574 SMILES Strings for Sodium channel protein type 1/10/11/2/3/4/5/8/9 subunit alpha

Compound Name
SMILES String
Fc1cc(O[C@@H]2CCCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@H]2CCCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3cc(Cl)cc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
CC(=O)N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3cc(Cl)cc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)c(Cl)c1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)c(Cl)c1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)c(F)c1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)c(F)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3c(Cl)cccc3Cl)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(CC3CCCCC3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Cn1nc(cc1CN1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)-c1ccccc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccnnc3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cccc4CNCc34)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(Cl)c(Cl)c3)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccc(Cl)c(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccc(Cl)c(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(F)cc3)C2)cc1F |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)cc1 |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)cc1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccccc3Cl)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccccc3Cl)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccccc3Cl)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cccc(Cl)c3)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(Cc3cccc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3cccc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(Cl)cc3Cl)C2)cc1F |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccc(Cl)cc3Cl)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(Cc3ccc(Cl)cc3Cl)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)cc1 |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)cc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(F)cc3C(F)(F)F)C2)cc1F |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)c(c1)C(F)(F)F |r|
Fc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)c(c1)C(F)(F)F |r|
Fc1ccc(cc1)N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1 |r|
Fc1ccc(cc1)N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1 |r|
Fc1ccc(N2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)c(Cl)c1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(C2)c2cc(Cl)cc(Cl)c2)cc1F |r|
Fc1cc(O[C@H]2CCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCN(Cc3ccccc3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(OCC2CC3CCC(C2)N3Cc2ccccc2Cl)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2CC3CCC(C2)N3Cc2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
Fc1cc(OCC2CC3CCC(C2)N3C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
C[C@H](N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H]1CC[C@H](CN1Cc1ccc(F)cc1Cl)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
Fc1cc(CN2CCC[C@@H](C2)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(CN2CCC[C@@H](C2)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(CN2CCC[C@H](C2)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(CN2CCC[C@H](C2)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(CN2CCC(CC2)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
C[Si](C)(C)CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
COCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
FC(F)S(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
Fc1cc(OCC2CN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)CCC(F)(F)F)C1CC1
Fc1cc(OCC2CN(C2)C(c2ccccc2)c2ccccc2)c(cc1C(=O)NS(=O)(=O)CC1CC1)C1CC1
CCCCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CN(Cc3ccccc3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CN(C2)C(c2ccccc2)c2ccccc2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CN(C1)C(c1ccccc1)c1ccccc1
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C)CN(C2)C(c2ccccc2)c2ccccc2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)C(c1ccccc1)c1ccccc1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CN(C1)C(c1ccccc1)c1ccccc1
CC(C)(C)OC(=O)N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3cccc(F)c3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3ccccc3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3cc(F)cc(Cl)c3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3ccc(c(F)c3)C(F)(F)F)C2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CN(Cc2cc(Cl)cc(Cl)c2)C1
CC(C)(C)OC(=O)N1CCC(COc2cc(F)c(cc2Cl)C(=O)NS(C)(=O)=O)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2ccccc2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccc(Cl)c(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2cccnc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2cccnc2)cc1F |r|
CC(C)Oc1ncc(CN2CC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)C2)cc1Cl
C[C@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1ccccc1 |r|
C[C@@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1ccccc1 |r|
CC(N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(F)cc(F)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccccc3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cccc(F)c3)CC2)cc1F
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(F)cc(F)c1
COCC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
COCC(N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cccc(Cl)c3)CC2)cc1F
Cc1ccc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)cc1
COc1ccc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccc(cc2)S(C)(=O)=O)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccc(cc2)S(C)(=O)=O)cc1F |r|
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
CC(N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](c1cc(cc(c1)Cl)Cl)N2CCC(CC2)COc3cc(c(cc3C4CC4)C(=O)NS(=O)(=O)C)F
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(C)c2cc(Cl)cc(Cl)c2)cc1F
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)cc3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)cc3Cl)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)cc3Cl)CC2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2cc(ccc2C(F)(F)F)C(F)(F)F)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2cccc(c2)C#N)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2cccc(c2)C#N)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccc(cc2)C#N)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccc(cc2)C#N)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccc(OC(F)(F)F)cc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccc(OC(F)(F)F)cc2)cc1F |r|
CC(C)Oc1ncc(cc1Cl)[C@@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1ccccc1 |r|
CC(C)Oc1ncc(cc1Cl)[C@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1ccccc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CCC(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccccn2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccccn2)cc1F |r|
C[C@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2cc(Cl)ccc2C(F)(F)F)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2cc(Cl)cc(Cl)c2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccccc2F)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccccc2F)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(cc3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccccc3F)CC2)cc1F
CC(C)Oc1ncc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)cc1Cl
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)S(=O)(=O)c2ccccc2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2ccc(F)cc2C(F)(F)F)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccc(cc2)C(F)(F)F)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3cc(Cl)cc(Cl)c3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(Cc3ccc(Cl)c(F)c3)C2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(=O)c2cc(Cl)cc(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)c(F)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2cc(Cl)cc(c2)C(F)(F)F)CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2cc(cc(Cl)c2F)C(F)(F)F)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccc(F)cc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccc(F)cc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)c(Cl)c3)CC2)cc1F
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cccc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccccc3C#N)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccccc2Cl)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccccc2Cl)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@@H](c2ccccc2)c2ccncc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)[C@H](c2ccccc2)c2ccncc2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2cccc(F)c2)cc1F
CCC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
CC(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(OC(F)(F)F)cc1
CC(N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1ccc(OC(F)(F)F)cc1
CCC(N1CC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccccc3C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)c(F)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)cc3)CC2)cc1F
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(F)cc(c1)C(F)(F)F |r|
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(F)cc(c1)C(F)(F)F |r|
COC[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C2(COC2)c2cc(Cl)cc(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)C2(COC2)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(CC2)C2(COC2)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C2(COC2)c2cc(Cl)cc(Cl)c2)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(CC1)C1(COC1)c1cc(Cl)cc(Cl)c1
CC(C)N(C(C)C)C(=O)CN1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
CC(C)N(C(C)C)C(=O)CN1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)c(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)c(Cl)c1 |r|
COc1ccc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)cc1Cl
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)cc1F
C[C@@H](N1CC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)c(c1)C(F)(F)F |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)c(c1)C(F)(F)F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)c(c3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cnc(OCC(F)(F)F)c(Cl)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccccc3Cl)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC(F)(F)C(F)F)CC2)cc1F
Fc1cc(OCC2CCN(CCC(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(CCC(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2cccc(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2cccc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2ccccc2)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2ccccc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H]2[C@@H](O)Cc3ccccc23)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H]2[C@H](O)Cc3ccccc23)cc1F |r|
COC[C@](C)(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC[C@@](C)(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@](C)(COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@](C)(COC)c2cc(Cl)cc(Cl)c2)cc1F |r|
COC(C)(C)[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
COC(C)(C)[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](c2cc(Cl)cc(Cl)c2)C(C)(C)OC)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](c2cc(Cl)cc(Cl)c2)C(C)(C)OC)cc1F |r|
CC(C)(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(C)(C)c2cc(Cl)cc(Cl)c2)cc1F
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)cc3Cl)CC2)cc1F
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(c3)C(F)(F)F)CC2)cc1F
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(c(Cl)c3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(C2)C(=O)c2cc(Cl)cc(Cl)c2)cc1F |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccccc1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccccc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](C(F)F)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](C(F)F)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](C(F)F)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](C(F)F)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)cc(c3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)c(c3)C(F)(F)F)CC2)cc1F
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(F)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(F)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2ccc(Cl)c(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2ccc(Cl)c(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@@H]2CCN(Cc3cc(Cl)cc(Cl)c3)C(=O)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2CCN(Cc3cc(Cl)cc(Cl)c3)C(=O)C2)cc1F |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1F |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1F |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
CC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3F)CC2)cc1F
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)cc1Cl |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)cc1Cl |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](C)c2ccc(F)cc2Cl)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](C)c2ccc(F)cc2Cl)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(c(F)c3)C(F)(F)F)CC2)cc1F
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(OC(F)(F)F)cc1 |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(OC(F)(F)F)cc1 |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cccc(F)c1 |r|
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cccc(F)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC3(CC3)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2cc(Cl)cc(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2ccccc2C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2ccccc2C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(=O)c2ccc(Cl)cc2Cl)cc1F
Fc1cc(OCC2CCN(CC2)C(=O)c2ccc(Cl)cc2Cl)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)cc1F
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cccc(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cccc(Cl)c1 |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)c(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](CO)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](CO)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)cc(Cl)c3)CC2)cc1F
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
C[C@@H](N1CCC(C)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
COC[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
COC[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(Cl)cc1Cl |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](C)c2ccc(Cl)cc2Cl)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](C)c2ccc(Cl)cc2Cl)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@H](COC)c2ccc(Cl)cc2Cl)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)[C@@H](COC)c2ccc(Cl)cc2Cl)cc1F |r|
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CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2cc(Cl)cc(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2ccccc2Cl)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2cccc(Cl)c2)cc1F
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C[C@@H](N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)c1ccc(F)cc1Cl |r|
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CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2cc(Cl)cc(Cl)c2)C(F)(F)F)cc1F
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CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2ccc(F)c(Cl)c2)C(F)(F)F)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)cc1F
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)cc1F
Fc1cc(OCCC2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
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Fc1cc(OCC2CCN(Cc3cc(cc(n3)C3CC3)C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
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C[C@@H]1CC[C@H](CN1Cc1ccc(F)cc1Cl)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1 |r|
C[C@H]1CC[C@H](CN1Cc1ccc(F)cc1Cl)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
C[C@H]1CC[C@H](CN1Cc1ccc(F)cc1Cl)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)N1CCC1 |r|
C[C@H]1CC[C@H](CN1Cc1ccc(F)cc1Cl)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(CC3(CCCC3)C(F)(F)F)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(CC3(CCC3)C(F)(F)F)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC3(CCCC3)C(F)(F)F)CC2)cc1F
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C[C@H]1[C@@H](CCCN1Cc1cc(Cl)cc(Cl)c1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@@H]2CCCN(Cc3ccc(F)cc3Cl)C2)cc1F |r|
Fc1ccc(CN2CCC[C@@H](COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)N3CCC3)C2)c(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@@H]2CCCN(Cc3cc(Cl)cc(Cl)c3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2CCCN(Cc3ccc(F)cc3Cl)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2CCCN(Cc3cc(Cl)cc(Cl)c3)C2)cc1F |r|
C[C@@H](N1CCC[C@H](COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC[C@H](COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)C1)c1cc(Cl)cc(Cl)c1 |r|
Fc1ccc(CN2CCC[C@H](COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)N3CCC3)C2)c(Cl)c1 |r|
Fc1ccc(CN2CCC[C@H](COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)C2)c(Cl)c1 |r|
C[C@@H]1CC[C@@H](COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CN1Cc1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1C[C@H](COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC[C@H]1C)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1C[C@H](COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC[C@H]1C)c1cc(Cl)cc(Cl)c1 |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@@H]2CC[C@@H](C)N(C2)[C@@H](C)c2cc(Cl)cc(Cl)c2)cc1F |r|
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@@H]2CC[C@@H](C)N(C2)[C@H](C)c2cc(Cl)cc(Cl)c2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)cc1F
Fc1cc(OCC2(F)CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)cc1F
C[C@H](N1CCC(F)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@H](N1CCC(F)(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@@H](N1CCC(F)(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2cccc(Cl)c2)c2cccc(Cl)c2)cc1F
C[C@@H](N1[C@H]2CC[C@@H]1C[C@@H](COc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)C2)c1cc(Cl)cc(Cl)c1 |r,THB:1:2:7.8.28:4.5|
Cc1nc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CC2)cs1
CC(C)c1nc(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CC2)cs1
CC(C)Nc1ccc(F)cc1CN1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
Cn1nc(c(CN2CCC(COc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CC2)c1Cl)C(F)(F)F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(CF)c2cc(Cl)cc(Cl)c2)cc1F
C[C@H](N1CCC(COc2cc(F)c(cc2C)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2ccccc2Cl)c2ccccc2Cl)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)cc1F
Fc1ccc(cc1)C(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1ccc(F)cc1
Fc1cc(OCC2CCN(Cc3ncccc3C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ncccc3C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2cc(Cl)c(Br)cc2F)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2cc(Cl)c(Br)cc2F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(Br)c(F)c2)cc1F
Fc1cc(ccc1Br)S(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccccc2C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccccc2C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(cc2)C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccc(cc2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2cccc(c2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)C2CCOCC2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)C2CCOCC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2)cc1F
Fc1cc(cc(F)c1F)S(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(F)c(Cl)c2)cc1F
Fc1ccc(cc1Cl)S(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Cc1cc(F)ccc1S(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1
Cc1cc(F)ccc1S(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc3ccccc3c2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccc3ccccc3c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)c2ccc(Br)c(Cl)c2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)c2ccc(Br)c(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(=O)(=O)C2COC2)cc1F
Fc1cc(OCC2CCN(CC2)S(=O)(=O)C2COC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)S(C)(=O)=O)cc1F
Fc1cc(OC[C@H]2C[C@@H]3CC[C@H](C2)N3Cc2cc(cc(Cl)c2F)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,THB:14:13:12.6.7:9.10|
Fc1cc(OC[C@H]2C[C@@H]3CC[C@H](C2)N3Cc2cc(ccc2Cl)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,THB:14:13:12.6.7:9.10|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2C[C@@H]3CC[C@H](C2)N3Cc2cc(cc(Cl)c2F)C(F)(F)F)cc1F |r,THB:24:23:22.16.17:19.20|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OC[C@H]2C[C@@H]3CC[C@H](C2)N3Cc2cc(ccc2Cl)C(F)(F)F)cc1F |r,THB:24:23:22.16.17:19.20|
Fc1cc(OCC2CCN(CC2)C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(CC2)C(c2cccc(Cl)c2)c2cccc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
C[C@H](N1CCC(COc2cc(F)c(cc2Cl)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2Cl)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCC(COc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)C2CC2)CC1)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)cc1F
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)C1CC1
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)c(Cl)cc1C(=O)NS(=O)(=O)N1CCC1
Fc1cc(OCC2CCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C#N
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3nc(no3)-c3ccccc3Cl)CC2)cc1F
Fc1cc(OCC2CCN(CC2)C(c2ccccc2)c2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2ccccc2)c2cc(Cl)cc(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Br)cc3Cl)CC2)cc1F
Fc1cc(OCC2CCN(Cc3ccc(Br)cc3Cl)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(cc3Cl)C3CC3)CC2)cc1F
Fc1cc(OCC2CCN(Cc3ccc(cc3Cl)C3CC3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(Cc3ccc(cc3Cl)C3CC3)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)C(c2ccc(F)cc2)c2ccc(F)cc2)cc1F
Fc1ccc(cc1)C(N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)N2CCC2)CC1)c1ccc(F)cc1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CN(C1)C(c1ccccc1)c1cc(Cl)cc(Cl)c1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)C(c1ccccc1)c1cc(Cl)cc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cc(Cl)cc(OC(F)(F)F)c3)C2)cc1F |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(C)c1 |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(Cl)c1 |r|
CC(C)(C)c1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)cc1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(cc3)-c3ccccc3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cc(Cl)ccc3O)C2)cc1F |r|
CCOc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(OCC)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc4OCCOc4c3)C2)cc1F |r|
COc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)cc1OC |r|
Cc1cc(F)ccc1CN1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
COc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(c(Cl)c3)C(F)(F)F)C2)cc1F |r|
COc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c(C)c1 |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)cc1Cl |r|
Cc1cc(C)cc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cccc(OC(F)(F)F)c3)C2)cc1F |r|
COc1cc(OC(F)(F)F)ccc1CN1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
Cc1ccc(CN2CCC[C@H](C2)Oc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)cc1C |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cc(Cl)cc(Cl)c3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccc(cc3Cl)S(C)(=O)=O)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3ccccc3-c3ccccc3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(Cc3cccc(c3)-c3ccccc3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(CC3CCC4(CCC4)CC3)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2CN(Cc3ccc(F)cc3Cl)CC(F)(F)C2)cc1F |r|
CS(=O)(=O)NC(=O)c1cc(Cl)c(O[C@H]2CN(Cc3ccc(F)cc3Cl)CC(F)(F)C2)cc1F |r|
COC[C@@H](N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CC3CCC(C2)N3Cc2cc(Cl)cc(Cl)c2)cc1F
C[C@H](N1C[C@@H]2C[C@@H](Oc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)[C@H]1C2)c1ccc(F)cc1Cl |r|
C[C@@H](N1C[C@@H]2C[C@@H](Oc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)[C@H]1C2)c1ccc(F)cc1Cl |r|
C[C@@H](N1C[C@@H](CC(C)(C)C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O)c1ccc(F)cc1Cl |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)c(Cl)cc3Cl)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)c(F)c(Cl)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)c(F)cc3F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)c(F)c(Cl)c3)CC2)cc1F
Fc1cc(OCC2(F)CCN(Cc3cc(Cl)ccc3C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCO[C@H](Cc3ccc(Cl)c(Cl)c3)C2)cc1F |r|
Fc1cc(CN2CCO[C@H](Cc3ccc(Cl)c(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1cc(CN2CCO[C@H](Cc3ccc(Cl)c(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCO[C@@H](Cc3ccc(Cl)c(Cl)c3)C2)cc1F |r|
Fc1cc(CN2CCO[C@@H](Cc3ccc(Cl)c(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCO[C@H](Cc3cc(Cl)cc(Cl)c3)C2)cc1F |r|
Fc1cc(CN2CCO[C@H](Cc3cc(Cl)cc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(CN2CCO[C@H](Cc3cc(Cl)cc(Cl)c3)C2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCO[C@H](Cc3ccc(F)cc3Cl)C2)cc1F |r|
Fc1ccc(C[C@@H]2CN(Cc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CCO2)c(Cl)c1 |r|
Fc1ccc(C[C@@H]2CN(Cc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)N3CCC3)CCO2)c(Cl)c1 |r|
CC1(C)CO[C@H](Cc2cc(Cl)cc(Cl)c2)CN1Cc1cc(F)c(cc1C1CC1)C(=O)NS(C)(=O)=O |r|
Fc1cc(CN2[C@H]3CC[C@@H]2CC(C3)Oc2cc(cc(Cl)c2F)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,TLB:4:5:7.8:10.12.11|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2[C@H]3CC[C@@H]2CC(C3)Oc2cc(cc(Cl)c2F)C(F)(F)F)cc1F |r,TLB:14:15:17.18:20.22.21|
CC1(CCN(Cc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)Oc1cc(c(Cl)cn1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|
Fc1cc(CN2CCC(CC2)Oc2ncc(Br)cc2Cl)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(CN2CCC(CC2)Oc2ncc(cc2Cl)C2CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(CN2[C@H]3CC[C@@H]2CC(C3)Oc2cc(Cl)cc(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,TLB:4:5:7.8:10.12.11|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(cn2)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(cn2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)OCc2ccc(F)cc2Cl)cc1F
Fc1ccc(COC2CCN(Cc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)N3CCC3)CC2)c(Cl)c1
Fc1ccc(COC2CCN(Cc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CC2)c(Cl)c1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1ncc(cc1Cl)C(F)(F)F
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C)CN(C2)c2ncc(cc2Cl)C(F)(F)F)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1ncc(Cl)cc1F
CCS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(C)CN(C2)c2ncc(Cl)cc2F)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1ccc(Cl)c(n1)C(F)(F)F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1cc(Cl)c(cn1)C(F)(F)F |$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1cc(Cl)ncc1C(F)(F)F |$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1ccc(cn1)C(F)(F)F |$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;$|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CN(C1)c1ccncc1C(F)(F)F |$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;$|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@@H]2CCCN(C2)c2ccc(cn2)C(F)(F)F)cc1F |r|
Fc1cc(O[C@@H]2CCCN(C2)c2ccc(cn2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2ccccn2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r|
Fc1cc(O[C@@H]2CCCN(C2)c2ccccn2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1 |r|
Fc1ccc(nc1)N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1 |r|
CC(C)(N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(=O)NS(=O)(=O)C1CC1)c1cc(Cl)cc(Cl)c1 |r|
Fc1cc(CN2[C@H]3CC[C@@H]2CC(C3)Oc2cc(Cl)cc(OC(F)(F)F)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1 |r,TLB:4:5:7.8:10.12.11|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccccc2C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccccc2C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(cc2)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(cc2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2cccc(c2)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2cccc(c2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(Cl)cc2)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(Cl)cc2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(F)cc2Cl)cc1F
OS(O)(NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(F)cc2Cl)cc1F)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(F)cc2)cc1F
Fc1ccc(OC2CCN(Cc3cc(F)c(cc3C3CC3)C(=O)NS(=O)(=O)C3CC3)CC2)cc1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(Cl)c(Cl)c2)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(Cl)c(Cl)c2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(Cl)cc2Cl)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(Cl)cc2Cl)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)N(S)C(=O)c1cc(C2CC2)c(CN2CCC(CF)(CC2)c2ccc(F)cc2)cc1F
FCC1(CCN(Cc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1ccc(F)cc1
COCC1(CCN(Cc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1ccc(F)cc1
COCC1(CCN(Cc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CC1)c1ccc(F)cc1
CS(=O)(=O)N(S)C(=O)c1cc(C2CC2)c(CN2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)cc1F
Fc1cc(CN2CCN(Cc3cc(Cl)cc(Cl)c3)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(Cl)c(c2)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2ccc(Cl)c(c2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2cc(c(Cl)cn2)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2cc(c(Cl)cn2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ncc(cc2Cl)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2ncc(cc2Cl)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CC1(COc2cc(F)c(cc2C2CC2)C(N)=O)CN(C1)c1cc(c(Cl)cn1)C(F)(F)F
NC(=O)c1cc(C2CC2)c(CN2CCN(CC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1F
NC(=O)c1cc(C2CC2)c(CN2[C@H]3CC[C@@H]2C[C@H](C3)Oc2cc(Cl)cc(Cl)c2)cc1F |r,THB:10:11:16.18.17:13.14|
CC(C)(N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(N)=O)c1cccc(Cl)c1 |r|
NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Sc2cc(Cl)cc(Cl)c2)cc1F
NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1F
NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)S(=O)c2cc(Cl)cc(Cl)c2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2cc(cc(Cl)c2F)C(F)(F)F)cc1F
Fc1cc(CN2CCC(CC2)Oc2cc(cc(Cl)c2F)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CC(C)(C)N1CCC[C@H](C1)Oc1cc(F)c(cc1C1CC1)C(N)=O |r|
CC(N1CCN(Cc2cc(F)c(cc2C2CC2)C(N)=O)CC1)c1cc(Cl)cc(Cl)c1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)c2cc(c(Cl)cn2)C(F)(F)F)cc1F
Fc1cc(OCC2CN(C2)c2cc(c(Cl)cn2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
NC(=O)c1cc(C2CC2)c(CN2CC(C2)Oc2cc(Cl)cc(Cl)c2)cc1F
NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2ccc(Cl)cc2Cl)cc1F
NC(=O)c1cc(C2CC2)c(CN2CCC(CC2)Oc2cc(Cl)cc(OC(F)(F)F)c2)cc1F
NC(=O)c1cc(C2CC2)c(CN2[C@H]3CC[C@@H]2C[C@@H](C3)Oc2cc(c(Cl)cn2)C(F)(F)F)cc1F |r,THB:10:11:16.18.17:13.14|
NC(=O)c1cc(C2CC2)c(CN2[C@H]3CC[C@@H]2C[C@@H](C3)Oc2ncc(cc2Cl)C(F)(F)F)cc1F |r,THB:10:11:16.18.17:13.14|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2cc(c(Cl)cn2)C(F)(F)F)cc1F
Fc1cc(OCC2CCN(CC2)c2cc(c(Cl)cn2)C(F)(F)F)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(CC1)c1cc(c(Cl)cn1)C(F)(F)F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(=O)(=O)C2CC2)CCN(CC1)c1cc(c(Cl)cn1)C(F)(F)F
NC(=O)c1cc(C2CC2)c(CN2C[C@@H]3C[C@H]2CN3S(=O)(=O)c2cc(Cl)cc(Cl)c2)cc1F |r|
NC(=O)c1cc(C2CC2)c(CN2[C@H]3CC[C@@H]2C[C@@H](C3)Oc2cc(Cl)cc(OC(F)(F)F)c2)cc1F |r,THB:10:11:18.17.16:13.14|
CC1(C)CN(Cc2cc(F)c(cc2C2CC2)C(N)=O)CCC1Oc1cc(c(Cl)cn1)C(F)(F)F
C[C@@H](N1C[C@@H]2C[C@H]1CN2Cc1cc(F)c(cc1C1CC1)C(N)=O)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1C[C@@H]2C[C@H]1CN2Cc1cc(F)c(cc1C1CC1)C(N)=O)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCN(Cc2cc(F)c(cc2C2CC2)C(N)=O)C[C@@H]1C)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCN(Cc2cc(F)c(cc2C2CC2)C(N)=O)C[C@@H]1C)c1cc(Cl)cc(Cl)c1 |r|
C[C@@H](N1CCN(Cc2cc(F)c(cc2C2CC2)C(N)=O)C[C@H]1C)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCN(Cc2cc(F)c(cc2C2CC2)C(N)=O)C[C@H]1C)c1cc(Cl)cc(Cl)c1 |r|
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(O[C@H]2CCCN(Cc3ccc(F)cc3Cl)C2)cc1F |r|
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(CC1)C(c1ccccc1)c1ccccc1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(Cc2ccc(Cl)c(Cl)c2)CC1
COc1cccc(CN2CCC(C)(COc3cc(F)c(cc3C3CC3)C(=O)NS(C)(=O)=O)CC2)n1
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(CC1)C(=O)c1cc(Cl)c(Cl)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CCN(CC1)C(=O)c1cc(Cl)ccc1Cl
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Cl)cc3C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(ccc3Cl)C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)cc1F
Fc1cc(OCC2CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)C1CC1)C1CC1
Fc1cc(OCC2CCN(Cc3cc(cc(Cl)c3Cl)C(F)(F)F)CC2)c(cc1C(=O)NS(=O)(=O)N1CCC1)C1CC1
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Br)cc3C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)cc3C(F)(F)F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Br)c(Cl)c3)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(F)c(Br)cc3F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(Br)cc3F)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(c3)C#N)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3ccc(F)c(c3)C#N)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CCN(CC2)c2cccc(n2)C(F)(F)F)cc1F
CC1(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CN(Cc2cc(cc(Cl)c2F)C(F)(F)F)C1
COC(=O)c1cc(C2CC2)c(OCC2CCN(Cc3cc(Cl)cc(Cl)c3C#N)CC2)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(CCN(Cc3cc(cc(Cl)c3F)C(F)(F)F)CC2)C#N)cc1F
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2(F)CCN(Cc3cc(cc(n3)C3CC3)C(F)(F)F)CC2)cc1F
C[C@@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)(CC1)C#N)c1cc(Cl)cc(Cl)c1 |r|
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)(CC1)C#N)c1cc(Cl)cc(Cl)c1 |r|