Compile Data Set for Download or QSAR
Report error Found 23 of ic50 data for complexid = 50000744
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.70nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
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PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136008(12-(3-hydroxypropyl)-9-isopropoxymethyl-6,7,12,13-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat brain Protein kinase CMore data for this Ligand-Target Pair
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PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50009723(CHEMBL329705 | 2,6-Diamino-hexanoic acid (1-tridec...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229926(CHEMBL319584)
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229931(CHEMBL100713)
Affinity DataIC50: 3.40E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229920(CHEMBL101142)
Affinity DataIC50: 3.60E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229930(CHEMBL97997)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229928(CHEMBL97998)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229921(CHEMBL99372)
Affinity DataIC50: 4.50E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229917(CHEMBL100289)
Affinity DataIC50: 4.50E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229932(CHEMBL97921)
Affinity DataIC50: 4.60E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229922(CHEMBL98968)
Affinity DataIC50: 4.80E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229924(CHEMBL99156)
Affinity DataIC50: 5.10E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229929(CHEMBL98337)
Affinity DataIC50: 5.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM83205((E,2S,3R)-2-azanyloctadec-4-ene-1,3-diol | cid_528...)
Affinity DataIC50: 5.70E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229927(CHEMBL319666)
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229916(CHEMBL322371)
Affinity DataIC50: 7.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229933(CHEMBL98542)
Affinity DataIC50: 7.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229915(CHEMBL101358)
Affinity DataIC50: 9.20E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229925(CHEMBL433408)
Affinity DataIC50: 1.02E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229923(CHEMBL317827)
Affinity DataIC50: 1.54E+5nMAssay Description:Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229919(CHEMBL101538)
Affinity DataIC50: 1.59E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229918(CHEMBL101731)
Affinity DataIC50: 2.99E+5nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed