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- 4BFR: discovery and optimization of pyrimidone indoline amide pi3kbeta inhibitors for the treatment of phosphatase and tensin homologue (pten)-deficient cancers (10.1021/JM401642Q )
- 4V0I: water network determines selectivity for a series of pyrimidone indoline amide pi3kbeta inhibitors over pi3k-delta (10.1021/ACS.JCIM.5B00641 )