ethyl-5,7-dimethyl-3-{4-[2-(2H-tetraz...)
Affinity DataIC50: 2.30nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50212853(CHEMBL274626)
Affinity DataIC50: 2.40nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230787(CHEMBL54421)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50212825(CHEMBL435855)
Affinity DataIC50: 3nMAssay Description:Competitive inhibition of Angiotensin II receptor binding of radiolabeled AII to rat adrenal glomerulosa tissue by 50%More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230792(CHEMBL56497)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230799(CHEMBL56333)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50228195(CHEBI:2719 | Angiotensin Ii)
Affinity DataIC50: 4nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230774(CHEMBL291955)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230762(CHEMBL56160)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50212843(CHEMBL267809)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230810(CHEMBL299064)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]-AII from the Angiotensin II receptor isolated from the liver of ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230764(CHEMBL299954)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50281823(SC-55634 | 4-Butyl-1-((1R,2R,6S)-2,6-dimethyl-cycl...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230767(CHEMBL56522)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50212845(CHEMBL274668)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50212849(CHEMBL430152)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50212952(CHEMBL46150)
Affinity DataIC50: 5nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50: 5.10nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50046078(5-[4'-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-biph...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50046078(5-[4'-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-biph...)
Affinity DataIC50: 5.60nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50049207(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataIC50: 6nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50212830(CHEMBL171524)
Affinity DataIC50: 6.40nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50281814(1,4-Dibutyl-3-{6-[2-(1H-tetrazol-5-yl)-phenyl]-pyr...)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230796(CHEMBL56690)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50145967(2-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-5-[2-(2H...)
Affinity DataIC50: 6.80nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50049209(5-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-2-[2-(2H...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50049209(5-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-2-[2-(2H...)
Affinity DataIC50: 6.90nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50212844(CHEMBL276689)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230772(CHEMBL59043)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50212954(CHEMBL295114)
Affinity DataIC50: 11nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50226528(CHEMBL284425)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration that gave 50 percent displacement of specific binding of [3H]AII (2 nM) to Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50229469(CHEMBL315094)
Affinity DataIC50: 12nMAssay Description:Inhibition of radioligand [3H]angiotensin II binding to angiotensin II receptor of rat adrenal cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50281822(SC-51895 | 1,4-Dibutyl-3-[2'-(1H-tetrazol-5-yl)-bi...)
Affinity DataIC50: 12nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 13nMAssay Description:Competitive inhibition of Angiotensin II receptor binding of radiolabeled AII to rat adrenal glomerulosa tissue by 50%More data for this Ligand-Target Pair
In DepthDetails

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