5231 SMILES Strings for P2X purinoceptor 7

Compound Name
SMILES String
FC(F)(F)c1cccc(C(=O)N2C3CCCC2c2nnc(-c4ncccn4)n2C3)c1Cl
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ncccn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.15.14|
FC(F)(F)c1cccc(C(=O)N2[C@@H]3CCC[C@H]2c2nnc(-c4ncccn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.15.14|
Fc1ccc(cc1)-c1nnc2C3CCCC(Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F
Fc1ccc(cc1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
Fc1ccc(cc1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
FC(F)(F)c1cccc(C(=O)N2C3CCCC2c2nnc(-c4cscn4)n2C3)c1Cl
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4cscn4)n2C3)c1Cl |r,THB:9:11:17.26.27:13.15.14|
FC(F)(F)c1cccc(C(=O)N2[C@@H]3CCC[C@H]2c2nnc(-c4cscn4)n2C3)c1Cl |r,THB:9:11:17.26.27:13.15.14|
Fc1ccc(nc1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
Fc1ccc(nc1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4cccnc4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.15.14|
Fc1cnc(nc1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
Fc1cnc(nc1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1ccc(Cl)cc1Cl |r,THB:19:18:10.17.16:14.12.13|
Cc1cccc(n1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
Cc1cccc(n1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.12.13|
COc1ccnc(c1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:11.18.17:15.13.14|
COc1ccnc(c1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:11.18.17:15.13.14|
FC(F)(F)c1cccc(C(=O)N2[C@@H]3CCC[C@H]2c2nnc(-c4ccc(Cl)cn4)n2C3)c1Cl |r,THB:9:11:17.28.29:13.14.15|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccccn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.14.15|
FC(F)(F)c1nccc(C(=O)N2[C@@H]3CCC[C@H]2c2nnc(-c4cccs4)n2C3)c1Cl |r,THB:9:11:17.26.27:13.14.15|
Cc1ccc(s1)-c1nnc2[C@@H]3CCC[C@H](Cn12)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:18:17:9.16.15:13.12.11|
Fc1ccc(cc1)-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:18:17:10.16.15:13.12|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccccn4)n2C3)c1Cl |r,THB:9:11:16.26.27:13.14|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cnccn4)n2C3)c1Cl |r,THB:9:11:16.26.27:13.14|
Fc1ccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccccn4)n2C3)c(Cl)c1C(F)(F)F |r,THB:5:7:12.22.23:9.10|
Cc1c(cccc1C(F)(F)F)C(=O)N1[C@H]2CC[C@@H]1c1nnc(-c3ccccn3)n1C2 |r,THB:11:13:18.28.29:15.16|
Fc1ccc(nc1)-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:18:17:10.16.15:12.13|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ncccn4)n2C3)c1Cl |r,THB:9:11:16.26.27:14.13|
Fc1ccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cnccn4)n2C3)c(Cl)c1Cl |r,THB:5:7:12.22.23:10.9|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cccnc4)n2C3)c1Cl |r,THB:9:11:16.26.27:14.13|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cscn4)n2C3)c1Cl |r,TLB:9:11:14.13:16.26.25|
Fc1cnc(nc1)-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,TLB:18:17:12.13:10.15.16|
Cc1cc([nH]n1)-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,TLB:17:16:11.12:9.14.15|
Fc1ccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cscn4)n2C3)c(Cl)c1C(F)(F)F |r,TLB:5:7:10.9:12.22.21|
Cc1c(cccc1C(F)(F)F)C(=O)N1[C@H]2CC[C@@H]1c1nnc(-c3cscn3)n1C2 |r,TLB:11:13:16.15:18.28.27|
Fc1c(Cl)ccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cscn4)n2C3)c1Cl |r,TLB:7:9:12.11:14.24.23|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccc(Cl)s4)n2C3)c1Cl |r,TLB:9:11:14.13:16.27.26|
Cc1nc(cs1)-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,TLB:17:16:11.12:9.14.15|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cncs4)n2C3)c1Cl |r,TLB:9:11:14.13:16.26.25|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccsc4)n2C3)c1Cl |r,TLB:9:11:14.13:16.26.25|
Cc1ncsc1-c1nnc2[C@H]3CC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:17:16:9.15.14:12.11|
FC(F)(F)c1nccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccc(Cl)s4)n2C3)c1Cl |r,THB:9:11:16.26.27:13.14|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4cccs4)n2C3)c1Cl |r,THB:9:11:16.25.26:13.14|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CC[C@@H]2c2nnc(-c4ccc[nH]4)n2C3)c1Cl |r,THB:9:11:16.25.26:13.14|
Cc1nc(ccc1F)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:11.18.17:15.14.13|
Cc1ccnc(c1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.17.16:14.13.12|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4cccnn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.14.15|
FC(F)(F)c1ccnc(c1)-c1nnc2[C@H]3CCC[C@@H](Cn12)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:22:21:13.20.19:17.16.15|
FC(F)(F)c1cccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccncn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.14.15|
Fc1c(ccnc1C(F)(F)F)C(=O)N1[C@H]2CCC[C@@H]1c1nnc(-c3ccccn3)n1C2 |r,THB:11:13:19.29.30:15.16.17|
FC(F)(F)c1nccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccccn4)n2C3)c1Cl |r,THB:9:11:17.27.28:13.14.15|
Fc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccccn4)n2C3)c(Cl)c1C(F)(F)F |r,THB:5:7:13.23.24:9.10.11|
Cc1c(cccc1C(F)(F)F)C(=O)N1[C@H]2CCC[C@@H]1c1nnc(-c3ccccn3)n1C2 |r,THB:11:13:19.29.30:15.16.17|
Fc1c(Cl)ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccccn4)n2C3)c1Cl |r,THB:7:9:15.25.26:11.12.13|
Fc1ccc(C(=O)N2[C@H]3CCC[C@@H]2c2nnc(-c4ccccn4)n2C3)c(Cl)c1Cl |r,THB:5:7:13.23.24:9.10.11|
Fc1ccc(cc1)-c1nnc2C(=O)N(Cc3cccc(c3Cl)C(F)(F)F)CCn12
Clc1cccc(CN2CCn3c(nnc3-c3cnccn3)C2=O)c1Cl
FC(F)(F)c1cccc(CN2CCn3c(nnc3-c3cnccn3)C2=O)c1Cl
CC(N1CCn2c(nnc2-c2cnccn2)C1=O)c1cccc(c1Cl)C(F)(F)F
Clc1cccc(Cl)c1CN1CCn2c(nnc2-c2cnccn2)C1=O
Fc1cccc(CN2CCn3c(nnc3-c3cnccn3)C2=O)c1F
CS(=O)(=O)c1cc(Cl)ccc1CN1CCn2c(nnc2-c2cnccn2)C1=O
Clc1cccc(CN2CCn3c(nnc3-c3ccccn3)C2=O)c1Cl
FC(F)(F)c1cccc(CN2CCn3c(nnc3-c3ccccn3)C2=O)c1Cl
CC1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(Cl)c1Cl
C[C@@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(Cl)c1Cl |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(Cl)c1Cl |r|
CC1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F
C[C@@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cc2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ccccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnc(C)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1ncco1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cocn1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cnco1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1ccn(C)n1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cnn(C)c1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cn[nH]c1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cc(C)[nH]n1 |r|
C[C@H]1Cn2c(nnc2-c2ncccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cc[nH]n1 |r|
C[C@H]1Cn2c(nnc2-c2cccnc2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1nccs1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cscn1 |r|
C[C@H]1Cn2c(nnc2-c2ccncn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ncc(F)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cc(CO)ccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1csc(C)n1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cncs1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1csc(n1)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1sc(C)nc1C |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1scnc1C |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1ccon1 |r|
C[C@H]1Cn2c(nnc2-c2ncc(Br)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cccnn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cncc(F)c2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cccc(C)n2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ccncc2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cccnc2C)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCC1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CC1 |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCCCC1 |r|
C[C@H]1Cn2c(nnc2-c2cncc(Cl)c2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCOCC1 |r|
C[C@H]1Cn2c(nnc2-c2nccc(n2)C(F)(F)F)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cccc(n2)C(F)(F)F)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2ccc(Cl)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cncc(C)c2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCN(C1)C(=O)OC(C)(C)C |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCCN(C1)C(=O)OC(C)(C)C |r|
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)C1CCCNC1 |r|
FC(F)(F)c1cccc(CN2C(Cn3c(nnc3-c3cnccn3)C2=O)C2CC2)c1Cl
FC(F)(F)c1cccc(CN2[C@@H](Cn3c(nnc3-c3cnccn3)C2=O)C2CC2)c1Cl |r|
FC(F)(F)c1cccc(CN2[C@H](Cn3c(nnc3-c3cnccn3)C2=O)C2CC2)c1Cl |r|
FC(F)(F)c1cccc(CN2C(Cn3c(nnc3-c3ncccn3)C2=O)C2CC2)c1Cl
FC(F)(F)c1cccc(CN2[C@@H](Cn3c(nnc3-c3ncccn3)C2=O)C2CC2)c1Cl |r|
FC(F)(F)c1cccc(CN2[C@H](Cn3c(nnc3-c3ncccn3)C2=O)C2CC2)c1Cl |r|
FC(F)(F)c1cccc(CN2C(Cn3c(nnc3-c3cccnc3)C2=O)C2CC2)c1Cl
FC(F)(F)c1cccc(CN2C(Cn3c(nnc3C2=O)-c2cc[nH]n2)C2CC2)c1Cl
Fc1ccc(nc1)-c1nnc2C(=O)N(Cc3cccc(c3Cl)C(F)(F)F)C(Cn12)C1CC1
Fc1cnc(nc1)-c1nnc2C(=O)N(Cc3cccc(c3Cl)C(F)(F)F)C(Cn12)C1CC1
CC[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
CC[C@H]1Cn2c(nnc2-c2ncccn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
CC[C@H]1Cn2c(nnc2-c2cccnc2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
CC[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1cc[nH]n1 |r|
CC[C@H]1Cn2c(nnc2-c2ncc(F)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
CC[C@H]1Cn2c(nnc2-c2ccc(F)cn2)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccc(F)cc1Cl |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccccc1 |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccccc1Cl |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccc(Cl)cc1S(C)(=O)=O |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccccc1OC(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cc2OCOc2cc1Cl |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1C)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1c(Cl)cccc1Cl |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1c(C)cccc1C |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cccc(c1)C(F)(F)F |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1ccccc1[N+]([O-])=O |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cc(ccc1Cl)[N+]([O-])=O |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)C(=O)N1Cc1cc(N)ccc1Cl |r|
CC(N1[C@@H](C)Cn2c(nnc2-c2cnccn2)C1=O)c1ccccc1 |r|
CC(N1[C@@H](C)Cn2c(nnc2-c2cnccn2)C1=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H](N1[C@@H](C)Cn2c(nnc2-c2cnccn2)C1=O)c1ccccc1 |r|
C[C@H](N1[C@@H](C)Cn2c(nnc2-c2cnccn2)C1=O)c1ccccc1 |r|
O=C1NCCn2c1nnc2-c1cnccn1
C[C@H]1CNC(=O)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
FC(F)(F)c1cccc(CN2C(CNC(=O)C2=O)C2CC2)c1Cl
CC[C@H]1CNC(=S)C(=O)N1Cc1cccc(c1Cl)C(F)(F)F |r|
CC(Br)c1cccc(c1Cl)C(F)(F)F
NNC(=O)c1ncccn1
NNC(=O)c1ccncn1
NNC(=O)c1cccnn1
Cc1cccc(n1)C(=O)NN
Cc1ncccc1C(=O)NN
NNC(=O)c1cccc(n1)C(F)(F)F
C[C@H]1Cn2c(nnc2C(=O)N1Cc1cccc(c1Cl)C(F)(F)F)-c1csc(n1)C(F)(F)F
C[C@H]1Cn2c(nnc2-c2cnccn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2cnccn2)-c2nnc(-c3cccc(Cl)c3Cl)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cc2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1cc[nH]n1 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1cocn1 |r|
C[C@H]1Cn2c(nnc2-c2ncccn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1nccs1 |r|
C[C@H]1Cn2cnnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2cccnn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1scnc1C |r|
C[C@H]1Cn2c(nnc2-c2cnc(C)cn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccncn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1cn[nH]c1 |r|
COc1ccnc(c1)-c1nnc2-c3nnc(-c4cccc(c4Cl)C(F)(F)F)n3[C@@H](C)Cn12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1cnn(C)c1 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1cnco1 |r|
CCc1nnc2-c3nnc(-c4cccc(c4Cl)C(F)(F)F)n3[C@@H](C)Cn12 |r|
C[C@H]1Cn2c(nnc2-c2cccc(n2)C(F)(F)F)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nccc(n2)C(F)(F)F)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2cc(ccn2)C(F)(F)F)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(Cl)cn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12)-c1ccc(C)s1 |r|
C[C@H]1Cn2c(nnc2-c2cccnc2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2cncc(C)c2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccccn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2cc(C)ccn2)-c2nnc(-c3cccc(c3Cl)C(F)(F)F)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cn2)-c2nnc(-c3cccc(Cl)c3Cl)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cn2)-c2nnc(-c3ccc(Cl)cc3Cl)n12 |r|
C[C@H]1Cn2c(nnc2-c2ccc(F)cn2)-c2nnc(-c3cccc(c3C)C(F)(F)F)n12 |r|
COc1ccnc(c1)-c1nnc2-c3nnc(-c4cccc(Cl)c4Cl)n3[C@@H](C)Cn12 |r|
COc1ccnc(c1)-c1nnc2-c3nnc(-c4ccc(Cl)cc4Cl)n3[C@@H](C)Cn12 |r|
COc1ccnc(c1)-c1nnc2-c3nnc(-c4cccc(c4C)C(F)(F)F)n3[C@@H](C)Cn12 |r|
FC(F)(F)c1cccc(-c2nnc3-c4nnc(-c5cnccn5)n4CCn23)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(N1CCc2ccccc2C1)c1nccs1
Cc1ncsc1C(CNC(=O)c1cc(ccc1F)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1nccs1
COc1ccc(cc1C(=O)NCC(N1CCC(F)(F)CC1)c1scnc1C)-c1ncc(F)cn1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cscn1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1cnccn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1cscn1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(CC1)Oc1ccccc1
Fc1cccc(Cl)c1C(=O)NCC(N1CCc2ccccc2C1)c1cscn1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1cccc(C)n1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCCOCC1)c1cscn1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cncs1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCc2ccccc2C1)c1cncs1
CN(CC(N1CCC(F)(F)CC1)c1scnc1C)C(=O)c1cc(ccc1Cl)-c1ncc(F)cn1
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1cncs1
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1cnccn1)N1CCC(F)(F)CC1
Cc1cccc(C)c1C(=O)NCC(N1CCOCC1)c1cncs1
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1cccc(C)n1)N1CCC(F)(F)CC1
Nc1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1cncs1
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1F)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Cc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1cncs1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C(F)(F)F
Cc1cccc(C)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cncs1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C(F)(F)F
Cc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cncs1
CCc1ncc(s1)C(CNC(=O)c1cc(ccc1F)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Nc1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cncs1
CCc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Nc1ccc(Cl)c(c1)C(=O)NCC(N1CCc2ccccc2C1)c1cncs1
CCc1ncc(s1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1cccc(C)c1C(=O)NCC(N1CCc2ccccc2C1)c1cncs1
Fc1cnc(nc1)-c1ccc(F)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CC1
Cc1cccc(Cl)c1C(=O)NCC(N1CCc2ccccc2C1)c1cncs1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CC1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cncs1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cncs2)c1OC
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCCOCC1
Cc1cccc(C)c1C(=O)NCC(N1CCC(CC1)OCc1ccccc1)c1cncs1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOC(C1)c1ccccc1C(F)(F)F
Cc1cccc(Cl)c1C(=O)NCC(N1CCC(CC1)OCc1ccccc1)c1cncs1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOC(C1)c1ccc(F)cc1F
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(CC1)OCc1ccccc1)c1cncs1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOC(C1)c1cnn(C)c1
Cc1cccc(C)c1C(=O)NCC(N1CCC(CC1)Oc1ccccc1)c1cncs1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCOC2(CCC2)C1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(CC1)Oc1ccccc1)c1cncs1
Cc1ncsc1C(CNC(=O)c1cc(ccc1F)-c1ncc(F)cn1)N1CCOC2(CCC2)C1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCc2ccccc2C1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1c(C)cccc1C)N1CCc2ccccc2C1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOC2(CCC2)C1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCOC(C1)c1cnn(C)c1
Cc1ncsc1C(CNC(=O)c1c(C)cccc1C)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1F)-c1ncc(F)cn1)N1CCOC(C1)c1cnn(C)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCOC(C1)c1ccc(F)cc1F
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1c(C)cccc1Cl)N1CCOC(C1)c1ccc(F)cc1F
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOCC1
Cc1ncsc1C(CNC(=O)c1c(C)cccc1C)N1CCOCC1
FC(F)c1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCOCC1
CC1CC(F)(F)CCN1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)c1scnc1C
Cc1ncc(s1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
CC1CC(F)(F)CCN1C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C
Cc1ncc(s1)C(CNC(=O)c1c(C)cccc1Cl)N1CCC(F)(F)CC1
FC1(F)CCN(CC1)C(CNC(=O)c1cccc2ncccc12)c1cnc(s1)C1CCC1
Cc1ncc(s1)C(CNC(=O)c1c(C)cccc1C)N1CCC(F)(F)CC1
Fc1cnc(nc1)-c1ccc(F)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CCC1
Cc1ncc(s1)C(CNC(=O)c1c(C)cccc1Cl)N1CCc2ccccc2C1
CCCc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1cnco1
CCCc1ncc(s1)C(CNC(=O)c1cccc2ncccc12)N1CCC(F)(F)CC1
Cc1cccc(C)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnco1
CCCc1ncc(s1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnco1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CCC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCc2ccccc2C1)c1cnco1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CCC1
Cc1cccc(C)c1C(=O)NCC(N1CCc2ccccc2C1)c1cnco1
OCc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ocnc2C)c1OC
CC1CC(F)(F)CCN1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)c1cnc(C)s1
Cc1ncoc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1ccc(cc1Cl)N1CCCS1(=O)=O)N1CCC(F)(F)CC1
Cc1ncoc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCOCC1
FC1(F)CCC(CC1)c1ncc(s1)C(CNC(=O)c1cccc2ncccc12)N1CCOCC1
COc1cccc(C(=O)NCC(N2CCc3ccccc3C2)c2ocnc2C)c1OC
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1cnc(s1)C1CCC(F)(F)CC1
Cc1ncoc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCc2ccccc2C1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CCC(F)(F)CC1
Cc1nc(C)c(o1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
CC(C)(C)c1ncc(s1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccccc1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1scnc1C1CC1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccccc1
Cc1ncsc1C(CNC(=O)c1cc2CCC(=O)Nc2cc1F)N1CCC(F)(F)CC1
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
FC1(F)CCN(CC1)C(CNC(=O)c1cccc2ncccc12)c1scnc1C1CC1
Cc1ncc(s1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccccc1
CC(C)(C)c1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(CC1)OCc1ccccc1)c1cnco1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1scnc1C1CC1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCCC(F)(F)C1
CC(C)(C)c1ncc(s1)C(CNC(=O)c1cccc2ncccc12)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CC(F)(F)C1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1cnc(s1)C1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCCC(F)(F)C1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(s1)C1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1scnc1C(F)(F)F
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Fc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1scnc1C(F)(F)F
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
Cc1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
FC(F)c1ncsc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCOCC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCOCC1
Cc1ncoc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCOCC2)c2ocnc2C)c1OC
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnco1
OC[C@@H](NC(=O)c1ccc2[nH]ccc2c1Cl)C1CCCCC1
OC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
OC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCCC1
OC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCC(F)(F)CC1
OC[C@@H](NC(=O)c1ccc2[nH]ccc2c1Cl)C1CCC(F)(F)CC1
Cn1ccc2c(Cl)c(ccc12)C(=O)NCC1(O)CCCCC1
Cn1ccc2c(Cl)c(ccc12)C(=O)N[C@H](CO)C1CCCCC1
OC[C@@H](NC(=O)c1ccc2[nH]cc(C=O)c2c1Cl)C1CCCCC1
OC1(CNC(=O)c2ccc3[nH]cc(C=O)c3c2Cl)CCCCC1
OCC(NC(=O)c1ccc2[nH]ccc2c1Cl)C1CCCCCC1
FC(F)(F)c1ncc(cn1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Clc1ccc(cn1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
FC(F)(F)c1ccc(cn1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
FC1(F)CCC(CNC(=O)c2ccc3[nH]ccc3c2Cl)(CC1)c1ccc(Cl)nc1
Clc1ccc(cc1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
FC(F)(F)c1ccc(cc1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Clc1c(ccc2[nH]ccc12)C(=O)NCC1(CCCCC1)c1cccnc1
Clc1c(ccc2[nH]ccc12)C(=O)NCC1(CCCC1)c1cccnc1
Clc1c(ccc2[nH]ccc12)C(=O)NCC1(CCCCCC1)c1cccnc1
Cc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
OC1(CNC(=O)c2ccc3NC(=O)Cc3c2Cl)CCCCCC1
Cc1cc2c(Cl)c(ccc2[nH]1)C(=O)NCC1(O)CCCCC1
CSc1c[nH]c2c(I)cc(C(=O)NCC3(O)CCCCC3)c(Cl)c12
Cc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
Cc1cc(C(=O)NCC2(O)CCCCCC2)c(Cl)c2cc[nH]c12
OC1(CNC(=O)c2ccc3[nH]cc(F)c3c2Cl)CCCCCC1
COc1c(ccc2[nH]ccc12)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2ccc3[nH]cc(Cl)c3c2Cl)CCCCC1
OC1(CNC(=O)c2cc([N+]([O-])=O)c3[nH]ccc3c2Cl)CCCCC1
COC(=O)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
OCC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Nc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
Cc1c[nH]c2ccc(C(=O)NCC3(O)CCCCCC3)c(Cl)c12
NC(=O)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
CNC(=O)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Clc1c(ccc2[nH]ccc12)C(=O)NCC1(CCCCC1)C#N
CC(C)(C)OC(=O)NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
OC1(CNC(=O)c2c(Cl)cc3[nH]ccc3c2Cl)CCC(F)(F)CC1
NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Cc1cc2[nH]ccc2c(Cl)c1C(=O)NCC1(O)CCCCC1
OC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCC1
OC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCCCC1
COC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
C[C@H](NC(=O)c1ccc2[nH]ccc2c1Cl)C1CCCCC1
C[C@@H](NC(=O)c1ccc2[nH]ccc2c1Cl)C1CCCCC1
CC(=O)NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
CS(=O)(=O)NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
CN(C)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Clc1c(ccc2[nH]ccc12)C(=O)NCC1(CCCCC1)NCc1ccccc1
Cc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2c(Br)c[nH]c12
COC(=O)CS(=O)(=O)NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
CC(C)Cc1cc(C(=O)NCC2(O)CCCCCC2)c(Cl)c2cc[nH]c12
COCCCc1cc(C(=O)NCC2(O)CCCCCC2)c(Cl)c2cc[nH]c12
CC(C)Cc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
COCCCc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
OCCS(=O)(=O)NC1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
Cc1c(ccc2[nH]ccc12)C(=O)NCC1(O)CCCCC1
Cc1ncc(cn1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCCCC1
COc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
Cc1ncc(cn1)C1(CNC(=O)c2ccc3[nH]ccc3c2Cl)CCC(F)(F)CC1
Cc1ncc(cn1)C1(CNC(=O)c2cc(C)c3[nH]ccc3c2Cl)CCC(F)(F)CC1
Cc1ncc(cn1)C1(CNC(=O)c2cc(C)c3[nH]ccc3c2Cl)CCCCC1
Cc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(C)c2cc[nH]c12
Cc1c(ccc2[nH]ccc12)C(=O)NCC1(O)CCC(F)(F)CC1
CCc1c(ccc2[nH]ccc12)C(=O)NCC1(O)CCC(F)(F)CC1
CC(=O)c1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CC(O)c1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CC(C)(O)c1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
Cc1cc(C(=O)NCC2(O)CCCCC2)c(c2cc[nH]c12)C(F)(F)F
Cc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(c2cc[nH]c12)C(F)(F)F
Cc1cc(C(=O)NCC2(O)CCCCC2)c(C)c2cc[nH]c12
CCc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
CCc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
Cc1c(cc(Cl)c2[nH]ccc12)C(=O)NCC1(O)CCCCC1
Cc1c(cc(Cl)c2[nH]ccc12)C(=O)NCC1(O)CCC(F)(F)CC1
COc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
COc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(C)c2cc[nH]c12
COc1cc(C(=O)NCC2(O)CCCCC2)c(C)c2cc[nH]c12
CCOc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
Oc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CCOc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CCCc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
CCCc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CC(C)(C)OCCOc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
CC(C)(C)OCCOc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
OCCOc1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
OCCOc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
CC(=O)c1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
CC(C)(O)c1cc(C(=O)NCC2(O)CCCCC2)c(Cl)c2cc[nH]c12
OC1(CNC(=O)c2cc(F)c3[nH]ccc3c2F)CCCCC1
OC1(CNC(=O)c2cc(F)c3[nH]ccc3c2F)CCC(F)(F)CC1
COc1cc(C(=O)NCC2(O)CCCCC2)c(F)c2cc[nH]c12
COc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(F)c2cc[nH]c12
CCOCCc1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
COC(C)(C)c1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c(Cl)c2cc[nH]c12
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccccc2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccccc2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccn[nH]2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncn3-c2cnccn2)c1Cl
C[C@H]1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1F)C(F)(F)F
CCC1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC(C)C1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccc(F)cc1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1ncn2-c1ncccc1F)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ncccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCOC(=O)C1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCOC(=O)C1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl
CCOC(=O)C1N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCOC(=O)C1N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
CCOC(=O)C1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCOC(=O)C1N(CCc2c1ncn2-c1cnccn1)C(=O)c1cccc(Cl)c1Cl
OCC1N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CN(C)CC1N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
FCC1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CN(C)C(=O)C1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCc3c(ncn3-c3ccccn3)C2C(=O)N2CCC2)c1Cl
FC(F)(F)c1cccc(C(=O)OCC2N(CCc3c2ncn3-c2ccccc2)C(=O)c2cccc(c2Cl)C(F)(F)F)c1Cl
Cc1nc2CN(CCc2n1-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1nc2CN(CCc2n1-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@@H]1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1F)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1ncn2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncn2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1(C)N(CCc2c1ncn2-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2Cc3ncn(c3C=C2)-c2cnccn2)c1Cl |c:19|
CCC1N(C=Cc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:4|
CC1N(C=Cc2c1ncn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nc(n2-c1ccccc1)C(F)(F)F
FC(F)(F)c1nc2CN(CCc2n1-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)ncn2-c1ccn[nH]1
Clc1cccc(C(=O)N2CCc3c(C2)ncn3-c2ccn[nH]2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nnn3-c2ccccc2)c1Cl
Clc1cccc(C(=O)C2CCc3c(C2)nnn3-c2ccccc2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nnn3-c2ccccn2)c1Cl
Fc1cnc(nc1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nnn3-c2ncccn2)c1Cl
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nnn2-c1ncccn1
Clc1cccc(C(=O)N2CCc3c(C2)nnn3-c2ncccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nnn3-c2ccn[nH]2)c1Cl
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nnn2-c1cnccn1
Clc1cccc(C(=O)N2CCc3c(C2)nnn3-c2cnccn2)c1Cl
Fc1ccc(nc1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(C=Cc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1N(CCc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
FC(F)(F)c1cccc(C(=O)N2C=Cc3c(nnn3-c3cnccn3)C2c2ccccc2)c1Cl |c:12|
FC(F)(F)c1cccc(C(=O)N2CCc3c(nnn3-c3cnccn3)C2c2ccccc2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3[nH]nnc3C2c2ccccc2)c1Cl
CC1N(C=Cc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(C=Cc2c1nnn2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1N(C=Cc2c1nnn2-c1ncccc1F)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1N(CCc2c1nnn2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ncccc1F)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc[nH]n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(C=Cc2c1nnn2-c1cc[nH]n1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
C[C@@H]1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
FC(F)(F)c1cccc(C(=O)N2Cc3nnn(c3C=C2)-c2cnccn2)c1Cl |c:19|
FC(F)(F)c1cccc(C(=O)N2Cc3nnn(c3C=C2)-c2ccccn2)c1Cl |c:19|
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nnn3-c2cnccn2)c1Cl
Cn1nc2CN(CCc2c1-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ccccn2)c1Cl
Fc1ccc(nc1)-c1n[nH]c2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Fc1cncc(c1)-c1n[nH]c2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2cccnc2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2cnccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ncccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ccccc2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ccccc2)c1Cl
Cn1nc(c2CCN(Cc12)C(=O)c1cccc(Cl)c1Cl)-c1ccccc1
Cn1nc2CN(CCc2c1-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
Clc1nccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ccccc2)c1Cl
Cn1nc2CN(CCc2c1-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1nc(c2CCN(Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F)-c1ccc(F)cc1
Cn1nc2CN(CCc2c1-c1cccnc1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1nc(c2CCN(Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F)-c1cccnc1
Cn1nc(c2CCN(Cc12)C(=O)c1cccc(Cl)c1Cl)-c1ccc(F)cc1
Fc1ccc(cc1)-c1n[nH]c2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1nc2CN(CCc2c1-c1cccnc1)C(=O)c1cccc(Cl)c1Cl
Cn1nc(c2CCN(Cc12)C(=O)c1cccc(Cl)c1Cl)-c1cccnc1
Cn1nc2CN(CCc2c1-c1cncnc1)C(=O)c1cccc(c1Cl)C(F)(F)F
Fc1ccc(cc1)-c1n[nH]c2CN(CCc12)C(=O)c1cccc(Cl)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)[nH]nc3-c2ccncc2)c1Cl
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccccn1
Fc1ccc(C(=O)N2CCc3c(C2)nnn3-c2ccccn2)c(Cl)c1
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccccn1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccccn1 |r|
CC1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ccccn1
CC1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nnn2-c1ccccn1
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncccc1F
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nnn2-c1ccccn1
COc1ccccc1-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
FCCOc1ccccc1-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1ccc(n1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1nccc1-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Fc1cc(Cl)ccc1C(=O)N1CCc2c(C1)nnn2-c1ccccn1
Fc1ccc(C(=O)N2CCc3c(C2)nnn3-c2ccccn2)c(Cl)c1Cl
Fc1ccnc(c1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1c(F)c(F)ccc1C(=O)N1CCc2c(C1)nnn2-c1ccccn1
C[C@H]1N(CCc2c1nnn2-c1cc[nH]n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
Fc1cccc(n1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
COc1ccnc(c1)-n1nnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1ccccn1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
C[C@@H]1N(CCc2c1nnn2-c1ccccn1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
C[C@H]1N(CCc2c1nnn2-c1cnccn1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
C[C@@H]1N(CCc2c1nnn2-c1cnccn1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
COc1ccc(nc1)-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cccc(F)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cccc(F)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1nnn2-c1cc(F)ccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(F)ccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
COc1ccnc(c1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
COc1ccnc(c1)-n1nnc2[C@@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1cc[nH]n1
C[C@H]1Cc2c(CN1C(=O)c1ccc(Cl)cc1F)nnn2-c1ncc(F)cn1 |r|
C[C@@H]1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1ncc(C)cc1C)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ncc(C)cc1C)C(=O)c1cccc(Cl)c1Cl
CC1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ncccc1F
C[C@@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ncccc1F |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ncccc1F |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncccc1F |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncccc1F |r|
C[C@@H]1N(CCc2c1nnn2-c1ccn(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1nnn2-c1ccn(CCF)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1ccn(CCF)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1cc(F)ccn1
CC1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cc(F)ccn1
CC1N(CCc2c1nnn2-c1cncnc1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@@H]1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1F)C(F)(F)F |r|
CC1N(C=Cc2c1nnn2-c1nc(C)cc(C)n1)C(=O)c1cccc(Cl)c1Cl |c:3|
CC1N(CCc2c1nnn2-c1cncc(C)n1)C(=O)c1cccc(Cl)c1Cl
C[C@H]1N(CCc2c1nnn2-c1nc(C)cc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1Cl)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CCc1nc2C(C)N(CCc2n1-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1Cc2c(CN1C(=O)c1ccnc(c1C)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1C)C(F)(F)F |r|
CC1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ccn[nH]1
C[C@H]1N(CCc2c1nnn2-c1ncc(F)cn1)C(=O)c1cccc(c1F)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl |r|
C[C@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl |r|
C[C@H]1N(CCc2c1ncn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncn2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1cc(F)ccn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1cc(F)ccn1 |r|
C[C@@H]1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1C)C(F)(F)F |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cc(F)ccn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cc(F)ccn1 |r|
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncc(F)cn1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CC1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ncc(F)cn1
C[C@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nnn2-c1ncc(F)cn1 |r|
CC1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1ncc(F)cn1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cnccn1
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cc[nH]n1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cnccn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1cnccn1 |r|
CC1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nnn2-c1ncc(F)cn1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nnn2-c1ncc(F)cn1 |r|
CC1Cc2c(CN1C(=O)c1ccc(Cl)c(F)c1Cl)nnn2-c1ncc(F)cn1
C[C@H]1Cc2c(CN1C(=O)c1ccc(Cl)c(F)c1Cl)nnn2-c1ncc(F)cn1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncccn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ncccn1 |r|
C[C@H]1N(CCc2c1n[nH]c2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(C=Cc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(Cl)c1Cl |c:3|
C[C@@H]1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1F)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CC1N(CCc2c1nnn2-c1ncc(F)c(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)cc(C)n1)C(=O)c1cccc(Cl)c1Cl
C[C@H]1Cc2c(CN1C(=O)c1cc(ccc1F)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CC1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(Cl)c1Cl
CC1NC(=NC=C1)n1nnc2[C@@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r,c:3,5|
C[C@H]1N(CCc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(C=Cc2c1nnn2-c1cncnc1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(Cl)c1Cl
CC1CN(C(C)c2nnn(c12)-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(nnn2-c2ccccc2)C(C)N1C(=O)c1cccc(c1Cl)C(F)(F)F
CC1CN(C(C)c2nnn(c12)-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(nnn2-c2ccc(F)cc2)C(C)N1C(=O)c1cccc(Cl)c1Cl
CC1Cc2c(nnn2-c2ccc(F)cc2)C(C)N1C(=O)c1cccc(c1Cl)C(F)(F)F
CC1CN(Cc2nnn(c12)-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
CC1CN(Cc2nnn(c12)-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1CN(Cc2nnn(c12)-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1CN(Cc2nnn(c12)-c1ccc(F)cc1)C(=O)c1cccc(Cl)c1Cl
COCCn1ccc(n1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1ncco1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cncc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1nc(C)cc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCc1cccnc1-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1ccc(C)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1ccc(F)cc1Cl
Clc1ccc(C(=O)N2CCc3c(C2)nnn3-c2ncccn2)c(Cl)c1
CCOc1cccnc1-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ncccc1C)C(=O)c1cccc(c1Cl)C(F)(F)F
COc1cccnc1-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1ccc(F)c(Cl)c1Cl
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1C)C(F)(F)F
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1ccccc1F
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)n(C)nc2-c1ccnn1C
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)[nH]nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1ccc(Cl)cc1Cl)[nH]nc2-c1ccn[nH]1
CC1N(CCc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(c1F)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1F)C(F)(F)F |r|
Fc1cc(Cl)ccc1C(=O)N1CCc2c(C1)nnn2-c1cnccn1
CC1N(CCc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1nnn2-c1cnccn1)C(=O)c1ccc(Cl)cc1F
CC1N(CCc2c1nnn2-c1ncccn1)C(=O)c1ccc(Cl)cc1F
Cc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nnn2-c1cnccn1
Clc1ccc(C(=O)N2CCc3c(C2)nnn3-c2cnccn2)c(Cl)c1
CC1N(CCc2c1nnn2-c1cnccn1)C(=O)c1cccc(c1C)C(F)(F)F
CC1N(CCc2c1nnn2-c1cnccn1)C(=O)c1ccc(Cl)cc1Cl
Fc1cc(Cl)ccc1C(=O)N1CCc2c(C1)nnn2-c1ncccn1
Cc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)nnn2-c1ncccn1
CC1N(CCc2c1nnn2-c1ncccn1)C(=O)c1cccc(c1C)C(F)(F)F
CC1N(CCc2c1nnn2-c1ncccn1)C(=O)c1ccc(Cl)cc1Cl
C[C@@H]1Cc2c(nnn2-c2ccc(F)cc2)[C@@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(nnn2-c2ccc(F)cc2)[C@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1Cc2c(nnn2-c2ccc(F)cc2)[C@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(nnn2-c2ccccc2)[C@@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccccc1 |r|
CC1N(CCc2nnn(c12)-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccccc1
C[C@H]1N(CCc2c1nnn2-c1ncccc1C)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1ncccc1C)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCCOc1cccnc1-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CCc1ccnc(n1)-n1nnc2[C@@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCc1cccnc1-n1nnc2C(C)N(CCc12)C(=O)c1cccc(c1)C(F)(F)F
C[C@@H]1Cc2c(nnn2-c2ccn[nH]2)[C@@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1Cc2c(nnn2-c2ccn[nH]2)[C@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)cc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ccc(C)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nn(COCC[Si](C)(C)C)c2-c1ncc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1N(CCc2c1nnn2-c1ncc(F)c(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1cc(F)cc(c1)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
CC1N(CCc2c1[nH]nc2C(F)(F)F)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1Cc2c(nnn2-c2ccn[nH]2)[C@@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ncc(F)cn1
Cc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)ncn2-c1ccc(F)cn1
Fc1ccc(nc1)-n1cnc2CN(CCc12)C(=O)c1ccc(Cl)cc1Cl
Fc1ccc(nc1)-n1cnc2CN(CCc12)C(=O)c1cccc(c1F)C(F)(F)F
Fc1ccc(nc1)-n1cnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CCOc1cccnc1-n1nnc2[C@@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCOc1cccnc1-n1nnc2[C@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(nnn2-c2ccn[nH]2)[C@H](C)N1C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(C=Cc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
Cn1nc2CN(CCc2c1-c1ccncc1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cn1nc2CN(CCc2c1-c1ccncc1)C(=O)c1cccc(Cl)c1Cl
Cn1nc2CN(CCc2c1-c1cncnc1)C(=O)c1cccc(Cl)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)n[nH]c3-c2cncnc2)c1Cl
Cc1nc2CN(CCc2n1-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
CCc1nc2CN(CCc2n1-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
C[C@@H]1N(CCc2c1nnn2-c1cncnc1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1N(CCc2c1nnn2-c1cncnc1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1ccc(C)cn1)C(=O)c1cccc(Cl)c1Cl
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ccn[nH]1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccn[nH]1 |r|
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cc(ccc1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1F)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1F)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1F)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cc(Cl)cc(c1)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cc(Cl)cc(c1)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cc(Cl)cc(c1)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccnc(c1F)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccnc(c1F)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccnc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(OC(F)(F)F)c1F
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cccc(OC(F)(F)F)c1F
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(OC(F)(F)F)c1
C[C@@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(OC(F)(F)F)c1 |r|
CC1N(CCc2c1nnn2-c1cccc(n1)C(F)(F)F)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cccc(n1)C(F)(F)F)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1nnn2-c1cc(C)c(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1ncc[nH]1)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(c1F)C(F)(F)F
C[C@@H]1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(c1F)C(F)(F)F |r|
CC1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(Cl)c1C
C[C@@H]1N(CCc2c1nnn2-c1cccc(C)n1)C(=O)c1cccc(Cl)c1Cl |r|
C[C@@H]1N(CCc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(Cl)c1Cl |r|
CC1N(C=Cc2c1nnn2-c1ncc[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |c:3|
C[C@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(Cl)c1Cl |r|
C[C@@H]1N(CCc2c1nnn2-c1cc(C)ccn1)C(=O)c1cccc(Cl)c1Cl |r|
CC1N(CCc2c1nnn2-c1cc(C)ncn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1nnn2-c1ccnc(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ccnc(C)n1)C(=O)c1ccnc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1ccnc(C)n1)C(=O)c1cccc(c1F)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)ncn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1cc(C)ncn1)C(=O)c1ccnc(c1Cl)C(F)(F)F
CCn1ccc(n1)-n1nnc2CN([C@@H](C)Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCn1ccc(n1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCn1nccc1-n1nnc2CN([C@@H](C)Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCn1ccc(n1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1ccnc(c1F)C(F)(F)F |r|
CCn1ccc(n1)-n1nnc2CN([C@@H](C)Cc12)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
CC(C)n1ccc(n1)-n1nnc2CN([C@@H](C)Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC(C)n1ccc(n1)-n1nnc2CN([C@@H](C)Cc12)C(=O)c1cccc(c1F)C(F)(F)F |r|
CC(C)n1ccc(n1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1cccc(c1F)C(F)(F)F |r|
CC(C)n1ccc(n1)-n1nnc2CN([C@@H](C)Cc12)C(=O)c1ccnc(c1Cl)C(F)(F)F |r|
CC(C)n1ccc(n1)-n1nnc2[C@H](C)N(CCc12)C(=O)c1ccnc(c1F)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnn2-c1ccsc1 |r|
C[C@@H]1N(CCc2c1nnn2-c1ccsc1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1Cl)C(F)(F)F)nnn2-c1cc[nH]n1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1ccnc(c1Cl)C(F)(F)F)nnn2-c1cc[nH]n1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1F)C(F)(F)F)nnn2-c1cc[nH]n1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1ccnc(c1F)C(F)(F)F)nnn2-c1cc[nH]n1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1O)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(OC(F)(F)F)c1F)nnn2-c1ncc(F)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1ncc(O)cn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1F)C(F)(F)F)nnn2-c1ncc(O)cn1 |r|
CC1N(CCc2c1n[nH]c2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1n[nH]c2-c1ncccn1)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1n[nH]c2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1n[nH]c2-c1cnccn1)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1n[nH]c2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1n[nH]c2-c1ccc(F)cc1)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1n[nH]c2-c1ccnn1C)C(=O)c1cccc(Cl)c1Cl
CC1N(CCc2c1n[nH]c2-c1ccnn1C)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1n[nH]c2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1cccnc1
Cc1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccncc1
Clc1cccc(C(=O)NCC(N2CCOCC2)c2cccnc2)c1Cl
Clc1cccc(C(=O)NCC(N2CCOCC2)c2ccncc2)c1Cl
Cc1cccc(C(=O)NCC(N2CCOCC2)c2cccnc2)c1C
Cc1cccc(C(=O)NCC(N2CCOCC2)c2ccncc2)c1C
Fc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
COc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCCC1
COc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Cc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(F)cc2)c1C
COc1ccc(cc1)C(CNC(=O)c1cccc(C)c1C)N1CCCCC1
COc1ccc(cc1)C(CNC(=O)c1cccc(C)c1C)N1CCOCC1
Cc1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(F)cc1
COc1ccc(cc1)C(CNC(=O)c1cc(C)ccc1Cl)N1CCCCC1
COc1ccc(cc1)C(CNC(=O)c1cc(C)ccc1Cl)N1CCOCC1
Cc1ccccc1C(=O)NCC(N1CCOCC1)c1ccc(F)cc1
COc1ccc(cc1)C(CNC(=O)c1ccccc1C)N1CCCCC1
COc1ccc(cc1)C(CNC(=O)c1ccccc1C)N1CCOCC1
Cc1ccc(cc1)C(CNC(=O)c1cc(C)ccc1Cl)N1CCOCC1
Cc1ccccc1C(=O)NCC(N1CCC(F)(F)CC1)c1ccc(Cl)cc1
Cc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(Cl)cc2)c1C
FC1(F)CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccc(Cl)cc1
Clc1ccc(cc1)[C@@H](CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1 |r|
Clc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(nc2)C2CC2)c1Cl
Cc1ccccc1C(=O)NC[C@@H](N1CCOCC1)c1ccc(Cl)cc1 |r|
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Cc1cccc(C(=O)NC[C@@H](N2CCOCC2)c2ccc(Cl)cc2)c1Cl
Clc1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Clc1cccc(C(=O)NCC(N2CCOCC2)c2cncnc2)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Fc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(c1Cl)C(F)(F)F)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(c1Cl)C(F)(F)F)N1CCOCC1
COc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Fc1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Fc1ccc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
Fc1ccccc1C(=O)NCC(N1CCOCC1)c1cnc(nc1)C(F)(F)F
Cc1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Clc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCOCC1
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
Fc1cccc(F)c1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCC1
COc1ccccc1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
Clc1ccc(cc1)C(CNC(=O)c1cc(ccc1Cl)C#N)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
CC(C)S(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(Cl)cc1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
Fc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Cc1ccc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ccc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1F)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
Fc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
CC1(C)CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C(F)(F)F
CC1(C)CCN(CC1)C(CNC(=O)c1cccc(F)c1Cl)c1cnc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCOCC1
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCCOCC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCCOCC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCCOCC1
COc1cccc(C(=O)NCC(N2CCOCC2)c2cnc(nc2)C(F)(F)F)c1Cl
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(nc2)C(F)(F)F)c1C
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(F)cc2)c1Cl
CC1CCN(C1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(C)nc1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CC(F)(F)C(F)(F)C1
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(Cl)cc2)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCCC(F)(F)C1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCCC(F)(F)C1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCC(F)(F)C1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCCC(F)(F)C1
FC1CCN(CC1)C(CNC(=O)c1ccccc1Cl)c1cnc(nc1)C(F)(F)F
FC1CCN(CC1)C(CNC(=O)c1c(Cl)cccc1Cl)c1cnc(nc1)C(F)(F)F
FC1CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCOCC1
Cn1cc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Cn1cc(cn1)C(CNC(=O)c1cc(F)cc(Cl)c1Cl)N1CCC(F)(F)CC1
Cn1cc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Fc1ccc(Cl)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCCCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCCC1
Fc1cc(Cl)c(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
Cn1cc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
FC(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(C)nc2)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)ccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cc(F)cc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)c1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCOCC1
FC1(F)CCN(CC1)C(CNC(=O)c1ccccc1Cl)c1cnc(nc1)C1CC1
FC1(F)CCN(CC1)C(CNC(=O)c1c(Cl)cccc1Cl)c1cnc(nc1)C1CC1
CCc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(OC(F)F)c1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
FC1(F)CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C1CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C1CC1
Cc1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCC(F)(F)CC1
CC1CCCN(C1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(C)nc1
Fc1cc(F)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
COc1ccc(F)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
CC(C)C1CCCCN1C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(C)nc1
CN(C)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CC2CCC1C2
CC1CCCCN1C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(C)nc1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCC(F)(F)CC1
Fc1cc(Cl)cc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
COc1ccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
COc1ccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1OC
COC1CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(C)nc1
Fc1cc(Cl)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
Cc1ncc(cn1)C(CNC(=O)c1cccc(OC(F)(F)F)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(=O)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCC(=O)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(Cl)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCC(Cl)CC1
Fc1cccc(C(=O)NCC(N2CCOCC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(nc2)C(F)F)c1Cl
Clc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Cc1ccc(Cl)c(c1)C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Cc1cccc(C(=O)NCC2(CCOCC2)c2ccc(Cl)cc2)c1C
COc1ccccc1C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Clc1ccc(cc1)C1(CNC(=O)c2c(Cl)cccc2Cl)CCOCC1
Cc1ccccc1C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Clc1cccc(C(=O)NCC2(CCCC2)c2cccnc2)c1Cl
Cc1ccc(Cl)c(c1)C(=O)NCC1(CCCC1)c1cccnc1
FC(F)(F)c1ccccc1C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Cc1ccccc1C(=O)NCC1(CCCC1)c1cccnc1
Fc1c(cccc1C(F)(F)F)C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Fc1c(Cl)cccc1C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
Fc1ccc(F)c(c1)C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
COc1ccc(cc1)C1(CNC(=O)c2cc(C)ccc2Cl)CCCC1
COc1ccc(cc1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCCC1
COc1ccc(cc1)C1(CNC(=O)c2ccccc2C)CCCC1
COc1ccc(cc1)C1(CNC(=O)c2cccc(C)c2C)CCCC1
CN1CCC(CNC(=O)c2cc(C)ccc2Cl)(CC1)c1ccccc1
CN1CCC(CNC(=O)c2ccccc2C)(CC1)c1ccccc1
Fc1cc(F)c(F)c(c1)C(=O)NCC1(CCOCC1)c1ccc(Cl)cc1
CN1CCC(CNC(=O)c2ccccc2C)(CC1)c1ccc(Cl)cc1
CC(C)CC(CNC(=O)c1cccc(Cl)c1Cl)c1ccc(C)nc1
CC(C)CC(CNC(=O)c1cccc(C)c1C)c1ccc(C)nc1
CC(C)CC(CNC(=O)c1ccccc1C)c1ccc(C)nc1
Cc1ccc(Cl)c(c1)C(=O)NCC1(CCOCC1)c1ccc(C)nc1
Clc1ccc(cc1)C1(CNC(=O)c2cc(Br)ccc2Cl)CCOCC1
Clc1ccc(cc1)C1(CNC(=O)c2ccccc2Cl)CCOCC1
Fc1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
Fc1ccc(cn1)C1(CNC(=O)c2c(F)cccc2Cl)CCC(F)(F)CC1
Cc1ccc(Cl)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Fc1ccc(cn1)C1(CNC(=O)c2cc(ccc2Cl)C(F)(F)F)CCC(F)(F)CC1
Fc1ccc(cn1)C1(CNC(=O)c2ccccc2F)CCC(F)(F)CC1
COc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(F)nc2)c1F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Fc1ccc(cn1)C1(CNC(=O)c2ccccc2Cl)CCC(F)(F)CC1
Cc1ccc(F)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Cc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(F)nc2)c1F
Fc1ccc(F)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Fc1ccc(cn1)C1(CNC(=O)c2cc(Cl)ccc2Cl)CCC(F)(F)CC1
COc1ccc(Cl)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Fc1ccc(cn1)C1(CNC(=O)c2cccc(F)c2F)CCC(F)(F)CC1
Clc1ccc(cc1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCOCC1
FC(F)(F)c1ccc(cc1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCOCC1
FC(F)(F)c1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCOCC1
FC1(F)CCC(CNC(=O)c2cccc(Cl)c2Cl)(CC1)c1ccc(nc1)C1CC1
COc1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C1(CNC(=O)c2ccccc2C#N)CCC(F)(F)CC1
CS(=O)(=O)c1ccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c(Cl)c1
Cc1ccccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CC1
CS(=O)(=O)c1ccccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Fc1cncc(c1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)CC1CC1
Cc1c(F)cccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
COc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1C
Cc1ccc(F)cc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Cc1ccc(cc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F)C(F)(F)F
Cc1c(Br)cccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Cc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Cc1c(cccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F)C#N
Clc1cncc(c1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
Clc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccccc1
Cc1ccc(C(CNC(=O)c2cccc(Cl)c2Cl)CC2CC2)c(C)n1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1(CC1)C(F)(F)F
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1(CC1)C(F)(F)F
FC(F)(F)C1(CC(CNC(=O)c2cccc(Cl)c2Cl)c2ccc(nc2)C2CC2)CC1
FC(F)C1(CC(CNC(=O)c2cccc(Cl)c2Cl)c2ccc(nc2)C2CC2)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(c1Cl)C(F)(F)F)CC1CC1
FC(F)C1(CC(CNC(=O)c2cccc(Cl)c2Cl)c2ccc(nc2)C(F)(F)F)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)CC1(CC1)C(F)(F)F
FC(F)(F)C1(CC(CNC(=O)c2ccccc2Cl)c2ccc(nc2)C2CC2)CC1
Fc1ccccc1C(=O)NCC(CC1(CC1)C(F)(F)F)c1ccc(nc1)C1CC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)CC1CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)CC1(CC1)C(F)(F)F
Fc1ccccc1C(=O)NCC(CC1(CC1)C(F)(F)F)c1ccc(nc1)C(F)(F)F
Cc1ncc(cn1)C1(CNC(=O)c2ccccc2Cl)CCC(F)(F)CC1
Cc1ncc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
CC(C)(O)c1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
CC(C)(O)c1ccc(cn1)C1(CNC(=O)c2ccccc2Cl)CCC(F)(F)CC1
COc1cccc(C(=O)NCC(CC2CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(CC1CC1)c1ccc(nc1)C(F)(F)F
COc1ccccc1C(=O)NCC(CC1CC1)c1ccc(nc1)C(F)(F)F
Fc1cccc(F)c1C(=O)NCC(CC1CC1)c1ccc(nc1)C(F)(F)F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(CC1CC1)c1ccc(nc1)C(F)(F)F
Cc1cn(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
Fc1cccc(C(=O)NCC(CC2CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1ccc(cn1)C(CNC(=O)c1ccccc1Cl)CC1CC1
CC(NC(=O)c1cccc(Cl)c1Cl)C1(CCC(F)(F)CC1)c1ccc(Br)nc1
FC(F)(F)c1ccc(cn1)C1(CNC(=O)c2ccccc2Cl)CCC(F)(F)CC1
Cc1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
COc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(C(=O)NCC2(CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1ccc(cn1)C1(CNC(=O)c2cccc(F)c2Cl)CCC(F)(F)CC1
Fc1c(Cl)cccc1C(=O)NCC1(CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Fc1ccc(cn1)C1(CNC(=O)c2cccc(Cl)c2F)CCC(F)(F)CC1
Fc1c(Cl)cccc1C(=O)NCC(CC1CC1)c1ccc(nc1)C(F)(F)F
Fc1ccc(C(=O)NCC(CC2CC2)c2ccc(nc2)C(F)(F)F)c(Cl)c1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)CC1CC1
CC(CNC(=O)c1ccccc1Cl)(CC1CC1)c1cnc(nc1)C(F)(F)F
CC(CNC(=O)c1cccc(F)c1Cl)(CC1CC1)c1cnc(nc1)C(F)(F)F
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)CC1CC1
Fc1cccc(C(=O)NCC(CC2CC2)c2cnc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(CC1CC1)c1cnc(nc1)C(F)(F)F
Clc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CCOCC1
Clc1ccc(cc1)C(CNC(=O)c1ccccc1Cl)C1CCOCC1
Fc1cccc(Cl)c1C(=O)NCC(C1CCOCC1)c1ccc(Cl)cc1
Fc1cccc(C(=O)NCC(C2CCOCC2)c2ccc(Cl)cc2)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)CC1CC1
FC(F)(F)c1ncc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCOCC1
FC(F)(F)c1ncc(cn1)C1(CNC(=O)c2ccccc2Cl)CCOCC1
Fc1cccc(Cl)c1C(=O)NCC1(CCOCC1)c1cnc(nc1)C(F)(F)F
COc1cccc(C(=O)NCC(CC2CC2)c2cnc(nc2)C(F)(F)F)c1Cl
COc1cccc(C(=O)NCC(CC2CC2)c2cnc(nc2)C(F)(F)F)c1C
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccncc1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)c1ccncc1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)c1ccncc1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)c1ccncc1
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)CC1CC1
FC(F)(F)c1ncc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCC(F)(F)CC1
CC(CNC(=O)c1cccc(Cl)c1Cl)(CC1CC1)c1cnc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)C1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)C1CCC(F)(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)CC1(CC1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)C1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)C1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)C1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)C1CCC(F)(F)CC1
Fc1cccc(C(=O)NCC(CC2(CC2)C(F)(F)F)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1(CC1)C(F)(F)F
Fc1cccc(C(=O)NCC(CC2(CC2)C(F)(F)F)c2ccc(nc2)C(F)(F)F)c1Cl
CC(C)(O)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)C1CCOCC1
Fc1cccc(Cl)c1C(=O)NCC(C1CCOCC1)c1cnc(nc1)C(F)(F)F
Fc1cccc(C(=O)NCC(C2CCOCC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)c1ccccc1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)c1ccccc1
CC(NC(=O)c1c(F)cccc1Cl)C1(CCOCC1)c1cnc(C)nc1
CC(NC(=O)c1cccc(F)c1Cl)C1(CCOCC1)c1cnc(C)nc1
Cc1ncc(cn1)C1(CNC(=O)c2cccc(Cl)c2Cl)CCOC1
Fc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccc(nc1)C(F)(F)F
Fc1ccc(cc1)C(CNC(=O)c1c(F)cccc1Cl)c1ccc(nc1)C(F)(F)F
Fc1ccc(cc1)C(CNC(=O)c1cccc(F)c1Cl)c1ccc(nc1)C(F)(F)F
Fc1ccc(cc1)C(CNC(=O)c1ccccc1Cl)c1ccc(nc1)C(F)(F)F
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)c1ccncc1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccncc1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)c1ccncc1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)c1ccncc1
Fc1ccc(cc1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C(F)(F)F
Fc1ccc(cc1)C(CNC(=O)c1ccccc1Cl)c1cnc(nc1)C(F)(F)F
CC(NC(=O)c1cccc(Cl)c1Cl)C1(CCC(F)(F)CC1)c1cnc(C)nc1
CC(NC(=O)c1ccccc1Cl)C1(CCC(F)(F)CC1)c1cnc(C)nc1
Fc1ccc(cc1)C(CNC(=O)c1c(F)cccc1Cl)c1cnc(nc1)C(F)(F)F
Fc1ccc(cc1)C(CNC(=O)c1cccc(F)c1Cl)c1cnc(nc1)C(F)(F)F
CC(NC(=O)c1c(F)cccc1Cl)C1(CCC(F)(F)CC1)c1cnc(C)nc1
CC(NC(=O)c1cccc(F)c1Cl)C1(CCC(F)(F)CC1)c1cnc(C)nc1
Fc1cccc(C(=O)NCC(C2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)C1CCC(F)(F)CC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)C1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(C1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
COCCC(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C(F)(F)F
Clc1cccc(C(=O)NCC(c2ccccc2)c2ccnnc2)c1Cl
Clc1ccc(C(=O)NCC(c2ccccc2)c2ccnnc2)c(Cl)c1
FC(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)CC1CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)CC1CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1cccc(F)c1Cl)CC1CC1
COc1cccc(C(=O)NCC(CC2CC2)c2ccc(nc2)C(F)F)c1Cl
CN(C)CC1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1ncn2-c1ccccn1)C(=O)c1cccc(c1F)C(F)(F)F |r|
Clc1cccc(C(=O)N2CCc3c(C2)nnn3-c2ccccc2)c1Cl
CC1N(CCc2c1nnn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCc2c1nnn2-c1nc(C)cc(C)n1)C(=O)c1cccc(Cl)c1Cl
CC1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nnn2-c1cc[nH]n1
CC1N(CCc2c1nnn2-c1nccc(C)n1)C(=O)c1cccc(Cl)c1Cl
Cc1nc2C3CCCC(Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(Cl)c1Cl
Cc1nc2C3CCCC(Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(F)c(Cl)c1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)cc1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1F)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(F)cc1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)cc1F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:21:20:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccc(Cl)cc1Cl |r,THB:21:20:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccc(F)cc1Cl |r,THB:21:20:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccc(F)c(Cl)c1Cl |r,THB:21:20:10.3.9:7.5.6|
Cc1nc2[C@@H]3CCC[C@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:21:20:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)cc1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(F)cc1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(F)c(Cl)c1Cl |r,THB:19:18:10.3.9:7.5.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(c1F)C(F)(F)F |r,THB:19:18:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccnc(c1F)C(F)(F)F |r,THB:19:18:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1ccc(Cl)cc1F |r,THB:19:18:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccn[nH]1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:19:18:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1ccc(F)c(Cl)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1cccc(c1F)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1ccnc(c1F)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1ccc(Cl)cc1F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnn(C)c1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ncccn1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ncccn1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ncccn1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ncccn1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ncccn1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnccn1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnccn1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnccn1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnccn1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1cnccn1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:20:19:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:21:20:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:21:20:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:21:20:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:21:20:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccc(F)cc1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:21:20:10.3.9:5.7.6|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccnn1C)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccnn1C)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccnn1C)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccnn1C)N3C(=O)c1cccc(Cl)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccnn1C)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccccn1)N3C(=O)c1ccnc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccccn1)N3C(=O)c1cccc(c1C)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccccn1)N3C(=O)c1cccc(c1Cl)C(F)(F)F |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccccn1)N3C(=O)c1ccc(Cl)c(F)c1Cl |r,THB:20:19:10.3.9:5.6.7|
Cc1nc2[C@H]3CCC[C@@H](Cc2c(n1)-c1ccccn1)N3C(=O)c1cccc(Cl)c1Cl |r,THB:20:19:10.3.9:5.6.7|
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccccc2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccccc2)c1Cl
CC1Cc2c(CN1C(=O)c1ccc(cc1C)C#N)nc(C)nc2-c1ccn[nH]1
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2cn[nH]c2)c1Cl
Cn1cc(cn1)-c1ncnc2CN(CCc12)C(=O)c1cccc(Cl)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccn[nH]2)c1Cl
Cc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccn[nH]2)c1Cl
Cc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)ncnc2-c1ccn[nH]1
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccccn2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2cnccn2)c1Cl
Cc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)ncnc2-c1cnccn1
Fc1cc(Cl)c(cc1F)C(=O)N1CCc2c(C1)ncnc2-c1cnccn1
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccn[nH]2)c1Cl
Cn1ccc(n1)-c1ncnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
Fc1c(Cl)ccc(C(=O)N2CCc3c(C2)ncnc3-c2ccn[nH]2)c1Cl
Fc1ccc(C(=O)N2CCc3c(C2)ncnc3-c2ccn[nH]2)c(Cl)c1
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-n2cccn2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-n2nccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-n2nccn2)c1Cl
Cc1nc2CN(CCc2c(n1)-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
Cc1nc2CN(CCc2c(n1)-c1ccc(F)cc1)C(=O)c1cccc(Cl)c1Cl
Nc1nc2CN(CCc2c(n1)-c1ccccc1)C(=O)c1cccc(Cl)c1Cl
Cc1nc2CN(CCc2c(n1)-c1ccccc1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(Cl)c1Cl
Cc1nc2CN(CCc2c(n1)-c1[nH]ncc1F)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-c1[nH]ncc1F)C(=O)c1cccc(Cl)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2nccs2)c1Cl
Clc1cccc(C(=O)N2CCc3c(C2)ncnc3-c2nccs2)c1Cl
Cc1nc2CN(CCc2c(n1)-c1[nH]ncc1C(F)(F)F)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2ccc[nH]2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-c2cscn2)c1Cl
Cc1nc2CN(CCc2c(n1)-c1cscn1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-n1nccn1)C(=O)c1cccc(c1)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-n1ccnn1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1ccc(Cl)c(F)c1Cl
CN(C)c1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
Nc1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)nc(nc3-c2ccn[nH]2)C2CC2)c1Cl
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
FC(F)(F)c1nc2CN(CCc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(CN1C(=O)c1cccc(C#N)c1C)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)ncnc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(N)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1ccc(F)c(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1
C[C@H]1Cc2c(CN1C(=O)c1ccc(F)c(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1ccc(F)c(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(Cl)c(F)c1Cl)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(Cl)c(F)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(Cl)c(F)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(C)nc2-c1ccnn1C
CC1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1F)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(F)c(Cl)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(Cl)cc1Cl)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(Cl)cc1Cl)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(Cl)cc1Cl)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(Cl)cc1F)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(Cl)cc1F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(Cl)cc1F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@@H]1Cc2c(CN1C(=O)c1ccc(F)cc1Cl)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(F)cc1Cl)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(F)cc1F)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1ccc(F)cc1F)nc(C)nc2-c1ccn[nH]1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccc(F)cc1F)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1ccc(Cl)cc1)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1ccccc1Cl)nc(C)nc2-c1ccn[nH]1
CCc1nc2CN(C(C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
CCc1nc2CN([C@H](C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCc1nc2CN([C@@H](C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC(C)c1nc2CN(C(C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC(C)c1nc2CN([C@H](C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC(C)c1nc2CN([C@@H](C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CCc1nc2CN(C(C)Cc2c(n1)-c1ccn[nH]1)C(=O)c1ccc(Cl)c(F)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-n2cnnc2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCc3c(C2)ncnc3-n2cncn2)c1Cl
Fc1c(cccc1C(F)(F)F)C(=O)N1CCc2c(C1)ncnc2-c1ccn[nH]1
CC1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(c1Cl)C(F)(F)F
C[C@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(c1Cl)C(F)(F)F |r|
C[C@@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(c1Cl)C(F)(F)F |r|
CC1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(Cl)c1Cl
C[C@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
C[C@@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(F)c(Cl)c1Cl |r|
CC1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(Cl)c(F)c1Cl
C[C@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(Cl)c(F)c1Cl |r|
C[C@@H]1N(CCc2c1ncnc2-c1ccn[nH]1)C(=O)c1ccc(Cl)c(F)c1Cl |r|
C[C@@H]1Cc2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nc(C)nc2-c1ccn(CCF)n1 |r|
COCCn1ccc(n1)-c1nc(C)nc2CN([C@@H](C)Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
COCCn1ccc(n1)-c1nc(C)nc2CN([C@H](C)Cc12)C(=O)c1cccc(c1Cl)C(F)(F)F |r|
Fc1cccc(n1)-c1ncnc2CN(CCc12)C(=O)c1ccc(F)c(Cl)c1Cl
Fc1cccc(n1)-c1ncnc2CN(CCc12)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1Cc2c(CN1C(=O)c1ccc(C)cc1C)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(C)c1C)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1ccc(F)cc1C)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(F)c1C)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(C)c1F)nc(C)nc2-c1ccn[nH]1
CC1Cc2c(CN1C(=O)c1cccc(OC(F)(F)F)c1F)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(OC(F)(F)F)c1)nc(C)nc2-c1ccn[nH]1 |r|
CC1Cc2c(CN1C(=O)c1cccc(F)c1Cl)nc(C)nc2-c1ccn[nH]1
C[C@@H]1Cc2c(CN1C(=O)c1cccc(F)c1Cl)nc(C)nc2-c1ccn[nH]1 |r|
COc1cccc(C(=O)N2Cc3nc(C)nc(-c4ccn[nH]4)c3CC2C)c1C
Cc1ncoc1C(CNC(=O)c1cc(ccc1Cl)-c1ncc(C)cn1)N1CCc2ccccc2C1
[2H]c1nc(C)c(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCC(F)(F)CC1
CC1CC(F)(F)CC(O)(CNC(=O)c2cn(CC(F)(F)F)c3cccc(Cl)c23)C1
C[C@H]1CCC[C@@](O)(CNC(=O)c2cn(CC(F)(F)F)c3cccc(Cl)c23)C1 |r|
C[C@@H]1CCC[C@](O)(CNC(=O)c2cn(CC(F)(F)F)c3cccc(Cl)c23)C1 |r|
OC1(CNC(=O)c2cn(CC(F)(F)F)c3cccc(Cl)c23)CCC(F)(F)CC1
FC(F)(F)Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
NCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
C[C@H]1CCC[C@@](O)(CNC(=O)c2cn(CCC(F)F)c3cccc(Cl)c23)C1 |r|
C[C@@H]1CCC[C@](O)(CNC(=O)c2cn(CCC(F)F)c3cccc(Cl)c23)C1 |r|
FC(F)CCn1cc(C(=O)NCC2CCCC(F)(F)C2)c2c(Cl)cccc12
OC1(CNC(=O)c2cn(CCC(F)F)c3cccc(Cl)c23)CCC(F)(F)CC1
FC(F)CCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
OC1(CNC(=O)c2cn(CCC(F)(F)F)c3cccc(Cl)c23)CCC(F)(F)CC1
FC(F)(F)CCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
COCCn1cc(C(=O)NC[C@]2(O)CCC[C@H](C)C2)c2c(Cl)cccc12 |r|
COCCn1cc(C(=O)NC[C@@]2(O)CCC[C@@H](C)C2)c2c(Cl)cccc12 |r|
COCCn1cc(C(=O)NCCC2(O)CCCC2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(CCC(F)(F)CC2)OC)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(O)CCCCC2O)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(O)CCCCC2)c2c(Cl)cccc12
COCCn1cc(C(=O)NC[C@]2(O)CCCC(F)(F)C2)c2c(Cl)cccc12 |r|
COCCn1cc(C(=O)NC[C@@]2(O)CCCC(F)(F)C2)c2c(Cl)cccc12 |r|
CCC1CCCC(O)(CNC(=O)c2cn(CCOC)c3cccc(Cl)c23)C1
COCCn1cc(C(=O)NCc2cccc3OCCOc23)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2ccccc2C(F)(F)F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2ccccc2F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2ccc(cc2)C(F)(F)F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2ccc3OCOc3c2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2ccco2)c2c(Cl)cccc12
COCCn1cc(C(=O)NC2COc3ccccc3C2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCCc2cccs2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCc2nc3ccccc3s2)c2c(Cl)cccc12
COCCn1cc(C(=O)NC(CO)c2cccc(c2)C(F)(F)F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC(C)c2ccccc2Cl)c2c(Cl)cccc12
COCCn1cc(C(=O)NCCc2ccc(F)cc2Cl)c2c(Cl)cccc12
COCCn1cc(C(=O)NCCc2ccccc2Cl)c2c(Cl)cccc12
COCCn1cc(C(=O)NCCc2ccc(Cl)cc2Cl)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(O)CCCC(F)(F)C2)c2c(Cl)cccc12
COCCn1cc(C(=O)N(C)CC2(CCOCC2)c2ccc(cc2)C(F)(F)F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(CCCCC2)c2ccccc2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
FC(F)(F)C(NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCC1
FC(F)(F)C(NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCCC1
Clc1cccc2n(cc(C(=O)NCC3(CCOCC3)N3CCN(CC3)c3ccccc3)c12)C1COC1
OC1(CCNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC1
CC1CC(O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCC1(F)F
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC(C1)C(F)(F)F
Clc1cccc2n(cc(C(=O)NCC3CCCCC3)c12)C1COC1
CC(O)(CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCC1
CC(C)(CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCC1
Clc1cccc2n(cc(C(=O)NCC3(CCCCC3)N3CCN(CC3)c3ccccc3)c12)C1COC1
FC(F)(F)[C@@H](NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCCC1 |r|
FC(F)(F)C1CCC(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CC1 |(6.53,3.69,;5.44,4.78,;5.84,6.27,;6.93,5.18,;3.95,4.38,;3.55,2.9,;2.07,2.5,;.98,3.59,;-.51,3.19,;-.91,1.7,;-2.4,1.3,;-3.49,2.39,;-2.8,-.19,;-1.89,-1.43,;-2.8,-2.68,;-2.4,-4.17,;-3.17,-5.5,;-1.83,-6.27,;-1.06,-4.94,;-4.26,-2.2,;-5.59,-2.97,;-6.93,-2.2,;-6.93,-.66,;-5.59,.11,;-5.59,1.65,;-4.26,-.66,;1.38,5.07,;2.86,5.47,)|
CC(C)(NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)[C@]12C[C@H]3C[C@H](C[C@H](C3)C1)C2 |r,THB:23:22:24.29.25:28|
Clc1cccc2n(cc(C(=O)NC3(CC3)C3CCCCC3)c12)C1COC1
FC(F)(F)C1CCCC(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC2(CC2)C1
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCCC1
Clc1cccc2n(cc(C(=O)NCC3C[C@@H]4CC[C@H]3C4)c12)C1COC1 |r,THB:12:13:16.17:19|
Clc1cccc2n(cc(C(=O)NC(C3CCCCC3)c3cccs3)c12)C1COC1
C[C@@H](NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)[C@]12C[C@H]3C[C@H](C[C@](O)(C3)C1)C2 |r,TLB:29:19:27:24.23.22,THB:1:19:24:27.21.22,1:19:27:24.23.22,29:23:27:19.20.28,22:23:27.21.20:28|
CC(NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)[C@]12C[C@H]3C[C@H](C[C@H](C3)C1)C2 |r,THB:22:21:23.28.24:27|
OC[C@H](NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)C1CCCCC1 |r|
CC1(C)CCCC(O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCCCC1
FC1(F)CCC[C@@H](CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1 |r|
FC1(F)CCC[C@H](CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1 |r|
Clc1cccc2n(cc(C(=O)NCC3CCCC4(CC4)C3)c12)C1COC1
FC1(F)CCCC(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1
Clc1cccc2n(cc(C(=O)NCC(C3CCCC3)c3ccccc3)c12)C1COC1
CC1(CCNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)OCCO1
Clc1cccc2n(cc(C(=O)NCCOC3CCCC3)c12)C1COC1
FC(F)(F)CCCNC(=O)c1cn(C2COC2)c2cccc(Cl)c12
Clc1cccc2n(cc(C(=O)NCC3CCCOC3)c12)C1COC1
Clc1cccc2n(cc(C(=O)NCC[C@@H]3C[C@H]4C[C@@H]3C=C4)c12)C1COC1 |r,c:20|
FC(F)CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12
FC(F)(F)CCNC(=O)c1cn(C2COC2)c2cccc(Cl)c12
CCOC(C)CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC1
Clc1cccc2n(cc(C(=O)NCCC3CCCC3)c12)C1COC1
CC1CCCC(O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1
O[C@]1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
O[C@@]1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCCC(F)(F)C1
O[C@@H]1CCCC[C@H]1CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12 |r|
O[C@@H]1CCCC[C@@H]1CNC(=O)c1cn(C2COC2)c2cccc(Cl)c12 |r|
CC1CC(F)(F)CC(O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1
C[C@H]1CCC[C@@](O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1 |r|
FC(F)(F)C1CC(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CC(F)(F)C1
OC1(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CCC(F)(F)CC1
C[C@@H]1CCC[C@](O)(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)C1 |r|
FC1(F)CCC(CNC(=O)c2cn(C3COC3)c3cccc(Cl)c23)CC1
FC(F)OCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CC1CC(O)(CNC(=O)c2cn(C3CCCO3)c3cccc(Cl)c23)CCC1(F)F
OC1(CNC(=O)c2cn(C3CCCO3)c3cccc(Cl)c23)CCC(F)(F)CC1
FC1(F)CCC(CNC(=O)c2cn(C3CCCO3)c3cccc(Cl)c23)CC1
OC1(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)CCCC(C1)C(F)(F)F
Clc1cccc2n(cc(C(=O)NCC3CCCCC3)c12)C1CCOC1
CC(O)(CNC(=O)c1cn(C2CCOC2)c2cccc(Cl)c12)C1CCCC1
CC(C)(CNC(=O)c1cn(C2CCOC2)c2cccc(Cl)c12)C1CCCC1
OC1(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)CCC(F)(F)CC1
Clc1cccc2n(cc(C(=O)NCC3C[C@@H]4CC[C@H]3C4)c12)C1CCOC1 |r,THB:12:13:16.17:19|
CC1CC(O)(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)CCC1(F)F
CC1(C)CCCC(O)(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)C1
Clc1cccc2n(cc(C(=O)NCCC3CCCC3)c12)C1CCOC1
CC(NC(=O)c1cn(C2CCOC2)c2cccc(Cl)c12)C1C[C@H]2CC[C@@H]1C2 |r,TLB:1:20:26:24.23|
OCCC(NC(=O)c1cn(C2CCOC2)c2cccc(Cl)c12)C1CCCCC1
CN(C)C(CNC(=O)c1cn(C2CCOC2)c2cccc(Cl)c12)C1CCCCC1
FC(F)(F)C1CCCC(CNC(=O)c2cn(C3CCCO3)c3cccc(Cl)c23)C1
C[C@@H]1CCC[C@](O)(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)C1 |r|
FC1(F)CCC(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)CC1
OC1(CNC(=O)c2cn(CC3CCO3)c3cccc(Cl)c23)CCC(F)(F)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCO3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3(CC3)OC(=O)c3ccccc3)c3cccc(Cl)c23)CC1
CC(C)(C)OC(=O)N1CC(C1)n1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12
CC(C)(C)OC(=O)N1CC(C1)n1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
OC1(CNC(=O)c2cn(C3CCNC3)c3cccc(Cl)c23)CCCC(F)(F)C1
CC(C)(C)OC(=O)N1CCC(C1)n1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CC(C)(C)OC(=O)N1CC[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
FC1(F)CCC(CNC(=O)c2cn(C[C@H]3CCN3)c3cccc(Cl)c23)CC1 |r|
OC1(CNC(=O)c2cn(CC3CCN3)c3cccc(Cl)c23)CCCC(F)(F)C1
OC1(CNC(=O)c2cn(CC3CNC3)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCC(CNC(=O)c2cn(C[C@H]3CNC(=O)O3)c3cccc(Cl)c23)CC1 |r|
FC1(F)CC(Cn2cc(C(=O)NCC3CCC(F)(F)CC3)c3c(Cl)cccc23)C1
CC(C)OCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
O[C@]1(CNC(=O)c2cn(C[C@@H]3CCCO3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
O[C@@]1(CNC(=O)c2cn(C[C@@H]3CCCO3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
OC1(CNC(=O)c2cn(C[C@H]3CCCO3)c3cccc(Cl)c23)CCC(F)(F)CC1 |r|
FC1(F)CCC(CNC(=O)c2cn(C[C@H]3CCCO3)c3cccc(Cl)c23)CC1 |r|
OC1(CNC(=O)c2cn(C[C@H]3CCCO3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
OC1(CNC(=O)c2cn(C[C@@H]3CCCO3)c3cccc(Cl)c23)CCC(F)(F)CC1 |r|
FC1(F)CCC(CNC(=O)c2cn(C[C@@H]3CCCO3)c3cccc(Cl)c23)CC1 |r|
OC1(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)CCCC(C1)C(F)(F)F
CCC1CCCC(O)(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)C1
CC1CC(F)(F)CC(O)(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)C1
OC1(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)CCCC(F)(F)C1
C[C@H]1CCC[C@@](O)(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)C1 |r|
FC(F)(F)C1CC(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)CC(F)(F)C1
OC1(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)CCC(F)(F)CC1
C[C@@H]1CCC[C@](O)(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)C1 |r|
FC1(F)CCC(CNC(=O)c2cn(CC3CCCO3)c3cccc(Cl)c23)CC1
OC1(CNC(=O)c2cn(CC3CCOC3)c3cccc(Cl)c23)CCCC(F)(F)C1
OC1(CNC(=O)c2cn(CC3CCOC3)c3cccc(Cl)c23)CCC(F)(F)CC1
FC1(F)CCC(CNC(=O)c2cn(CCOC3CC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3COCCO3)c3cccc(Cl)c23)CC1
CN1CC[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
CC1(Cn2cc(C(=O)NCC3CCC(F)(F)CC3)c3c(Cl)cccc23)CCN1
CC(C)(C)OC(=O)N1CCC[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
FC1(F)CCC(CNC(=O)c2cn(C[C@H]3CCCN3)c3cccc(Cl)c23)CC1 |r|
OC1(CNC(=O)c2cn(CC3CCCN3)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCCC(CNC(=O)c2cn(CC3CCCN3)c3cccc(Cl)c23)C1
CC1CC(CNC(=O)c2cn(CC3CCCN3)c3cccc(Cl)c23)CC(F)(F)C1
CC(C)(C)OC(=O)N1CCCC1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
OC1(CNC(=O)c2cn(CC3CCNC3)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCC(CNC(=O)c2cn(CC3CCNC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(C[C@H]3CCC(=O)N3)c3cccc(Cl)c23)CC1 |r|
CCN(C)C(=O)Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CC(C)(C)OC(=O)N1CCOCC1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
OC1(CNC(=O)c2cn(CC3CCCCO3)c3cccc(Cl)c23)CCC(F)(F)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCCCO3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCOCC3)c3cccc(Cl)c23)CC1
CC(C)(C)OC(=O)N1CCC[C@H]1Cn1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
CN1CCCC1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
FC1(F)CCC(CNC(=O)c2cn(C3CN(C3)C3CC3)c3cccc(Cl)c23)CC1
OC1(CNC(=O)c2cn(C3CC4(CNC4)C3)c3cccc(Cl)c23)CCC(F)(F)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCCCN3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCCNC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3CCNCC3)c3cccc(Cl)c23)CC1
O[C@]1(CNC(=O)c2cn(CCN3CCCC3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
O[C@@]1(CNC(=O)c2cn(CCN3CCCC3)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
OC1(CNC(=O)c2cn(CCN3CCCC3)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCC(CNC(=O)c2cn(CCN3CCCC3)c3cccc(Cl)c23)CC1
CN1CC(F)(F)C[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
CC(=O)N1CC[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
CN1[C@@H](Cn2cc(C(=O)NCC3CCC(F)(F)CC3)c3c(Cl)cccc23)CCC1=O |r|
CN1CCOC(Cn2cc(C(=O)NCC3CCC(F)(F)CC3)c3c(Cl)cccc23)C1
CN1CCOCC1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
FC1(F)CCC(CNC(=O)c2cn(CC(=O)N3CCCC3)c3cccc(Cl)c23)CC1
O[C@]1(CNC(=O)c2cn(CCN3CCCC3=O)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
O[C@@]1(CNC(=O)c2cn(CCN3CCCC3=O)c3cccc(Cl)c23)CCCC(F)(F)C1 |r|
OC1(CNC(=O)c2cn(CCN3CCCC3=O)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCC(CNC(=O)c2cn(CCN3CCCC3=O)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC(=O)N3CCOCC3)c3cccc(Cl)c23)CC1
CC(C)N1CC[C@H]1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
OC1(CNC(=O)c2cn(CCN3CCCCC3)c3cccc(Cl)c23)CCCC(F)(F)C1
FC1(F)CCC(CNC(=O)c2cn(CCN3CCCCC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC(=O)N3CCCCC3)c3cccc(Cl)c23)CC1
CC(C)N1CCCC1Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
FC1(F)CCC(CNC(=O)c2cn(CC3CCCN3C3CC3)c3cccc(Cl)c23)CC1
OCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(cccc12)C(F)(F)F
COCCn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(cccc12)C(F)(F)F
CC(C(=O)N(C)C)n1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CC(C)N(C)C(=O)Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CN(C)C(=O)Cn1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12
CCN(CC)C(=O)Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
CN(C)C(=O)Cn1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
Cc1nc2CN(CCc2c(n1)-n1nccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
[O-]S(=O)(=O)c1cc(c2c(NC(=O)c3ccc(NC(=O)c4ccc(NC(=O)Nc5ccc(cc5)C(=O)Nc5ccc(cc5)C(=O)Nc5ccc(c6cc(cc(c56)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O)cc4)cc3)ccc(c2c1)S([O-])(=O)=O)S([O-])(=O)=O
Cc1ccc(cc1NC(=O)c1cccc(NC(=O)Nc2cccc(c2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c3cc(cc(c23)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O)c1)C(=O)Nc1ccc(c2cc(cc(c12)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccccc1)S(=O)(=O)c1cccc2cnccc12 |r|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=C)NNc1c(Cl)cncc1Cl |TLB:7:1:8.5.4:10,THB:2:1:8:4.3.10,2:3:8:11.1.7,7:5:10:11.1.2,0:1:8.5.4:10,0:1:8:4.3.10|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1ccnc2ccccc12 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1cnc2ccccc2c1 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1ccc2ccccc2n1 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1ccnc2c(Cl)cccc12 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1ncnc2ccccc12 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1ncnc2nc[nH]c12 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1nc(Cl)nc2nc[nH]c12 |TLB:7:1:10:8.4.5,THB:0:1:10:8.4.5,2:1:8:10.3.4,2:3:8:11.1.7,7:5:10:11.1.2|
Cc1ncc(cn1)[C@@H](CNC(=O)c1cccc(Cl)c1Cl)CC1CC1 |r|
FC(F)(F)c1ncc(cn1)[C@@H](CNC(=O)c1cccc(Cl)c1Cl)C1CCOCC1 |r|
Fc1cccc(Cl)c1C(=O)NC[C@H](C1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F |r|
Fc1cccc(Cl)c1C(=O)NC[C@@H](C1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F |r|
COc1ccc(F)c(c1)C(=O)NCC1(CCC(F)(F)CC1)c1ccc(F)nc1
Clc1cccc(C(=O)NC2CC2)c1Cl
[O-][n+]1cccc2C(COc12)NC(=O)Cc1cccc(c1Cl)C(F)(F)F
[O-][n+]1ccc2C(COc2c1)NC(=O)Cc1cccc(c1Cl)C(F)(F)F
Clc1ccc(CC(=O)NC2COc3ncccc23)c(Cl)c1
Fc1ccc(CC(=O)NC2COc3ncccc23)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2ncccc12
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1CCOc2ncccc12
Clc1ccc(CC(=O)NC2CCOc3ncccc23)c(Cl)c1
O=C(Cc1ccccc1C#N)NC1COc2ncccc12
Cc1ccccc1CC(=O)NC1COc2ncccc12
COc1ccccc1CC(=O)NC1COc2ncccc12
O=C(Cc1ccc(cc1)C#N)NC1COc2ncccc12
Cc1ccc(CC(=O)NC2COc3ncccc23)cc1
Clc1ccc(CC(=O)NC2COc3ncccc23)cc1
FC(F)(F)c1ccc(CC(=O)NC2COc3ncccc23)cc1
Fc1ccc(CC(=O)NC2COc3ncccc23)c(F)c1
Fc1ccc(CC(=O)NC2COc3ncccc23)c(c1)C(F)(F)F
COc1ccc(CC(=O)NC2COc3ncccc23)c(OC)c1
COc1ccc(CC(=O)NC2COc3ncccc23)c(F)c1
Clc1ccc(CC(=O)NC2COc3ncccc23)cc1Cl
Fc1cc(F)c(CC(=O)NC2COc3ncccc23)c(F)c1
CC(C(=O)NC1COc2ncccc12)c1ccc(Cl)cc1
Clc1ccc(c(Cl)c1)C1(CC1)C(=O)NC1COc2ncccc12
Fc1ccc(c(Cl)c1)C1(CCCC1)C(=O)NC1COc2ncccc12
CC(C)(C(=O)NC1COc2ncccc12)c1ccc(Cl)cc1
Clc1ccc(CCC(=O)NC2COc3ncccc23)c(Cl)c1
CCc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2ncccc12
FC(F)(F)c1cc(Cl)cc(Cl)c1CC(=O)NC1COc2ncccc12
FC(F)(F)c1cccc(CC(=O)NC2COc3ncccc23)c1Cl
FC(F)(F)c1cc(Cl)ccc1CC(=O)NC1COc2ncccc12
O=C(Cc1ccc(Oc2ccccc2)cc1)NC1COc2ncccc12
Clc1cc(Cl)c(CC(=O)NC2COc3ncccc23)c(c1)C#N
Fc1ccc(CC(=O)NC2CCOc3ncccc23)c(Cl)c1
Clc1cc(Cl)c(CC(=O)NC2COc3ncccc23)c(c1)C1CC1
Cc1c(Cl)cc(c(CC(=O)NC2COc3ncccc23)c1F)C(F)(F)F
Fc1cc(CC(=O)NC2COc3ncccc23)c(Cl)cc1Cl
Cc1ccc(F)c(CC(=O)NC2COc3ncccc23)c1Cl
FC(F)(F)c1ccc(Cl)cc1CC(=O)NC1COc2ncccc12
Clc1ccccc1CC(=O)NC1CCOc2ncccc12
O=C(Cc1ccc(cc1)C#N)NC1CCOc2ncccc12
FC(F)(F)c1ccc(CC(=O)NC2CCOc3ncccc23)cc1
FC(F)(F)c1cccc(CC(=O)NC2CCOc3ncccc23)c1
O=C(Cc1ccc(Oc2ccccc2)cc1)NC1CCOc2ncccc12
FC(F)(F)c1cccc(CC(=O)NC2CCOc3ncccc23)c1Cl
Fc1cccc(Cl)c1CC(=O)NC1CCOc2ncccc12
Fc1ccc(CC(=O)NC2CCOc3ncccc23)c(F)c1
Fc1ccc(CC(=O)NC2CCOc3ncccc23)c(c1)C(F)(F)F
FC(F)(F)c1cc(Cl)ccc1CC(=O)NC1CCOc2ncccc12
Clc1cccc(CC(=O)NC2CCOc3ncccc23)c1Cl
Clc1ccc(CC(=O)NC2CCOc3ncccc23)cc1Cl
FC(F)(F)c1cc(Cl)cc(Cl)c1CC(=O)NC1CCOc2ncccc12
Fc1cc(CC(=O)NC2CCOc3ncccc23)c(Cl)cc1Cl
Clc1ccc(c(Cl)c1)C1(CC1)C(=O)NC1CCOc2ncccc12
Fc1ccc(c(Cl)c1)C1(CCCC1)C(=O)NC1CCOc2ncccc12
Clc1ncccc1CC(=O)NC1CCOc2ncccc12
Cc1ccc(OCC(=O)NC2CCOc3ncccc23)c(C)n1
Cc1cc(CC(=O)NC2CCOc3ncccc23)on1
Cc1ccnn1CC(=O)NC1CCOc2ncccc12
CC(C(=O)NC1CCOc2ncccc12)c1ccc(Cl)cc1
Clc1ccc(CCC(=O)NC2CCOc3ncccc23)c(Cl)c1
Clc1cccc(CC(=O)NC2COc3ncccc23)c1Cl
Fc1ccc(Cl)c(Cl)c1CC(=O)NC1COc2ncccc12
Fc1cccc(c1CC(=O)NC1COc2ncccc12)C(F)(F)F
Fc1cc(CC(=O)NC2COc3ncccc23)ccc1OC(F)(F)F
Fc1cc(Cl)cc(Cl)c1CC(=O)NC1CCOc2ncccc12
FC(F)(F)c1ccc(Cl)c(Cl)c1CC(=O)NC1COc2ncccc12
FC(F)(F)c1ccc(Cl)c(CC(=O)NC2COc3ncccc23)c1Cl
Clc1c(CC(=O)NC2COc3ncccc23)cccc1C#N
Fc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2ncccc12
Fc1c(Cl)ccc(Cl)c1CC(=O)NC1COc2ncccc12
Fc1ccc(F)c(CC(=O)NC2COc3ncccc23)c1Cl
OCC(C(=O)NC1COc2ncccc12)c1ccc(Cl)cc1Cl
NC(=O)c1cccc(CC(=O)NC2COc3ncccc23)c1Cl
Clc1ccc(C(CN2CCCC2)C(=O)NC2COc3ncccc23)c(Cl)c1
Fc1ccc(CCCC(=O)NC2COc3ncccc23)cc1
Clc1ccc(CC(=O)NC2COc3cnccc23)c(Cl)c1
CCC(C(=O)NC1COc2ncccc12)c1ccc(Cl)cc1Cl
CC(C(=O)NC1COc2ncccc12)c1ccc(Cl)cc1Cl
FC(F)(F)c1cccc(CC(=O)NC2COc3cnccc23)c1Cl
FC(F)(F)c1ccc(CC(=O)NC2COc3ncccc23)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2cnccc12
Fc1c(CC(=O)NC2COc3ncccc23)cccc1C(F)(F)F
CC(C(=O)NC1COc2ncccc12)c1cccc(c1Cl)C(F)(F)F
Clc1cc(ccc1CC(=O)NC1COc2ncccc12)C#N
FC(F)(F)c1c(Cl)cccc1CC(=O)NC1COc2ncccc12
Cc1nccc2C(COc12)NC(=O)Cc1ccc(Cl)cc1Cl
OCc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2ncccc12
Clc1ccc(CC(=O)NC2COc3c2ccnc3C2CC2)c(Cl)c1
COc1nccc2C(COc12)NC(=O)Cc1ccc(Cl)cc1Cl
Clc1ccc(CC(=O)NC2COc3c2ccnc3Cl)c(Cl)c1
Fc1ccc(CC(=O)NC2COc3ncccc23)c(Cl)c1C#N
FC(F)(F)Oc1cccc(CC(=O)NC2COc3ncccc23)c1Cl
FC(F)(F)c1cccc(CC(=O)NC2COc3nnccc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2nnccc12
CC(=O)c1cccc(CC(=O)NC2COc3ncccc23)c1Cl
Clc1ccc(CC(=O)NC2COc3ncccc23)c(Cl)c1C#N
FC(F)(F)c1c(CC(=O)NC2COc3ncccc23)cccc1C#N
FC(F)c1cccc(CC(=O)NC2COc3ncccc23)c1Cl
FC(F)(F)c1cccc(CC(=O)NC2COc3cnc(Cl)cc23)c1Cl
Clc1ccc(CC(=O)NC2COc3cnc(Cl)cc23)c(Cl)c1
Cc1cc2C(COc2cn1)NC(=O)Cc1cccc(c1Cl)C(F)(F)F
Cc1cncc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
Clc1cc2CCC(C(=O)NC3COc4ncccc34)c2c(Cl)c1
Cc1cncc2OCC(NC(=O)Cc3c(C)cc(Cl)cc3Cl)c12
FC(F)(F)c1cccc(CC(=O)NC2COc3cncc(C4CC4)c23)c1Cl
Cc1ccc2C(COc2n1)NC(=O)Cc1c(C)cc(Cl)cc1Cl
Cc1ccc2C(COc2n1)NC(=O)Cc1cccc(c1Cl)C(F)(F)F
COc1cc(C)nc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
CCOc1cc(C)nc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
Cc1ccnc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
Cc1ccnc2OCC(NC(=O)Cc3c(C)cc(Cl)cc3Cl)c12
COc1ccnc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
Clc1ccc(OCC(=O)NC2COc3ncccc23)c(Cl)c1
Clc1ccc(OCC(=O)NC2COc3ncccc23)cc1Cl
Cc1ccc(OCC(=O)NC2COc3ncccc23)c(C)c1
FC(F)(F)c1cccc(CC(=O)NC2COc3nc(Cl)ccc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2nc(Cl)ccc12
Clc1ccc2C(CCc2c1)C(=O)NC1COc2ncccc12
Clc1ccc2CC(Cc2c1)C(=O)NC1COc2ncccc12
Cc1cc(Cl)cc(Cl)c1CC(=O)NC1COc2nccc(c12)C(F)(F)F
FC(F)(F)c1ccnc2OCC(NC(=O)Cc3cccc(c3Cl)C(F)(F)F)c12
Clc1ccc(CNC(=O)C2COc3ncsc23)cc1
Clc1ccc(CNC(=O)C2COc3ncsc23)c(Cl)c1
Fc1ccc(CNC(=O)C2COc3ncsc23)c(Cl)c1
Clc1ccc(CNC(=O)C2COc3ncsc23)cc1Cl
Clc1cc(Cl)c(CNC(=O)C2COc3ncsc23)c(Br)c1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncsc12
Clc1ccc(CCNC(=O)C2COc3ncsc23)c(Cl)c1
Clc1ccc(CCCNC(=O)C2COc3ncsc23)c(Cl)c1
OC[C@@H](NC(=O)C1COc2ncsc12)c1ccc(Cl)cc1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncsc12
Clc1cc2CCC(NC(=O)C3COc4ncsc34)c2c(Cl)c1
Clc1cc(Cl)c(CNC(=O)C2COc3ncsc23)c(c1)C1CC1
FC(F)(F)c1cccc(CNC(=O)C2COc3ncsc23)c1Cl
FC(F)(F)c1c(Cl)cccc1CNC(=O)C1COc2ncsc12
OCCOCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncsc12
O=C(NCc1ccc(Oc2ccccc2)cc1)C1COc2ncsc12
Clc1ccc(CNC(=O)C2CCc3ncsc23)c(Cl)c1
Fc1ccc(CNC(=O)C2CCc3ncsc23)c(Cl)c1
Clc1cc(Cl)c(CNC(=O)C2CCc3ncsc23)c(Br)c1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCc2ncsc12
Clc1ccc(CCNC(=O)C2CCc3ncsc23)c(Cl)c1
Clc1c(CNC(=O)C2CCc3ncsc23)cccc1C#N
Clc1ccc(CCCNC(=O)C2CCc3ncsc23)c(Cl)c1
OC[C@@H](NC(=O)C1CCc2ncsc12)c1ccc(Cl)cc1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCc2ncsc12
COc1cc(Cl)cc(Cl)c1CNC(=O)C1CCc2ncsc12
Clc1cc2CCC(NC(=O)C3CCc4ncsc34)c2c(Cl)c1
FC(F)(F)c1cccc(CNC(=O)C2CCc3ncsc23)c1Cl
Fc1cc(CNC(=O)C2CCc3ncsc23)ccc1OC(F)(F)F
CN(Cc1ccc(Cl)cc1)C(=O)C1CCOc2ncsc12
Clc1ccc(CNC(=O)C2CCOc3ncsc23)c(Cl)c1
Fc1ccc(CNC(=O)C2CCOc3ncsc23)c(Cl)c1
Clc1cccc(CNC(=O)C2CCOc3ncsc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2ncsc12
Clc1ccc(CCNC(=O)C2CCOc3ncsc23)c(Cl)c1
Clc1c(CNC(=O)C2CCOc3ncsc23)cccc1C#N
FC(F)(F)c1ccc(CNC(=O)C2CCOc3ncsc23)cc1
Clc1ccc(CCCNC(=O)C2CCOc3ncsc23)c(Cl)c1
OC[C@@H](NC(=O)C1CCOc2ncsc12)c1ccc(Cl)cc1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2ncsc12
Clc1cc2CCC(NC(=O)C3CCOc4ncsc34)c2c(Cl)c1
FC(F)(F)c1cccc(CNC(=O)C2CCOc3ncsc23)c1Cl
OCCOc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2ncsc12
Fc1cc(CNC(=O)C2CCOc3ncsc23)ccc1OC(F)(F)F
O=C(NCc1ccc(Oc2ccccc2)cc1)C1CCOc2ncsc12
Clc1ccc(CNC(=O)C2CCCc3ncsc23)cc1
CN(Cc1ccc(Cl)cc1)C(=O)C1CCCc2ncsc12
Cc1c(Cl)cccc1CNC(=O)C1CCCc2ncsc12
Nc1nc2CCCC(C(=O)NCc3ccc(Cl)cc3Cl)c2s1
Cc1nc2CCCC(C(=O)NCc3ccc(Cl)cc3Cl)c2s1
Clc1ccc(CNC(=O)C2CCCc3nc(Br)sc23)c(Cl)c1
Clc1ccc(CNC(=O)C2CCCc3ncsc23)c(Cl)c1
Fc1ccc(CNC(=O)C2CCCc3ncsc23)c(Cl)c1
Clc1cccc(CNC(=O)C2CCCc3ncsc23)c1Cl
O=C(NC1CCc2ccccc12)C1CCCc2ncsc12
C[C@@H](NC(=O)C1CCCc2ncsc12)c1ccc(Cl)cc1Cl
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2nc(sc12)-c1ccccc1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2nc(sc12)C(F)(F)F
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2nc(N)sc12
Cc1nc2CCCC(C(=O)NCc3c(C)cc(Cl)cc3Cl)c2s1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2nc(Br)sc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2ncsc12
Clc1ccc(CCNC(=O)C2CCCc3ncsc23)c(Cl)c1
OC[C@@H](NC(=O)C1CCCc2ncsc12)c1ccc(Cl)cc1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2ncsc12
FC(F)(F)c1cccc(CNC(=O)C2CCCc3nc(Br)sc23)c1Cl
FC(F)(F)c1cccc(CNC(=O)C2CCCc3ncsc23)c1Cl
COCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCc2ncsc12
Fc1cc(CNC(=O)C2CCCc3ncsc23)ccc1OC(F)(F)F
O=C(NCc1ccc(Oc2ccccc2)cc1)C1CCCc2ncsc12
Nc1nc2CCCCC(C(=O)NCc3ccc(Cl)cc3Cl)c2s1
Clc1ccc(CNC(=O)C2CCCCc3ncsc23)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCCc2nc(N)sc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCCCc2ncsc12
OC[C@@H](NC(=O)C1CCCCc2ncsc12)c1ccc(Cl)cc1Cl
OCC(NC(=O)C1COc2ncsc12)C1CCCCCC1
Clc1ccc(cn1)C1(CNC(=O)C2COc3ncsc23)CCCCC1
Cc1ncc(cn1)C(CNC(=O)C1COc2ncsc12)N1CCC(F)(F)CC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)C1COc2ncsc12)N1CCOCC1
OC[C@@H](NC(=O)C1CCc2ncsc12)C1CCCCC1
Cc1ncc(cn1)C(CNC(=O)C1CCc2ncsc12)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)C1CCc2ncsc12)N1CCC(F)(F)CC1
OC[C@@H](NC(=O)C1CCOc2ncsc12)C1CCCCC1
Cc1ncc(cn1)C(CNC(=O)C1CCOc2ncsc12)N1CCOCC1
FC1(F)CCN(CC1)C(CNC(=O)C1CCOc2ncsc12)c1ccc(Cl)nc1
C[C@@H](NC(=O)C1CCCc2ncsc12)C1CCCCC1
OC[C@@H](NC(=O)C1CCCc2ncsc12)C1CCCCC1
Clc1ccc(cn1)C1(CNC(=O)C2CCCc3ncsc23)CCCCC1
FC1(F)CCC(CNC(=O)C2CCCc3ncsc23)(CC1)c1ccc(Cl)nc1
FC(F)(F)c1ncc(cn1)C(CNC(=O)C1CCCc2ncsc12)N1CCOCC1
OC[C@@H](NC(=O)C1CCCCc2ncsc12)C1CCCCC1
OC[C@@H](NC(=O)C1COc2ncccc12)C1CCCCC1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
Clc1ccc(CNC(=O)C2COc3ncccc23)c(Cl)c1
OC[C@@H](NC(=O)C1COc2ncccc12)c1ccc(Cl)cc1Cl
OC[C@@H](NC(=O)[C@H]1CCOc2ncccc12)C1CCCCC1
OC[C@@H](NC(=O)[C@H]1CCOc2ncccc12)c1ccc(Cl)cc1Cl
OC1(CNC(=O)C2CCOc3ncccc23)CCCCC1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)COc2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCOc2ncccc12
OCC(NC(=O)C1COc2ncccc12)C1CCCCCC1
Fc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
FC(F)(F)c1cccc(CNC(=O)C2COc3ncccc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2ncccc12
Clc1ccc(cn1)C1(CNC(=O)C2CCOc3ncccc23)CCCCC1
FC1(COc2ncccc12)C(=O)NCc1cccc(Cl)c1Cl
Clc1cc(Cl)c(CNC(=O)C2COc3ncccc23)c(c1)C1CC1
CCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
Clc1cc(Cl)c(CNC(=O)C2COc3ncccc23)c(C=C)c1
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
COc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
Cc1ncc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCOCC1
Cc1c(Cl)cccc1CNC(=O)C1CCOc2ncccc12
Fc1ccc(CNC(=O)C2CCOc3ncccc23)c(Cl)c1
O=C(NCc1ccc(Oc2ccccc2)cc1)C1CCOc2ncccc12
Clc1cccc(CNC(=O)C2CCOc3ncccc23)c1Cl
Clc1ccc(CNC(=O)C2CCOc3ncccc23)cc1
FC(F)(F)c1ccc(CNC(=O)C2CCOc3ncccc23)cc1
CN(Cc1ccc(Cl)cc1)C(=O)C1CCOc2ncccc12
Clc1ccc(CCNC(=O)C2CCOc3ncccc23)c(Cl)c1
Clc1ccc(CNC(=O)C2CCOc3ncccc23)c(Cl)c1
FC(F)(F)c1cccc(CNC(=O)C2CCOc3ncccc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2c1ccc[n+]2[O-]
Cc1c(Cl)cccc1CNC(=O)C1COc2ncccc12
Fc1ccc(CNC(=O)C2COc3ncccc23)c(Cl)c1
O=C(NCc1ccc(Oc2ccccc2)cc1)C1COc2ncccc12
Clc1cccc(CNC(=O)C2COc3ncccc23)c1Cl
Clc1ccc(CNC(=O)C2COc3ncccc23)cc1
FC(F)(F)c1ccc(CNC(=O)C2COc3ncccc23)cc1
CN(Cc1ccc(Cl)cc1)C(=O)C1COc2ncccc12
Clc1ccc(CCNC(=O)C2COc3ncccc23)c(Cl)c1
OCCOc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCOc2ncccc12
OCC(NC(=O)C1CCOc2ncccc12)C1CCCCCC1
Fc1cc(CNC(=O)C2CCOc3ncccc23)ccc1OC(F)(F)F
O=C(NCC1(CCCCC1)c1ccccc1)C1CCOc2ncccc12
FC(F)(F)c1cccc(CNC(=O)C2(F)COc3ncccc23)c1Cl
Clc1c(CNC(=O)C2COc3ncccc23)cccc1C#N
Fc1cc(CNC(=O)C2COc3ncccc23)ccc1OC(F)(F)F
Clc1ccc(c(Cl)c1)C1(CC1)NC(=O)C1CCOc2ncccc12
FC(F)(F)c1ncc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCOCC1
Clc1cc(ccc1CNC(=O)C1COc2ncccc12)C#N
FC(F)(F)c1ncc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCC(F)(F)CC1
NC(=O)C1(CCCC1)NC(=O)C1COc2ncccc12
O=C(NC1CC1c1ccccc1)C1COc2ncccc12
O[C@@H]1Cc2ccccc2[C@@H]1NC(=O)[C@@H]1COc2ncccc12
NC(=O)C1CCCCC1NC(=O)C1COc2ncccc12
FC1(F)CCC(CNC(=O)C2CCOc3ncccc23)(CC1)c1ccc(Cl)nc1
FC(F)(F)c1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
O=C(N[C@@H]1CCc2ccccc12)[C@@H]1COc2ncccc12
C[C@@H](NC(=O)C1COc2ncccc12)c1ccc(Cl)cc1Cl
COCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
FC(F)(F)c1c(Cl)cccc1CNC(=O)C1COc2ncccc12
FC1(F)CCN(CC1)C(CNC(=O)C1COc2ncccc12)c1ccc(Cl)nc1
Clc1cc2CCC(NC(=O)C3COc4ncccc34)c2c(Cl)c1
FC(F)(F)c1ccc(cc1)C(CNC(=O)C1COc2ncccc12)N1CCC(F)(F)CC1
Clc1cc(Cl)c(CNC(=O)C2COc3ncccc23)c(Br)c1
COc1ccc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCOCC1
O=C(NC1CC(=O)c2ccccc12)C1COc2ncccc12
Cc1ccc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCOCC1
O=C(NCC(N1CCOCC1)c1cnc(nc1)C1CC1)C1COc2ncccc12
FC(F)(F)c1ccc(cn1)C(CNC(=O)C1COc2ncccc12)N1CCOCC1
OCCOCc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2ncccc12
Clc1cc2C(CCc2c(Cl)c1)NC(=O)C1COc2ncccc12
Clc1ccc2C(CCc2c1)NC(=O)C1COc2ncccc12
Clc1cccc2CCC(NC(=O)C3COc4ncccc34)c12
FC(F)(F)c1ccc(CNC(=O)C2COc3ncccc23)c(Cl)c1
Clc1ccc(CCCNC(=O)C2COc3ncccc23)c(Cl)c1
O=C(N[C@@H]1CCCc2ccccc12)C1COc2ncccc12
Clc1cccc2CCC[C@@H](NC(=O)C3COc4ncccc34)c12
Brc1cccc2CCC(NC(=O)C3COc4ncccc34)c12
Clc1cc(Cl)c(CNC(=O)C2COc3ncccc23)c(Cl)c1
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1COc2c1ccc[n+]2[O-]
Clc1cc2CC(NC(=O)C3COc4ncccc34)C(=O)c2c(Cl)c1
OCc1cc(Cl)ccc1CNC(=O)C1COc2ncccc12
OCc1cccc(Cl)c1CNC(=O)C1COc2ncccc12
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(c1Cl)C(F)(F)F)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1cccc(c1Cl)C(F)(F)F)N1CCOCC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
Fc1cccc(F)c1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
CS(=O)(=O)c1ccc(Cl)c(c1)C(=O)NCC(N1CCOCC1)c1ccc(Cl)cc1
COc1ccccc1C(=O)NCC(N1CCOCC1)c1ccc(nc1)C(F)(F)F
Clc1ccc(cc1)C(CNC(=O)c1cc(ccc1Cl)C#N)N1CCOCC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
Fc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(nc2)C(F)(F)F)c1Cl
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1ccc(nc1)C(F)(F)F
Cc1ccc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ccc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
Fc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
COc1cccc(C(=O)NCC(N2CCOCC2)c2cnc(nc2)C(F)(F)F)c1Cl
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(nc2)C(F)(F)F)c1C
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(F)cc2)c1Cl
COc1cccc(C(=O)NCC(N2CCOCC2)c2ccc(Cl)cc2)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCCC(F)(F)C1
Cc1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCCC(F)(F)C1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCCC(F)(F)C1
FC1CCN(CC1)C(CNC(=O)c1ccccc1Cl)c1cnc(nc1)C(F)(F)F
FC1CCN(CC1)C(CNC(=O)c1c(Cl)cccc1Cl)c1cnc(nc1)C(F)(F)F
FC1CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C(F)(F)F
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)CC1
Cn1cc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Cn1cc(cn1)C(CNC(=O)c1cc(F)cc(Cl)c1Cl)N1CCC(F)(F)CC1
Cn1cc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Fc1ccc(Cl)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCCCC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCCCC1
Fc1cc(Cl)c(Cl)c(c1)C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
Cn1cc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
FC(F)c1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCOCC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(C)nc2)c1Cl
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)ccc(F)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cc(F)cc(Cl)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)c1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCOCC1
FC(F)c1ncc(cn1)C(CNC(=O)c1cccc(F)c1Cl)N1CCOCC1
FC1(F)CCN(CC1)C(CNC(=O)c1ccccc1Cl)c1cnc(nc1)C1CC1
FC1(F)CCN(CC1)C(CNC(=O)c1c(Cl)cccc1Cl)c1cnc(nc1)C1CC1
CCc1ncc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
Cc1ncc(cn1)C(CNC(=O)c1cccc(OC(F)F)c1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
CCc1ncc(cn1)C(CNC(=O)c1c(F)cccc1Cl)N1CCC(F)(F)CC1
FC1(F)CCN(CC1)C(CNC(=O)c1cccc(Cl)c1Cl)c1cnc(nc1)C1CC1
Fc1cccc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C1CC1
Fc1cc(F)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
COc1ccc(F)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c1Cl
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1ccc(Cl)cc1Cl)N1CCC(F)(F)CC1
Fc1cc(Cl)cc(Cl)c1C(=O)NCC(N1CCC(F)(F)CC1)c1cnc(nc1)C(F)(F)F
COc1ccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
COc1ccc(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1OC
Fc1cc(Cl)c(C(=O)NCC(N2CCC(F)(F)CC2)c2cnc(nc2)C(F)(F)F)c(Cl)c1
Cc1ncc(cn1)C(CNC(=O)c1cccc(OC(F)(F)F)c1Cl)N1CCC(F)(F)CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1ccccc1Cl)N1CCC(F)(F)CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1cccc(Cl)c1Cl)N1CCC(F)(F)CC1
FC(F)c1ccc(cn1)C(CNC(=O)c1c(Cl)cccc1Cl)N1CCC(F)(F)CC1
COc1cccc(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(nc2)C(F)F)c1Cl
CC1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC(N1C=Cc2c(ncn2-c2ccc(F)cn2)C1C)c1cccc(c1Cl)C(F)(F)F |c:3|
CC1C(CCc2c1nnn2-c1ncc(F)c(C)n1)C(=O)c1cccc(c1Cl)C(F)(F)F
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccc(F)cc1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1cccc(F)c1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccccc1F
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1cc(F)cc(F)c1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(F)cc1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccc(F)c1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccccc1F
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(F)cc(F)c1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(F)c(F)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccc(F)cc1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1cccc(F)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1cc(F)cc(F)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccc(F)c(F)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccc(F)cc1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1cccc(F)c1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccccc1F
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccc(F)c(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccccc1F
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccc(F)c(F)c1
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccc(F)cc1
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccccc1F
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccc(Cl)cc1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccc(F)c(F)c1
Cc1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(Cl)cc1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccc(Cl)cc1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccccc1F
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccc(Cl)cc1
Cc1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1cc(F)cc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccccc1F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1cc(F)cc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)OCc1ccc(F)c(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(Cl)cc1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(F)cc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)OCc1ccccc1F
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1ccc(Cl)cc1
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1cccc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1cccc2ncccc12)N1CCC(CC1)Oc1cc(F)cc(F)c1
Cc1ncsc1C(CN)N1CCC(CC1)Oc1ccccc1
CC1Cc2c(CN1C(=O)c1cccc(c1C)C(F)(F)F)nnn2C1=NN=CC1 |c:28,t:26|
C[C@H]1CC2=C(CN1C(=O)c1cccc(c1)C(F)(F)F)NNN2c1ncc(F)cn1 |r,c:3|
COCCn1cc(C(=O)NC(CO)c2cccc(c2Cl)C(F)(F)F)c2c(Cl)cccc12
COCCn1cc(C(=O)NCC2(CCOCC2)c2ccc(cc2)C(F)(F)F)c2c(Cl)cccc12
CC(NC(=O)c1cn(C2COC2)c2cccc(Cl)c12)[C@]12C[C@H]3C[C@H](C[C@](O)(C3)C1)C2 |r|
FC1(F)CCC(CNC(=O)c2cn(CC3CCCN3)c3cccc(Cl)c23)CC1
FC(F)(F)C1CCCC(CNC(=O)c2cn(C3CCOC3)c3cccc(Cl)c23)C1
OC1(Cn2cc(C(=O)NCC3CCC(F)(F)CC3)c3c(Cl)cccc23)CC1
CN1CC(C1)n1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12
CN1CC(C1)n1cc(C(=O)NCC2CCC(F)(F)CC2)c2c(Cl)cccc12
FC1(F)CCC(CNC(=O)c2cn(C3CCNC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(C[C@@H]3CCN3)c3cccc(Cl)c23)CC1 |r|
FC1(F)CCC(CNC(=O)c2cn(CC3CCOC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(C[C@@H]3CCCN3)c3cccc(Cl)c23)CC1 |r|
FC1(F)CCC(CNC(=O)c2cn(CC(=O)N3CCC3)c3cccc(Cl)c23)CC1
FC1(F)CCC(CNC(=O)c2cn(CC3COCCN3)c3cccc(Cl)c23)CC1
OC1(CNC(=O)c2cn(CC3COCCN3)c3cccc(Cl)c23)CCC(F)(F)CC1
CN1CCC[C@H]1Cn1cc(C(=O)NCC2(O)CCC(F)(F)CC2)c2c(Cl)cccc12 |r|
FC1(F)CCC(CNC(=O)c2cn(C3CC4(CNC4)C3)c3cccc(Cl)c23)CC1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(CCc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C#N
COc1cn(Cc2ccccc2C)c(Nc2cccc(c2Cl)C(F)(F)F)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(=O)NC1CCOCC1
COC(=O)Nc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(N)cn1Cc1ccccc1
Cc1nc2cc(C)c(Nc3cc(=O)n(C)c(=O)n3Cc3cc(F)c(F)c(F)c3)cc2s1
COc1cn(Cc2ccccc2)c(NC2C[C@@H]3CC[C@H]2C3)nc1=O |r|
COc1cccc(Cn2cc(OC)c(=O)nc2Nc2cccc(Cl)c2C)c1
Cc1c(Cl)cccc1Nc1nc(=O)ccn1CCc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cccc3CCCc23)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3OCCc23)nc1=O
COc1cn(Cc2ccccc2)c(NCc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(OCc2ccccc2)cn1Cc1ccccc1
COc1cn(Cc2ccccc2F)c(Nc2cc(C)c(C)cc2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1F
COc1cn(Cc2ccccc2)c(Nc2cncc(Cl)c2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1
COc1cn(Cc2ccccc2)c(NC2CCc3ccccc3C2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3CCCCc23)nc1=O
COc1cn(Cc2ccc(Cl)cc2)c(Nc2cc(C)c(C)cc2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(Cl)cc1
CCOC(=O)c1cn(Cc2ccccc2)c(Nc2cc(C)c(C)cc2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(O)cn1Cc1ccccc1
Cc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccccc2)C(O)=O)cc1C
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1)N1CCCS1(=O)=O
Cc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccccc2)C(N)=O)cc1C
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)cc2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccccc2C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(c2)C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(cc2)C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(N[C@@H]2CCc3ccccc23)nc1=O |r|
COc1cn(Cc2ccc(F)c(Cl)c2)c(N[C@@H]2CCCc3ccccc23)nc1=O |r|
COc1cn(Cc2cc(F)c(F)cc2F)c(Nc2cccc(Cl)c2C)nc1=O
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
Cc1cc2OCCOc2cc1Nc1nc(=O)c(F)cn1Cc1ccccc1
Cc1cc2OCCOc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1
Cc1cc2OCCOc2cc1Nc1nc(=O)c(Cl)cn1Cc1ccccc1
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)cc1C
COc1cn(Cc2ccccc2)c(Nc2ccccc2SC)nc1=O
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)cc1C
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3[nH]c(=O)ccc23)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)c1C
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c1
COc1cn(Cc2cc(C)cc(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)cc1OC
CCc1ccccc1CNc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
COc1cn(Cc2ccc(F)c(C)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(SC)c2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3[nH]ccc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3occc23)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc3sccc23)nc1=O
COc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
COc1cc(Cn2cc(OC)c(=O)nc2Nc2cccc(Cl)c2C)ccc1F
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
Fc1cc(F)cc(Cn2cc(F)c(=O)nc2Nc2cccc3c2cc[nH]c3=O)c1
Cc1cc(Nc2nc(=O)c(Cl)cn2Cc2cc(F)cc(F)c2)c2cc[nH]c2c1
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
COc1cn(Cc2ccsc2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3OCOc3cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3nc(C)sc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(cc(C)c2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3ncccc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3ncccc3cc2C)nc1=O
Cc1nc2cc(C)c(Nc3nc(=O)c(Cl)cn3Cc3ccccc3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3ccccc3)cc2s1
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1C
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(Cl)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3oc(C)cc3c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2c(C)cc3oc(C)cc3c2C)nc1=O
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)c1
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1)-c1ncco1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc3ncsc3c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc3nc(C)sc3c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3CCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc3COCc3c2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3COCc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3C=CCOc3cc2C)nc1=O |c:20|
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3CCCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2c(C)ccc(C)c2F)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3scnc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3cc[nH]c3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Oc2cc(ccc2C)-c2ncco2)nc1=O
COc1cc(C)c(Nc2cc(=O)c(OC)cn2Cc2ccccc2)cc1C
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2ncco2)cc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C#N)cc1=O
COc1ccc(C)c(Oc2cc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Oc2cc(ccc2C)-c2ncco2)cc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Oc2cc3sc(C)nc3cc2C)cc1=O
COc1cnc(Nc2cccc(Cl)c2C)n(Cc2ccccc2)c1=O
COc1cc(C)c(Nc2ncc(OC)c(=O)n2Cc2ccc(F)c(Cl)c2)cc1C
COc1cnc(Nc2cc(ccc2C)N2CCCC2=O)n(Cc2ccc(F)c(Cl)c2)c1=O
COc1cnc(Nc2cc3sc(C)nc3cc2C)n(Cc2ccc(F)c(Cl)c2)c1=O
COc1cnc(Nc2cc(C)cc3[nH]ccc23)n(Cc2ccc(F)c(Cl)c2)c1=O
Cc1c(Cl)cccc1Nc1cc(=O)n(C)c(=O)n1Cc1ccccc1
COc1cc(C)c(Nc2cc(=O)n(C)c(=O)n2Cc2cc(F)c(F)c(F)c2)cc1C
Cn1ccc2c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(Cl)c3)cccc12
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
Cc1cc2COCc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)cc1F
COc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)n1
COc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1C(C)C
Fc1cc(Cn2cc(F)c(=O)nc2Nc2cccc3C(=O)CCCc23)cc(F)c1F
Fc1cc(Cn2cc(F)c(=O)nc2Nc2ccccc2C=C)cc(F)c1F
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1)-c1nnco1
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)nc1OC(F)F
Cc1nc2cc(C)c(Nc3nc(=O)c(C)nn3Cc3cc(F)c(F)c(F)c3)cc2s1
COc1cc(C)c(Nc2nc(=O)c(C)nn2Cc2cc(F)cc(F)c2)cc1OC
Cc1c(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)ccc2[nH]ccc12
COc1cc(C)c(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=NC#N
Cc1ccc(C)c(Nc2nc(=NO)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1ccc(F)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COc1ccc(F)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)c1F
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3COCc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1C
Cc1c(Cl)cccc1Nc1nc(=O)ccn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(F)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(Cl)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(C)cn1Cc1ccccc1
Cc1ccccc1Cn1cc(O)c(=O)nc1Nc1cccc(c1Cl)C(F)(F)F
Cc1c(Cl)cccc1Nc1nc(=O)c(OCC(F)(F)F)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(O)=O
Cc1c(Cl)cccc1Nc1nc(=O)c(NC(=O)OC(C)(C)C)cn1Cc1ccccc1
CCOC(=O)Cc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(CCO)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(O)=O)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(N)=O)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(Br)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)-c1ccccc1
COc1cn(Cc2ccccc2)c(NCc2cccc(c2Cl)C(F)(F)F)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(c2Cl)C(F)(F)F)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(c2Cl)C(F)(F)F)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2F)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1
COc1cn(Cc2ccccc2C)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(C)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(C)cc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(c2)C#N)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3CNCCc23)nc1=O
COc1ccccc1Cn1cc(OC)c(=O)nc1Nc1cccc(Cl)c1C
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccc(F)cc1)C#N
COc1cn(Cc2ccccc2)c(Nc2ccccc2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccccc2C)nc1=O
COc1cn(Cc2ccccc2)c(NCc2ccccc2C(F)(F)F)nc1=O
COc1cn(Cc2ccccc2)c(NCc2ccccc2Oc2ccc(C)cc2)nc1=O
COc1cn(Cc2ccccc2)c(NCc2ccccc2N(C)C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)N2CCCS2(=O)=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(Cl)cc2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(Cl)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(NC2CCc3ccccc23)nc1=O
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(=O)NCC#N
COCCNC(=O)c1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(=O)NCCS(C)(=O)=O
CCNC(=O)c1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)ccc2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(F)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2c(Cl)cccc2Cl)nc1=O
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cccc(c2C)C(F)(F)F)nc1=O
COC(=O)c1cccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1C
COc1cn(Cc2ccccc2)c(Nc2ccccc2C(F)(F)F)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(F)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(c2C)-n2cccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(C)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)C(F)(F)F)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(=O)NCC(F)(F)F
COc1cn(CCCc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
CN(C)C(=O)c1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
CCc1cc(Br)ccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(NCc2ccccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3occc23)nc1=O
CCc1ccccc1Nc1nc(=O)c(Cl)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2ccc(C)cc2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(Br)cn1Cc1ccccc1
Cc1cccc(Nc2nc(=O)c(Br)cn2Cc2ccccc2)c1C
CCCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cccc(CO)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(=O)OC(C)(C)C
Cc1cccc(Nc2nc(=O)c(cn2Cc2ccccc2)C(O)=O)c1Cl
COc1ccccc1CNc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1ccccc1CNc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1Cl
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cccc3n(C)ccc23)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccccc2Cc2ccccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccccc2Cl)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(Cl)cc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1cccc(Nc2nc(=O)c(F)cn2Cc2ccccc2)c1C
COc1cn(Cc2ccccc2)c(Nc2cccc(OC(C)C)c2C)nc1=O
COc1c(C)cccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(NCc2c(C)cccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(Cl)c(Cl)c2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(OC(F)F)c2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
CCc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1CC
CCOc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(Oc3ccccc3)c2C)nc1=O
Cc1cccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)cc2)c1C
CCc1ccccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(C)c2C)nc1=O
CC(C)Oc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)C(C)C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Br)ccc2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)cc(Cl)c2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)ccc2Cl)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)c1
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccccc1)N1CCCS1(=O)=O
COC(=O)c1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1
COc1ccc(Cl)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1
Cc1cccc(C)c1Nc1nc(=O)c(F)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)c(Cl)cc2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)[N+]([O-])=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(O)ccc2Cl)nc1=O
CCc1ccccc1Nc1nc(=O)c(F)cn1Cc1ccccc1
Cc1cccc(Nc2nc(=O)c(Cl)cn2Cc2ccccc2)c1C
CCc1cc(Cl)ccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(C)c(C)cc2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2F)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccccc2Cl)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(Cl)cc2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(N[C@@H]2CCCc3ccccc23)nc1=O |r|
CCc1ccc(Cl)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2cccc(F)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1cccc(F)c1
COc1cn(Cc2ccccc2)c(Nc2cc(CO)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2Cl)C(N)=O)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccccc2)cc1OC
COc1cn(Cc2ccccc2)c(Nc2ccc(Br)cc2Cc2ccccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(OC(C)C)cc2C)nc1=O
COc1cn(Cc2ccccc2Cl)c(Nc2cc(C)c(C)cc2C)nc1=O
CCc1cc2CCCc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1Cl
COc1cn(Cc2ccccc2)c(Nc2cccc(Oc3ccccn3)c2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
COc1cn(Cc2ccccc2)c(N[C@@H]2CCc3ccccc23)nc1=O |r|
COc1cn(Cc2ccccc2)c(Nc2ccc(cc2C)N2CCOCC2)nc1=O
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc1C
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)cc2)cc1OC
CCc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(CC)c1
CCc1ccc(CC)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1
CCc1c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cccc1OC
CCc1c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)cccc1OC
CCc1c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cccc1OC
CCc1c(Cl)cccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(cn1Cc1ccccc1)C(F)(F)F
COc1cn(Cc2ccccc2)c(Nc2cccc(N(C)C)c2C)nc1=O
Cc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccccc2)C(=O)NC2CCOCC2)cc1C
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc1C
COc1cn(Cc2ccccc2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(F)cn1Cc1cccc(Cl)c1
Cc1cccc(Nc2nc(=O)c(F)cn2Cc2cccc(Cl)c2)c1C
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(Cl)c(F)c1
CN(C)C(=O)CNC(=O)c1cn(Cc2ccccc2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C(C)C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1C
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1C
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)N2CCCS2(=O)=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c(C)c1
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
Cc1c(Cl)cccc1NC(=O)Cc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-n2cccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(CO)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(cc2C)N(C)C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)c(C)c1
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cc1C
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(F)c1
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)cc1C
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)cc1C
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cc1C
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)cc1C
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1cccc(F)c1
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
CCc1cc(C)c(C)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1ccccc1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)cc1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(F)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)cc1OC
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(CO)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(Cl)c(F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1C
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)cc1C
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)cc1C
Cc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccccc2)C(=O)NCc2ccccc2)cc1C
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(F)c2F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccc(Cl)c(F)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccc(Cl)c(Cl)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)cc(C)c2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1cn(Cc2ccccc2OC(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(OC(F)(F)F)c2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)cc2)cc1C
Cc1cc(C)c(Nc2nc(=O)c(Cl)cn2Cc2ccccc2)cc1C
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cccc(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(Cl)cn2Cc2ccccc2)cc1OC
COc1cn(Cc2c(F)cccc2F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(C)c2C)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1ccccc1)N1CCCS1(=O)=O
CCc1c(Nc2nc(=O)c(F)cn2Cc2ccc(F)cc2)cc(OC)cc1OC
CCc1c(Nc2nc(=O)c(F)cn2Cc2cccc(Cl)c2)cc(OC)cc1OC
CCc1c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc(OC)cc1OC
COc1cn(Cc2cc(Cl)cc(Cl)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccccc2)cc1C
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)cc2)cc1C
COc1cn(Cc2ccccc2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
COc1cn(Cc2cccc(F)c2)c(Nc2cccc(C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(C)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(C)c2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cn(Cc2cc(F)ccc2F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)cc2F)c(Nc2cccc(Cl)c2C)nc1=O
CNC(=O)Cc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
CN(C)C(=O)Cc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(C)ccc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(C)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)ccc2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)NCCO)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)NC2CCOCC2)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)N2CCOCC2)cn1Cc1ccccc1
COCCNC(=O)Cc1cn(Cc2ccccc2)c(Nc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)NCc2ccccc2)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)NC2COC2)cn1Cc1ccccc1
Cc1c(Cl)cccc1Nc1nc(=O)c(CC(=O)NCC#N)cn1Cc1ccccc1
COc1cc(C)c(Nc2nc(=O)c(Cl)cn2Cc2ccc(F)c(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(Cl)cn2Cc2cccc(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cccc(Cl)c2)cc1C
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc1C
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1cccc(Cl)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(Cl)cn1Cc1ccccc1
COCc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1C
COCc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1C
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(F)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(F)c(F)cc2C)nc1=O
CCc1c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc(OC)cc1OC
CCc1c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cc(OC)cc1OC
CCc1c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc(OC)cc1OC
COc1cn(Cc2ccccc2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
Cc1cc2OCCOc2cc1Nc1nc(=O)c(F)cn1Cc1cccc(Cl)c1
Cc1cc2OCCOc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1C
COc1cn(Cc2cccc(Cl)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1)-c1nnco1
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)cc1C
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Br)ccc2C)nc1=O
CCc1ccc(Cl)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
CCc1ccc(Cl)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1ccc(Cl)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)c1C
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c1C
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
CCc1cc(F)ccc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(N(C)C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(N(C)C)c2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc(C)c2C)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c1C
COc1cc(C)c(Nc2nc(=O)c(Cl)cn2Cc2ccc(F)cc2)cc1OC
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c1
COc1c(C)ccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1C
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)N2CCN(CC2)C(=O)OC(C)(C)C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)N2CCN(CC2)C(=O)OC(C)(C)C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(c(F)cc2C)S(=O)(=O)Nc2ccccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2nc3ncccc3o2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2nc3ncccc3o2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(C)c(OC)c2C)nc1=O
CCc1cc(F)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccccc2OC(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2COC(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)c(Cl)cc2C)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1C
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(Cl)c(Cl)cc2C)nc1=O
COc1cc(F)cc(Cn2cc(OC)c(=O)nc2Nc2cccc(Cl)c2C)c1
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c1C
COc1cn(Cc2ccccc2)c(Nc2cccc(SC)c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(SC)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(N(C)C)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)ccc2C)nc1=O
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)ccc2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1C
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)cc1OC
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(NCc2cccc(Cl)c2C)nc1=O
CCc1ccccc1CNc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c1
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(c2C)C(F)(F)F)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(c2C)C(F)(F)F)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(c2C)C(F)(F)F)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1c(Cl)cccc1Nc1nc(=O)c(Cl)cn1Cc1ccc(F)c(F)c1
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)cc1Cl
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3sccc23)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)c1C
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)C(C)(C)C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C(C)(C)C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)cc(C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c1C
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)cc1Cl
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(SC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc(OC(C)C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc(OC(C)C)c2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
COc1c(C)ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c1C
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(Cl)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccc(cc2C)N2CCOCC2)nc1=O
COc1cn(Cc2cc(C)cc(C)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(CN3CCCC3)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-n2c(C)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-n2c(C)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3[nH]c(cc23)-c2ccccc2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccc(OC(C)C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(OC(C)C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(OC(C)C)cc2C)nc1=O
COc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c(C)cc1Cl
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
COc1c(C)ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1C
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(Cl)c(Cl)cc2C)nc1=O
CCc1cc(Cl)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(cc2C)N2CCOCC2)nc1=O
COc1ccc(Cl)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
CCc1cc(Cl)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(SC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(cc2C)N2CCOCC2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(c(C)cc2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)N2CCCS2(=O)=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)c1C
COc1cn(Cc2cccc(Cl)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(Cl)cc2C)nc1=O
CCc1ccc(F)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)cc1
CCc1ccc(F)cc1Nc1nc(=O)c(OC)cn1Cc1cccc(Cl)c1
CCc1ccc(F)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)c(F)c(F)c1
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc(C)c2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)ccc2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1C
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)c(F)c(F)c1
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(Cl)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(CO)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc3[nH]ncc3cc2C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COc1cn(Cc2cc(F)cc(c2)C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)cc1C
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1C
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(c(F)cc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(c(F)cc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(c(F)cc2C)-c2cccn(C)c2=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(Cl)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(Cl)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccccc2Cc2ccccn2)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3[nH]c(C)cc23)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(CO)c(C)cc2C)nc1=O
COc1cc(C)cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1C
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc3[nH]c(=O)ccc23)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(c(C)cc2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc(SC)c2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(OC(F)F)cc2C)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c(C)c1
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2ccc(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2ccc(C)c(OC)c2C)nc1=O
CCc1cc(Cl)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2ccc(cc2C)N2CCOCC2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)cc1Cl
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3[nH]ccc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3[nH]ccc3cc2C)nc1=O
CCc1ccc(Br)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2ccc(cc2C)N(C)C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1C
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c1
COc1cn(Cc2ccccc2)c(Nc2ccc(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(OC(F)(F)F)cc2C)nc1=O
CCc1cc(Br)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
CCc1cc(Br)ccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1C
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC(C)C)ccc2C)nc1=O
COc1cn(Cc2ccc(c(F)c2)C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
COc1cn(Cc2ccc(F)c(c2)C(F)(F)F)c(Nc2cccc(Cl)c2C)nc1=O
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1Cl
COc1ccc(Cl)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3occc23)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)c1C
COc1cn(Cc2cccc(F)c2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2cccc(F)c2)c(Nc2cc(C)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-n2cccc2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-n2cccc2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-n2cccc2)nc1=O
CCc1cc(Br)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2ccc(C)o2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2ccc(C)o2)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(OC(F)F)c2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)c1C
COc1cn(Cc2ccc(F)cc2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2cnccn2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2cnccn2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(Cl)c(Cl)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)cc1Cl
CCc1ccc(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)c(F)c(F)c1
CCc1ccccc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c(C)c1
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc(SC)c2C)nc1=O
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1Cl
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2cnccn2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccccc2C)nc1=O
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1F
CCc1cc2OCOc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1cc2OCOc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc3c2cc[nH]c3=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2cccnc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2cccnc2)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1cc(F)cc(F)c1)-c1nnco1
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1)N1CCCC1=O
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1cc(F)cc(F)c1)N1CCCC1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cccc(SC)c2C)nc1=O
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c2cc[nH]c2c1
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc3OCCOc3cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3OC(F)(F)Oc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(F)cc2C)nc1=O
CCOc1cn(Cc2ccccc2)c(Nc2cc(C)c(OC)cc2C)nc1=O
CCOc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(OC)cc2C)nc1=O
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1C
CCOc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)cc(OC)c2C)nc1=O
CCOc1cn(Cc2ccccc2)c(Nc2cc(C)cc(OC)c2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc1F
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1F
COc1cn(Cc2ccccc2)c(Nc2cc3OCOc3cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)cc1F
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)C(C)=C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C(C)=C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2c(C)cccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3OC(F)(F)Oc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3OC(F)(F)Oc3cc2C)nc1=O
CCc1cc2OC(F)(F)Oc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1cc2OC(F)(F)Oc2cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
CCc1cc2OC(F)(F)Oc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)C(C)(C)O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)C(C)(C)O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2ccnn2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2ccnn2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)N2CCOCC2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)N2CCOCC2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)N2CCOCC2)nc1=O
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)c(C)c1
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)N2CCOCC2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3OCOc3cc2C)nc1=O
CCc1cc2OCOc2cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3nc(C)sc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3nc(C)sc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)C(C)=C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)C(C)=C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)C(C)=C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2cscn2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2cscn2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2cscn2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2cscn2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(cc(C)c2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(cc(C)c2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(cc(C)c2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(cc(C)c2C)S(C)(=O)=O)nc1=O
CCOc1cn(Cc2ccccc2)c(Nc2cc(OC)c(OC)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3nc(C)sc3cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc(C)c2F)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1Cl
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2cccnc2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2cccnc2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2cccnc2)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2ccc(C)o2)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)-c2ccc(C)o2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2ccc(C)o2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc3ncccc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc3ncccc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc3ncccc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C(C)(C)O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(ccc2C)C(C)(C)O)nc1=O
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1C
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(Cl)c3)cc2s1
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c(C)cc1F
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c(C)cc1F
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)cc1F
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2ccnn2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(ccc2C)-c2ccnn2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2ccnn2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)C(C)(C)O)nc1=O
Cc1nc2cc(C)c(Nc3nc(=O)c(Cl)cn3Cc3ccc(F)c(Cl)c3)cc2s1
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c(C)cc1C
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)cc1C
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c(C)cc1C
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c(C)cc1C
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)cc1C
CCOc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC)c(OC)cc2C)nc1=O
CCc1cc2OCCOc2cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1cc2OCCOc2cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(F)c1
CCc1cc2OCCOc2cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3occc3c2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(OCC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(Cl)cc2F)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)-c2cscn2)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)N2CCCC2=O)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1F
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C)c(OCC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(OCC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(Cl)s2)c(Nc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(Cl)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(Cl)c(F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(Cl)c(F)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(Cl)c(F)cc2C)nc1=O
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(Cl)c1
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1ccc(F)c(F)c1
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(Cl)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(Cl)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(Cl)cc3[nH]ccc23)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(Cl)cc3[nH]ccc23)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3OC(F)(F)C(F)(F)Oc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3OC(F)(F)C(F)(F)Oc3c2C)nc1=O
COc1nc2ccc(Nc3nc(=O)c(OC)cn3Cc3ccc(F)c(Cl)c3)c(C)c2s1
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)-c2ccccc2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)-c2ccccc2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)-c2ccccc2)nc1=O
COc1nc2ccc(Nc3nc(=O)c(OC)cn3Cc3cc(F)cc(F)c3)c(C)c2s1
COc1ncccc1-c1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1
COc1ncccc1-c1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(Cl)cn1Cc1ccc(F)c(Cl)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(Cl)cn1Cc1ccc(F)c(F)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(Cl)cn1Cc1cc(F)cc(F)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(Cl)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(Cl)cn2Cc2ccc(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(Cl)cn2Cc2cc(F)cc(F)c2)c(C)c1
COc1ccc(Cl)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(Cl)c1
COc1cc(Cl)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1)-c1ncco1
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1)-c1ncco1
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1ccc(F)c(Cl)c1)-c1ncco1
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1ccc(F)c(F)c1)-c1ncco1
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1cc(F)cc(F)c1)-c1ncco1
COc1cn(Cc2ccccc2)c(Nc2ccc3ncsc3c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3ncsc3c2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3nc(C)sc3c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc3nc(C)sc3c2C)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1)-c1cscn1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3CCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3CCOc3cc2C)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1)-c1cscn1
CCOc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1F
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(OC(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OC(F)F)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OC(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OC(F)F)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OC(F)F)c(C)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3n(C)c(=O)ccc23)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3n(C)c(=O)ccc23)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(ccc2C)N2CCCC2)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)N2CCCC2)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(ccc2C)N2CCCC2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(F)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(F)c(Cl)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(OC3CC3)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC3CC3)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(OC3CC3)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cc(OC3CC3)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(OC3CC3)ccc2C)nc1=O
CCOc1cn(Cc2ccccc2)c(Nc2cc(OC)c(OC)cc2CC)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)-n2cccc2)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(Oc3ccccn3)ccc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(Oc3ccccn3)ccc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(Oc3ccccn3)ccc2C)nc1=O
COc1cn(Cc2ccc(F)cc2)c(Nc2cc(Oc3ccccn3)ccc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(Oc3ccccn3)ccc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2cccc3c2ccn(C)c3=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cccc3c2ccn(C)c3=O)nc1=O
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2cccc3c2ccn(C)c3=O)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2cccc3c2ccn(C)c3=O)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cccc3c2ccn(C)c3=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3COCc3cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc3COCc3c2C)nc1=O
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)c(F)c(F)c1
CCOc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(OC)c(OC)cc2CC)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc3COCc3c2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc3CCCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2cc(C#C)c(F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C#C)c(F)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3CCCOc3cc2C)nc1=O
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2ccccc2)c(C)cc1F
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1F
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c(C)cc1F
CCOc1cc(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(OC(F)(F)F)cc2C)nc1=O
COc1cn(Cc2ccccc2)c(Nc2c(C)ccc(C)c2F)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2c(C)ccc(C)c2F)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2c(C)ccc(C)c2F)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3C(=O)CCOc3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)N2CCOCC2)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OCC(F)(F)F)ccc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(Oc3ccnc(F)c3)cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3sc(nc3cc2C)C(F)F)nc1=O
COc1ccc(C)cc1Nc1nc(=O)c(OC)cn1Cc1cc(F)c(F)c(F)c1
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cc2s1
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3cc[nH]c3cc2C)nc1=O
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OCF)cc2C)nc1=O
COc1ccc(Nc2cc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(F)cc2C)cc1=O
COc1ccc(C)c(Nc2cc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(OC(F)F)cc2C)cc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(C)c(Cl)cc2C)cc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(Cl)cc2C)cc1=O
COc1cn(Cc2ccccc2)c(Nc2cc(C)c(OC(F)F)cc2C)cc1=O
COc1ccc(C)c(Nc2cc(=O)c(OC)cn2Cc2ccccc2)c1
COc1cc(C)c(Nc2cc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1C
COc1ccc(Cl)c(Nc2cc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(ccc2C)C(F)(F)F)cc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2ccc(cc2C)C#N)cc1=O
COc1ccc(Nc2cc(=O)c(OC)cn2Cc2ccccc2)c(C)c1
COc1cc(C)c(Nc2c(Cl)c(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1C
COc1cnc(Nc2cccc(Cl)c2C)n(Cc2cccc(Cl)c2)c1=O
COc1cnc(Nc2cccc(Cl)c2C)n(Cc2ccc(F)c(Cl)c2)c1=O
COc1cnc(Nc2cccc(Cl)c2C)n(Cc2ccc(F)c(F)c2)c1=O
COc1cnc(Nc2cc(C)c(Cl)cc2C)n(Cc2ccccc2)c1=O
COc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)cc1Cl
Cc1ccc(OC(F)F)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Fc1cc(Cn2cc(F)c(=O)nc2Nc2cccc3NCCc23)cc(F)c1F
COCc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c1
Cc1ccc(OCC2CC2)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
CCOc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c1
CCOc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c1
COc1nc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1C
Cc1cc2OCCc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
CCOc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c1
COc1nc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1C
COc1nc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc1C
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1Cl
CCOc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1nc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)cc1C
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(F)c3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3ccc(F)cc3)cc2s1
Cc1ccc(CO)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1ccc(CO)cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1ccc(CO)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1ccc(CO)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1nc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1nc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cn1ccc2c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cccc12
Cn1ccc2c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(F)c3)cccc12
Cn1ccc2c(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)cccc12
Fc1cc(F)cc(Cn2cc(F)c(=O)nc2Nc2cccc3[nH]ccc23)c1
Fc1cc(Cn2cc(F)c(=O)nc2Nc2cccc3[nH]ccc23)cc(F)c1F
Fc1ccc(Cn2cc(F)c(=O)nc2Nc2cccc3[nH]ccc23)cc1Cl
Fc1ccc(Cn2cc(F)c(=O)nc2Nc2cccc3[nH]ccc23)cc1F
Cc1cc2COCc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc2COCc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1cc2COCc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
CCOc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
CCOc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1F
CCOc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)cc1F
CCOc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)n1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)n1
CCOc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1F
Cc1cc(OC(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1cc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1cc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc2OCCc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
CCOc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)c1
CCOc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)n1
COc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c(C)cc1F
COc1cc(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c(C)cc1F
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1)N1CC2CCC1C2
Cc1cc2cc(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)c(C)cc2[nH]1
Cc1cc2cc(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(Cl)c3)c(C)cc2[nH]1
Cc1cc2cc(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(F)c3)c(C)cc2[nH]1
Cc1cc2cc(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)c(C)cc2[nH]1
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
CCOc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc1F
CCOc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1F
CCOc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)cc1F
Cc1cc(OC(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc(OC(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1cc(OC(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
COc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c1
COc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c1
COc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c1
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1C(C)C
Cc1cc2OCCc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1cc2OCCc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Fc1cc(F)cc(Cn2cc(F)c(=O)nc2Nc2cccc3NCCc23)c1
Cc1nc2cc(Cl)c(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)cc2o1
Cc1nc2cc(Cl)c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(F)c3)cc2o1
Cc1nc2cc(Cl)c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(Cl)c3)cc2o1
Cc1nc2cc(Cl)c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cc2o1
COC(=O)\C=C\c1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)c(F)c(F)c2)c1
CCOC(=O)c1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC)cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C(N)=O)cc1C
Cc1ccccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COc1cc(C)c(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C#N)cc1C
COCc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(F)c2)c1
COCc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)c1
COCc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1F
Cc1nc2cc(C)c(Nc3nc(=O)c(CCO)cn3Cc3cc(F)c(F)c(F)c3)cc2s1
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2ccc(F)c(Cl)c2)cc1CO
Cc1nc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Cc1nc2[nH]ccc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc2[nH]ncc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1cc2[nH]ncc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
Cc1cc2[nH]ncc2cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc2[nH]ncc2cc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(F)c1
Fc1cc(Cn2cc(F)c(=O)nc2Nc2cccc3cnccc23)cc(F)c1F
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccccc2C)nc1=O
Cc1ccccc1Nc1nc(=O)c(C)cn1Cc1cc(F)c(F)c(F)c1
COc1ccc(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C(O)=O)c(C)c1
COc1ccc(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C(N)=O)c(C)c1
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1F
Cc1cc(OC(F)(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
Cc1cc(OC(F)(F)F)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COc1ccc(Nc2nc(=O)c(CCO)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
Oc1cccc2c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cccc12
CN1CCc2c(C1)cccc2Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
CCOC(=O)c1cn(Cc2ccc(F)c(F)c2)c(Nc2cc(C)c(OC)cc2C)nc1=O
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1CO
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1CO
COc1ccc(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C#N)c(C)c1
Cc1cc(C)c(Nc2nc(=O)c(Br)cn2Cc2cc(F)cc(F)c2)cc1C
Oc1cccc2c(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)cccc12
Oc1cccc2c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(F)c3)cccc12
Oc1cccc2c(Nc3nc(=O)c(F)cn3Cc3ccc(F)c(Cl)c3)cccc12
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)nc1F
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)nc1F
Cc1c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)ccc2[nH]ccc12
Cc1c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)ccc2[nH]ccc12
CCOC(=O)c1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
CCOC(=O)c1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC)c(F)cc2C)nc1=O
COc1ccc(C)c(Nc2nc(=O)c(cn2Cc2cc(F)cc(F)c2)C#N)c1
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC(F)F)cc2C)nc1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OCCO)ccc2C)nc1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3COCc3cc2C)nc1=O
Cc1cc2COCc2cc1Nc1nc(=O)c(CCO)cn1Cc1cc(F)c(F)c(F)c1
COc1ccc(C)c(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C(O)=O)c1
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)-c2ncco2)nc1=O
Cc1cc2COCc2cc1Nc1nc(=O)c(cn1Cc1cc(F)c(F)c(F)c1)C#N
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(ccc2C)-c2nnco2)nc1=O
Cc1cc(ccc1Nc1nc(=O)c(C)cn1Cc1cc(F)c(F)c(F)c1)N1CCOCC1
COc1cc(F)c(Nc2nc(=O)c(C)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
Cc1ccc(cc1Nc1nc(=O)ccn1Cc1cc(F)c(F)c(F)c1)S(C)(=O)=O
COc1cc(C)c(Nc2nc(=O)c(C)c(C)n2Cc2cc(F)cc(F)c2)cc1OC
Cc1nc2cc(C)c(Nc3nc(=O)cc(C)n3Cc3cc(F)c(F)c(F)c3)cc2s1
Cc1cc(F)c(cc1Nc1nc(=O)ccn1Cc1cc(F)c(F)c(F)c1)-c1cccn(C)c1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC)ccc2C)nc1=O
COc1cc(Cl)c(Nc2nc(=O)c(C)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc(OC)cc2C)nc1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc3sc(C)nc3cc2C)nc1=O
COCc1cc(=O)nc(Nc2cc(OC)c(OC)cc2C)n1Cc1cc(F)cc(F)c1
Cc1ccc(cc1Nc1nc(=O)c(C)cn1Cc1cc(F)c(F)c(F)c1)-c1cccn(C)c1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC)c(OC)cc2C)nc1=O
Cc1ccc(OCCO)cc1Nc1nc(=O)c(C)cn1Cc1cc(F)c(F)c(F)c1
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(Cl)c(OC)cc2C)nc1=O
COCc1cc(=O)nc(Nc2cc(OC)c(OC)cc2C)n1Cc1cc(F)c(F)c(F)c1
Cc1cc(F)c(cc1Nc1nc(=O)c(C)cn1Cc1cc(F)c(F)c(F)c1)-c1cccn(C)c1=O
Cc1cc(ccc1Nc1nc(=O)ccn1Cc1cc(F)c(F)c(F)c1)N1CCOCC1
COc1cc(C)c(Nc2nc(=O)ccn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(C)c(Nc2nc(=O)c(cn2Cc2cc(F)c(F)c(F)c2)C#N)c1
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(CO)ccc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(C)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(Nc2nc(=O)c(C)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)cc3[nH]ccc23)nc1=O
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(C)c(OC)cc2C)nc1=O
Cc1ccc(cc1Nc1nc(=O)c(Cl)cn1Cc1cc(F)c(F)c(F)c1)-c1nnco1
COc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccc(F)c(F)c2)C(N)=O)cc1C
COc1cc(C)c(Nc2nc(=O)ccn2Cc2ccc(F)c(Cl)c2)cc1OC
COc1cc(C)c(Nc2nc(=O)c(cn2Cc2ccc(F)c(F)c2)C#N)cc1C
Cc1cc(Nc2nc(=O)ccn2Cc2cc(F)c(F)c(F)c2)c2cc[nH]c2c1
Fc1cc(Cn2cc(Cl)c(=O)nc2Nc2cccc3C(=O)CCCc23)cc(F)c1F
COCc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
Cc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
Cc1cn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
COc1cc(Nc2nc(=O)ccn2Cc2ccc(F)c(Cl)c2)c(C)c(OC)c1
COc1ccc(Nc2nc(=O)cc(C)n2Cc2cc(F)c(F)c(F)c2)c(C)c1
Cc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
Cc1c(Nc2nc(=O)ccn2Cc2cc(F)c(F)c(F)c2)ccc2[nH]ccc12
Cc1c(Nc2nc(=O)ccn2Cc2ccc(F)c(Cl)c2)ccc2[nH]ccc12
Cc1c(Nc2nc(=O)ccn2Cc2cc(F)cc(F)c2)ccc2[nH]ccc12
Fc1cc(Cn2cc(F)c(=O)nc2Nc2cccc3OCCCc23)cc(F)c1F
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1Cl
CCc1ccccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1c(CO)cccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COCc1cccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1C
COCCOc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1C
Cc1c(F)cccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1nc2cc(Cl)c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)cc2o1
Cc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(Cl)c1
Cc1cccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1F
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(Cl)c1
COc1cc(Cl)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
Cc1cccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1C
CCc1ccc(Cl)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
CCc1ccc(OC)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(Cl)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
Cc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1ccc(Cl)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Cl)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
CCc1cc(OC)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1nc2ccc(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)c(C)c2s1
Cc1nc2ccc(Nc3nc(=O)c(F)cn3Cc3cc(F)c(F)c(F)c3)c(C)c2s1
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1C
CCOc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1C
Cc1c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)ccc2scnc12
Cc1c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)ccc2scnc12
COCCOc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
Cc1ccc(OCCO)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)cc1Cl
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1Cl
CCc1cc(F)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(Cl)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(OC(F)F)c(C)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
CCc1cc(F)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1C)S(C)(=O)=O
Cc1c(F)cccc1Nc1nc(=O)c(F)cn1Cc1ccc(F)c(Cl)c1
CCc1cc(OC)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
CCOc1ccc(F)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
CCOc1ccc(Cl)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
CCc1ccc(F)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1c(Cl)cccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
CCc1cc(OC)c(OC)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1)-c1cccn(C)c1=O
CN1C=CC=C(C1=C)c1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F |c:2,4|
CCOc1c(C)cccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(Cl)cc1F
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(Cl)cc1F
CCc1ccc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)cc1F
CCc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)c1
COCCn1ccc2c(C)c(Nc3nc(=O)c(F)cn3Cc3cc(F)cc(F)c3)ccc12
Cc1cc(C)c(OC(F)F)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(CF)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
COc1cc(C)c(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c1
Cc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)nc1OC(F)F
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)nc1OC
Cc1cc(CO)ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1cc(ccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1)C(F)F
Cc1cc(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1F
COc1cc(Cl)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1F
Cc1ccc(CF)cc1Nc1nc(=O)c(F)cn1Cc1cc(F)cc(F)c1
CN(C)c1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)c1
CN(C)c1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(OC)c1C
Cc1cc(F)c(C)c(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c1F
COc1ccc(C)c(Nc2nc(=O)c(CO)nn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)c(CO)nn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COc1cc(C)c(Nc2nc(=O)c(CF)nn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(C)c(Nc2nc(=O)c(nn2Cc2cc(F)c(F)c(F)c2)C(O)=O)c1
COc1ccc(Nc2nc(=O)c(nn2Cc2cc(F)c(F)c(F)c2)C(O)=O)c(C)c1
COc1cc(C)c(Nc2nc(=O)c(nn2Cc2cc(F)c(F)c(F)c2)C(O)=O)cc1OC
CCOC(=O)c1nn(Cc2cc(F)c(F)c(F)c2)c(Nc2cc(OC)c(OC)cc2C)nc1=O
Cc1ccc(F)cc1Nc1nc(=O)c(CO)nn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(CO)cc1Nc1nc(=O)c(C)nn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(CO)cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1
COc1cc(C)c(Nc2nc(=O)c(CO)nn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1cc(F)c(Nc2nc(=O)c(C)nn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1cc(F)c(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(Nc2nc(=O)c(C)nn2Cc2cc(F)c(F)c(F)c2)c(C)n1
Cc1nc2cc(C)c(Nc3nc(=O)c(C)nn3Cc3cc(F)cc(F)c3)cc2s1
Cc1nn(Cc2cc(F)c(F)c(F)c2)c(Nc2ccc3[nH]ccc3c2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(Cl)nn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(Nc2nc(=O)c(Cl)nn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COc1cc(C)c(Nc2nc(=O)c(C)nn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(Nc2nc(=O)cnn2Cc2ccc(Cl)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2cc(F)cc(Cl)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2ccc(F)c(Cl)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2cc(F)cc(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2ccc(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2ccc(F)cc2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2cccc(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2ccccc2F)c(C)c1
COc1ccc(Nc2nc(=O)cnn2Cc2ccccc2)c(C)c1
COc1ccc(Nc2nc(=O)c(C)nn2Cc2cc(F)c(F)c(F)c2)c(C)c1
COc1cc(C)c(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)cc1Cl
COc1cc(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)c(C)cc1Cl
Cc1cc2COCc2cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1
COc1ccc(C)c(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)cnn2Cc2cc(F)c(F)c(F)c2)c(C)c1
Cc1nc2cc(C)c(Nc3nc(=O)cnn3Cc3cc(F)c(F)c(F)c3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=NC#N)c(F)cn3Cc3cc(F)c(F)c(F)c3)cc2s1
COc1cc(C)c(Nc2nc(=NC#N)c(OC)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1cc(C)c(Nc2nc(=NC#N)c(F)cn2Cc2cc(F)c(F)c(F)c2)cc1OC
CN=c1nc(Nc2cc(C)ccc2C)n(Cc2cc(F)c(F)c(F)c2)cc1F
CON=c1nc(Nc2cc3sc(C)nc3cc2C)n(Cc2cc(F)c(F)c(F)c2)cc1F
CON=c1nc(Nc2cc(C)ccc2C)n(Cc2cc(F)c(F)c(F)c2)cc1F
Cc1ccc(C)c(Nc2nc(=NC#N)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
Cc1ccc(C)c(Nc2nc(=N)c(F)cn2Cc2cc(F)c(F)c(F)c2)c1
O=c1cc2OCC(c3ccccc3)n2c(Nc2cccc3ncccc23)n1
Cc1c(Cl)cccc1Nc1nc(=O)cc2COCC(c3ccccc3)n12
Cc1ccccc1Nc1nc(=O)cc2CCCC(c3ccccc3)n12
COc1c2OCCC(c3ccccc3)n2c(Nc2cccc(Cl)c2C)nc1=O
COc1c2CCC(c3ccccc3)n2c(Nc2cc3sc(C)nc3cc2C)nc1=O
CCc1nc(OC)ccc1Nc1nc(=O)cc2CCC(c3cc(F)cc(F)c3)n12
COc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4)n23)c(C)n1
COc1ccc(Nc2nc(=O)c(C=C)c3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
Cc1nc2cc(C)c(Nc3nc(=O)cc4NCC(c5ccccc5)n34)cc2s1
Cc1cc2COCc2cc1Nc1nc(=O)c(F)c2CCC(c3cc(F)cc(F)c3)n12
CN1CC(c2ccccc2)n2c1cc(=O)nc2Nc1cc(C)c(C)cc1C
CCN1C2=NCC(N2C(Nc2cc(C)c(C)cc2C)=NC1=O)c1ccccc1 |c:20,t:3|
CN1C2=NCC(N2C(Nc2cc(ccc2C)C#N)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)c1F |t:7,13|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)cc1F |t:6,12|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)c(C)cc1F |t:6,12|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)c(C)c1F |t:7,13|
CCc1nc(OC)ccc1NC1=NC(=O)N(C)C2=NCC(N12)c1cc(F)c(F)c(F)c1 |t:12,18|
COCCOc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:12,18|
CN1C2=NCC(N2C(Nc2cc(CO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
COc1nc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)cc1F |t:8,14|
CN1C2=NCC(N2C(Nc2cc3COCc3cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:21,t:2|
CN1C2=NCC(N2C(Nc2cc(CO)c(F)cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:20,t:2|
CN1C2=NCC(N2C(Nc2cc(OCCO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:21,t:2|
CCc1ccc(CO)cc1NC1=NC(=O)N(C)C2=NCC(N12)c1cc(F)c(F)c(F)c1 |t:12,18|
CN1C2=NCC(N2C(NCc2ccccc2)=NC1=O)c1cc(F)c(F)c(F)c1 |c:17,t:2|
CN1C2=NCC(N2C(Nc2cc(OC(F)F)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:21,t:2|
COCc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:10,16|
Cc1c(Cl)cccc1Nc1nc(=O)cc2OCC(c3ccccc3)n12
Cc1c(Cl)cccc1Nc1nc(=O)cc2CCCC(c3ccccc3)n12
Cc1c(Cl)cccc1Nc1nc(=O)cc2OCCC(c3ccccc3)n12
Cc1c(Cl)cccc1Nc1nc(=O)cc2CCC(c3ccccc3)n12
Cc1c(Cl)cccc1Nc1nc(=O)cc2CCC(c3cccc(Cl)c3)n12
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1OC
Cc1cc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)cc1Cl
Cc1cc(Nc2nc(=O)cc3CCC(c4ccc(F)c(Cl)c4)n23)c(C)cc1Cl
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)c(Cl)c4)n23)cc1OC
COc1ccc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)c1
Cc1ccccc1Nc1nc(=O)cc2CCC(c3ccccc3)n12
COc1ccc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c1
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)cc4)n23)cc1OC
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4cccc(F)c4)n23)cc1OC
COc1ccc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1OC
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1C
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4cc(F)c(F)c(F)c4)n23)cc1OC
COc1cc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)cc1F
COc1ccc(Nc2nc(=O)cc3CCC(c4ccc(F)cc4)n23)c(C)c1
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1F
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)c(F)c4)n23)cc1OC
Cc1nc2cc(C)c(Nc3nc(=O)cc4CCC(c5ccc(F)cc5)n34)cc2s1
COc1cc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)cc1Cl
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1Cl
Cc1nc2cc(C)c(Nc3nc(=O)cc4CC[C@@H](c5ccccc5)n34)cc2s1 |r|
COc1cc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cn1
COc1cc(C)c(Nc2nc(=O)c(OC)c3CCC(c4ccccc4)n23)cc1C
COc1cc(Nc2nc(=O)cc3CCC(c4ccc(F)cc4)n23)c(C)cc1Cl
COc1ccc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)n1
COc1cc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)cn1
COc1c2CCC(c3ccc(F)cc3)n2c(Nc2cc3sc(C)nc3cc2C)nc1=O
COc1ccc(Nc2nc(=O)cc3CCC(c4ccc(F)c(Cl)c4)n23)c(C)c1
COc1ccc(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)c(C)c1
CCc1cc(Nc2nc(=O)cc3CCC(c4ccccc4)n23)c(C)cc1OC
Cc1cc2COCc2cc1Nc1nc(=O)cc2CCC(c3ccccc3)n12
COc1ccc(Nc2nc(=O)cc3CCC(c4ccc(F)c(F)c4)n23)c(C)c1
COc1ccc(Nc2nc(=O)cc3CCC(c4cc(F)c(F)c(F)c4)n23)c(C)c1
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4ccccc4)n23)cc1C
COc1cc(Nc2nc(=O)c(OC)c3CCC(c4ccccc4)n23)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)c3CCC(c4ccccc4)n23)c(C)cc1F
COc1ccc(Nc2nc(=O)c(F)c3CCC(c4ccccc4)n23)c(C)c1
COc1ccc(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
COc1ccc(Nc2nc(=O)cc3CCC(c4cc(F)c(F)c(F)c4)n23)c(C)n1
COc1ccc(Nc2nc(=O)cc3CCC(c4cccc(F)c4)n23)c(C)c1
COc1ccc(Nc2nc(=O)cc3CCC(c4cccc(Cl)c4)n23)c(C)c1
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)cc1C
COc1ccc(Nc2nc(=O)c(OC)c3CCC(c4ccccc4)n23)c(C)c1
Cc1nc2cc(C)c(cc2s1)\N=c1/[nH]c(=O)cc2CCC(c3cc(F)cc(F)c3)n12
Cc1nc2cc(C)c(cc2s1)\N=c1/[nH]c(=O)c(F)c2CCC(c3ccc(F)cc3)n12
CCOc1ccc(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
Cc1cc(OC(F)F)ccc1\N=c1/[nH]c(=O)cc2CCC(c3cc(F)cc(F)c3)n12
Cc1cc(OC(F)F)ccc1\N=c1/[nH]c(=O)c(F)c2CCC(c3ccc(F)cc3F)n12
Cc1nc2cc(C)c(Nc3nc(=O)c(F)c4CCC(c5ccc(F)cc5F)n34)cc2s1
COc1ccc(C)c(Nc2nc(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c1
COc1ccc(C)c(c1)\N=c1/[nH]c(=O)cc2CCC(c3cc(F)cc(F)c3)n12
COc1cc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(C)cc1F
COc1cc(\N=c2/[nH]c(=O)cc3CCC(c4cc(F)cc(F)c4)n23)c(C)cc1F
COc1ccc(Nc2nc(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(C)c1
Cc1cc(\N=c2/[nH]c(=O)cc3CCC(c4ccccc4)n23)c(C)cc1OC(F)F
Cc1cc2COCc2cc1Nc1nc(=O)cc2CCC(c3cc(F)cc(F)c3)n12
Cc1cc2COCc2cc1Nc1nc(=O)cc2CCC(c3ccc(F)cc3)n12
COc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(C)n1
COc1ccc(\N=c2/[nH]c(=O)cc3CCC(c4ccc(F)cc4)n23)c(C)n1
COc1cnc(C)c(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)c1
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4cc(F)cc(F)c4)n23)cc1F
Cc1cc2COCc2cc1\N=c1/[nH]c(=O)c(F)c2CCC(c3ccc(F)cc3F)n12
Cc1cc2COCc2cc1\N=c1/[nH]c(=O)c(F)c2CCC(c3ccc(F)cc3)n12
CCOc1ccc(\N=c2/[nH]c(=O)cc3CCC(c4ccc(F)cc4F)n23)c(CC)n1
CCOc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(CC)n1
Cc1nc(OC(F)F)ccc1Nc1nc(=O)c(F)c2CCC(c3ccc(F)cc3)n12
COc1cnc(C)c(c1)\N=c1/[nH]c(=O)c(F)c2CCC(c3ccc(F)cc3)n12
COc1cnc(C)c(c1)\N=c1/[nH]c(=O)cc2CCC(c3ccc(F)cc3)n12
CCOc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4)n23)c(C)n1
CCOc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(C)n1
CCOc1nc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)cc4F)n23)cc1F
CCOc1nc(C)c(Nc2nc(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)cc1F
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)cc4F)n23)cc1F
COc1ccc(Nc2nc(=O)c(Cl)c3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
COc1ccc(Nc2nc(=O)c(Br)c3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
COc1ccc(Nc2nc(=O)c(C)c3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
Cc1[nH]c(=O)c(F)cc1Nc1nc(=O)cc2CCC(c3ccc(F)cc3F)n12
COc1ccc(Nc2nc(=O)c(c3CCC(c4cc(F)cc(F)c4)n23)-c2ccccc2)c(C)n1
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4cc(F)c(F)c(F)c4)n23)cc1F
CCc1c2CCC(c3cc(F)cc(F)c3)n2c(Nc2ccc(OC)nc2C)nc1=O
COc1ccc(Nc2nc(=O)c(F)c3CCC(c4ccc(F)cc4F)n23)c(C)n1
COc1nc(C)c(Nc2nc(=O)cc3CCC(c4ccc(F)c(Cl)c4)n23)cc1F
COc1ccc(\N=c2/[nH]c(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c(C)n1
CCOc1ccc(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c(CC)n1
COc1ccc(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c(C)c1
COc1ccc(C)c(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c1
COc1cc(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c(C)cc1F
Cc1nc2cc(C)c(Nc3nc(=O)c(F)c4CCC(c5cc(F)cc(F)c5)n34)cc2s1
CN1CC(c2ccccc2)n2c1cc(=O)nc2Nc1cc2sc(C)nc2cc1C
COc1ccc(Nc2nc(=O)cc3N(C)CC(c4ccccc4)n23)c(C)c1
COc1ccc(C)c(Nc2nc(=O)cc3N(C)CC(c4ccccc4)n23)c1
COc1ccc(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c(C)c1F
CCN1C2=NCC(N2C(Nc2cc(C)c(C)cc2C)=NC1=O)c1ccc(F)cc1 |c:20,t:3|
CCN1C2=NCC(N2C(Nc2ccc(C)nc2C)=NC1=O)c1ccc(F)cc1 |c:19,t:3|
CN1C2=NCC(N2C(Nc2cc(nn2C)C2CC2)=NC1=O)c1ccc(F)cc1 |c:20,t:2|
CN1C2=NCC(N2C(Nc2ccc(C)nc2C)=NC1=O)c1cc(F)cc(F)c1 |c:18,t:2|
CN1C2=NCC(N2C(Nc2ccc(C)nc2C)=NC1=O)c1ccc(F)c(F)c1 |c:18,t:2|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)c(F)c2)c(C)nc1OC |t:6,12|
CCN1C2=NCC(N2C(Nc2ccc(OC)nc2C)=NC1=O)c1ccc(F)cc1 |c:20,t:3|
CCN1C2=NCC(N2C(Nc2cc(OC)c(OC)nc2C)=NC1=O)c1ccc(F)cc1 |c:22,t:3|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)c(C)n1 |t:7,13|
CN1C2=NCC(N2C(Nc2ccc(C)nc2C)=NC1=O)c1ccc(F)cc1 |c:18,t:2|
COc1cc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)cc1OC |t:8,14|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c(C)c1 |t:7,13|
COc1cnc(C)c(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)c1
COc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)c(F)c2)c1 |t:9,15|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)c(F)c2)c(C)c1 |t:7,13|
COc1cc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)c(F)c2)cc1OC |t:8,14|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)c(F)c2)c(C)n1 |t:7,13|
COc1cc(Nc2nc(=O)cc3NCC(c4cc(F)cc(F)c4)n23)c(C)cc1F
COc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)c1 |t:9,15|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2ccc(F)cc2)c(C)c1 |t:7,13|
COc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c1 |t:9,15|
COc1cc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)cc1OC |t:8,14|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c(C)nc1OC |t:6,12|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)c1 |t:7,13|
COc1nc(C)c(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)cc1C
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c(C)c1F |t:7,13|
CCN1C2=NCC(N2C(Nc2cc(OC)c(OC)cc2C)=NC1=O)c1ccc(F)cc1 |c:22,t:3|
CCN1C2=NCC(N2C(Nc2cc(OC)ccc2C)=NC1=O)c1ccc(F)cc1 |c:20,t:3|
CCN1C2=NCC(N2C(Nc2ccc(OC)cc2C)=NC1=O)c1ccc(F)cc1 |c:20,t:3|
COc1nc(C)c(Nc2nc(=O)c(F)c3CCC(c4cc(F)cc(F)c4)n23)cc1F
COc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:9,15|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)n1 |t:7,13|
COc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c(C)n1 |t:7,13|
CN1C2=NCC(N2C(Nc2cc(ccc2C)C#N)=NC1=O)c1cc(F)cc(F)c1 |c:19,t:2|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)cc(F)c2)c(C)cc1F |t:6,12|
COc1cc(C)c(Nc2nc(=O)c(F)c3N(C)CC(c4ccc(F)cc4)n23)cc1OC
COc1cc(C)c(Nc2nc(=O)nc3NCC(c4cc(F)c(F)c(F)c4)n23)cc1OC
CCc1nc(OC)ccc1NC1=NC(=O)N(C)C2=NCC(N12)c1cc(F)cc(F)c1 |t:12,18|
CN1C2=NCC(N2C(Nc2cc3sc(C)nc3cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:22,t:2|
CCOc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)cc1F |t:7,13|
COc1nc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)cc1C |t:8,14|
COc1ccc(Nc2nc(=O)c(F)c3N(C)CC(c4ccc(F)cc4)n23)c(C)n1
COc1ccc(Nc2nc(=O)c(F)c3NCC(c4cc(F)c(F)c(F)c4)n23)c(C)n1
CCOc1ccc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(CC)n1 |t:8,14|
COc1ccc(C)c(Nc2nc(=O)c(F)c3NCC(c4cc(F)c(F)c(F)c4)n23)c1
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)nc1OC |t:6,12|
COCCOc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(Cc4ccccc4)N23)c1 |t:12,18|
COc1cc(C)c(Nc2nc(=O)n(C)c3ncn(Cc4ccccc4)c23)cc1OC
CN1C2=NCC(N2C(Nc2cc(OCCO)c(F)cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:22,t:2|
COc1ccc(C)c(Nc2nc(=O)n(C)c3ncn(Cc4ccccc4)c23)c1
COc1ccc(Nc2nc(=O)n(C)c3ncn(Cc4ccccc4)c23)c(C)c1
CN1C2=NCC(N2C(Nc2cc(CO)cnc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
CN1C2=NCC(Cc3ccccc3)N2C(Nc2cc(C)ccc2C)=NC1=O |c:26,t:2|
Cc1ccc(CO)cc1NC1=NC(=O)NC2=NCC(N12)c1cc(F)c(F)c(F)c1 |t:11,16|
CN1C2=NCC(Cc3ccccc3)N2C(Nc2cc(CO)ccc2C)=NC1=O |c:27,t:2|
CCc1ccc(CO)cc1NC1=NC(=O)NC2=NCC(N12)c1cc(F)c(F)c(F)c1 |t:12,17|
CN1C2=NCC(N2C(Nc2cc(CCCO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:21,t:2|
COc1nc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)cc1CO |t:8,14|
CCc1ccc(CO)cc1NC1=NC(=O)N(C)C2=NCC(Cc3ccccc3)N12 |t:12,18|
CN1C2=NCC(N2C(Nc2cc(CC(F)(F)CO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:23,t:2|
CN1C2=NCC(N2C(Nc2cc(O[C@@H]3C[C@H](CO)C3)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |r,wU:13.13,15.16,c:25,t:2,(6.94,2.82,;5.61,2.05,;5.61,.51,;6.76,-.52,;6.13,-1.93,;4.6,-1.77,;4.28,-.26,;2.94,.51,;1.61,-.26,;.28,.51,;.28,2.05,;-1.06,2.82,;-1.06,4.36,;-2.39,5.13,;-2.79,6.62,;-4.28,6.22,;-5.61,6.99,;-6.94,6.22,;-3.88,4.73,;-2.39,2.05,;-2.39,.51,;-1.06,-.26,;-1.06,-1.8,;2.94,2.05,;4.28,2.82,;4.28,4.36,;3.57,-2.91,;2.06,-2.59,;1.03,-3.74,;-.48,-3.42,;1.51,-5.2,;.48,-6.35,;3.01,-5.52,;3.49,-6.99,;4.04,-4.38,)|
CN1C2=NCC(N2C(Nc2cc(O[C@H]3C[C@H](CO)C3)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |r,wU:15.16,wD:13.13,c:25,t:2,(6.94,2.82,;5.61,2.05,;5.61,.51,;6.76,-.52,;6.13,-1.93,;4.6,-1.77,;4.28,-.26,;2.94,.51,;1.61,-.26,;.28,.51,;.28,2.05,;-1.06,2.82,;-1.06,4.36,;-2.39,5.13,;-2.79,6.62,;-4.28,6.22,;-5.61,6.99,;-6.94,6.22,;-3.88,4.73,;-2.39,2.05,;-2.39,.51,;-1.06,-.26,;-1.06,-1.8,;2.94,2.05,;4.28,2.82,;4.28,4.36,;3.57,-2.91,;2.06,-2.59,;1.03,-3.74,;-.48,-3.42,;1.51,-5.2,;.48,-6.35,;3.01,-5.52,;3.49,-6.99,;4.04,-4.38,)|
CN1C2=NCC(N2C(Nc2cc3n(CCO)ncc3cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:24,t:2|
Cc1ccc(cc1NC1=NC(=O)N(CCO)C2=NCC(N12)c1cc(F)c(F)c(F)c1)C#N |t:9,17|
CN1C2=NCC(N2C(Nc2cc(OC[C@H]3C[C@H](O)C3)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |r,wU:16.17,wD:14.14,c:25,t:2,(5.21,1.12,;3.88,.35,;3.88,-1.19,;5.02,-2.22,;4.4,-3.63,;2.87,-3.47,;2.55,-1.96,;1.21,-1.19,;-.12,-1.96,;-1.46,-1.19,;-1.46,.35,;-2.79,1.12,;-2.79,2.66,;-4.12,3.43,;-4.12,4.97,;-3.03,6.06,;-4.12,7.15,;-4.12,8.69,;-5.21,6.06,;-4.12,.35,;-4.12,-1.19,;-2.79,-1.96,;-2.79,-3.5,;1.21,.35,;2.55,1.12,;2.55,2.66,;1.83,-4.61,;.33,-4.29,;-.7,-5.44,;-2.21,-5.12,;-.23,-6.9,;-1.26,-8.05,;1.28,-7.22,;1.76,-8.69,;2.31,-6.08,)|
CN1C2=NCC(N2C(Nc2cc(C=O)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
CN1C2=NCC(N2C(Nc2cc(Oc3ccccn3)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:25,t:2|
CN1C2=NCC(N2C(Nc2cc(CCO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:20,t:2|
CN1C2=NCC(N2C(Nc2cc(CO)ccc2C)=NC1=O)c1cc(F)nc(F)c1 |c:19,t:2|
CN1C2=NCC(N2C(NCc2ccccc2F)=NC1=O)c1cc(F)c(F)c(F)c1 |c:18,t:2|
CN1C2=NCC(N2C(NCc2cccc(F)c2)=NC1=O)c1cc(F)c(F)c(F)c1 |c:18,t:2|
CN1C2=NCC(N2C(NCc2ccc(F)cc2)=NC1=O)c1cc(F)c(F)c(F)c1 |c:18,t:2|
CN1C2=NCC(N2C(Nc2cc(OCCS(C)(=O)=O)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:24,t:2|
CN1C2=NCC(N2C(Nc2cc(OCC#N)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:21,t:2|
COCCc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:11,17|
COCC(F)(F)Oc1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:14,20|
CN1C2=NCC(N2C(Nc2cc(OC(F)(F)CO)ccc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:23,t:2|
COCC(F)(F)c1ccc(C)c(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c1 |t:13,19|
CN1C2=NCC(N2C(Nc2cc(ccc2C)C(F)(F)CO)=NC1=O)c1cc(F)c(F)c(F)c1 |c:22,t:2|
COc1ccc(cc1)[C@@H](C)NC1=NC(=O)N(C)C2=NCC(N12)c1cc(F)c(F)c(F)c1 |r,t:12,18|
CN1C2=NCC(N2C(Nc2ccc(cc2C)C#N)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
COc1cc(NC2=NC(=O)N(C)C3=NCC(N23)c2cc(F)c(F)c(F)c2)c(C)cc1C#N |t:6,12|
CN1C2=NCC(N2C(Nc2cc(ccc2F)C#N)=NC1=O)c1cc(F)c(F)c(F)c1 |c:19,t:2|
CN1C2=NCC(N2C(Nc2cc(C#N)c(F)cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:20,t:2|
CN1C2=NCC(N2C(Nc2cc(cc(F)c2C)C#N)=NC1=O)c1cc(F)c(F)c(F)c1 |c:20,t:2|
CN1C2=NCC(N2C(Nc2cc(ccc2C)C2=NCCO2)=NC1=O)c1cc(F)c(F)c(F)c1 |c:23,t:2,18|
CN1C2=NCC(N2C(Nc2cc(C3=NCCO3)c(F)cc2C)=NC1=O)c1cc(F)c(F)c(F)c1 |c:24,t:2,13|
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(=O)c2ncccc12
FC(F)(F)c1cccc(CNC(=O)C2CCC(=O)c3ncccc23)c1Cl
Clc1cccc(CNC(=O)C2CCC(=O)c3ncccc23)c1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(=O)c2ncccc12
O=C(NCC1CCCCCC1)C1CCC(=O)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(O)c2ncccc12
OC1CCC(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
OC1CCC(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(O)c2ncccc12
COCc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(O)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CC(=C)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(=O)c2ncccc12
FC(F)(F)c1cccc(CNC(=O)C2(F)CCC(=O)c3ncccc23)c1Cl
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(=O)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(O)CCC(=O)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CC(=O)c2ncccc12
FC(F)(F)c1cccc(CNC(=O)C2CC(=O)c3ncccc23)c1Cl
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(O)c2ncccc12
OC1CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
OCc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(O)c2ncccc12
OC1CCC(F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12
OC1CCC(F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12
COCc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(O)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(O)CCC(O)c2ncccc12
OC1CCC(O)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CC(O)c2ncccc12
OC1CC(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
OC1CC(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12
OC1CC(F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(CC(O)=O)c2ncccc12
OC(=O)CC1CCC(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
NC(=O)CC1CCC(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(O)(CO)c2ncccc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(O)(CO)c2ncccc12
OCC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
OCC1(O)CCC(F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12
OCC1(O)CCC(F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12
OCC1(O)CC(F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12
COCC1(O)CCC(F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12
COCC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
COC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
COC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CCC(O)(CN)c2ncccc12
CNCC1(O)CCC(C(=O)NCc2c(C)cc(Cl)cc2Cl)c2cccnc12
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1(F)CCC(O)(CN)c2ncccc12
CNCC1(O)CCC(F)(C(=O)NCc2c(C)cc(Cl)cc2Cl)c2cccnc12
CN(C)CC1(O)CCC(F)(C(=O)NCc2c(C)cc(Cl)cc2Cl)c2cccnc12
NCC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
CNCC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
CN(C)CC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
OC1CN(C[C@]2(O)CC[C@@](F)(C(=O)NCc3ccc(Cl)cc3Cl)c3cccnc23)C1 |r|
OC1CN(C[C@]2(O)CC[C@@](F)(C(=O)NCc3ccc(F)cc3Cl)c3cccnc23)C1 |r|
COC1CN(C[C@]2(O)CC[C@@](F)(C(=O)NCc3ccc(F)cc3Cl)c3cccnc23)C1 |r|
CC1(O)CN(C[C@]2(O)CC[C@@](F)(C(=O)NCc3ccc(F)cc3Cl)c3cccnc23)C1 |r|
COC1(C)CN(C[C@]2(O)CC[C@@](F)(C(=O)NCc3ccc(F)cc3Cl)c3cccnc23)C1 |r|
OCCNC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CN(CCO)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CC1(O)CCC(F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12
N[C@]1(CO)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
N[C@@]1(CO)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
F[C@]1(CC[C@]2(COCC(=O)N2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
F[C@]1(CC[C@@]2(COCC(=O)N2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@H]1CC[C@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)C1CC[C@H](O)c2ncccc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2c(F)cc(F)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(F)cc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(F)cc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(Br)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(Br)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2ccc(F)c(F)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@H](C(=O)NCc2ccc(F)c(F)c2Cl)c2cccnc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@H]1C[C@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@@H]1CC[C@@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@H]1CC[C@@H](O)c2ncccc12 |r|
O[C@H]1CC[C@H](C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@@H](C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@H](C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@H](C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@H](C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@H](C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@H](C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@H](C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@@H]1CC[C@H](C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@@H]1CC[C@@H](C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@@H]1CC[C@H](C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@@H]1C[C@@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@H]1C[C@@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@@]1(F)CC[C@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@H](O)c2ncccc12 |r|
O[C@H]1CC[C@](F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@@]1(F)CC[C@H](O)c2ncccc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@H](O)c2ncccc12 |r|
O[C@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@](F)(C(=O)NCc2c(Cl)cc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2C(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2C(F)F)c2cccnc12 |r|
O[C@H]1CC[C@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2ccc(Br)cc2Cl)c2cccnc12 |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@@H](O)c2ncccc12)c1ccc(Cl)cc1Cl |r|
O[C@H]1CC[C@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
Cc1cccc(Cl)c1CNC(=O)[C@]1(F)CC[C@@H](O)c2ncccc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2cc(F)c(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@@](F)(C(=O)NCc2c(Cl)ccc(Cl)c2Cl)c2cccnc12 |r|
Cc1ccc(CNC(=O)[C@]2(F)CC[C@@H](O)c3ncccc23)c(Cl)c1 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@@]1(F)CC[C@@H](O)c2ncccc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@@]1(F)CC[C@@H](O)c2ncccc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2c(Cl)cccc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cccc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
Cc1ccc(F)c(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c1Cl |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(F)cc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2c(Cl)cc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2C(F)F)c2cccnc12 |r|
OCc1cc(F)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(Br)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Br)cc2Cl)c2cccnc12 |r|
C[C@@H](NC(=O)[C@@]1(F)CC[C@@H](O)c2ncccc12)c1ccc(Cl)cc1Cl |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2C(F)(F)F)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
Cc1cccc(Cl)c1CNC(=O)[C@@]1(F)CC[C@@H](O)c2ncccc12 |r|
Cc1cccc(Cl)c1CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2cc(F)c(F)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(F)c(F)cc2Cl)c2cccnc12 |r|
O[C@@H]1CC[C@](F)(C(=O)NCc2c(Cl)ccc(Cl)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)ccc(Cl)c2Cl)c2cccnc12 |r|
Cc1ccc(CNC(=O)[C@@]2(F)CC[C@@H](O)c3ncccc23)c(Cl)c1 |r|
Cc1ccc(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c(Cl)c1 |r|
C[C@H](NC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)c1ccc(Cl)c(Cl)c1Cl |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(F)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)ccc(F)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cccc2Cl)c2cccnc12 |r|
COc1ccc(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c(Cl)c1 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(Cl)ccc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(c2F)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(F)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ncc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(F)c2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cccc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(F)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(Br)ccc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Br)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)c(F)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(Cl)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cccc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(Cl)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@@H]2CCCc3ccccc23)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(Cl)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCC2(CCCCC2)N2CCOCC2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)ccc(Cl)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ncc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccccc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@@H]2CCc3ccccc23)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)c(Cl)c2)c2cccnc12 |r|
COc1cccc(Cl)c1CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccccc2C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(F)c(F)c(F)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(cc2F)C#N)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(F)cc(Cl)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(F)ccc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(Cl)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)c(F)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(OC(F)(F)F)cc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cccc(F)c2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(ccc2Cl)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2)c2cccnc12 |r|
COc1ccc(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c(c1)C(F)(F)F |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(Cl)cc(Cl)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2nc(cs2)-c2ccc(Cl)cc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccccc2CN2CCOCC2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@H]2C[C@@H]2c2ccccc2)c2cccnc12 |r|
Cc1ccc(Cl)c(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c1F |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cccc2F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@H]2CCCc3ccccc23)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCCOc2cccc(c2)C(F)(F)F)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCC2(CC2)c2ccc(F)cc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2cc(F)cc(F)c2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@@H]2C[C@H]2c2ccccc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccccc2F)c2cccnc12 |r|
COc1cccc(CNC(=O)[C@]2(F)CC[C@H](O)c3ncccc23)c1Cl |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@H]2CCC[C@@H]2OCc2ccccc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)N[C@H]2CCc3ccccc23)c2cccnc12 |r|
CC(C)(C)CCNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCCOc2ccccc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NC2COc3cc(Cl)cc(Cl)c23)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NC2CCOc3cc(Cl)cc(Cl)c23)c2cccnc12 |r|
CC(NC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)C12CC3CC(CC(C3)C1)C2 |r,TLB:20:21:19.18.24:25,24:19:26:23.25.22,24:23:26:20.19.18,THB:20:19:25:26.21.22|
O[C@H]1CC[C@@](F)(C(=O)NCC(N2CCC(F)(F)CC2)c2ccc(Cl)cc2)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NC2COc3ccccc3C2)c2cccnc12 |r|
CC(CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)c1ccc(Cl)cc1 |r|
O[C@H]1CC[C@@](F)(C(=O)NCC(N2CCOCC2)c2ccccc2)c2cccnc12 |r|
Cc1ncsc1C(CNC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)N1CCC(F)(F)CC1 |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)c1ccc(F)cc1Cl |r|
O[C@H]1CC[C@@](F)(C(=O)NC2CC2c2ccc(Cl)cc2Cl)c2cccnc12 |r|
C[C@H](NC(=O)[C@]1(F)CC[C@H](O)c2ncccc12)c1ccc(F)cc1Cl |r|
O[C@H]1CC[C@@](F)(C(=O)NCC2(CCOCC2)c2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cc(F)cnc12 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cc(F)cnc12 |r|
Cc1cnc2[C@@H](O)CC[C@@](F)(C(=O)NCc3ccc(Cl)cc3Cl)c2c1 |r|
Cc1cnc2[C@@H](O)CC[C@@](F)(C(=O)NCc3ccc(F)cc3Cl)c2c1 |r|
O[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2ccc[n+]([O-])c12 |r|
FC(F)(F)c1cccc(CNC(=O)[C@@]2(F)CCC(=O)c3ncccc23)c1Cl |r|
FC(F)(F)c1cccc(CNC(=O)[C@]2(F)CCC(=O)c3ncccc23)c1Cl |r|
F[C@]1(CCC(=O)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
Fc1ccc(CNC(=O)[C@]2(F)CCC(=O)c3ncccc23)c(Cl)c1 |r|
Fc1cccc(CNC(=O)[C@]2(F)CCC(=O)c3ncccc23)c1Cl |r|
Fc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CCC(=O)c2ncccc12 |r|
F[C@]1(CCC(=O)c2ncccc12)C(=O)NCc1cccc(Cl)c1Cl |r|
FC(F)(F)c1ccc(CNC(=O)[C@]2(F)CCC(=O)c3ncccc23)c(Cl)c1 |r|
Fc1ccc(CNC(=O)[C@]2(F)CCC(=O)c3ncccc23)c(F)c1F |r|
F[C@]1(CCC(=O)c2ncccc12)C(=O)NCc1ncc(Cl)cc1Cl |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
C[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
C[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2CO)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2c(Cl)cc(F)cc2CO)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(F)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)c(F)c2F)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(Cl)c2F)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2F)c2cccnc12 |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@](C)(O)c2ncccc12)c1ccc(F)cc1Cl |r|
C[C@H](NC(=O)[C@]1(F)CC[C@](C)(O)c2ncccc12)c1ccc(F)cc1Cl |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCc2ncc(Cl)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NC2CC2c2ccc(Cl)cc2Cl)c2cccnc12 |r|
C[C@]1(O)CC[C@@](F)(C(=O)NCC2(CCCCC2)N2CCOCC2)c2cccnc12 |r|
C[C@@]1(O)CC[C@@](F)(C(=O)NCC2(CCCCC2)N2CCOCC2)c2cccnc12 |r|
Cc1cnc2c(c1)[C@@](F)(CC[C@]2(C)O)C(=O)NCc1ccc(F)cc1Cl |r|
CN(CCO)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
CN(CCO)C[C@@]1(O)CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC1CN(C[C@@]2(O)CC[C@](F)(C(=O)NCc3ccc(Cl)cc3Cl)c3cccnc23)C1 |r|
O[C@@]1(CC#N)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@]1(CC#N)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
O[C@]1(CC#N)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@](O)(CC#N)c2ncccc12 |r|
OCc1cc(F)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@](O)(CC#N)c2ncccc12 |r|
O[C@@]1(CF)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
O[C@@]1(CF)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CSC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
CSC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OCCSC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CN1CCO[C@]2(CC[C@@](F)(C(=O)NCc3ccc(Cl)cc3Cl)c3cccnc23)C1 |r|
F[C@]1(CC[C@]2(CNC(=O)O2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
F[C@]1(CC[C@@]2(CNC(=O)O2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
F[C@@]1(CC[C@]2(CNC(=O)CO2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
F[C@]1(CC[C@]2(CNC(=O)CO2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
F[C@]1(CC[C@@]2(CNC(=O)CO2)c2ncccc12)C(=O)NCc1ccc(Cl)cc1Cl |r|
CS(=O)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CS(=O)(=O)C[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
CS(=O)(=O)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
CS(=O)(=O)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OCCS(=O)(=O)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OCCS(=O)(=O)C[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OC[C@@]1(O)CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2Cl)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
OC[C@@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
OCc1cc(Cl)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@](O)(CO)c2ncccc12 |r|
OCc1cc(F)cc(Cl)c1CNC(=O)[C@]1(F)CC[C@@](O)(CO)c2ncccc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)c(F)c2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(Cl)c2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(F)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)c(F)c2F)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)c(Cl)c2F)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2F)c2cccnc12 |r|
Cc1cnc2c(c1)[C@@](F)(CC[C@@]2(O)CO)C(=O)NCc1ccc(Cl)cc1Cl |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@@](O)(CO)c2ncccc12)c1ccc(Cl)cc1Cl |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@@](O)(CO)c2ncccc12)c1ccc(F)cc1Cl |r|
C[C@@H](NC(=O)[C@]1(F)CC[C@](O)(CO)c2ncccc12)c1ccc(F)cc1Cl |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCc2ncc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NC2CC2c2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC[C@]1(O)CC[C@@](F)(C(=O)NCC2(CCOCC2)c2ccc(Cl)cc2Cl)c2cccnc12 |r|
CO[C@H]1CC[C@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2CO)c2cccnc12 |r|
CO[C@@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2CO)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2Cl)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(cc2Cl)C(F)(F)F)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(F)cc2F)c2cccnc12 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
OCCO[C@H]1CC[C@@](F)(C(=O)NCc2c(Cl)cc(Cl)cc2CO)c2cccnc12 |r|
OCCO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
OCCO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)c(F)c2F)c2cccnc12 |r|
OCCO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2F)c2cccnc12 |r|
OCCO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(F)cc2F)c2cccnc12 |r|
OCCO[C@@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OCC(O)CO[C@H]1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
CS(=O)(=O)C1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OCCS(=O)(=O)C1CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
F[C@H]1CC[C@](F)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
F[C@H]1CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
F[C@H]1CC[C@](F)(C(=O)NCc2cccc(Cl)c2Cl)c2cccnc12 |r|
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc3sc(C)nc3cc2C)cc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Oc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(NCc2cccc(Cl)c2C)nc1=O
Cc1c(Cl)cccc1Nc1nc(=O)c(OOC(C)(C)C)cn1Cc1ccccc1
COc1cn(Cc2ccccc2)c(Nc2cccc(C)c2Cl)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)cc1C
COc1cn(Cc2ccccc2)c(Oc2cc(C)c(C)cc2C)nc1=O
COc1cn(Cc2cccc(OC(F)F)c2)c(Nc2cccc(Cl)c2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)cc1C
CCc1cc(OC)ccc1Nc1nc(=O)c(OC)cn1Cc1cc(F)cc(Cl)c1
COc1cn(Cc2ccccc2)c(Nc2cc(c(C)cc2C)S(C)(=O)=O)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2cc(c(C)cc2C)S(C)(=O)=O)nc1=O
CCc1ccc(F)cc1Nc1nc(=O)c(OC)cn1Cc1ccccc1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(F)c2)c1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1
CCOc1ccc(C)c(Nc2nc(=O)c(OC)cn2Cc2cc(F)cc(Cl)c2)c1
COc1cn(Cc2ccc(F)c(F)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(Cl)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cn(Cc2cc(F)cc(F)c2)c(Nc2ccc(C)cc2C)nc1=O
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccccc2)cc1Cl
COc1cc(C)c(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)cc1Cl
COc1cn(Cc2cccc(Cl)c2)c(Nc2cccc(c2C)C(F)(F)F)nc1=O
COc1cc(Nc2nc(=O)c(OC)cn2Cc2cccc(F)c2)c(C)cc1Cl
COc1cc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)cc2)c(C)cc1Cl
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2cccc(Cl)c2)c1C
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(F)c2)c1C
COc1cccc(Nc2nc(=O)c(OC)cn2Cc2ccc(F)c(Cl)c2)c1C
COc1cn(Cc2cc(F)c(F)c(F)c2)c(Cc2cccc3[nH]c(=O)ccc23)nc1=O
COC1CN(Cc2ccc(F)c(F)c2)C(Nc2cc(c(C)cc2C)S(C)(=O)=O)=NC1=O |c:29|
COc1cn(Cc2ccccc2)c(Nc2cc(cc(C)c2C)[N+]([O-])=O)nc1=O
COc1cn(Cc2ccccc2)c(Nc2ccc(C)cc2F)nc1=O
COc1cn(Cc2ccc(F)c(Cl)c2)c(Nc2c(C)cc3COCc3c2C)nc1=O
CCOc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)cc(F)c2)c(C)cc1F
COc1cc(C)c(Nc2nc(=O)cc(C)n2Cc2cc(F)c(F)c(F)c2)cc1OC
COc1ccc(NC2=NC(=O)CC(C)N2Cc2cc(F)c(F)c(F)c2)c(C)c1 |t:7|
Cc1cc(F)c(cc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1)-c1cccn(C)c1=O
COCC1(O)CCC(F)(C(=O)NCc2c(C)cc(Cl)cc2Cl)c2cccnc12
OC1CC(C1)N[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r,wU:10.11,6.6,wD:10.12,6.7,(-1.73,-6.93,;-2.13,-5.45,;-3.46,-4.68,;-2.69,-3.34,;-1.36,-4.11,;-3.09,-1.86,;-2,-.77,;-.91,-1.86,;-.67,0,;-.67,1.54,;-2,2.31,;-.67,3.08,;-2,3.85,;-3.33,4.62,;-.67,4.62,;.67,3.85,;2,4.62,;2,6.16,;3.33,6.93,;4.67,6.16,;6,6.93,;4.67,4.62,;3.33,3.85,;3.33,2.31,;-3.33,1.54,;-4.67,2.31,;-6,1.54,;-6,0,;-4.67,-.77,;-3.33,0,)|
OC1CC(C1)N[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r,wU:10.11,6.6,wD:10.12,6.7,(-1.73,-6.93,;-2.13,-5.45,;-3.46,-4.68,;-2.69,-3.34,;-1.36,-4.11,;-3.09,-1.86,;-2,-.77,;-.91,-1.86,;-.67,0,;-.67,1.54,;-2,2.31,;-.67,3.08,;-2,3.85,;-3.33,4.62,;-.67,4.62,;.67,3.85,;2,4.62,;2,6.16,;3.33,6.93,;4.67,6.16,;6,6.93,;4.67,4.62,;3.33,3.85,;3.33,2.31,;-3.33,1.54,;-4.67,2.31,;-6,1.54,;-6,0,;-4.67,-.77,;-3.33,0,)|
COC1CC(C1)N[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r,wU:11.12,7.7,wD:11.13,7.8,(-.24,-7.13,;-1.73,-6.73,;-2.13,-5.25,;-3.46,-4.48,;-2.69,-3.14,;-1.36,-3.91,;-3.09,-1.66,;-2,-.57,;-.91,-1.66,;-.67,.2,;-.67,1.74,;-2,2.51,;-.67,3.28,;-2,4.05,;-3.33,4.82,;-.67,4.82,;.67,4.05,;2,4.82,;2,6.36,;3.33,7.13,;4.67,6.36,;6,7.13,;4.67,4.82,;3.33,4.05,;3.33,2.51,;-3.33,1.74,;-4.67,2.51,;-6,1.74,;-6,.2,;-4.67,-.57,;-3.33,.2,)|
CC1(O)CC(C1)N[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r,wU:11.12,7.7,wD:11.13,7.8,(-2.9,-6.86,;-2.13,-5.52,;-.79,-6.29,;-3.46,-4.75,;-2.69,-3.42,;-1.36,-4.19,;-3.09,-1.93,;-2,-.84,;-.91,-1.93,;-.67,-.07,;-.67,1.47,;-2,2.24,;-.67,3.01,;-2,3.78,;-3.33,4.55,;-.67,4.55,;.67,3.78,;2,4.55,;2,6.09,;3.33,6.86,;4.67,6.09,;6,6.86,;4.67,4.55,;3.33,3.78,;3.33,2.24,;-3.33,1.47,;-4.67,2.24,;-6,1.47,;-6,-.07,;-4.67,-.84,;-3.33,-.07,)|
COC1(C)CC(C1)N[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r,wU:12.13,8.8,wD:12.14,8.9,(.54,-5.52,;-.79,-6.29,;-2.13,-5.52,;-2.9,-6.86,;-3.46,-4.75,;-2.69,-3.42,;-1.36,-4.19,;-3.09,-1.93,;-2,-.84,;-.91,-1.93,;-.67,-.07,;-.67,1.47,;-2,2.24,;-.67,3.01,;-2,3.78,;-3.33,4.55,;-.67,4.55,;.67,3.78,;2,4.55,;2,6.09,;3.33,6.86,;4.67,6.09,;6,6.86,;4.67,4.55,;3.33,3.78,;3.33,2.24,;-3.33,1.47,;-4.67,2.24,;-6,1.47,;-6,-.07,;-4.67,-.84,;-3.33,-.07,)|
OCCNN[C@]1(O)CC[C@@](F)(C(=O)NCc2ccc(F)cc2Cl)c2cccnc12 |r|
Cc1cc(Cl)cc(Cl)c1CNC(=O)[C@@H]1CC[C@H](O)c2ncccc12 |r|
CN(CCO)C[C@@]1(C)CC[C@](F)(C(=O)NCc2ccc(Cl)cc2Cl)c2cccnc12 |r|
OC1CN(CC2(O)CC[C@](F)(C(=O)NCc3ccc(Cl)cc3Cl)c3cccnc23)C1 |r|
CO[C@H]1CC[C@@](F)(C(=O)NCc2c(F)cc(Cl)cc2CO)c2cccnc12 |r|
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccnc1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccncc1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccncc1F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncccc1F
Cc1cc(COC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)no1
Cc1noc(C)c1COC1CCN(CC1)C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C(F)F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccs1
Cc1nsc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nc(Cl)cs1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nc(ns1)C1CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc(c1)C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccnc1C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccnc1C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nc2ccccc2s1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nc2ccccc2o1
COCCc1nsc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nc(no1)-c1ccccc1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nnnn1-c1ccccc1
Cc1cnc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)nc1
Cc1ccc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)nn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(F)cn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(F)ncn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccc(F)nn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc(F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccnc1F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccnc(F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncccc1C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccc(n1)C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cnccc1C#N
Cc1nc(F)cc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
Cc1c(F)ncnc1OC1CCN(CC1)C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C(F)F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccc(n1)C(F)(F)F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(ncn1)C(F)(F)F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccn2nccc12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc2nncn12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccn2cnnc12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncccc1Cl
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccnc2cccnc12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccc2ncccc12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccncc1C#N
Cn1ncc2c(OC3CCN(CC3)C(CNC(=O)c3c(F)cccc3Cl)c3scnc3C(F)F)ncnc12
Cc1nnc2c(OC3CCN(CC3)C(CNC(=O)c3c(F)cccc3Cl)c3scnc3C(F)F)nccn12
Cc1nsc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)c1C#N
Cc1cc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)nc(F)n1
Cc1cnc(F)nc1OC1CCN(CC1)C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C(F)F
Cc1ncnc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)c1F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc(n1)-n1cccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncccc1C(F)(F)F
COc1nccc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
COc1ccnc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
COc1cc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)ncn1
Cc1nc(C)c(F)c(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ncnc2ccccc12
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cnccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccnn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccc(F)n1
Cc1cc(OC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)ccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1nccc(Cl)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cncc(Cl)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cccc(Cl)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccncn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(ccn1)C#N
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccnc(F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1cc(F)ccn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nccs2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nc(Cl)cs2)CC1
Cc1nsc(OCC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nc(ns2)C2CC2)CC1
Cc1cccc(OCC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)n1
Cc1ccnc(OCC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)c1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cccnc2C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cncc(c2)C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nccnc2C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nc3ccccc3s2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nnnn2-c2ccccc2)CC1
Cc1cccnc1OCC1CCN(CC1)C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C(F)F
Cc1cnc(OCC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)nc1
Cc1ccc(OCC2CCN(CC2)C(CNC(=O)c2c(F)cccc2Cl)c2scnc2C(F)F)nn1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccc(F)cn2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cc(F)ncn2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccc(F)nn2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cncc(F)n2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nccnc2F)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccnc(F)n2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ncccc2C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cccc(n2)C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccnc(c2)C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cnccc2C#N)CC1
Cc1c(F)ncnc1OCC1CCN(CC1)C(CNC(=O)c1c(F)cccc1Cl)c1scnc1C(F)F
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nccc(n2)C(F)(F)F)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cc(ncn2)C(F)(F)F)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2nccn3nccc23)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccn3nccc3n2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cncc3nncn23)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ncccc2Cl)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccncc2C#N)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cccc(F)n2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2ccnc(F)c2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(COc2cc(F)ccn2)CC1
FC(F)c1ncsc1C(CNC(=O)c1c(F)cccc1Cl)N1CCC(CC1)Oc1ccnc(c1)C#N
N=C(NCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
S=C(NCC12CC3CC(CC(C3)C1)C2)Nc1ccccc1 |TLB:3:4:7:11.10.9,THB:5:6:9:13.4.12,5:4:7.6.11:9,12:4:7:11.10.9,12:10:7:13.5.4|
O=C(NCc1ccncc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
O=C(NCc1cccnc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
O=C(NCCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:12:13:16:20.19.18,THB:14:15:18:22.13.21,14:13:16.15.20:18,21:13:16:20.19.18,21:19:16:22.14.13|
O=C(NCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:15:16:20:14.13.19,THB:15:14:20:16.21.17,17:16:13:18.20.19,17:18:13:16.21.15|
N#C\N=C(/NCC12CC3CC(CC(C3)C1)C2)Nc1ccccc1 |TLB:5:6:9:13.12.11,THB:7:8:11:15.6.14,7:6:9.8.13:11,14:6:9:13.12.11,14:12:9:15.7.6|
S=C(NCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
O=C(NCc1ccccn1)NCC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
O=C(NCC12CC3CC(CC(C3)C1)C2)Nc1ccccc1 |TLB:3:4:7:11.10.9,THB:5:6:9:13.4.12,5:4:7.6.11:9,12:4:7:11.10.9,12:10:7:13.5.4|
C[C@H]1Cc2c(CN1C(=O)c1cn[nH]c1C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
[H][C@]1(C)Cc2c(CN1C(=O)c1ccnc(c1C)C(F)(F)F)nnn2-c1ncc(F)cn1 |r|
c1cc(c(cc1CCCNCCCO)C(=O)NCC23CC4CC(C2)CC(C4)C3)Cl
COc1ccc(cc1)C(=O)C1=C(O)C(=O)N(C1C1CCCCC1)c1ccc(cc1)-c1ccon1 |c:11|
CCOc1ccc(Nc2ccc(cc2)C(=C2\C=C/C(/C=C2C)=[N+](/CC)Cc2cccc(c2)S([O-])(=O)=O)\c2ccc(cc2C)N(CC)Cc2cccc(c2)S([O-])(=O)=O)cc1 |c:17,20|
O=Cc1cn(nn1)-c1ccccc1
CCCCCCCCCC(=O)OCc1cn(nn1)-c1ccc(Cl)cc1
Clc1cccc(c1Cl)-n1nnnc1NCc1ccccc1Oc1ccccn1
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc3ncccc23)C(C)(C)C)cc1OC |w:11.10|
OCc1cnn(n1)-c1ccccc1
CCOCc1cn(nn1)-c1ccc(Cl)cc1
O\N=C\c1cnn(n1)-c1ccccc1
COc1ccc(cc1)-n1cc(CO)nn1
CCCCOCc1cn(nn1)-c1cc(Cl)ccc1Cl
COC[C@H](O)Cn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O |r|
Clc1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:15:16:19:23.21.22,THB:21:20:17:23.22.24,21:22:19.20.25:17,24:22:19:25.16.17,24:16:19:23.21.22|
O=C(CC12CC3CC(CC(C3)C1)C2)Nc1cccc2nc(ccc12)-c1ccccc1 |TLB:2:3:6:10.8.9,THB:8:7:4:10.9.11,8:9:6.7.12:4,11:9:6:12.3.4,11:3:6:10.8.9|
OCc1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:16:17:20:24.22.23,THB:22:21:18:24.23.25,22:23:20.21.26:18,25:23:20:26.17.18,25:17:20:24.22.23|
COC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(Br)cc2)c1=O |THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
COc1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:16:17:20:24.22.23,THB:22:21:18:24.23.25,22:23:20.21.26:18,25:23:20:26.17.18,25:17:20:24.22.23|
OCCCNCCCc1ccc(Cl)c(c1)C(=O)NCC1C2CC3CC(C2)CC1C3
COC(=O)c1cc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(OC)cc2)c1=O |THB:17:16:13:19.18.20,17:18:15.16.21:13,20:18:15:21.12.13,20:12:15:19.17.18|
CCOC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(OC)cc2)c1=O |THB:17:16:13:19.18.20,17:18:15.16.21:13,20:18:15:21.12.13,20:12:15:19.17.18|
[O-][N+](=O)c1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)C1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Clc1cccc(-c2nnnn2Cc2cccnc2)c1Cl
N[C@H]1CCN(Cc2ccc(Cl)c(c2)C(=O)NCC2C3CC4CC(C3)CC2C4)C1 |r,wU:1.0,TLB:23:22:26:19.18.17,23:18:21.22.24:26,THB:17:18:21:24.25.26,17:25:21:19.23.18,16:17:21.22.24:26,(18.99,-10.68,;17.45,-10.69,;16.69,-12.03,;15.18,-11.72,;15,-10.2,;13.66,-9.44,;13.64,-7.9,;14.97,-7.12,;14.95,-5.57,;13.6,-4.82,;13.58,-3.28,;12.29,-5.61,;12.3,-7.15,;10.95,-4.85,;10.93,-3.31,;9.63,-5.64,;8.28,-4.88,;6.96,-5.67,;6.95,-7.21,;5.54,-7.55,;4.21,-7.06,;3.01,-8.35,;4.52,-7.93,;5.93,-8.49,;4.52,-6.33,;5.56,-5.09,;4.2,-5.57,;16.4,-9.55,)|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)NNc1c(Cl)cncc1Cl |TLB:12:9:4:2.7.1,7:1:4.5.8:10,0:1:4:8.9.10,THB:7:5:10:2.1.11,6:5:10:2.1.11,11:1:4:8.9.10,11:9:4:2.7.1|
CN(C)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
COC(=O)c1cc2c(NC(=O)CC3CCCCC3)cccc2n(Cc2ccc(OC)cc2)c1=O
COC(=O)c1cc2c(NC(=O)C3CCCCC3)cccc2n(Cc2ccc(OC)cc2)c1=O
COC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(F)cc2)c1=O |THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
Clc1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:9:10:13:17.15.16,THB:15:14:11:17.16.18,15:16:13.14.19:11,18:16:13:19.10.11,18:10:13:17.15.16|
Clc1ccc2c(NC(=O)CC3CCCCC3)cccc2n1
Nc1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:15:16:19:23.21.22,THB:21:20:17:23.22.24,21:22:19.20.25:17,24:22:19:25.16.17,24:16:19:23.21.22|
OC(=O)c1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Oc1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:15:16:19:23.21.22,THB:21:20:17:23.22.24,21:22:19.20.25:17,24:22:19:25.16.17,24:16:19:23.21.22|
COC(=O)c1ccc(cc1)-c1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:18:19:22:26.24.25,THB:24:23:20:26.25.27,24:25:22.23.28:20,27:25:22:28.19.20,27:19:22:26.24.25|
COC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(OC)cc2)c1=O |THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
CCCOC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(OC)cc2)c1=O |THB:18:17:14:20.19.21,18:19:16.17.22:14,21:19:16:22.13.14,21:13:16:20.18.19|
COC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(cc2)[N+]([O-])=O)c1=O |THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
COC(=O)c1cc2c(NC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n(Cc2ccc(Cl)cc2)c1=O |THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
c1ccc2c(c1)C(=O)C=C(C2=O)O
OC1=C(C(=O)c2ccccc2C1=O)c1ccc(cc1)C#N |t:1|
COc1cccc(c1)C1=C(O)C(=O)c2ccccc2C1=O |c:9|
OC1=C(C(=O)c2ccccc2C1=O)c1cccc(F)c1 |t:1|
Cc1ccc(cc1)C1=C(O)C(=O)c2ccccc2C1=O |c:8|
OC1=C(C(=O)c2ccccc2C1=O)c1ccccc1 |t:1|
OC1=C(Br)C(=O)c2ccccc2C1=O |c:1|
COc1ccc(cc1)C1=C(O)C(=O)c2ccccc2C1=O |c:9|
OC1=C(I)C(=O)c2ccccc2C1=O |c:1|
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(N)cc1)S(=O)(=O)c1cccc2cnccc12
Clc1ccccc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:18:13:20:17.19.16,18:17:20:13.12.14,THB:16:17:12:15.20.14,16:15:12:17.19.18|
COc1cccc(Cn2cnnc2-c2cccc(Cl)c2Cl)c1
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(cc1)C#N)S(=O)(=O)c1cccc2cnccc12
CN(C)CCn1nc(C)c(CC(=O)NCc2ccc(F)cc2Cl)c1C
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(Cc2ccc(F)cc2)CC1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(C)cc1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1cccc(Cl)c1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(F)cc1)S(=O)(=O)c1cccc2cnccc12
Cc1nn(C)c(C)c1CC(=O)NCc1ccc(F)cc1Cl
Cc1nn(c(C)c1CC(=O)NCc1ccc(F)cc1Cl)-c1ccc(Cl)cc1
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1
Clc1cccc(-c2nncn2[C@H]2CCc3ccccc23)c1Cl
CSc1ccccc1Cn1cnnc1-c1cccc(c1Cl)C(F)(F)F
Clc1cccc(-c2ccnn2Cc2ccccc2)c1Cl
CN(Cc1ccc(Cl)cc1)CC12CC3CC(CC(C3)C1)C2 |THB:16:15:12:18.17.19,20:15:18:11.12.19|
COc1ccc(Cl)c(NC(=O)CC23CC4CC(CC(C4)C2)C3)c1 |TLB:21:12:19:16.15.17,THB:20:12:15:18.19.17,20:18:12.13.21:15,21:16:12.13.20:19|
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(Cc2ccccc2)CC1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(cc1)[N+]([O-])=O)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1cccc(C)c1C)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(Cl)c(Cl)c1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccccc1Cl)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(Cl)cc1)S(=O)(=O)c1cccc2cnccc12
COc1cccc(-c2nnnn2Cc2cccnc2)c1OC
Cc1cccc(-c2nnnn2Cc2cccnc2)c1C
Cc1nn(c(C)c1Cc1nnc(Cc2ccc(Cl)cc2Cl)o1)-c1ccccc1
Oc1cn(CC(=O)NCc2ccc(F)cc2Cl)c(=O)n1-c1ccccc1
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(F)cc1Cl
Cc1nn(c(C)c1CC(=O)NC(C)(C)c1ccccc1)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1cccc(Cl)c1Cl)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccc(Cl)cc1Cl)-c1ccccc1
COc1ccccc1Cn1cnnc1-c1cccc(Cl)c1Cl
Clc1cccc(-c2nncn2[C@@H]2CCc3ccccc23)c1Cl
CC(c1ccccc1)n1cnnc1-c1cccc(Cl)c1Cl
FC(F)(F)c1cccc(Cn2cnnc2-c2cccc(Cl)c2Cl)c1
CSc1ccccc1Cn1cnnc1-c1cccc(Cl)c1Cl
Cc1ccccc1Cn1cnnc1-c1cccc(Cl)c1Cl
Clc1cccc(-c2nnnn2Cc2ccccc2)c1Cl
Clc1ccc(NC(=O)CC23CC4CC(CC(C4)C2)C3)cc1 |THB:14:13:10:16.15.17,18:13:16:9.10.17|
CC(NC(=O)c1ccc(Cl)cc1)C12CC3CC(CC(C3)C1)C2 |THB:17:16:13:19.18.20,21:16:19:12.13.20|
COc1cccc(NC(=O)CC23CC4CC(CC(C4)C2)C3)c1C |TLB:20:11:18:15.14.16,THB:19:11:14:17.18.16,19:17:11.12.20:14,20:15:11.12.19:18|
Clc1ccc(C(=O)NCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:12:13:17:11.10.16,THB:14:15:10:13.18.12,14:13:10:15.17.16,12:11:17:13.18.14|
Clc1ccc(C(=O)NCC23CC4CC(C2)CC(CNC(=O)c2ccc(Cl)cc2Cl)(C4)C3)c(Cl)c1 |TLB:14:9:29:13.15.12,12:13:30:11.10.29,12:11:30:13.15.14,THB:14:13:9.30.10:29|
FC(F)(F)c1ccc(Cn2cnnc2-c2cccc(Cl)c2Cl)cc1
COc1ccc(C)c(NC(=O)CC23CC4CC(CC(C4)C2)C3)c1 |TLB:21:12:19:16.15.17,THB:20:12:15:18.19.17,20:18:12.13.21:15,21:16:12.13.20:19|
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(I)cc1)S(=O)(=O)c1cccc2cnccc12
Clc1cccc(c1Cl)-n1ncnc1Cc1ccccc1
Cc1nn(c(C)c1NC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccc(F)cc1Cl)-c1ncccn1
Clc1cccc(-c2cncn2Cc2ccccc2)c1Cl
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccc(cc1)C(C)=O)S(=O)(=O)c1cccc2cnccc12
CN(Cc1ccc(F)cc1Cl)C(=O)Cc1c(C)nn(c1C)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccc(F)cc1Cl)-c1ccc(cc1)C(N)=O
CC(C)(c1ccccc1)n1cnnc1-c1cccc(Cl)c1Cl
Cc1nn(CCO)c(C)c1CC(=O)NCc1ccc(F)cc1Cl
Cc1nn(cc1CC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
COc1ccc(cc1)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)N(C)S(=O)(=O)c1cccc2cnccc12
Cc1nc(sc1CC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
CN(CC12CC3CC(CC(C3)C1)C2)C(=O)c1ccc(Cl)cc1 |THB:8:7:4:10.9.11,12:7:10:3.4.11|
COC[C@H](O)Cn1c(=O)cnn(-c2ccc(C)c(NC(=O)C3=CN(C)C(=O)C[C@H]3c3ccc(F)cc3)c2)c1=O |r,t:21|
CN1C=C([C@@H](NC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1C)-n1ccccc1=O |r,c:2|
Cc1cc(Cl)c(OCCO)cc1NC(=O)C1=CNC(=O)C[C@H]1c1ccc(F)cc1 |r,t:16|
COc1cc(C)c(C)c(NC(=O)C2=CNC(=O)C[C@H]2c2ccc(F)cc2)c1 |r,t:12|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(c(F)cc1C)-c1ccnn(C)c1=O |r,c:2|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1C)-c1ccnn(C)c1=O |r,c:2|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1C)-c1ccn[nH]c1=O |r,c:2|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1C)-c1ccnn(CCO)c1=O |r,c:2|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1C)-n1ncccc1=O |r,c:2|
COc1cc(Br)c(CC(=O)N2C=CC(=O)CC2c2ccccc2)cc1OC |c:11|
COc1cc(Br)c(NC(=O)N2C=CC(=O)CC2c2ccccc2)cc1OC |c:11|
COc1cc(I)c(CC(=O)N2C=CC(=O)C[C@H]2c2ccccc2)cc1OC |r,c:11|
COc1cc(I)c(CC(=O)N2C=CC(=O)C[C@@H]2c2ccccc2)cc1OC |r,c:11|
COc1cc(Br)c(NC(=O)N2C=CC(=O)C[C@H]2c2ccc(F)cc2)cc1OC |r,c:11|
COc1cc(Br)c(NC(=O)C2=CNC(=O)C[C@H]2c2cccc(F)c2)cc1OC |r,t:10|
OCCOc1cc(NC(=O)N2C=CC(=O)C[C@H]2c2ccc(F)cc2)c(Br)cc1Cl |r,c:11|
Cc1cc(Cl)c(OCCO)cc1NC(=O)N1C=CC(=O)C[C@H]1c1ccc(F)cc1 |r,c:17|
CN1C=C([C@@H](CC1=O)c1ccc(F)cc1)C(=O)Nc1cc(ccc1F)-c1ccn[nH]c1=O |r,c:2|
Cc1cc2cnn(CCO)c2cc1NC(=O)C1=CNC(=O)C[C@H]1c1ccc(F)cc1 |r,t:18|
COc1cc(I)c(CC(=O)N2C=CC(=O)CC2c2ccccc2)cc1OC |c:11|
COc1cc(C)c(NC(=O)N2C=CC(=O)C[C@H]2c2ccc(F)cc2)cc1OC |r,c:11|
COc1cc(NC(=O)N2C=CC(=O)C[C@@H]2c2ccccc2)c(Br)cc1Cl |r,c:9|
COc1cc(NC(=O)N2C=CC(=O)C[C@H]2c2ccc(F)cc2)c(Br)cc1Cl |r,c:9|
COc1cc(NC(=O)N2C=CC(=O)C[C@H]2c2ccccc2)c(Br)cc1Cl |r,c:9|
COc1cc(NC(=O)N2C=CC(=O)C[C@H]2c2ccc(F)cc2)c(Br)cc1F |r,c:9|
FC(F)(F)c1cccc(c1)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
BrC12CC3CC(C1)CC(C3)(C2)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1 |TLB:9:8:4.3.2:6,0:1:4:8.7.9,THB:9:3:6:8.7.10,10:8:4:2.1.6,10:1:4:8.7.9,11:8:4:2.1.6,11:8:4.3.2:6|
O=C(CC1CC2CCC1C2)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Fc1cc(Cl)ccc1C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Brc1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Clc1cccc(c1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Fc1ccc(CN2CCN(CC2)c2cc(=O)[nH]c(=O)n2Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)cc1
O=C(CC1CCCCC1)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Clc1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Fc1cc(ccc1Cl)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Clc1ccccc1C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C12CC3CC1CC(C2)C3 |TLB:40:39:44:41.42,42:41:45.43.44:38,THB:42:43:38:40.41|
Clc1ccc(cc1Cl)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1 |TLB:10:9:4.3.2:7,THB:10:3:7:9.8.11,11:9:4:2.1.7,11:1:4:9.8.10,12:9:4.3.2:7,0:1:4:9.8.10|
O=C(C1CC2CCC1C2)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C12CC3CC(CC(C3)C1)C2 |TLB:44:39:46:43.42.45,44:43:46:40.39.38,THB:38:37:40.39.44:42,38:39:42:37.46.45,1:37:40.39.44:42|
O=C(CC12CC3CC(CC(C3)C1)C2)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1 |TLB:10:5:12:9.8.11,10:9:12:6.5.4,THB:8:7:4:10.9.11,8:9:6.7.12:4|
O=c1cc(N2CCN(Cc3ccccc3)CC2)n(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)c(=O)[nH]1
O=C(C1CCCCC1)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(Cc1ccccc1)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Clc1ccc(Br)cc1C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
Fc1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)c1ccccc1
Fc1ccc(cc1F)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
c1ccc(cc1)CC(=O)Nc2ccc(c(c2)S(=O)(=O)N)Oc3cccc(c3)Cl
CN1[C@@H](CCC1=O)C(=O)NCc1cccc(c1F)C(F)(F)F
CN1[C@@H](CCC1=O)C(=O)NCc1cccc(c1I)C(F)(F)F |r|
CN1[C@@H](CCC1=O)C(=O)NCc1cccc(c1Br)C(F)(F)F |r|
CN1[C@@H](CCC1=O)C(=O)NCc2cccc(c2Cl)C(F)(F)F
C[C@H]1CCC[C@@](O)(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CC[C@@H](F)C2)C1 |r|
C[C@@H]1CCC[C@@](O)(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CC[C@H](C2)C(C)(C)O)C1 |r|
COCCOc1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
OC1(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CC[C@H](F)C2)CCCC(F)(F)C1 |r|
OCCC1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
CN(C)[C@H]1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1 |r|
OCCNC1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
FC1(F)CCC(CNC(=O)c2c(Cl)ccc3nc(ccc23)C2CCCC2)CC1
OCCNc1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
CC1(C)OB(OC1(C)C)C1=CCCC1 |t:10|
F[C@@H]1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1 |r|
F[C@@H]1CCN(C1)c1ccc2c(C(=O)NCC3CCCC(F)(F)C3)c(Cl)ccc2n1 |r|
O[C@@]1(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CC[C@@H](F)C2)CCCC(F)(F)C1 |r|
FC1(F)CCC(CNC(=O)c2c(Cl)ccc3ncccc23)CC1
COCCNc1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
CN(C)[C@@H]1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1 |r|
F[C@H]1CCN(C1)c1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1 |r|
C[C@@H]1CCC[C@@](O)(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CCC(C2)N(C)C)C1 |r|
FC1(F)CCC(CNC(=O)c2c(Cl)ccc3nc(ccc23)N2CCCC2)CC1
FC1(F)CCC(CNC(=O)c2c(Cl)ccc3nc(ccc23)C2=CCCC2)CC1 |t:23|
CCCCc1cn(nn1)C1=CC(=O)c2cccc(O)c2C1=O |t:10|
Oc1cccc2C(=O)C=C(C(=O)c12)n1cc(CCCCl)nn1 |c:8|
c1cc2c(ccc(n2)NCCNCCO)c(c1)NC(=O)CC34CC5CC(C3)CC(C5)C4
O=C([C@@H]1Cc2ccc(cc2CN1S(=O)(=O)c1cccc2ccccc12)S(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ccccc1
COc1ccccc1[C@H]1N(C(=O)C([O-])=C1C(=O)C(C)C)c1ccc(cc1)-c1ccsc1 |r,c:14|
CCc1nnc2[C@H](N(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
Clc1ccc(cn1)C1(CNC(=O)c2c(Cl)ccc3[nH]ccc23)CCCCC1
C[C@H]1CC[C@@](O)(CNC(=O)c2cc(C3CCOC3)n3cccc(Cl)c23)CC1 |r,wU:1.0,wD:4.4,(57.38,-40.18,;56.24,-39.15,;54.77,-39.61,;53.64,-38.58,;53.97,-37.08,;53.96,-35.54,;52.82,-36.05,;51.36,-36.52,;50.22,-35.49,;50.54,-33.98,;48.75,-35.96,;47.5,-35.06,;46.26,-35.96,;44.79,-35.5,;43.54,-36.41,;42.3,-35.51,;42.77,-34.04,;44.31,-34.04,;46.73,-37.42,;45.96,-38.75,;46.73,-40.08,;48.27,-40.08,;49.03,-38.75,;50.57,-38.75,;48.27,-37.43,;55.43,-36.6,;56.57,-37.64,)|
Clc1ccc(cn1)C1(CNC(=O)C2CCCc3[nH]ccc23)CCCCC1
Cc1ncc(s1)C(CNC(=O)c1cc(ccc1Cl)-c1ncc(F)cn1)N1CCCC(F)(F)C1
CN(C)C(=O)CCNc1ccc2c(C(=O)NCC3CCC(F)(F)CC3)c(Cl)ccc2n1
FC(F)(F)c1cccc(C(=O)N2CCn3cnnc3[C@H]2c2ccccc2)c1Cl |r|
CC(C)(C)c1nnc2[C@H](N(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1cccc(C(=O)N2CCn3c(nnc3[C@H]2c2ccccc2)C2CC2)c1Cl |r|
CCCCc1nnc2[C@H](N(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1nnc2[C@H](N(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)ccc2[nH]ccc12)N1CCOCC1
Cc1nnc2[C@H](N(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F)c1ccccc1 |r|
[H][C@]12OC(C)(C)O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12
[H][C@]12O[C@H](O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12)c1ccccc1
[H][C@]12OCO[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12
[H][C@]12OC(C)(C)O[C@@]1([H])[C@@H](O[C@@H]2C(=O)N[C@@H](CCC(O)=O)C(O)=O)n1cnc2c(N)ncnc12 |r|
[H][C@]12OC3(CCCCC3)O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12
[H][C@]12OC3(CCCCC3)O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)CP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12
[H][C@]12OC(C)(C)O[C@@]1([H])[C@@H](O[C@@H]2COC(=O)c1cc(C(O)=O)c(cc1C(O)=O)C(O)=O)n1cnc2c(N)ncnc12 |r|
[H][C@]12O[C@@H](O[C@@]1([H])[C@@H](O[C@@H]2COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1cnc2c(N)ncnc12)c1ccccc1
OCCCNCCCc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2
CC(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
CNC(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(cc1)N(C)C
[O-][N+](=O)c1ccc(cc1)C(=O)N1CCC(CC1)c1nc2cc(OS(=O)(=O)c3cccc4cnccc34)ccc2[nH]1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C#N)cc1
CNC(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
CCN(CC)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CN(C)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C#N)cc1
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3ccncc23)cc1)C(=O)N1CCN(CC1)c1ccccc1)S(=O)(=O)c1cccc2cnccc12 |r|
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)c1nc2cc(OS(=O)(=O)c3cccc4cnccc34)ccc2[nH]1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OC(=O)c2cccc3cnccc23)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OC(=O)c2ccccc2)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccs2)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OC(=O)c2cccs2)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(Br)c2)cc1
[O-][N+](=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C(=O)NC2CC2)cc1
COc1ccc(cc1OC)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)c1ccc(Oc2ccccc2)cc1
[O-][N+](=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CC(C)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)c1ccc(cc1)C#N
CS(=O)(=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C#N)cc1
CNC(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(cc1)S(C)(=O)=O
CNC(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(cc1)[N+]([O-])=O
CNC(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(OC)cc1
[O-][N+](=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C(=O)NC2CC2)cc1
COc1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C(=O)NC2CC2)cc1
[O-][N+](=O)c1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CN(C)c1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CN(C)c1ccc(cc1)C(=O)N1CCC(CC1)c1nc2cc(OS(=O)(=O)c3cccc4cnccc34)ccc2[nH]1
[O-][N+](=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C#N)cc1
CN(C)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C(=O)NC2CC2)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3ccccc23)cc1
CCN(CC)C(=O)c1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
COc1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C#N)cc1
CS(=O)(=O)c1ccc(cc1)C(=O)N1CCN(CC1)c1cc(=O)[nH]c(=O)n1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
COc1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1ccc2cc(OS(=O)(=O)c3cccc4cnccc34)ccc12
CS(=O)(=O)c1ccc(cc1)C(=O)N1CCC(CC1)c1nc2cc(OS(=O)(=O)c3cccc4cnccc34)ccc2[nH]1
FC(F)(F)c1cc(ccc1Cl)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2ccccc2)cc1
Nc1cccc(c1)S(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CC(C)(O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CS(=O)(=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc(c2)C(=O)NC2CC2)cc1
CN(C)c1cccc(c1)C(=O)N1CCC(CC1)n1cncc1-c1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CS(=O)(=O)Oc1ccc(cc1)-c1cncn1C1CCN(CC1)C(=O)c1ccc(Cl)c(c1)C(F)(F)F
Oc1ccc(Cl)cc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1ccccc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1c(Cl)cccc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1cc(Cl)ccc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1c(F)cccc1C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1c(ccc2ccccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F
Oc1ccc(Cl)cc1C(=O)Nc1cccc(c1)C(F)(F)F
Oc1ccc(Cl)cc1C(=O)Nc1ccc(cc1)C(F)(F)F
Oc1ccc(Cl)cc1C(=O)Nc1cc(cc(c1)C(F)(F)F)[N+]([O-])=O
Oc1ccc(Cl)cc1C(=O)Nc1cc(Cl)cc(Cl)c1
Oc1ccc(Cl)cc1C(=O)Nc1cc(F)cc(F)c1
Oc1ccc(Cl)cc1C(=O)Nc1cccc(Cl)c1
FC(F)(F)c1cccc(CNC(=O)[C@@H]2CCC(=O)N2c2cccs2)c1Cl |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2cscn2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2nccs2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2ccoc2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2ccco2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2ccsc2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2cccs2)c(Cl)c1 |r|
CN1[C@@H](CCC1=O)C(=O)NCc1ccc(Cl)cc1Cl
Clc1ccc(CNC(=O)C2CN(C(=O)C2)c2cccs2)c(Cl)c1
Clc1ccc(CNC(=O)[C@@H]2COC(=O)N2c2cccs2)c(Cl)c1 |r|
CN1CCN(CC1)\C=C1/C[C@H](N(C1=O)c1cccs1)C(=O)NCc1ccc(Cl)cc1Cl |r|
Clc1ccc(CNC(=O)[C@@H]2C\C(=C/N3CCOCC3)C(=O)N2)c(Cl)c1 |r|
COC(=O)[C@@H]1C\C(=C/NCc2ccc(Cl)cc2Cl)C(=O)N1C(=O)OC |r|
O\N=C1/C[C@H](N(C1=O)c1cccs1)C(=O)NCc1ccc(Cl)cc1Cl |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2Cc2ccccc2Cl)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2Cc2ccccc2)c(Cl)c1 |r|
Clc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2ccccc2)c(Cl)c1 |r|
CN1[C@@H](COC1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CNC1=O)C(=O)NCc1ccc(Cl)cc1Cl |r|
CN1[C@@H](CC(C)(C)C1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(C1=O)c1cccnc1C)C(=O)NCc1ccc(Cl)cc1Cl |r|
Clc1ccc(C(=O)Cn2cnc3c(Cl)ncnc23)c(Cl)c1
Clc1ccc(cc1)C(=O)Cn1cnc2c(Cl)ncnc12
Clc1ccc(C(=O)Cn2cnc3c(ncnc23)-c2ccccc2)c(Cl)c1
Clc1ccc(C(=O)Cn2cnc3c(Cl)nc(Cl)nc23)c(Cl)c1
Clc1ccccc1S(=O)(=O)n1cnc2c(Cl)nc(Cl)nc12
Cn1c2ncn(c2c(=O)n(C)c1=O)S(=O)(=O)c1ccccc1Cl
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CCc2ccccc2)CC1)S(=O)(=O)c1cccc2cnccc12
COc1ccccc1N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)N(C)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)C(=O)c1ccc(F)cc1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1cccc(c1)C(F)(F)F)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccccc1C)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccccn1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ccccc1F)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(Cc2ccc(cc2)[N+]([O-])=O)CC1)S(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCN(CC1)c1ncccn1)S(=O)(=O)c1cccc2cnccc12
Cc1ccccc1N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)NS(=O)(=O)c1cccc2cnccc12
Fc1ccc(cc1)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)NS(=O)(=O)c1cccc2cnccc12
CN([C@@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C(=O)N1CCC(Cc2ccccc2)CC1)S(=O)(=O)c1cccc2cnccc12
CC(C)Oc1ccc(Nc2nc(=O)n(CC(C)(C)C(O)=O)c(=O)n2Cc2ccc(Cl)cc2)cc1F
CC(C)Oc1ccc(Nc2nc(=O)n(CCC(O)=O)c(=O)n2Cc2ccc(C)cc2)cc1Cl
COc1cc(C(C)C)c(Oc2cnc(NC(CO)CO)nc2N)cc1I
C[C@@H](Cn1c(=O)[nH]\c(=N/c2ccc(Oc3ccsn3)cc2)n(Cc2ccc(Cl)cc2)c1=O)C(O)=O |r|
C[C@@H](Cn1c(=O)[nH]\c(=N/c2ccc(Oc3ccccn3)cc2)n(Cc2ccc(Cl)cc2)c1=O)C(O)=O |r|
C[C@@H](Cn1c(=O)[nH]\c(=N/c2ccc(Oc3ccnc(F)c3)cc2)n(Cc2ccc(Cl)cc2)c1=O)C(O)=O |r|
CCCN1CCN(C(C1)c1ccccc1)C(=O)c1ccccc1Cl
CN1CCN(CC1c1ccccc1)C(=O)c1ccccc1Cl
CCN1CCN(CC1c1ccccc1)C(=O)c1ccccc1Cl
FC(F)(F)CCN1CCN(CC1c1ccccc1)C(=O)c1cccc(Cl)c1Cl
Clc1ccccc1NC(=O)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccccc1Cl
COc1ccc(cc1OC)C(=O)N1CCN(CC1c1ccccc1)c1c(Nc2ccccc2C)c(=O)c1=O
COc1ccc(cc1OC)C(=O)N1CCN(CC1c1ccccc1)c1c(Nc2cccc3ncccc23)c(=O)c1=O
COc1ccc(NC(=O)N2CCN(CC2c2ccccc2)c2c(Nc3ccccc3C)c(=O)c2=O)cc1OC
Cc1ccccc1Nc1c(N2CCN(C(C2)c2ccccc2)C(=O)Nc2ccc(Cl)cc2)c(=O)c1=O
Cc1ccccc1Nc1c(N2CCN(C(C2)c2ccccc2)C(=O)Nc2ccccc2Cl)c(=O)c1=O
COc1ccc(NC(=O)N2CCN(CC2)c2c(Nc3ccccc3C)c(=O)c2=O)cc1OC
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccc(N)cc2)c(=O)c1=O
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccc(F)cc2)c(=O)c1=O
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccc(Cl)cc2)c(=O)c1=O
Cc1ccc(NC(=O)N2CCN(CC2)c2c(Nc3ccccc3C)c(=O)c2=O)cc1
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccccc2)c(=O)c1=O
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccc(cc2)C(C)(C)C)c(=O)c1=O
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)Nc2ccc(cc2)[N+]([O-])=O)c(=O)c1=O
COC(=O)c1ccc(NC(=O)N2CCN(CC2)c2c(Nc3ccccc3C)c(=O)c2=O)cc1
Cc1ccccc1Nc1c(N2CCN(CC2)C(=O)NC2CCCCC2)c(=O)c1=O
CC(C)(C)c1ccc(NC(=O)N2CCN(CC2)c2c(Nc3cccc4ncccc34)c(=O)c2=O)cc1
c1ccc(cc1)N2CCN(CC2)C3(CCOCC3)CNC(=O)c4cccnc4Sc5ccccc5
CC1=C(C=C)\C(NC1=O)=C\c1[nH]c(Cc2[nH]c(\C=C3/NC(=O)C(C)=C3C=C)c(C)c2CCC(O)=O)c(CCC(O)=O)c1C |c:1,24|
C[C@H](N\C(Nc1cccc2ncccc12)=N\C#N)c1ccccc1 |r|
FC(F)(F)c1nc(sc1C(=O)NC[C@H](N1CCOCC1)c1ccc(Cl)cc1)-c1ncccn1 |r|
FC(F)(F)c1nc(sc1C(=O)NC[C@@H](N1CCOCC1)c1ccc(Cl)cc1)-c1ncccn1 |r|
OCCn1cc(C(=O)NCC2CCCCCC2)c2ccccc12
FC(F)(F)c1cccc(-c2nnnn2Cc2cccnc2)c1Cl
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCC(F)(F)CC1
CCOc1ccc(Nc2ccc(cc2)C(=C2\C=C/C(/C=C2C)=[N+](/CC)Cc2cccc(c2)S([O-])(=O)=O)\c2ccc(cc2C)N(CC)Cc2cccc(c2)S(O)(=O)=O)cc1 |c:17,20|
CN(C)CCN1CCN(CCC(=O)Nc2nc3c(C)cccc3s2)CC1
CN(C)CCCN1CCN(CCC(=O)Nc2nc3c(C)cccc3s2)CC1
Cc1cccc2sc(NC(=O)CCN3CCN(CC3)c3ccccn3)nc12
Cc1cccc2sc(NC(=O)CCN3CCN(CC3)c3ccncc3)nc12
Cc1cccc2sc(NC(=O)CCN3CCN(CC3)c3ncccn3)nc12
COc1ccc(cc1)C(=O)O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1OC(=O)c1ccc(OC)cc1)n1cnc2c(N)ncnc12 |r|
c1nc(c2c(n1)n(cn2)[C@H]3[C@@H]([C@@H]([C@H](O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)F)N
N[C@@H]1[C@H](O)[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]1n1cnc2c(N)ncnc12 |r|
CO[C@@H]1[C@H](O)[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]1n1cnc2c(N)ncnc12 |r|
c1nc(c2c(n1)n(cn2)[C@H]3[C@H]([C@@H]([C@H](O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)N
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cnc2c(Cl)ncnc12 |r|
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cnc2c(S)ncnc12 |r|
CNc1c2c(ncn1)n(cn2)[C@H]3[C@@H]([C@@H]([C@H](O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O
CCCCNc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |r|
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cnc2c(Nc3ccccc3)ncnc12 |r|
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cnc2c(NCc3ccccc3)ncnc12 |r|
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1cnc2c3nccn3cnc12 |r|
Nc1ncnc2n([C@@H]3O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]3O)c(N=[N+]=[N-])nc12 |r|
O[C@@H]1[C@@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)O[C@H]([C@@H]1O)n1c2ncncc2[nH]c1=O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](OC(=O)c2ccccc2)[C@H]1OC(=O)c1ccccc1 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](OC(=O)c2cccc3ccccc23)[C@H]1OC(=O)c1cccc2ccccc12 |r|
Oc1ccccc1NC(=S)NC(=O)C12CC3CC(CC(C3)C1)C2 |TLB:20:19:22:16.15.14,20:15:22:19.21.18,THB:18:19:22.17.16:14,18:17:19.21.20:14|
Oc1ccc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)cc1 |TLB:18:17:20:14.13.12,18:13:20:17.19.16,THB:16:17:20.15.14:12,16:15:17.19.18:12|
Oc1c(Cl)cc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)cc1Cl |TLB:19:18:21:15.14.13,19:14:21:18.20.17,THB:17:18:21.16.15:13,17:16:18.20.19:13|
FC(F)(F)c1cc(Br)cc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)c1 |TLB:23:22:25:19.18.17,23:18:25:22.24.21,THB:21:22:25.20.19:17,21:20:22.24.23:17|
NS(=O)(=O)c1ccccc1NC(=S)NC(=O)C12CC3CC(CC(C3)C1)C2 |TLB:23:22:25:19.18.17,23:18:25:22.24.21,THB:21:22:25.20.19:17,21:20:22.24.23:17|
[O-][N+](=O)c1ccc(Cl)c(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)c1 |TLB:22:21:24:18.17.16,22:17:24:21.23.20,THB:20:21:24.19.18:16,20:19:21.23.22:16|
COc1ccc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)cc1OC |TLB:19:18:21:15.14.13,19:14:21:18.20.17,THB:17:18:21.16.15:13,17:16:18.20.19:13|
Brc1ccc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)cc1 |TLB:18:17:20:14.13.12,18:13:20:17.19.16,THB:16:17:20.15.14:12,16:15:17.19.18:12|
Cc1ccc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)c(Br)c1 |TLB:18:17:20:14.13.12,18:13:20:17.19.16,THB:16:17:20.15.14:12,16:15:17.19.18:12|
Clc1ncccc1NC(=S)NC(=O)C12CC3CC(CC(C3)C1)C2 |TLB:20:19:22:16.15.14,20:15:22:19.21.18,THB:18:19:22.17.16:14,18:17:19.21.20:14|
CC1=CCC(=C\C1=N\C(=O)C1=CC=C\C(C1)=N/C(=O)/N=C1/CC(=CC=C1)C(=O)\N=C1\CC(=CC=C1C)C(=O)\N=C1/CC=C(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O)C(=O)\N=C1/CC=C(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O |c:4,13,24,26,34,36,45,72,t:1,11|
Nc1c2C(=O)c3ccccc3C(=O)c2c(Nc2ccc(Nc3nc(Cl)nc(Nc4cccc(c4)S(O)=O)n3)c(c2)S(O)(=O)=O)cc1S(O)(=O)=O
O=C(NC(=S)Nc1cccc2cccnc12)C12CC3CC(CC(C3)C1)C2 |TLB:23:22:25:19.18.17,23:18:25:22.24.21,THB:21:22:25.20.19:17,21:20:22.24.23:17|
CC(C)c1ccc(NC(=S)NC(=O)C23CC4CC(CC(C4)C2)C3)c(Br)c1 |TLB:20:19:22:16.15.14,20:15:22:19.21.18,THB:18:19:22.17.16:14,18:17:19.21.20:14|
Oc1ccc(NC(=S)NC(=O)c2ccc3OCOc3c2)cc1
NS(=O)(=O)c1cccc(NC(=S)NC(=O)c2ccc3OCOc3c2)c1
NS(=O)(=O)c1ccc(CCNC(=S)NC(=O)c2ccc3OCOc3c2)cc1
FC(F)(F)c1cc(Br)cc(NC(=S)NC(=O)c2ccc3OCOc3c2)c1
FC(F)(F)c1ccc(Br)c(NC(=S)NC(=O)c2ccc3OCOc3c2)c1Br
Oc1c(Cl)cc(NC(=S)NC(=O)c2ccc3OCOc3c2)cc1Cl
[O-][N+](=O)c1ccc(NC(=S)NC(=O)c2ccc3OCOc3c2)cc1
CC(C)c1ccc(NC(=S)NC(=O)c2ccc3OCOc3c2)c(Br)c1
Clc1ncccc1NC(=S)NC(=O)c1ccc2OCOc2c1
O=C(NC(=S)Nc1cccc2cccnc12)c1ccc2OCOc2c1
O=C(NNc1cccc2ncccc12)C12CC3CC(CC(C3)C1)C2 |TLB:1:14:17:21.20.19,THB:15:16:19:23.14.22,15:14:17.16.21:19,22:14:17:21.20.19,22:20:17:23.15.14|
C[C@@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1cc(O[11CH3])ccn1 |r|
C[C@H]1Cc2c(CN1C(=O)c1ccnc(c1[18F])C(F)(F)F)nnn2-c1ncccn1 |r|
COc1ccc(CC(=O)NC(N\C(Nc2cccc3ncccc23)=N\C#N)C(C)(C)C)cc1O[11CH3]
FC(F)(F)c1cccc(CNC(=O)[C@@H]2CCC(=O)N2CC[18F])c1Cl |r|
[11CH3]Oc1ccc(Cl)c(c1)C(=O)NCC12CC3(F)CC(F)(CC(F)(C3)C1)C2 |TLB:17:18:24:23.15.14,16:15:20.18.25:24,19:18:24:23.15.14,12:13:20:23.17.15,THB:17:15:20.18.25:24,14:15:20:25.13.24,14:13:20:23.17.15,16:15:20:25.13.24|
[18F]c1ccc(CN\C(Nc2cccc3ncccc23)=N\C#N)cc1
O=c1[nH]c2ccccc2n1CCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
O=C(C(c1ccccc1)c1ccccc1)N1CCN(CCCn2c3ccccc3[nH]c2=O)CC1
Cc1ccc(cc1)S(=O)(=O)N1CCN(CCCn2c3ccccc3[nH]c2=O)CC1
[O-][N+](=O)c1ccc(cc1)S(=O)(=O)N1CCN(CCCn2c3ccccc3[nH]c2=O)CC1
Fc1ccc(cc1)S(=O)(=O)N1CCN(CCCn2c3ccccc3[nH]c2=O)CC1
O=c1[nH]c2ccccc2n1CCCN1CCN(CC1)C1c2ccccc2CCc2ccccc12
OC(C1CCN(CCCn2c3ccccc3[nH]c2=O)CC1)(c1ccccc1)c1ccccc1
O=c1[nH]c2ccccc2n1CCCN1CCC(CC1)=C(c1ccccc1)c1ccccc1 |(-7.26,4.38,;-6.9,2.89,;-7.9,1.71,;-7.09,.4,;-7.53,-1.08,;-6.47,-2.19,;-4.97,-1.83,;-4.54,-.36,;-5.6,.76,;-5.48,2.3,;-4.16,3.1,;-2.81,2.37,;-1.5,3.17,;-.14,2.44,;1.17,3.24,;2.52,2.51,;2.56,.97,;1.25,.16,;-.1,.9,;3.92,.24,;3.96,-1.3,;5.31,-2.04,;5.35,-3.58,;4.04,-4.38,;2.69,-3.65,;2.65,-2.11,;5.23,1.04,;6.59,.31,;7.9,1.11,;7.86,2.65,;6.5,3.39,;5.19,2.58,)|
O=c1[nH]c2ccccc2n1CCN1CCN(CC1)C(c1ccccc1)c1ccccc1
O=c1[nH]c2ccccc2n1CCCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
O=c1[nH]c2ccccc2n1CCCCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
O=c1[nH]c2ccccc2n1C\C=C\CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1cnc2ccccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
Cc1nc2ccccc2n1CCCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1c(nc2ccccc12)-c1ccccc1)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
Cc1cc2ncn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c2cc1C
C(CCn1ncc2ccccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1ccc2ncccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1ccc2cnccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1ccc2ccncc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1ccc2cccnc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1nnc2ccccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1ccc2ccccc12)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1cncn1)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
Cc1nnnn1CCCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
C(CCn1nnnc1-c1ccccc1)CN1CCN(CC1)C(c1ccccc1)c1ccccc1
Cc1nccn1CCCCN1CCN(CC1)C(c1ccccc1)c1ccccc1
Cc1cccc2n(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)ccc12
Cc1ccc2ccn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c2c1
Cc1cccc2ccn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c12
COc1ccc2n(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)ccc2c1
N#Cc1cn(CCCCN2CCN(CC2)C(c2ccccc2)c2ccccc2)c2ccccc12
N#Cc1ccc2n(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)ccc2c1
COC(=O)c1cccc2ccn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c12
Fc1cccc2n(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)ccc12
Fc1ccc2n(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)ccc2c1
Fc1ccc2ccn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c2c1
Fc1cc2ccn(CCCCN3CCN(CC3)C(c3ccccc3)c3ccccc3)c2cc1F
C[C@H](NC(NC#N)=Nc1cccc2ncccc12)c1ccccc1 |r,w:7.7|
C[C@@H](CO)n1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2c1=O |r,TLB:16:17:21:15.20.14,20:15:22:19.18.21,20:19:22:16.15.14,THB:16:15:22.17.18:21|
C[C@H](CO)n1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2c1=O |r,TLB:16:17:21:15.20.14,20:15:22:19.18.21,20:19:22:16.15.14,THB:16:15:22.17.18:21|
COc1ccc(Cl)c(c1)C(=O)NCC12CC3(F)CC(F)(CC(F)(C3)C1)C2 |TLB:17:18:24:23.15.14,16:15:20.18.25:24,19:18:24:23.15.14,12:13:20:23.17.15,THB:17:15:20.18.25:24,14:15:20:25.13.24,14:13:20:23.17.15,16:15:20:25.13.24|
COc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:12:13:16:20.19.18,THB:14:15:18:22.13.21,14:13:16.15.20:18,21:13:16:20.19.18,21:19:16:22.14.13|
COc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(F)(C3)C1)C2 |TLB:20:19:16.17.23:14,16:17:22:21.15.14,THB:16:15:22:17.18.23,18:19:16.17.23:14,18:17:22.19.21:14|
COc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(F)(CC(F)(C3)C1)C2 |TLB:22:20:24:15.16.14,22:15:24:19.20.23,16:17:22.15.14:23,THB:18:17:22.15.14:23,16:15:24.17.19:23,21:20:24:15.16.14|
Cc1ccc(cc1)C1(CNC(=O)c2cc(CO[N+]([O-])=O)ccc2Cl)CCCCC1
[O-][N+](=O)OCc1ccc(cc1)C1(CNC(=O)c2ccccc2Cl)CCCCC1
O=C(NCC1CCCCCCC1)C1CCC(=O)c2ncccc12
OC1CC[C@](O)(C(=O)NCc2cccc(c2Cl)C(F)(F)F)c2cccnc12 |r|
COc1ccc(C)c(Nc2nc(=O)cnn2Cc2cncc(F)c2)c1
COc1cc(Nc2nc(=O)c(F)cn2Cc2cc(F)c(F)c(F)c2)c(C)c(F)c1OC
Cn1nccc1Nc1nc(=O)c(F)cn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(CO)cc1Nc1nc(=O)ccn1Cc1cc(F)c(F)c(F)c1
Cc1c(F)cc(CO)cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1
Cc1ccc(cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1)-c1ncco1
Cc1ccc(cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1)N1CCCC1=O
Cc1ccc(OCCO)cc1Nc1nc(=O)cnn1Cc1cc(F)c(F)c(F)c1
Cc1cc(Nc2nc(=O)c3[nH]cnc3n2Cc2ccccc2)c(C)cc1Cl
COc1ccc(Nc2nc(=O)c3[nH]cnc3n2Cc2ccc(F)c(F)c2)c(C)c1
Cc1nc2cc(C)c(Nc3nc(=O)c4[nH]cnc4n3Cc3ccc(F)cc3)cc2s1
Cc1nc2cc(C)c(Nc3nc(=O)c4[nH]cnc4n3Cc3ccc(C)cc3)cc2s1
COc1nc(C)c(Nc2nc(=O)c3[nH]cnc3n2Cc2ccc(F)c(F)c2)cc1C
CCc1cccc(Nc2nc(=O)c3[nH]cnc3n2Cc2ccc(F)cc2)c1CC
COc1cnc(C)c(Nc2nc(=O)c3CCCc3n2Cc2cc(F)c(F)c(F)c2)c1
COc1ccc(Nc2nc(=O)c3onc(C)c3n2Cc2ccc(F)c(F)c2)c(C)c1
COc1ccc(Nc2nc(=O)c3nn(C)cc3n2Cc2cc(F)c(F)c(F)c2)c(C)c1
Fc1cccc(Cl)c1Cc1nsc(=O)n1CC1CCC(F)(F)CC1
Fc1cccc(Cl)c1Cc1noc(=O)n1CC1CCC(F)(F)CC1
Fc1cccc(Cl)c1Cc1noc(=O)n1CC1CCC(CC1)C(F)(F)F |(-2.29,-5.48,;-3.62,-4.71,;-4.95,-5.48,;-6.29,-4.71,;-6.29,-3.18,;-4.96,-2.4,;-4.96,-.86,;-3.62,-3.17,;-2.29,-2.4,;-2.29,-.86,;-3.53,.04,;-3.06,1.5,;-1.52,1.5,;-.75,2.84,;-1.04,.04,;.45,-.36,;1.53,.73,;1.14,2.22,;2.22,3.31,;3.71,2.91,;4.11,1.42,;3.02,.33,;4.8,4,;4.4,5.48,;6.29,3.6,;5.89,5.09,)|
CC1CC(F)(F)CCN1Cn1c(Cc2c(F)cccc2Cl)noc1=O
FC1(F)CCC(Cn2c(Cc3ccccc3Cl)noc2=O)CC1
FC1(F)CCC(Cn2c(Cc3ccc(Cl)cc3Cl)noc2=O)CC1
Cc1noc(C)c1Cc1noc(=O)n1CC1CCC(F)(F)CC1
COc1ccc(Cc2noc(=O)n2CC2CCC(F)(F)CC2)cc1
Cc1ncccc1Cc1noc(=O)n1CC1CCC(F)(F)CC1
FC1(F)CCC(Cn2c(CN3CCC(F)(F)CC3)noc2=O)CC1
FC1(F)CCC(Cn2c(CN3CCOc4ccccc34)noc2=O)CC1
Fc1cccc(Cl)c1Cc1noc(=O)n1CC1CC2CCC1C2
Fc1cccc(Cl)c1Cc1noc(=O)n1CC1CCCCCC1
CC1=C(Cn2cc(COCc3ccco3)nn2)C(=O)c2ccccc2C1=O |c:1|
CC1=C(C(c2ccccc2)n2cc(COCc3ccco3)nn2)C(=O)c2ccccc2C1=O |c:1|
CC1=C(C(c2ccc(cc2)[N+]([O-])=O)n2cc(COCc3ccco3)nn2)C(=O)c2ccccc2C1=O |c:1|
CC1=C(C(c2ccc(Cl)cc2)n2cc(COCc3ccco3)nn2)C(=O)c2ccccc2C1=O |c:1|
CC(CO)n1ccc2c(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c(C)ccc2c1=O
CS(=O)(=O)Nc1cccc(c1)-c1ccc(Cl)c(c1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
COc1ccc(cc1OC)-c1ccc(Cl)c(c1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)c1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)Nc1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
Nc1cccc(c1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
Clc1ccnc(c1)-n1cc(CNC(=O)c2cnc(s2)-c2cccc(NS(=O)(=O)N3CCOCC3)c2)nn1
Clc1ccnc(c1)-n1cc(CNC(=O)c2cnc(s2)-c2cccc(NS(=O)(=O)C3CC3)c2)nn1
Clc1ccnc(c1)-n1cc(CNC(=O)c2cnc(s2)-c2ccc(NS(=O)(=O)N3CCOCC3)cc2)nn1
CC(C)S(=O)(=O)c1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)c1ccc(cc1)-c1nc(cs1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)c1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Br)ccn1
CS(=O)(=O)c1ccc(cc1)-c1nc(cs1)C(=O)NCc1cn(nn1)-c1cc(Br)ccn1
CS(=O)(=O)c1ccc(cc1)-c1nc(cs1)C(=O)NCc1cn(nn1)-c1ccc(Br)cn1
CS(=O)(=O)c1ccc(cc1)-c1nc(cs1)C(=O)NCc1cn(nn1)-c1cccc(Br)n1
Clc1ccnc(c1)-n1cc(CNC(=O)c2cc(ccc2Cl)-c2cccc3ncccc23)nn1
CS(=O)(=O)c1ccc(cc1)-c1ccc(Cl)c(c1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
Clc1ccnc(c1)-n1cc(CNC(=O)c2cc(ccc2Cl)-c2cccc3cc[nH]c23)nn1
CC(C)Cc1ccc(cc1)-c1ccc(Cl)c(c1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
Nc1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)c1ccc(cc1)-c1csc(n1)C(=O)NCc1cn(nn1)-c1cc(Cl)ccn1
CS(=O)(=O)c1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cc(F)ccn1
CS(=O)(=O)c1ccc(cc1)-c1ncc(s1)C(=O)NCc1cn(nn1)-c1cccc(Br)n1
Oc1cccc2C(=O)C=C(C(=O)c12)n1cc(CCCl)nn1 |c:8|
Clc1ccc(CNC(=O)C2CCC(=O)N2c2ccoc2)c(Cl)c1
Ic1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Brc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Clc1ccc(CN2CCN(CC2)C(=O)CNS(=O)(=O)c2cccc3cnccc23)cc1
[O-][N+](=O)c1ccc(cc1)N1CCN(CC1)C(=O)CCNS(=O)(=O)c1cccc2cnccc12
Clc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2ccccc12)N1CCN(CC1)c1ccccc1
[O-][N+](=O)c1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccccc1N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2ccccc12
Fc1ccc(N2CCN(CC2)C(=O)CNS(=O)(=O)c2cccc3cnccc23)c(F)c1
CN(CC(=O)N1CCN(CC1)c1ccccc1F)S(=O)(=O)c1cccc2cnccc12
Fc1ccccc1N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1cccc(c1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccc(CN2CCN(CC2)C(=O)CNS(=O)(=O)c2cccc3cnccc23)cc1
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1cccc2ccccc12
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCCN(Cc2ccccc2)CC1
O=C(CCNS(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ccccc1
Cc1ccc(CN2CCN(CC2)C(=O)CNS(=O)(=O)c2cccc3cnccc23)cc1
CN(CC(=O)N1CCN(Cc2ccccc2)CC1)S(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ccccc1
Cc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(Cc2ccccc2)CC1
Nc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccc(F)c(c1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1cccc(N2CCN(CC2)C(=O)CNS(=O)(=O)c2cccc3cnccc23)c1F
O=C(CNS(=O)(=O)c1cccc2ccccc12)N1CCN(CC1)c1cccc2ccccc12
Fc1ccc(cc1F)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ncccn1
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ccc(cc1)C#N
CC(=O)c1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Cc1ccccc1N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2ccccc12)N1CCN(Cc2ccccc2)CC1
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CCc2ccccc2)CC1
CN(CC(=O)N1CCN(CC1)c1ccc(F)cc1)S(=O)(=O)c1cccc2cnccc12
Fc1ccccc1N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cccnc12
COc1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccccc1N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2ncccc12
Fc1ccc(cc1)N1CCN(CC1)C(=O)CCNS(=O)(=O)c1cccc2ccccc12
FC(F)(F)c1ccc(cc1)N1CCN(CC1)C(=O)CNS(=O)(=O)c1cccc2cnccc12
Fc1ccc(cc1)N1CCN(CC1)C(=O)CCNS(=O)(=O)c1cccc2cnccc12
O=C(CNS(=O)(=O)c1cccc2cnccc12)N1CCN(CCCc2ccccc2)CC1
O=C(CNS(=O)(=O)c1cccc2ccccc12)N1CCN(CCc2ccccc2)CC1
Clc1ccc(CC2CCCNC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |w:6.5,TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(NC2CCCNC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |w:6.5,TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(OC2CCNCC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1cc(CN2CCCCC2)ccc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1cnc(OC2CCCNC2)nc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(CN2CCNCC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(O[C@@H]2CCCNC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(NC2CCNCC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(CC2CCNCC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(cc1C(=O)NCC12CC3CC(CC(C3)C1)C2)N1CCNCC1 |TLB:10:11:14:18.16.17,THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
Clc1ccc(O[C@H]2CCCNC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
Clc1ccc(CN2C[C@@H]3C[C@H]2CN3)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:18:19:22:26.24.25,THB:24:23:20:26.25.27,24:25:22.23.28:20,27:25:22:28.19.20,27:19:22:26.24.25|
Clc1ccc(cc1C(=O)NCC12CC3CC(CC(C3)C1)C2)C1CCNCC1 |TLB:10:11:14:18.16.17,THB:16:15:12:18.17.19,16:17:14.15.20:12,19:17:14:20.11.12,19:11:14:18.16.17|
Cc1nnc(OC2CCNCC2)cc1C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:18:21:25.23.24,THB:23:22:19:25.24.26,23:24:21.22.27:19,26:24:21:27.18.19,26:18:21:25.23.24|
C[C@H](c1ccc2ccccc2c1)Nc3cc(nc4n3nc(n4)C5CC5)N6CCN(CC6)C(=O)N
CN([C@@H](Cc1ccc(OS(=O)(=O)c2ccc(C)cc2)cc1)C(=O)N1CCN(CC1)C(=O)c1ccccc1)C(=O)OCc1ccccc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)OC(C)(C)C)cc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(CBr)cc2)cc1)NC(=O)OCc1ccccc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1)NC(=O)OCc1ccccc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(cc2)C#N)cc1)NC(=O)OCc1ccccc1
C[C@H]1CN(CCN1C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(C)cc2)cc1)NC(=O)OCc1ccccc1)C(=O)c1ccccc1
C[C@@H]1CN(CCN1C(=O)c1ccccc1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(C)cc2)cc1)NC(=O)OCc1ccccc1
C[C@H]1CN(CCN1C(=O)c1ccccc1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(C)cc2)cc1)NC(=O)OCc1ccccc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccc(F)cc2)cc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(I)cc2)cc1)NC(=O)OCc1ccccc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccccc2)cc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(Br)cc2)cc1)NC(=O)OCc1ccccc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccc(cc2)C(F)(F)F)cc1
Cc1cc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccccc2)cc(C)c1OS(=O)(=O)c1ccccc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)NS(=O)(=O)c1cccc2cnccc12
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(F)cc2)cc1)NC(=O)OCc1ccccc1
CN(C)c1ccc(cc1)C(=O)N1CCN(CC1)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(C)cc2)cc1)NC(=O)OCc1ccccc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccc(Br)cc2)cc1
C[C@H]1CN(CCN1C(=O)c1ccc(cc1)N(C)C)C(=O)[C@H](Cc1ccc(OS(=O)(=O)c2ccc(cc2)C#N)cc1)NC(=O)OCc1ccccc1
[O-][N+](=O)c1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)c2ccccc2)cc1
Cc1ccc(cc1)S(=O)(=O)Oc1ccc(C[C@@H](NC(=O)OCc2ccccc2)C(=O)N2CCN(CC2)C(=O)OC(C)(C)C)cc1
CN(C)Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1 |w:10.10|
CC(C)C1CN(CCN1C(NC#N)=Nc1ccccc1C)C(=O)Nc1ccc(Cl)cc1 |w:13.14|
COc1ccc(CC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)cc1OC |w:25.27|
Clc1ccc(NC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2cccc3[nH]ccc23)cc1 |w:24.26|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2[nH]ncc12)C(=O)Nc1cccc(F)c1 |w:13.14|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2nc(C)ccc12)C(=O)Nc1ccc(Cl)cc1 |w:13.14|
CN(C(=O)N1CCN(CC1c1ccccc1)C(NC#N)=Nc1ccccc1C)c1ccc(Cl)cc1 |w:20.22|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2NCCCc12)C(=O)Nc1cccc(F)c1 |w:13.14|
Cc1ccccc1N=C(C[N+]([O-])=O)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1 |w:7.7|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)S(=O)(=O)c1ccc(Cl)cc1 |w:7.7|
Cc1ccccc1N=C(NC(N)=O)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1 |w:7.7|
CC(C)C1CN(CCN1C(=O)Nc1ccc(Cl)cc1)C(NC#N)=Nc1ccccc1C |w:23.25|
Cc1ccccc1NC(=O)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2ncccc12)C(=O)Nc1ccc(Cl)cc1 |w:13.14|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2[nH]ccc12)C(=O)Nc1ccc(Cl)cc1 |w:13.14|
CC(C)C1CN(CCN1C(=O)Nc1ccc(Cl)cc1)C(NC#N)=Nc1cccc2ncccc12 |w:23.25|
COc1ccc(NC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)cc1OC |w:25.27|
Cn1cnc2c(cccc12)N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1 |w:10.11|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Nc1ccc(Cl)cc1 |w:7.7|
Clc1ccc(NC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2cccnc2)cc1 |w:24.26|
Cc1ccccc1N=C(NC#N)N1CCN(Cc2ccc(Cl)cc2)C(C1)c1ccccc1 |w:7.7|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2occc12)C(=O)Nc1cccc(F)c1 |w:13.14|
CC(C)C1CN(CCN1C(NC#N)=Nc1cccc2CNCCc12)C(=O)Nc1ccc(Cl)cc1 |w:13.14|
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(Cl)nc3)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cccc(Cl)c3)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(F)cc3C(F)(F)F)c(OC)ccc12
COc1ccc2c(CC=C)c3-c4cc5OCOc5cc4CC[n+]3cc2c1OC
CCc1c2-c3cc4OCOc4cc3CC[n+]2cc2c(OC)c(OC)ccc12
COc1cc(Cc2c3-c4cc5OCOc5cc4CC[n+]3cc3c(OC)c(OC)ccc23)cc(OC)c1
COc1ccc2c(Cc3c(F)cccc3Cl)c3-c4cc5OCOc5cc4CC[n+]3cc2c1OC
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccccc3C)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cc(C)ccc3C)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cc(C)ccc3[N+]([O-])=O)c(OC)ccc12
CC[C@H]1[C@@H]2N(CCc3cc4OCOc4cc23)Cc2c1ccc(OC)c2OC |r|
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cccc(c3C)[N+]([O-])=O)c(OC)ccc12
COc1cc2CC[n+]3cc4c(OC)c(OC)ccc4c(CC4CCCCC4)c3-c2cc1OC
CCCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OC)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccccc3C(F)(F)F)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(OCc4ccccc4)cc3)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(Br)cc3)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(cc3)C(C)(C)C)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cc(OC)c(OC)cc3[N+]([O-])=O)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3cc(ccc3OC)[N+]([O-])=O)c(OC)ccc12
CCCC(I)c1c2-c3cc4OCOc4cc3CC[n+]2cc2c(OC)c(OC)ccc12
CCc1c2-c3cc(OC)c(OC)cc3CC[n+]2cc2c(OCc3ccc(cc3)-c3ccccc3)c(OC)ccc12
COc1cc(C(C)C)c(Oc2cnc(N)nc2N)cc1I
NC1=[NH+]C2(O)C(N1)OC1NC(=[NH2+])NC11C(OC3C(CNC(=O)c4cc(Br)c(Br)[nH]4)C(CNC(=O)c4cc(Br)c(Br)[nH]4)C4C5(O)NC(=[NH2+])NC5OC5NC(=[NH2+])NC345)C(CNC(=O)c3cc(Br)c(Br)[nH]3)C(CNC(=O)c3cc(Br)c(Br)[nH]3)C21 |t:1|
NC1=N[C@]2(O)[C@H](N1)O[C@@H]1N=C(N)N[C@@]11[C@@H](O[C@H]3[C@H](CNC(=O)c4cc(Br)c(Br)[nH]4)[C@@H](CNC(=O)c4cc(Br)c(Br)[nH]4)[C@@H]4[C@]5(O)N=C(N)N[C@@H]5O[C@@H]5N=C(N)N[C@]345)[C@H](CNC(=O)c3cc(Br)c(Br)[nH]3)[C@@H](CNC(=O)c3cc(Br)c(Br)[nH]3)[C@@H]21 |r,t:1,10,48,56|
CC(C)(C)OC(=O)N1CCC(CCn2cc3N(C[C@@H](Cc4ccccc4)NC(=O)c3n2)C(=O)C2CC2)CC1 |r|
CC(C)(C)OC(=O)N1CCC(CCn2cc3N(C[C@H](Cc4ccccc4)NC(=O)c3n2)C(=O)C2CC2)CC1 |r|
O=C(OC[C@H]1CNc2cn(CCc3ccccc3)nc2C(=O)N1)c1cccc2cnccc12 |r|
Cn1cc(C(=O)OC[C@H]2CN(Cc3ccc(cc3)[N+]([O-])=O)c3cn(CCc4ccccc4)nc3C(=O)N2)c2ccccc12 |r|
Cc1cc(O)ccc1CN1C[C@H](COC(=O)c2cn(C)c3ccccc23)NC(=O)c2nn(CCc3ccccc3)cc12 |r|
Cn1cc(C(=O)OC[C@H]2CN(Cc3ccccc3)c3cn(CCc4ccccc4)nc3C(=O)N2)c2ccccc12 |r|
Cc1ccc(CN2C[C@H](COC(=O)c3cccc4cnccc34)NC(=O)c3nn(CCc4ccccc4)cc23)cc1 |r|
Cc1cc(CN2C[C@H](COC(=O)c3cccc4cnccc34)NC(=O)c3nn(CCc4ccccc4)cc23)ccc1O |r|
Cn1cc(CN2C[C@H](COC(=O)c3cn(C)c4ccccc34)NC(=O)c3nn(CCc4ccccc4)cc23)c2ccccc12 |r|
Cn1cc(C(=O)OC[C@H]2CN(Cc3ccc(Cl)cc3)c3cn(CCc4ccccc4)nc3C(=O)N2)c2ccccc12 |r|
Cc1ccc(CN2C[C@H](COC(=O)c3cn(C)c4ccccc34)NC(=O)c3nn(CCc4ccccc4)cc23)cc1 |r|
Cn1cc(C(=O)OC[C@H]2CN(Cc3ccc(Br)cc3)c3cn(CCc4ccccc4)nc3C(=O)N2)c2ccccc12 |r|
Fc1ccc(CN2C[C@H](COC(=O)c3cccc4cnccc34)NC(=O)c3nn(CCc4ccccc4)cc23)cc1 |r|
O=C(OC[C@H]1CN(Cc2ccccc2)c2cn(CCc3ccccc3)nc2C(=O)N1)c1cccc2cnccc12 |r|
OC1(CNC(=O)c2cc(ccc2Cl)-c2ccc(F)cn2)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ccc(Cl)cn2)CCCCCC1
Cc1ccc(nn1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2cccc(n2)C#N)CCCCCC1
OCc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
Cc1cnc(cn1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
Cc1cnc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCC(F)(F)C1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ccccn2)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCCCC1F
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCC(F)(F)CC1
COc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ccc(cn2)C#N)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ncc(F)cn2)CCCC1
Cc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
CCCCCNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
Cc1ccc(cc1C(=O)NCC1(O)CCCCCC1)-n1ncc(=O)[nH]c1=O
CCC(CC)CNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
COC[C@@H](O)Cn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O |r|
CCCCCCNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
CCn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O
CC(C)Cn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O
COCCn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O
OC1(CNC(=O)c2cc(ccc2Cl)-n2ncc(=O)[nH]c2=O)CCCCCC1
Cn1c(=O)cnn(-c2ccc(Cl)c(c2)C(=O)NCC2(O)CCCCCC2)c1=O
Clc1ccccc1CCNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
OC1(CNC(=O)c2cc(ccc2Cl)-n2ncc(=O)[nH]c2=O)CCCCC1
CCCCC(CC)CNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
Clc1ccc(cc1C(=O)NCCc1ccccc1)-n1ncc(=O)[nH]c1=O
CCCOCCNC(=O)c1cc(ccc1Cl)-n1ncc(=O)[nH]c1=O
Clc1ccc(cc1C(=O)NCC1CCOCC1)-n1ncc(=O)[nH]c1=O
Clc1ccc(cc1C(=O)NCC1CCCCC1)-n1ncc(=O)[nH]c1=O
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2cc(F)cc(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(=O)N3CCCCC3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)cc2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2CC2CCCC2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(=O)N3CCOCC3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3cccc(OC(F)(F)F)c3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2cc(F)c(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(=O)N3[C@@H](C)CCC[C@H]3C)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)cc2F)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CC[C@H](C)[C@@H]1CN2C(=N1)N(CC)C(=O)c1nc(-c3ccc(F)cc3)n(Cc3ccc(F)c(F)c3)c21 |r,c:7|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C#N)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)nc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccnc(c3)C(F)(F)F)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(F)(F)F)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(C#N)c(F)c3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(=O)N3CCC(F)(F)CC3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)C#N)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3cccs3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)c(c3)C#N)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CC(C)[C@@H]1CN2C(=N1)N(C(C)C)C(=O)c1nc(-c3ccc(F)cc3)n(Cc3ccccc3)c21 |r,c:6|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccccc3F)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)c1ccc(F)cc1 |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(N)nc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccccc2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(OC(F)(F)F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)N3CCOCC3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CC(C)[C@@H]1CN2C(NC(=O)c3nc(-c4ccc(F)cc4)n(Cc4ccccc4)c23)=N1 |r,c:32|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)C1CCCC1 |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)C1CC1 |r,t:3|
CCN1C2=NC3(CCc4ccccc34)CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC3(CCC3)CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccccc2)C1=O)C(C)C |r,t:4|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)N3CCCCC3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccccn2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)(C)C |r,t:3|
CCN1C2=NC3(CCc4ccccc34)CN2c2c(nc(Cc3ccccc3)n2Cc2ccccc2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(F)cc3)n2Cc2ccncc2)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(nc3)C(=O)N3CCCC(F)(F)C3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCn1c(CC(=O)NCc2c(C)cccc2Cl)c(C)nc1-c1ccc(F)cc1F
Cc1nc(-c2ccc(F)cc2F)n(C)c1CC(=O)NCc1cccc(Cl)c1C
CCn1c(CC(=O)NCc2cccc(Cl)c2C)c(C)nc1-c1ccccc1
CCn1c(CC(=O)NCc2ccc(F)c(F)c2F)c(C)nc1-c1ccc(F)cc1F
Cc1nc(-c2ccccc2)n(C)c1CC(=O)NCc1c(C)cccc1Cl
CCn1c(CC(=O)NCc2ccc(F)c(F)c2F)c(C)nc1-c1ccccc1
Cc1nc(-c2ccccc2)n(C)c1CC(=O)NCc1ccc(F)c(F)c1F
Cc1nc(-c2ccc(F)cc2F)n(C)c1CC(=O)NCc1ccc(F)cc1Cl
Cc1nc(-c2ccccc2)n(C)c1CC(=O)NCc1ccc(F)cc1Cl
CCn1c(CC(=O)NCc2c(C)cccc2Cl)c(C)nc1-c1ccccc1
Cc1nc(-c2ccccc2)n(C)c1CC(=O)NCc1cccc(Cl)c1C
Cc1c(Cl)cccc1CNC(=O)Cc1cnc(-c2ccc(F)cc2F)n1C
CCn1c(CC(=O)NCc2ccc(F)cc2Cl)c(C)nc1-c1ccc(F)cc1F
CCn1c(CC(=O)NCc2ccc(F)cc2Cl)c(C)nc1-c1ccccc1
Cn1c(CC(=O)NCc2ccc(F)cc2Cl)cnc1-c1ccc(F)cc1F
CCn1c(CC(=O)NCc2ccc(F)cc2Cl)cnc1-c1ccc(F)cc1F
Cc1nc(-c2ccc(F)cc2F)n(C)c1CC(=O)NCc1ccc(F)c(F)c1F
CCn1c(CC(=O)NCc2cccc(Cl)c2C)c(C)nc1-c1ccc(F)cc1F
CC(=O)Nc1cccc(Nc2ncnc(n2)N2CCC(CC2)OCc2ccc(OC(F)(F)F)cc2)c1C
COc1ccc(nn1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
Clc1ccccc1CCNC(=O)c1cc(ccc1Cl)-c1n[nH]c(=O)[nH]c1=O
COc1ccc(nn1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Cc1ccc(nn1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
CC(O)c1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Cc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Clc1ccccc1CCNC(=O)c1cc(ccc1Cl)-c1ccccn1
NC(=O)c1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Clc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Cn1ccc(n1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
Cc1cc(nn1C[C@@H](O)CN)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1 |r|
Clc1ccccc1CCNC(=O)c1cc(ccc1Cl)-c1cccnc1
Cc1cc(n[nH]1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
Cc1cc(nn1C[C@H](O)CN)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1 |r|
Cn1nccc1-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2ccc(=O)[nH]n2)CCCCCC1
FC(F)(F)c1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCCc1ccccc1Cl
Clc1ccccc1CCNC(=O)c1cc(ccc1Cl)-c1ccncc1
OC1(CNC(=O)c2cc(ccc2Cl)-c2cnoc2)CCCCCC1
Cc1nc(cs1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2c[nH]cn2)CCCCCC1
OC1(CNC(=O)c2cc(ccc2Cl)-c2cc[nH]n2)CCCCCC1
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2cccc(F)c2F)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(F)cc3F)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)cc2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(OC(F)(F)F)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2cccc(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(OC)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccccc2F)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(F)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)c(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(cc3)C(F)(F)F)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccc(C)cc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3cccc(OC(F)(F)F)c3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3cccc(F)c3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3cccc(c3)C(F)(F)F)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3cccc(C)c3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2cc(F)ccc2F)C1=O)C(C)C |r,t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)cc2F)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccccc3F)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccccc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2cc(F)cc(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)cc2F)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)cc2)C1=O |t:3|
CCN1C(=O)c2nc(-c3ccc(cc3)-c3ccccc3)n(Cc3ccc(F)c(F)c3)c2N2CCC(C)(C)N=C12 |t:41|
CCN1C2=NC3(CN2c2c(nc(-c4ccc(cc4)-c4ccccc4)n2Cc2ccc(F)c(F)c2)C1=O)CCCCC3 |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=N[C@@H](CN2c2c(nc(-c3ccc(cc3)-c3ccccc3)n2Cc2cc(F)cc(F)c2)C1=O)C(C)C |r,t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3cc(F)cc(F)c3)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CCN1C2=NC(C)(C)CN2c2c(nc(-c3ccc(nc3)-c3ccccc3OC)n2Cc2ccc(F)c(F)c2)C1=O |t:3|
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)C(Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)NS(=O)(=O)c1cccc2cnccc12
Cc1ccccc1NC(=O)CC12CC3CC(CC(C3)C1)C2 |TLB:20:11:18:15.14.16,THB:20:15:11.12.19:18,16:17:12:15.20.14,16:15:12:17.19.18|
Clc1ccccc1NC(=O)CC12CC3CC(CC(C3)C1)C2 |TLB:20:11:18:15.14.16,THB:20:15:11.12.19:18,16:17:12:15.20.14,16:15:12:17.19.18|
Clc1cc(Cl)cc(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:19:14:21:18.20.17,19:18:21:14.13.15,THB:20:12:15:18.19.17,20:18:12.21.13:15|
CN(CC12CC3CC(CC(C3)C1)C2)C(=O)c1ccccc1Cl |TLB:10:5:12:9.11.8,10:9:12:5.4.6,THB:8:7:4:9.11.10,8:9:4:7.12.6|
CC(NC(=O)c1ccccc1Cl)C12CC3CC(CC(C3)C1)C2 |TLB:19:18:21:13.14.15,19:14:21:20.18.17,THB:17:18:13:21.16.15,17:16:13:20.18.19|
Cc1ccc(cc1NC(=O)c2cccc(c2)NC(=O)Nc3cccc(c3)C(=O)Nc4cc(ccc4C)C(=O)Nc5ccc(c6c5c(cc(c6)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O)C(=O)Nc7ccc(c8c7c(cc(c8)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CO[P@](O)(=O)O[P@@](O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)CP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1OC(=O)c1ccc(cc1)-c1ccccc1
Cc1c(c(c(c(n1)/N=N/c2ccc(cc2S(=O)(=O)O)S(=O)(=O)O)COP(=O)(O)O)C=O)O
CCOc1ccc(Nc2ccc(cc2)[C+](c2ccc(cc2C)N(CC)Cc2cccc(c2)S([O-])(=O)=O)c2ccc(cc2C)N(CC)Cc2cccc(c2)S([O-])(=O)=O)cc1
[O-]S(=O)(=O)c1cc(ccc1\C=C\c1ccc(cc1S([O-])(=O)=O)N=C=S)N=C=S
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccccc1 |w:7.7|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccc(Cl)cc1 |w:7.7|
COc1ccc(CC(=O)N2CCN(C(C2)c2ccccc2)C(NC#N)=Nc2ccccc2C)cc1OC |w:25.27|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1cccnc1 |w:7.7|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccncc1 |w:7.7|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccc2ccccc2c1 |w:7.7|
COc1ccc(CCCC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)cc1OC |w:27.29|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(cc1OC)C(=O)N1CCN(CC1c1ccccc1)C(NC#N)=Nc1ccccc1C |w:28.31|
COc1ccc(CCC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)cc1OC |w:26.28|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1cnc[nH]1 |w:7.7|
COc1ccc(CC(=O)N2CCN([C@@H](C2)C(C)C)C(NC#N)=Nc2ccccc2C)cc1OC |w:22.23|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1cccs1 |w:7.7|
Cc1ccn(CC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)n1 |w:24.26|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1c[nH]c2ccccc12 |w:7.7|
COc1ccc(cc1OC)C(=O)N1CCN(CC1c1ccccc1)C(NC#N)=Nc1cccc2ncccc12 |w:28.31|
Cc1cc(CC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)on1 |w:23.25|
COc1ccc(CC(=O)N2C(C)CN(CC2C)C(NC#N)=Nc2ccccc2C)cc1OC |w:21.22|
COc1ccc(CC(=O)N2CCN([C@H](CC(C)C)C2)C(NC#N)=Nc2ccccc2C)cc1OC |w:23.24|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)CC12CC3CC(CC(C3)C1)C2 |w:7.7,TLB:36:27:34:30.31.32,26:27:34:30.31.32,THB:36:31:28.27.35:34,32:31:28:35.33.34,32:33:28:30.36.31|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccco1 |w:7.7|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccoc1 |w:7.7|
Cc1ccnn1CC(=O)N1CCN(CC1c1ccccc1)C(NC#N)=Nc1ccccc1C |w:25.28|
Cc1cc(CC(=O)N2CCN(CC2c2ccccc2)C(NC#N)=Nc2ccccc2C)no1 |w:23.25|
Cc1ccccc1N=C(NC#N)N1CCN(C(C1)c1ccccc1)C(=O)Cc1ccsc1 |w:7.7|
COc1ccc(CC(=O)N2CCN(CC2C(C)(C)C)C(NC#N)=Nc2ccccc2C)cc1OC |w:23.24|
Nc1c(cc(Nc2ccc(c(Nc3nc(Cl)nc(Cl)n3)c2)S([O-])(=O)=O)c2C(=O)c3ccccc3C(=O)c12)S([O-])(=O)=O
Clc1cncc(Cl)c1NNC(=O)CC1CCCCCC1
Clc1cncc(Cl)c1NNC(=O)CCC1CCCCC1
Clc1cncc(Cl)c1NNC(=O)C1C2CC3CC(C2)C(Br)C1C3 |TLB:22:21:16.15.14:18,20:19:16:14.13.18,20:19:16.15.14:18,THB:10:12:16.15.14:18,22:15:18:19.21.12,20:19:16.15.22:13.18.12,12:21:16:14.13.18,12:13:16:19.22.21|
Clc1cncc(Cl)c1NNC(=O)CCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)C1C2CC3CC(C2)CC1C3 |TLB:10:12:14:18.16.17,THB:16:15:12:18.17.19,16:17:14.15.21:12,19:17:14:21.20.12,19:20:14:18.16.17,(.23,-.82,;1.57,-1.59,;1.57,-3.13,;2.9,-3.9,;4.24,-3.13,;4.23,-1.58,;5.56,-.8,;2.9,-.82,;2.89,.72,;4.22,1.5,;4.22,3.04,;2.88,3.8,;5.55,3.81,;6.95,3.33,;7.76,1.77,;7.86,3.33,;8.86,4.47,;7.99,5.85,;7.86,4.42,;6.56,6.37,;5.55,5.24,;6.37,3.85,)|
Clc1cncc(Cl)c1NNC(=O)C1Cc2ccccc12
Clc1cncc(Cl)c1NNC(=O)CC1CC2CCC1C2 |TLB:12:13:19:16.17|
Clc1cncc(Cl)c1NNC(=O)C1CC2CCC1C2 |TLB:10:12:18:15.16|
Clc1cncc(Cl)c1NNC(=O)C12CC3CC1CC(C2)C3 |THB:17:18:13:15.16,17:16:13:19.20.18|
Clc1cncc(Cl)c1NNC(=O)CC1C2CC3CC(C2)CC1C3 |TLB:12:13:15:19.17.18,THB:17:16:13:19.18.20,17:18:15.16.22:13,20:18:15:22.21.13,20:21:15:19.17.18,(-10.48,.47,;-9.14,-.3,;-9.14,-1.85,;-7.81,-2.62,;-6.47,-1.85,;-6.48,-.3,;-5.15,.48,;-7.81,.47,;-7.82,2.01,;-6.49,2.78,;-6.49,4.32,;-7.83,5.09,;-5.16,5.1,;-3.82,4.33,;-3.81,2.84,;-5.01,1.57,;-3.51,1.99,;-2.11,1.42,;-1.09,2.7,;-2.49,2.35,;-1.08,4.23,;-2.48,4.81,;-3.52,3.57,)|
Clc1cncc(Cl)c1NNC(=O)CCCC1CCCCC1
Clc1cncc(Cl)c1NNC(=O)CC1CCCCC1
Clc1cncc(Cl)c1NNC(=O)CCC1CCCC1
Clc1cncc(Cl)c1NNC(=O)CCc1cccc2ccccc12
Clc1cncc(Cl)c1NNC(=O)C1Cc2ccccc2C1
Clc1cncc(Cl)c1NNC(=O)C1CCc2ccccc2C1
Clc1cncc(Cl)c1NNC(=O)OCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)CCCCCCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)CCCCCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)CCCCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)CCCc1ccccc1
Clc1cncc(Cl)c1NNC(=O)Cc1ccccc1
Clc1ccc(CC(=O)NNc2c(Cl)cncc2Cl)c(Cl)c1
Clc1ccc(CC(=O)NNc2c(Cl)cncc2Cl)cc1
COc1ccc(CCC(=O)NNc2c(Cl)cncc2Cl)cc1
Cc1ccc(CCC(=O)NNc2c(Cl)cncc2Cl)cc1
Clc1ccc(CCC(=O)NNc2c(Cl)cncc2Cl)cc1
Fc1ccc(CCC(=O)NNc2c(Cl)cncc2Cl)cc1
Cc1cccc(C)c1NNC(=O)CCc1ccccc1
Clc1cccc(Cl)c1NNC(=O)CCc1ccccc1
Cc1ccc(COC(=O)N2c3ccccc3Oc3ccccc23)cc1
CCCN(CCC)C(=O)N1c2ccccc2Oc2ccccc12
OC1(c2ccccc2)c2ccccc2N(Cc2ccccc2)c2ccccc12
Cc1ccc(cc1)S(=O)(=O)N1c2ccccc2Oc2ccccc12
O=C(NCCc1ccccc1)N1c2ccccc2Oc2ccccc12
CC(C)OC(=O)N1c2ccccc2Oc2ccccc12
O=C(OCc1ccccc1)N1c2ccccc2Oc2ccccc12
COC(=O)NNC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
CC(=O)NNC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
CN1CC(=O)N(C(CCc2ccncc2)COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)C1=O
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2CCCC2=O)cc1
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2CCCS2(=O)=O)cc1
CN(NC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O)C(C)=O
CN1C(=O)N(C(CCc2ccncc2)COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)C(=O)C1(C)C
NC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
COC(=O)N(C)NC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2CCCCC2=O)cc1
CN(C)C(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)n2c(O)csc2=O)cc1
CN(C)C(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)N2C(=O)CCCC2=O)cc1
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccc(cc2)C(=O)N2CCCC2)N2C(=O)CCCC2=O)cc1
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccc(cc2)C(=O)N2CCCC2)N2C(=O)CCC2=O)cc1
CN(C)C(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)N2C(=O)CCC2=O)cc1
CNC(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)N2C(=O)CCC2=O)cc1
CNC(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)n2c(O)csc2=O)cc1
CC1(C)NC(=O)N(C(CCc2ccncc2)COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)C1=O
CNC(=O)c1ccc(CCC(COc2ccc(cc2)-c2cccc(c2)[N+]([O-])=O)N2C(=O)CCCC2=O)cc1
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2CCCOC2=O)cc1
Oc1c[nH]c(=O)n1C(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
[O-][N+](=O)c1cccc(c1)-c1ccc(OCC(CCc2ccncc2)N2C(=O)CCNC2=O)cc1
Oc1csc(=O)n1C(CCc1ccc(cc1)C(=O)N1CCCC1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
Clc1ccc(Cl)c(c1)-c1nnnn1Cc1cccnc1
Fc1ccc(-c2nnnn2Cc2cccnc2)c(Cl)c1Cl
Fc1c(cccc1C(F)(F)F)-c1nnnn1Cc1cccnc1
Cc1ncccc1Cn1nnnc1-c1cccc(Cl)c1Cl
Clc1cccc(-c2nnnn2Cc2ccncc2)c1Cl
Fc1cccc(-c2nnnn2Cc2cccnc2)c1C(F)(F)F
Cc1nc(C)c(Cn2nnnc2-c2cccc(Cl)c2Cl)s1
C(c1ccccc1)n1nnnc1-c1ccncc1
Fc1ccc(c(Cl)c1Cl)-n1nnnc1Cc1cccnc1
Clc1cccc(C(=O)NCC23CC4CC(CC(C4)C2)C3)c1Cl |TLB:13:14:18:12.11.17,17:12:19:16.18.15,17:16:19:12.11.13,THB:13:12:18:14.19.15|
Clc1cccc(c1Cl)-n1nnnc1Cc1cccnc1
Fc1ccc(c(Cl)c1C(F)(F)F)-n1nnnc1Cc1cccnc1
Clc1ccc(cc1Cl)-c1nnnn1Cc1cccnc1
C(c1cccnc1)n1nnnc1-c1ccccc1
C(c1ccccc1)n1nnnc1-c1cccc2cccnc12
Clc1ccc(-c2nnnn2Cc2cccnc2)c(Cl)c1Cl
FC(F)(F)c1cccc(c1Cl)-n1nnnc1Cc1cccnc1
Cc1ccccc1Cn1nnnc1-c1cccc(C)c1C
Cc1c(C)c(ccc1N1CCCC1)-c1nnnn1Cc1ccccc1
Clc1cccc(c1)-c1nnnn1Cc1cccnc1
Clc1ccccc1-c1nnnn1Cc1cccnc1
Cc1ccccc1Cn1nnnc1-c1cccc(Cl)c1Cl
Clc1cccc(-c2nnnn2Cc2ccccn2)c1Cl
COc1cccc(-c2nnnn2Cc2ccccc2Cl)c1OC
Clc1cccc(-c2nnnn2CCc2cccnc2)c1Cl
Cc1noc(C)c1Cn1nnnc1-c1cccc(Cl)c1Cl
C(c1ccccc1)n1nnnc1-c1cccc2ncccc12
CSc1ccccc1CNc1ncnn1-c1cccc(Cl)c1Cl
CCOc1ccccc1CNc1ncnn1-c1cccc(Cl)c1Cl
COc1ccc(CNc2ncnn2-c2cccc(Cl)c2Cl)cc1
COc1ccccc1CNc1ncnn1-c1cccc(Cl)c1Cl
Cc1ccc(CNc2ncnn2-c2cccc(Cl)c2Cl)cc1
Cc1cccc(CNc2ncnn2-c2cccc(Cl)c2Cl)c1
Clc1cccc(c1Cl)-n1ncnc1NCc1ccccc1
Clc1cccc(c1Cl)-n1ncnc1Nc1ccccc1N1CCOCC1
FC(F)(F)Oc1ccccc1Nc1ncnn1-c1cccc(Cl)c1Cl
COc1ccccc1Nc1ncnn1-c1cccc(Cl)c1Cl
CCc1ccccc1Nc1ncnn1-c1cccc(Cl)c1Cl
Cc1ccccc1Nc1ncnn1-c1cccc(Cl)c1Cl
Cc1nnc(NCc2cccnc2-c2ccsc2)n1-c1cccc(Cl)c1Cl |(12.13,-22.48,;13.28,-23.5,;14.78,-23.17,;15.56,-24.5,;14.53,-25.65,;14.86,-27.16,;16.21,-27.9,;17.56,-27.15,;17.59,-25.62,;18.94,-24.88,;20.26,-25.68,;20.22,-27.22,;18.87,-27.96,;18.84,-29.5,;20.06,-30.44,;19.54,-31.89,;18,-31.85,;17.57,-30.37,;13.12,-25.03,;11.79,-25.8,;11.8,-27.36,;10.45,-28.13,;9.12,-27.36,;9.13,-25.81,;7.79,-25.04,;10.45,-25.04,;10.44,-23.5,)|
Clc1cccc(c1Cl)-n1cnnc1NCc1cccnc1-c1ccsc1
Clc1cccc(c1Cl)-n1cnnc1NCc1cccnc1N1CCCC1
Clc1cccc(c1Cl)-n1cnnc1NCc1cccnc1
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1-c1ccsc1
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1N1CCOCC1
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1N1CCCC1
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1N1CCC1
Clc1cccc(c1Cl)-n1ncnc1NCc1ccncc1
Clc1cccc(c1Cl)-n1ncnc1NCc1ccccc1Oc1cccnc1
COc1cccc(CNc2ncnn2-c2cccc(Cl)c2Cl)c1OC
COc1cccc(CNc2ncnn2-c2cccc(Cl)c2Cl)c1
Cc1ccccc1CNc1ncnn1-c1cccc(Cl)c1Cl
CCOc1ccccc1Nc1ncnn1-c1cccc(Cl)c1Cl
Clc1cccc(c1Cl)-n1ncnc1Nc1ccccc1
NC(=O)CN1CCCN(CC1)c1ncccc1CNc1nncn1-c1cccc(Cl)c1Cl
Clc1cccc(c1Cl)-n1cnnc1NCc1cccnc1Oc1cccnc1
Cc1ncccc1CNc1nncn1-c1cccc(Cl)c1Cl
Clc1cccc(c1Cl)-n1ncnc1NCc1cccnc1Oc1cccnc1
Cc1ncccc1CNc1ncnn1-c1cccc(Cl)c1Cl
Cc1cccc(CNc2ncnn2-c2cccc(Cl)c2Cl)c1C
CC(C)N1CCCN(CC1)c1ncccc1CNc1nncn1-c1cccc(Cl)c1Cl
CS(=O)(=O)c1ccccc1CNc1ncnn1-c1cccc(Cl)c1Cl
CCCCCCC(=O)NNc1ccccc1C
CC1(CC2CC1C=C2)C(=O)NNc1cccc2ncccc12 |c:7,TLB:0:1:4:7.6,THB:8:1:4:7.6|
CC1CCC(C)(C(=O)NNc2cccc3ncccc23)C1(C)C
Fc1ccc(cc1)C1(CCCCC1)C(=O)NNc1cccc2ncccc12
Fc1cccc(c1)C1(CCCCC1)C(=O)NNc1cccc2ncccc12
Fc1ccccc1C1(CCCCC1)C(=O)NNc1cccc2ncccc12
COc1ccc(cc1)C1(CCCCC1)C(=O)NNc1cccc2ncccc12
OC12CC3CC(C1)CC(C3)(C2)C(=O)NNc1cccc2ncccc12 |TLB:9:8:4.3.2:6,11:8:4:2.1.6,11:8:4.3.2:6,THB:9:3:6:8.7.10,0:1:4:8.7.9,10:8:4:2.1.6,10:1:4:8.7.9|
CCC12CC3CC(C1)CC(C3)(C2)C(=O)NNc1cccc2ncccc12 |TLB:10:9:5.4.3:7,12:9:5:3.2.7,12:9:5.4.3:7,THB:10:4:7:9.8.11,1:2:5:9.8.10,11:9:5:3.2.7,11:2:5:9.8.10|
ClC12CC3CC(C1)CC(C3)(C2)C(=O)NNc1cccc2ncccc12 |TLB:9:8:4.3.2:6,11:8:4:2.1.6,11:8:4.3.2:6,THB:9:3:6:8.7.10,10:8:4:2.1.6,10:1:4:8.7.9,0:1:4:8.7.9|
O=C(CC12CC3CC(CC(C3)C1)C2)NNc1cccc2ncccc12 |TLB:6:7:5.4.10:11,THB:6:5:7.12.8:11,8:7:4:10.9.11,8:9:6.7.12:4|
O=C(NNc1cccc2ncccc12)C12CC3CC1CC(C2)C3 |TLB:19:18:22.20.21:15,THB:19:20:15:17.18|
Clc1ccc2c(NNC(=O)C34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:8:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
O=C(NNc1cccc2cnccc12)C12CC3CC(CC(C3)C1)C2 |TLB:1:14:17:21.20.19,THB:15:16:19:23.14.22,15:14:17.16.21:19,22:14:17:21.20.19,22:20:17:23.15.14|
O=C(NNc1cccnc1)C12CC3CC(CC(C3)C1)C2 |TLB:1:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
O=C(NNc1ccccn1)C12CC3CC(CC(C3)C1)C2 |TLB:1:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
Clc1ccc(NNC(=O)C23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:7:9:12:16.15.14,THB:10:11:14:18.9.17,10:9:12.11.16:14,17:9:12:16.15.14,17:15:12:18.10.9|
Clc1cccc(NNC(=O)C23CC4CC(CC(C4)C2)C3)c1Cl |TLB:8:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
c1ccc(c(c1)NNC(=O)C23CC4CC(C2)CC(C4)C3)Cl
Fc1ccc(NNC(=O)C23CC4CC(CC(C4)C2)C3)cc1 |TLB:7:9:12:16.15.14,THB:10:11:14:18.9.17,10:9:12.11.16:14,17:9:12:16.15.14,17:15:12:18.10.9|
Fc1cccc(NNC(=O)C23CC4CC(CC(C4)C2)C3)c1 |TLB:8:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
Fc1ccccc1NNC(=O)C12CC3CC(CC(C3)C1)C2 |TLB:9:11:14:18.17.16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11|
O=C(NNc1ccccc1)C12CC3CC(CC(C3)C1)C2 |TLB:1:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
Cc1ccc(C)c(NNC(=O)C23CC4CC(CC(C4)C2)C3)c1 |TLB:9:11:14:18.17.16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11|
COc1ccc(NNC(=O)C23CC4CC(CC(C4)C2)C3)cc1 |TLB:8:10:13:17.16.15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
Cc1ccccc1NNC(=O)C12CC3CC(CC(C3)C1)C2 |TLB:9:11:14:18.17.16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11|
Cc1ccccc1NNC(=O)C1(CCCC1)c1ccccc1
Cc1ccccc1NNC(=O)C1CCCCCC1
Cc1ccccc1NNC(=O)CC1CCCCC1
Cc1ccccc1NNC(=O)C1(C)CCCCC1
CC(C)CCC(=O)NNc1ccccc1C
CC1(C)C2CCC1(C(=O)NNc1cccc3ncccc13)C(=O)C2 |THB:22:21:5.4:1|
CC1(C)C(C(=O)NNc2cccc3ncccc23)C1(C)C
Cc1ccccc1NNC(=O)C1CCCCC1
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc(C)c2)C(C)(C)C)cc1OC |w:11.10|
Cc1ccccc1NC(NC#N)=NC(NC(=O)Cc1ccccc1)C(C)(C)C |w:12.13|
COc1ccc(cc1OC)C(=O)NC(N=C(NC#N)Nc1ccccc1C)C(C)(C)C |w:14.14|
Cc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccnc2C)C(C)(C)C)cc1F |w:10.9|
CC(C)(C)C(NC(=O)CCCc1cccnc1)N=C(NC#N)Nc1cccc2ncccc12 |w:17.17|
COc1cc(OC)cc(c1)C(=O)NC(NC(Nc1cccnc1C)=NC#N)C(C)(Cl)Cl |w:24.26|
O=C(CC12CC3CC(CC(C3)C1)C2)Nc1ccc2[nH]ncc2c1 |TLB:6:7:5.10.4:11,THB:8:7:4:10.9.11,8:9:6.7.12:4,6:5:7.8.12:11|
COc1ccc(CC(=O)NC(NC(=S)Nc2ccccc2C)C(Cl)(Cl)Cl)cc1OC
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cc(F)ccc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccccc1NC(NC#N)=NC(NC(=O)Cc1ccc(OC)c(OC)c1)C(C)(C)C |w:13.14|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccccc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2c(F)cccc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccc(F)cc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc3cnccc23)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccc(F)cc2)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc(F)c2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NCc2ccccc2Cl)NC#N)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccc(F)c(F)c2)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc3cccnc23)C(C)(C)C)cc1OC |w:11.10|
Cc1ccccc1NC(NC#N)=NC(NC(=O)Cc1ccc2OCOc2c1)C(C)(C)C |w:12.13|
COc1cc(CC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc(OC)c1 |w:10.9|
COc1cc(OC)cc(c1)C(=O)NC(N=C(NC#N)Nc1ccccc1C)C(C)(C)C |w:14.14|
COc1ccc(cc1)C(=O)NC(N=C(NC#N)Nc1ccccc1C)C(C)(C)C |w:12.12|
COc1ccc(CCC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1OC |w:12.11|
CSc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccnc2C)C(C)(C)C)cc1 |w:11.10|
Cc1ncccc1NC(NC#N)=NC(NC(=O)Cc1ccc(F)cc1)C(C)(C)C |w:12.13|
COc1ccc(CCCC(=O)NC(N=C(NC#N)Nc2cccnc2C)C(C)(C)C)cc1 |w:13.12|
Cc1ncccc1NC(NC#N)=NC(NC(=O)CCCCc1ccccc1)C(C)(C)C |w:12.13|
CC(C)(C)C(NC(=O)Cc1ccc(cc1)C#N)N=C(NC#N)Nc1cccc2ncccc12 |w:17.17|
COc1ccc(NC(NC(NC(=O)c2ccc(Cl)cc2)C(C)(Cl)Cl)=NC#N)c(OC)n1 |w:24.25|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cc(Cl)ccc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2c(F)cc(F)cc2F)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccnc2OC)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccnc2C)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cc(F)cc(F)c2)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc(F)c2)C(C)(C)C)cc1OC |w:11.10|
CSc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1 |w:11.10|
COc1ccc(CCCC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1 |w:13.12|
Cc1ccccc1NC(NC#N)=NC(NC(=O)CCCc1ccccc1)C(C)(C)C |w:12.13|
Cc1ncccc1NC(NC#N)=NC(NC(=O)Cc1ccc(Cl)cc1)C(C)(C)C |w:12.13|
CC(C)(C)C(NC(=O)Cc1ccc2OCCOc2c1)N=C(NC#N)Nc1cccc2ncccc12 |w:19.20|
CC(C)(C)C(NC(=O)Cc1cccc2ccccc12)N=C(NC#N)Nc1cccc2ncccc12 |w:19.20|
COc1ccc(CC(=O)NC(NC(Nc2cccnc2OC)=NC#N)C(C)(Cl)Cl)cc1OC |w:22.23|
COc1ncccc1NC(NC(NC(=O)c1ccc(Cl)cc1)C(C)(Cl)Cl)=NC#N |w:26.28|
CC(Cl)(Cl)C(NC(Nc1cccnc1Cl)=NC#N)NC(=O)c1ccc(Cl)cc1 |w:15.16|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cc(C)ccc2C)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccc(C)cc2)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1 |w:11.10|
COc1ccc(CCC(=O)NC(N=C(NC#N)Nc2ccccc2C)C(C)(C)C)cc1 |w:12.11|
CC(C)(C)C(NC(=O)Cc1ccc(Cl)cc1)N=C(NC#N)Nc1cccc2ncccc12 |w:16.16|
CSc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccc3ncccc23)C(C)(C)C)cc1 |w:11.10|
COc1cc(OC)cc(c1)C(=O)NC(NC(Nc1cccnc1OC)=NC#N)C(C)(Cl)Cl |w:25.27|
Cc1ccccc1NC(NC#N)=NC(NC(=O)Cc1ccc(Cl)cc1)C(C)(C)C |w:12.13|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2ccccc2Cl)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(NC(NC#N)=NC(NC(=O)Cc2ccc(OC)c(OC)c2)C(C)(C)C)c(OC)n1 |w:11.11|
CCCCCC(=O)NC(N=C(NC#N)Nc1ccccc1C)C(C)(C)C |w:9.8|
COc1ccc(CC(=O)NC(N=C(NC#N)Nc2cccnc2Cl)C(C)(C)C)cc1OC |w:11.10|
COc1ccc(CCC2=N[C@@H]([C@@H](N2)c2ccccc2)c2ccccc2)cc1 |t:8|
Cc1ccccc1CCC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:10|
Clc1ccccc1CCC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:10|
Clc1ccc(CCC2=N[C@@H]([C@@H](N2)c2ccccc2)c2ccccc2)cc1 |t:7|
Fc1ccccc1CC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:9|
Fc1ccc(CC2=N[C@@H]([C@@H](N2)c2ccccc2)c2ccccc2)cc1 |t:6|
Fc1cccc(CNC2=NC(C(N2)c2ccccc2)c2ccccc2)c1 |t:8|
CN(CCO)CCc1cc(C(=O)NCC23CC4CC(CC(C4)C2)C3)c(Cl)cn1 |TLB:15:14:17.16.21:19,21:16:23:20.19.22,21:20:23:17.16.15,13:14:17.16.21:19,THB:15:16:19:23.14.22,22:14:17:21.20.19,22:20:17:23.15.14,13:14:17:21.20.19|
OCCCNCCOc1cc(C(=O)NCC23CC4CC(CC(C4)C2)C3)c(Cl)cn1 |TLB:16:15:18.17.22:20,22:17:24:21.20.23,22:21:24:18.17.16,14:15:18.17.22:20,THB:16:17:20:24.15.23,23:15:18:22.21.20,23:21:18:24.16.15,14:15:18:22.21.20|
OCCCNc1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2n1 |TLB:15:14:17.16.21:19,21:16:23:20.19.22,21:20:23:17.16.15,13:14:17.16.21:19,THB:15:16:19:23.14.22,22:14:17:21.20.19,22:20:17:23.15.14,13:14:17:21.20.19|
OCCN1CCN(Cc2ccc3c(NC(=O)CC45CC6CC(CC(C6)C4)C5)c(Cl)ccc3n2)CC1 |TLB:18:17:20.19.24:22,24:19:26:23.22.25,24:23:26:20.19.18,16:17:20.19.24:22,THB:18:19:22:26.17.25,25:17:20:24.23.22,25:23:20:26.18.17,16:17:20:24.23.22|
Cc1ccc2nc(CCNCCCO)ccc2c1NC(=O)CC12CC3CC(CC(C3)C1)C2 |TLB:23:22:25.24.29:27,29:24:31:28.27.30,29:28:31:25.24.23,21:22:25.24.29:27,THB:23:24:27:31.22.30,30:22:25:29.28.27,30:28:25:31.23.22,21:22:25:29.28.27|
OC(=O)C1CCCN(C1)c1ccc2c(C(=O)NCC34CC5CC(CC(C5)C3)C4)c(Cl)ccc2n1 |TLB:19:18:21.20.25:23,25:20:27:24.23.26,25:24:27:21.20.19,17:18:21.20.25:23,THB:19:20:23:27.18.26,26:18:21:25.24.23,26:24:21:27.19.18,17:18:21:25.24.23|
OC(=O)CCNC1CCCN(C1)c1ccc2c(C(=O)NCC34CC5CC(CC(C5)C3)C4)c(Cl)ccc2n1 |TLB:22:21:24.23.28:26,28:23:30:27.26.29,28:27:30:24.23.22,20:21:24.23.28:26,THB:22:23:26:30.21.29,29:21:24:28.27.26,29:27:24:30.22.21,20:21:24:28.27.26|
OC(=O)c1cccc(c1)-c1ccc2c(C(=O)NCC34CC5CC(CC(C5)C3)C4)c(Cl)ccc2n1 |TLB:19:18:21.20.25:23,25:20:27:24.23.26,25:24:27:21.20.19,17:18:21.20.25:23,THB:19:20:23:27.18.26,26:18:21:25.24.23,26:24:21:27.19.18,17:18:21:25.24.23|
Clc1ccc2nc(ccc2c1C(=O)NCC12CC3CC(CC(C3)C1)C2)N1CCCC(C1)NCCc1nnn[nH]1 |TLB:16:15:18.17.22:20,22:17:24:21.20.23,22:21:24:18.17.16,14:15:18.17.22:20,THB:16:17:20:24.15.23,23:15:18:22.21.20,23:21:18:24.16.15,14:15:18:22.21.20|
OCCCNc1ccc2c(NC(=O)CC3CCCCC3)c(Cl)ccc2n1
CC1CCC(CC(=O)Nc2cccc3ncccc23)CC1 |(-5,-10.97,;-4.29,-11.38,;-4.29,-12.21,;-3.58,-12.62,;-2.86,-12.21,;-2.15,-12.62,;-1.43,-12.21,;-1.43,-11.39,;-.72,-12.63,;-.01,-12.21,;.71,-12.63,;1.42,-12.22,;1.42,-11.39,;.71,-10.98,;.7,-10.16,;-.01,-9.75,;-.72,-10.17,;-.72,-10.99,;-.01,-11.39,;-2.86,-11.38,;-3.58,-10.97,)|
Clc1ccc2ncccc2c1C(=O)NCC1CCCCC1
CS(=O)(=O)NC(=O)NCCCc1ccc2c(C(=O)NCC3CCCCC3)c(Cl)ccc2n1
OC(=O)c1ccccc1-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
OC(=O)C1CCN(CC1)c1ncccc1-c1ccc(Cl)c(c1)C(=O)NCC1CCCCCC1
OC1CCN(C1)c1ccc2c(NC(=O)CNc3cccc(c3)C#N)c(Cl)ccc2n1
OC1CCN(C1)c1ccc2c(NC(=O)CSc3ccccc3)c(Cl)ccc2n1
CC(CC(=O)Nc1c(Cl)ccc2nc(C)ccc12)c1ccccc1
Clc1ccc(CCC(=O)Nc2c(Cl)ccc3nc(ccc23)N2CCNCC2)c(Cl)c1
Clc1ccc(cc1C(=O)NCC12CC3CC(CC(C3)C1)C2)-n1ncc(=O)[nH]c1=O |TLB:12:11:14.13.18:16,18:13:20:17.16.19,18:17:20:14.13.12,10:11:14.13.18:16,THB:12:13:16:20.11.19,19:11:14:18.17.16,19:17:14:20.12.11,10:11:14:18.17.16|
Cc1ccc(nc1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCC(C)(C)C1
Cc1cc(n[nH]1)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCC(C)(C)C1
CN(C)CCNC(=O)Cn1nc(cc1C)-c1ccc(Cl)c(c1)C(=O)NCC1(O)CCCCCC1
CC(C)C(CO)n1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2c1=O |TLB:16:15:18.17.22:20,22:17:24:21.20.23,22:21:24:18.17.16,14:15:18.17.22:20,THB:16:17:20:24.15.23,14:15:18:22.21.20,23:15:18:22.21.20,23:21:18:24.16.15|
OCC(CO)n1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)cccc2c1=O |TLB:15:14:17.16.21:19,21:16:23:20.19.22,21:20:23:17.16.15,13:14:17.16.21:19,THB:15:16:19:23.14.22,13:14:17:21.20.19,22:14:17:21.20.19,22:20:17:23.15.14|
O=C(CC12CC3CC(CC(C3)C1)C2)Nc1cccc2c1ccn(CC1CCCN1)c2=O |TLB:4:3:6.5.10:8,10:5:12:9.8.11,10:9:12:6.5.4,2:3:6.5.10:8,THB:4:5:8:12.3.11,2:3:6:10.9.8,11:3:6:10.9.8,11:9:6:12.4.3|
CC(C(N)=O)n1ccc2c(NC(=O)CC34CC5CC(CC(C5)C3)C4)c(Cl)ccc2c1=O |TLB:15:14:17.16.21:19,21:16:23:20.19.22,21:20:23:17.16.15,13:14:17.16.21:19,THB:15:16:19:23.14.22,13:14:17:21.20.19,22:14:17:21.20.19,22:20:17:23.15.14|
FC(F)(F)c1cc(CC(=O)Nc2cccc3c2ccn(C2CCNC2)c3=O)ccc1Cl
OCCn1ccc2c(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c(Cl)ccc2c1=O
O=C(CC1CCCCCC1)Nc1cccc2c1ccn(C1CCNC1)c2=O
OC1CNCC1n1ccc2c(NC(=O)Cc3ccc(F)c(c3)C(F)(F)F)cccc2c1=O
OCCn1ccc2c(NC(=O)Cc3ccc(Cl)c(c3)C(F)(F)F)cccc2c1=O
Fc1c(CC(=O)Nc2c(Cl)ccc3c2ccn(C2CC2)c3=O)cccc1C(F)(F)F
CCS(=O)(=O)N1CCc2c(C1)ccc(C)c2NC(=O)Cc1ccc(c(F)c1)C(F)(F)F
Fc1cc(CC(=O)Nc2cccc3CN(CCc23)C(=O)C2CCCN2)ccc1C(F)(F)F
CC1(C)C2CCC(C2)(C(=O)NNc2ccccc2)C1=C |THB:19:18:4.5:7|
Clc1ccc(cc1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:10:11:14:17.18.16,THB:19:11:14:17.18.16,19:17:11.20.12:14,16:17:12:15.20.14,16:15:12:17.19.18|
Clc1ccccc1C(=O)NC12CC3CC(CC(C3)C1)C2 |TLB:13:14:18:12.11.17,THB:13:12:18:14.19.15,15:16:11:14.19.13,15:14:11:16.18.17|
Fc1cccc(CNC2=NC(C(N2)c2cccc(F)c2)c2cccc(F)c2)c1 |t:8|
Cc1cccc(c1)C1NC(NCc2cccc(F)c2)=NC1c1cccc(C)c1 |c:20|
CC1(NC(NCc2cccc(F)c2)=NC1c1cccc(F)c1)c1cccc(F)c1 |c:13|
Fc1cccc(CSC2=NC(C(N2)c2ccccc2)c2ccccc2)c1 |t:8|
CC(=O)NC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
COC(=O)NC(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
CNCC(O)c1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:17:16:19.18.23:21,23:18:25:22.21.24,23:22:25:19.18.17,15:16:19.18.23:21,THB:17:18:21:25.16.24,24:16:19:23.22.21,24:22:19:25.17.16,15:16:19:23.22.21|
CNCC(O)Cc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:18:17:20.19.24:22,24:19:26:23.22.25,24:23:26:20.19.18,16:17:20.19.24:22,THB:18:19:22:26.17.25,25:17:20:24.23.22,25:23:20:26.18.17,16:17:20:24.23.22|
OC(=O)c1ccc(cc1)-c1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:21:20:23.22.27:25,27:22:29:26.25.28,27:26:29:23.22.21,19:20:23.22.27:25,THB:21:22:25:29.20.28,28:20:23:27.26.25,28:26:23:29.21.20,19:20:23:27.26.25|
OC(=O)c1cncc(c1)-c1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:21:20:23.22.27:25,27:22:29:26.25.28,27:26:29:23.22.21,19:20:23.22.27:25,THB:21:22:25:29.20.28,28:20:23:27.26.25,28:26:23:29.21.20,19:20:23:27.26.25|
C(Cc1ccccc1)C1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:9|
N1[C@H]([C@H](N=C1c1ccccc1)c1ccccc1)c1ccccc1 |c:3|
C(CC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1)Cc1ccccc1 |t:2|
C(CCc1ccccc1)CC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:11|
CC(CC1=NC(C(N1)c1ccccc1)c1ccccc1)c1ccccc1 |t:3|
CC(C)(CC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1)c1ccccc1 |t:4|
C1C(Cc2ccccc12)C1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:11|
Clc1cccc(-c2nnnn2Cc2c(Cl)cccc2Cl)c1Cl
Cc1ccccc1CC1=N[C@@H]([C@@H](N1)c1ccccc1)c1ccccc1 |t:9|
Clc1cccc(CCC2=N[C@@H]([C@@H](N2)c2ccccc2)c2ccccc2)c1 |t:8|
Fc1cccc(CC2=N[C@@H]([C@@H](N2)c2ccccc2)c2ccccc2)c1 |t:7|
Fc1cccc(CNC2=NC(C(N2)c2ccccc2Cl)c2ccccc2Cl)c1 |t:8|
Fc1cccc(COC2=NC(C(N2)c2ccccc2)c2ccccc2)c1 |t:8|
COC(=O)N(C)C(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
CN(C(CN1CCN(CC1)c1ccccc1)Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)S(=O)(=O)c1cccc2cnccc12
CN(C)CC(O)Cc1ccc(Cl)c(c1)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:19:18:21.20.25:23,25:20:27:24.23.26,25:24:27:21.20.19,17:18:21.20.25:23,THB:19:20:23:27.18.26,26:18:21:25.24.23,26:24:21:27.19.18,17:18:21:25.24.23|
CC(CO)n1ccc2c(NC(=O)Cc3ccc(Cl)c(c3)C(F)(F)F)cccc2c1=O
C[C@H](CN1CCN(CC1)C(C)=O)NC(=O)c1cc2c(nn(C)c2s1)-c1ccccc1 |r|
CCCc1nc(oc1C(=O)NC(C)CN1CCN(CC1)c1ncccn1)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1nn(Cc2cccnc2)c(C)c1CC(=O)NCc1ccc(F)cc1Cl
Cc1nn(Cc2ccccc2)c(C)c1CC(=O)NCc1ccc(F)cc1Cl
COc1ccc(cc1)-n1nc(C)c(CC(=O)NCc2ccc(F)cc2Cl)c1C
Cc1sc(nc1CC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1oc(nc1CC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1c(CC(=O)NCc2ccc(F)cc2Cl)cnn1-c1ccccc1
Cc1nn(c(C)c1CNC(=O)Cc1ccc(F)cc1Cl)-c1ccccc1
Cc1nn(c(C)c1C(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ncccc1C)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NC1CCCCCC1)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1cc(Cl)cc(Cl)c1)-c1ccccc1
COc1ccccc1CNC(=O)Cc1c(C)nn(c1C)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccccc1Cl)-c1ccccc1
Cc1nn(c(C)c1CC(=O)NCc1ccccc1)-c1ccccc1
Cc1n[nH]c(C)c1CC(=O)NCc1ccccc1Cl
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(F)cc1F
Cc1noc(C)c1CC(=O)NCc1cccc(c1Cl)C(F)(F)F
Cc1noc(C)c1CC(=O)NCc1ccc(Cl)cc1Cl
Cn1ncc(F)c1CC(=O)NCc1cccc(c1Cl)C(F)(F)F
Cc1cnn(C)c1CC(=O)NCc1cccc(c1Cl)C(F)(F)F
Cc1cnn(C)c1CC(=O)NCc1ccc(Cl)cc1Cl
Cc1n[nH]c(C)c1CC(=O)NCc1cccc(c1Cl)C(F)(F)F
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(Cl)c(c1)C(F)(F)F
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(F)cc1C(F)(F)F
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(Cl)cc1Cl
Cc1n[nH]c(C)c1CC(=O)NCc1ccc(Cl)cc1
Cc1n[nH]c(C)c1CC(=O)NCc1cccc(Cl)c1
Cc1noc(C)c1CCC(=O)NCc1ccc(F)cc1Cl
Cc1cc(CCC(=O)NCc2ccc(F)cc2Cl)n(C)n1
Cc1cnn(C)c1CCC(=O)NCc1ccc(F)cc1Cl
Cc1cn[nH]c1CCC(=O)NCc1ccc(F)cc1Cl
Cc1[nH]nc(c1CCC(=O)NCc1ccc(F)cc1Cl)C(F)(F)F
Cc1[nH]nc(c1CCC(=O)NCc1ccc(F)cc1Cl)-c1ccccc1
Cc1[nH]nc(c1CCC(=O)NCc1ccc(F)cc1Cl)C(C)(C)C
CC(C)Cc1n[nH]c(C)c1CCC(=O)NCc1ccc(F)cc1Cl
CC(C)c1n[nH]c(C(C)C)c1CCC(=O)NCc1ccc(F)cc1Cl
CCc1n[nH]c(CC)c1CCC(=O)NCc1ccc(F)cc1Cl
CCN1[C@@H](CCC1=O)C(=O)NCc1ccc(Cl)cc1Cl |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CC(=O)N1CCC[C@H]1C(=O)NCc1ccc(F)cc1Cl |r|
CCN1[C@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CCN1[C@@H](CCCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CC(C)N1[C@@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CN(C(=O)c1cc(Cl)c(=O)n(Cc2c(Cl)cccc2Cl)c1)c1ccccc1
CN1[C@@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CCCN1[C@@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
CC(C)CN1[C@@H](CCC1=O)C(=O)NCc1ccc(F)cc1Cl |r|
Fc1ccc(CNC(=O)[C@@H]2CCC(=O)N2C2CCC2)c(Cl)c1 |r|
Fc1ccc(CNC(=O)[C@@H]2CCC(=O)N2C2CCCC2)c(Cl)c1 |r|
Fc1ccc(CNC(=O)[C@@H]2CCC(=O)N2c2ccccc2)c(Cl)c1 |r|
CCN1[C@@H](CCC1=O)C(=O)NCC12CC3CC(CC(C3)C1)C2 |r,TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
CCN1[C@@H](CCC1=O)C(=O)NCc1ccc(Cl)cc1 |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1ccccc1C(F)(F)F |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1ccccc1Cl |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1cccc(c1)C(F)(F)F |r|
CCN1[C@@H](CCC1=O)C(=O)NCc1cccc(Cl)c1Cl |r|
CN1[C@@H](CN(C1=O)c1cccc(C)n1)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(C2CCN(C)CC2)C1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(CCN2CCOCC2)C1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(C1=O)c1ccnc(C)c1)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1C[C@H](N(C)C1=O)C(=O)NCc1cccc(Cl)c1Cl |r|
CN1[C@@H](CN(C1=O)c1cccnc1C)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](COCC1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CNC1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(C1=O)c1cn(C)cn1)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1C[C@H](N(C)C1=O)C(=O)NCc1ccc(Cl)cc1Cl |r|
CN1[C@@H](CNC1=O)C(=O)NCc1cccc(Cl)c1Cl |r|
CN1[C@@H](CC(F)(F)C1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1[C@@H](CN(C1=O)c1nccn1C)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
CN1C[C@H](N(C)C1=O)C(=O)NCc1cccc(c1Cl)C(F)(F)F |r|
Clc1cccc(c1Cl)-n1nnnc1NCc1ccccc1N1CCOCC1
FC(F)Oc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
CCOc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
CC(C)Oc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Clc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Clc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
Clc1ccc(CNc2nnnn2-c2cccc(Cl)c2Cl)cc1
FC(F)(F)c1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
FC(F)(F)c1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
FC(F)(F)c1ccc(CNc2nnnn2-c2cccc(Cl)c2Cl)cc1
FC(F)(F)Oc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
FC(F)(F)Oc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
FC(F)(F)Oc1ccc(CNc2nnnn2-c2cccc(Cl)c2Cl)cc1
COc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1OC
Clc1cccc(c1Cl)-n1nnnc1NCc1cccc2OCOc12
Clc1cccc(c1Cl)-n1nnnc1NCc1cccc2OCCc12
Cc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1C
Fc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1F
Fc1ccc(F)c(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
Fc1ccc(Cl)cc1CNc1nnnn1-c1cccc(Cl)c1Cl
Fc1ccc(F)c(CNc2nnnn2-c2cccc(Cl)c2Cl)c1Cl
Clc1cccc(c1Cl)-n1nnnc1N[C@@H]1CCc2ccccc12 |r|
Clc1cccc(c1Cl)-n1nnnc1N[C@H]1CCc2ccccc12 |r|
Clc1cccc(c1Cl)-n1nnnc1NC1COc2ccccc12
CC(C)(Nc1nnnn1-c1cccc(Cl)c1Cl)c1ccccc1
C[C@@H](Nc1nnnn1-c1cccc(Cl)c1Cl)c1ccccc1 |r|
CN(Cc1ccccc1)c1nnnn1-c1cccc(Cl)c1Cl
CS(=O)(=O)c1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
COc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Clc1cccc(c1Cl)-n1nnnc1NCc1ccccc1
Cc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Cc1ccccc1Nc1nnnn1-c1cccc(Cl)c1Cl
Fc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Fc1ccc(CNc2nnnn2-c2cccc(Cl)c2Cl)cc1
Clc1cccc(c1Cl)-n1nnnc1NCc1ccccc1C#N
CSc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
CN(C)c1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
C[C@H](Nc1nnnn1-c1cccc(Cl)c1Cl)c1ccccc1 |r|
COc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
Fc1cccc(CNc2nnnn2-c2cccc(Cl)c2Cl)c1
CCN(CC)CCOc1ccccc1CNc1nnnn1-c1cccc(Cl)c1Cl
Cc1ccc(F)cc1Cn1cnnc1-c1cccc(Cl)c1Cl
Clc1cccc(Cn2cnnc2-c2cccc(Cl)c2Cl)c1Cl
Clc1cccc(c1Cl)-n1nncc1Cc1ccccc1
FC(F)(F)c1ccccc1Cn1cnnc1-c1cccc(Cl)c1Cl
Clc1cccc(-c2nncn2Cc2ccccc2)c1Cl
Fc1ccc(cc1Cn1cnnc1-c1cccc(Cl)c1Cl)C(F)(F)F
Clc1cccc(-c2nncn2Cc2cccc3ccccc23)c1Cl
Clc1cccc(-c2ncnn2Cc2ccccc2)c1Cl
CS(=O)(=O)c1ccccc1Cn1cnnc1-c1cccc(c1Cl)C(F)(F)F
Fc1ccc(c(Cn2cnnc2-c2cccc(Cl)c2Cl)c1)C(F)(F)F
Clc1ccc(Cn2cnnc2-c2cccc(Cl)c2Cl)c(Cl)c1
COc1cccc(Cn2cnnc2-c2cccc(Cl)c2Cl)c1OC
Clc1cccc(-c2cnnn2Cc2ccccc2)c1Cl
Clc1ccc(Cl)c(Cn2cnnc2-c2cccc(Cl)c2Cl)c1
FC(F)c1ccccc1Cn1cnnc1-c1cccc(Cl)c1Cl
C[C@H](CN)n1ccc2c(NC(=O)Cc3ccc(c(F)c3)C(F)(F)F)c(C)ccc2c1=O |r|
Cc1c(c(c(c(n1)/N=N/c2ccc(cc2)C(=O)O)COP(=O)(O)O)C=O)O
Cc1nc(N=Nc2cc(c3cc(cc(c3c2)S(O)(=O)=O)[N+]([O-])=O)S(O)(=O)=O)c(CO[P+](O)(O)[O-])c(C=O)c1O |w:4.3|
O=C(NC1(C2CC3CC(C2)CC1C3)C(=O)NC1CC1)c1ccccc1 |TLB:2:3:5.6.12:9.8.10,2:3:5:9.8.7,13:3:5:9.8.7,THB:13:3:5.6.12:9.8.10,7:6:3:9.8.10,7:8:3:5.6.12,10:11:5:9.8.7,10:8:5:3.12.11,(22.9,-26.25,;22.14,-24.91,;20.6,-24.91,;19.84,-23.58,;18.44,-23.02,;16.93,-23.44,;18.13,-22.16,;18.12,-20.68,;19.47,-20.2,;18.43,-21.43,;20.87,-20.78,;20.86,-22.31,;19.46,-22.65,;19.06,-24.9,;19.83,-26.24,;17.52,-24.9,;16.75,-26.23,;15.41,-27.01,;16.74,-27.78,;22.91,-23.58,;24.45,-23.6,;25.23,-22.27,;24.46,-20.93,;22.91,-20.93,;22.14,-22.26,)|
CC(C)N(C(C)C)C(=O)N1c2ccccc2C=Cc2ccccc12 |c:17|
CCCN(CCC)C(=O)N1c2ccccc2C=Cc2ccccc12 |c:17|
O=C(N1CCCC1)N1c2ccccc2C=Cc2ccccc12 |c:16|
O=C(N1CCCCC1)N1c2ccccc2C=Cc2ccccc12 |c:17|
O=C(NC1CCCCC1)N1c2ccccc2C=Cc2ccccc12 |c:18|
CCN(CC)C(=O)N1c2ccccc2C=Cc2ccccc12 |c:15|
CC(C)(C)OC(=O)N1CCC(CN2C(=O)C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)N(Cc3cccc4cnccc34)C2=O)CC1
O=C1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)N(CC2CCN(Cc3ccccc3)CC2)C(=O)N1Cc1cccc2cnccc12
CC(C)(C)OC(=O)N1CCC(CN2C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C(=O)N(Cc3cccc4cnccc34)C2=O)CC1
O=C1N[C@@H](Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)N1Cc1cccc2cnccc12 |r|
CC(C)(C)OC(=O)N1CCC(CN2C(=O)N[C@@H](Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C2=O)CC1 |r|
O=C1NC(=O)N(Cc2cccc3cnccc23)C1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C1NC(=O)N(CC2CCN(Cc3ccccc3)CC2)C1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
CC(C)(C)OC(=O)N1CCC(CN2C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C(=O)NC2=O)CC1
CC(C)(C)OC(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
O=C1NC(=O)N(C1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C1CCN(Cc2ccccc2)CC1
O=C(N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O)c1ccccc1
O=C(N1CCC(CN2C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C(=O)NC2=O)CC1)c1ccccc1
CC(C)(C)OC(=O)N1CCC(CCN2C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C(=O)NC2=O)CC1
O=C1NC(=O)N(CCC2CCN(Cc3ccccc3)CC2)C1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1
O=C(N1CCC(CCN2C(Cc3ccc(OS(=O)(=O)c4cccc5cnccc45)cc3)C(=O)NC2=O)CC1)c1ccccc1
CCC(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
CC(C)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
CC(C)(C)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
CCCC(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
CC(C)CC(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
O=C(C1CCCCC1)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
O=C(N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O)C12CC3CC(CC(C3)C1)C2 |TLB:45:36:43:39.40.41,THB:41:40:37:43.42.44,41:42:39.40.45:37,45:40:43:36.37.44,1:36:43:39.40.41|
O=C1NC(=O)N(C1Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)C1CCN(CC23CC4CC(CC(C4)C2)C3)CC1 |TLB:42:33:40:36.37.38,THB:38:37:34:40.39.41,38:39:36.37.42:34,42:37:40:33.34.41,32:33:40:36.37.38|
O=C(CC12CC3CC(CC(C3)C1)C2)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O |TLB:12:3:10:6.7.8,THB:8:7:4:10.9.11,8:9:6.7.12:4,12:7:10:3.4.11,2:3:10:6.7.8|
BrC12CC3CC(C1)CC(C3)(C2)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O |TLB:4:5:2.3.9:10,9:8:6:2.3.4,THB:9:3:6:8.10.7|
CC12CC3CC(C)(C1)CC(C3)(C2)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O |TLB:4:5:11:2.3.10,12:9:2:7.5.4,6:5:2:9.11.10,6:5:11:2.3.10,THB:4:3:7.5.8:11,8:5:2:9.11.10,8:9:2:7.5.4|
O=C(N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O)C12CC3CC1CC(C2)C3 |TLB:39:38:40.41:43,THB:39:40:43:37.38.44,41:42:37:39.40|
O=C(CC1CC2CCC1C2)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
COc1ccc(cc1OC)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Clc1ccccc1C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Clc1cccc(c1)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Clc1ccc(cc1)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Fc1ccc(cc1)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
O=C([C@@H]1Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2CN1S(=O)(=O)c1cccc2cnccc12)N1CCN(CC1)c1ccccc1
Fc1ccc(cc1F)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Clc1ccc(cc1Cl)C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
Fc1cc(Cl)ccc1C(=O)N1CCC(CC1)N1C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)C(=O)NC1=O
CN1C(=O)C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)N(C2CCN(CC2)C(=O)c2ccc(Cl)c(c2)C(F)(F)F)C1=O
CCN1C(=O)C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)N(C2CCN(CC2)C(=O)c2ccc(Cl)c(c2)C(F)(F)F)C1=O
CCCN1C(=O)C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)N(C2CCN(CC2)C(=O)c2ccc(Cl)c(c2)C(F)(F)F)C1=O
CC(C)N1C(=O)C(Cc2ccc(OS(=O)(=O)c3cccc4cnccc34)cc2)N(C2CCN(CC2)C(=O)c2ccc(Cl)c(c2)C(F)(F)F)C1=O
Oc1csc(=O)n1C(CCc1ccncc1)COc1ccc(cc1)-c1cccc(c1)[N+]([O-])=O
C[S+]([O-])c1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccccn1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnc2-c1cnccn1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1cnccn1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnc2-c1ccc(F)cc1 |r|
C[C@@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccc(F)cc1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccc(F)cc1 |r|
C[C@@H]1N(CCn2c1nnc2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl |r|
C[C@H]1N(CCn2c1nnc2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl |r|
CC1Cn2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnc2-c1ccccc1
CC1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccccc1
CC1N(CCn2c1nnc2-c1cnccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCn2c1nnc2-c1ccccn1)C(=O)c1cccc(c1F)C(F)(F)F
CC1CN(Cc2nnc(-c3ccc(F)cc3)n12)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1CN(Cc2nnc(-c3ccc(F)cc3)n12)C(=O)c1cccc(Cl)c1Cl
CC1Cn2c(CN1C(=O)c1cccc(c1Cl)C(F)(F)F)nnc2-c1ccc(F)cc1
CC1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccc(F)cc1
CC1N(CCn2c1nnc2-c1ccc(F)cc1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCn2c1nnc2-c1ccccn1)C(=O)c1cccc(c1Cl)C(F)(F)F
CC1N(CCn2c1nnc2-c1ccccn1)C(=O)c1cccc(Cl)c1Cl
Fc1ccc(cc1)-c1nnc2CN(CCn12)C(=O)c1cccc(c1Cl)C(F)(F)F
FC(F)(F)c1cccc(C(=O)N2CCn3c(C2)nnc3-c2ccccn2)c1Cl
Clc1cccc(C(=O)N2CCn3c(C2)nnc3-c2ccccn2)c1Cl
FC(F)(F)c1cccc(C(=O)N2CCn3c(C2)nnc3-c2cnccn2)c1Cl
Clc1cccc(C(=O)N2CCn3c(C2)nnc3-c2cnccn2)c1Cl
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1cccc(F)n1 |r|
COc1ccnc(c1)-c1nnc2CN([C@@H](C)Cn12)C(=O)c1cccc(Cl)c1Cl |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ccc(F)cn1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1ncc(F)cn1 |r|
C[C@H]1Cn2c(CN1C(=O)c1cccc(Cl)c1Cl)nnc2-c1cc(F)ccn1 |r|
FC(F)(F)c1cccc(CN2CCc3c(nnn3-c3cnccn3)C2=O)c1Cl
COc1cccc(C(=O)N2Cc3nc(C)nc(-c4ccn[nH]4)c3CC2C)c1F
O[C@@H]1CCN(C1)c1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1 |r|
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)ccc2nc(NC3CC3)ccc12)N1CCC(F)(F)CC1
O[C@H]1CCN(C1)c1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1 |r|
FC(F)(F)c1ncc(cn1)C(CNC(=O)c1c(Cl)ccc2nc(ccc12)N1CCOCC1)N1CCC(F)(F)CC1
CNc1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1
CN1CCN(CC1)c1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1
OC1CCN(CC1)c1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1
Nc1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1
OCCNc1ccc2c(C(=O)NCC(N3CCC(F)(F)CC3)c3cnc(nc3)C(F)(F)F)c(Cl)ccc2n1
FC(F)(F)c1ccccc1NNC(=O)C12C3C=CC4C3C3C(C=CC13)C24 |c:17,24,TLB:17:18:15.14:21.20,17:18:15:24.20,12:14:16.17:19,THB:21:25:16.17:19,21:25:15:24.20,24:14:16.17:19,20:19:16.17:14.25|
FC(F)(F)c1ccc(NNC(=O)C23C4C=CC5C4C4C(C=CC24)C35)c(Cl)c1 |c:14,21,TLB:15:16:13.12:19.18,15:16:13:22.18,10:12:14.15:17,THB:19:23:14.15:17,19:23:13:22.18,22:12:14.15:17,18:17:14.15:12.23|
Clc1ccccc1NNC(=O)C12C3C=CC4C3C3C(C=CC13)C24 |c:14,21,TLB:14:15:12.11:18.17,14:15:12:21.17,9:11:13.14:16,THB:18:22:13.14:16,18:22:12:21.17,21:11:13.14:16,17:16:13.14:11.22|
FC(F)(F)c1ccccc1NNC(=O)C12C3CCC4C3C3C(CCC13)C24 |TLB:17:18:15.14:21.20,17:18:15:24.20,12:14:16.17:19,THB:21:25:16.17:19,21:25:15:24.20,24:14:16.17:19,20:19:16.17:14.25|
CC12CC3CC1(C)CC3(C2)C(=O)NNc1ccccc1Cl |TLB:2:1:7:3.4,4:3:9:7.5,THB:2:3:7:9.1,0:1:7:3.4|
Clc1ccccc1NNC(=O)C12C3CCC4C3C3C(CCC13)C24 |TLB:14:15:12.11:18.17,14:15:12:21.17,9:11:13.14:16,THB:18:22:13.14:16,18:22:12:21.17,21:11:13.14:16,17:16:13.14:11.22|
N#C\N=C(\NCCc1ccccc1)NC12CC3CC(CC(C3)C1)C2 |TLB:13:14:17:21.20.19,THB:15:16:19:23.14.22,15:14:17.16.21:19,22:14:17:21.20.19,22:20:17:23.15.14,13:14:17.16.21:19|
Fc1ccc(N\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)cc1 |TLB:8:9:12.11.16:14,THB:10:11:14:18.9.17,10:9:12.11.16:14,17:9:12:16.15.14,17:15:12:18.10.9|
N#C\N=C(\NCc1ccccn1)NCC12CC3CC(CC(C3)C1)C2 |TLB:13:14:17:21.20.19,THB:22:20:17:15.23.14,22:14:17:21.20.19,19:20:15:17.18.23,19:18:15:21.22.20|
N#C\N=C(\NCc1ccncc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:13:14:17:21.20.19,THB:22:20:17:15.23.14,22:14:17:21.20.19,19:20:15:17.18.23,19:18:15:21.22.20|
N#C\N=C(/NCCC12CC3CC(CC(C3)C1)C2)Nc1ccccc1 |TLB:6:7:10:14.13.12,THB:8:9:12:16.7.15,8:7:10.9.14:12,15:7:10:14.13.12,15:13:10:16.8.7,6:7:10.9.14:12|
Fc1ccc(CN\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)cc1 |TLB:9:10:13:17.16.15,THB:18:16:13:11.19.10,18:10:13:17.16.15,15:16:11:13.14.19,15:14:11:17.18.16|
COc1cccc(N\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)c1 |TLB:10:11:14.13.18:16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11|
COc1ccc(CN\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)cc1 |TLB:10:11:14:18.17.16,THB:19:17:14:12.20.11,19:11:14:18.17.16,16:17:12:14.15.20,16:15:12:18.19.17|
COc1cccc(CN\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)c1 |TLB:11:12:15:19.18.17,THB:20:18:15:13.21.12,20:12:15:19.18.17,17:18:13:15.16.21,17:16:13:19.20.18|
COc1ccccc1CN\C(NCC12CC3CC(CC(C3)C1)C2)=N\C#N |TLB:12:13:16:20.19.18,THB:21:19:16:14.22.13,21:13:16:20.19.18,18:19:14:16.17.22,18:17:14:20.21.19|
N#C\N=C(/NCC12CC3CC(CC(C3)C1)C2)Nc1ccncc1 |TLB:5:6:9.8.13:11,THB:7:8:11:15.6.14,7:6:9.8.13:11,14:6:9:13.12.11,14:12:9:15.7.6|
N#C\N=C(/NCC12CC3CC(CC(C3)C1)C2)Nc1cccnc1 |TLB:5:6:9.8.13:11,THB:7:8:11:15.6.14,7:6:9.8.13:11,14:6:9:13.12.11,14:12:9:15.7.6|
Fc1cccc(N\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)c1 |TLB:9:10:13.12.17:15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
Fc1ccccc1N\C(NCC12CC3CC(CC(C3)C1)C2)=N\C#N |TLB:10:11:14.13.18:16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11|
COc1ccc(N\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)cc1 |TLB:9:10:13.12.17:15,THB:11:12:15:19.10.18,11:10:13.12.17:15,18:10:13:17.16.15,18:16:13:19.11.10|
COc1ccccc1N\C(NCC12CC3CC(CC(C3)C1)C2)=N\C#N |TLB:11:12:15.14.19:17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12|
N#C\N=C(/NCCC12CC3CC(CC(C3)C1)C2)NCc1ccccc1 |TLB:6:7:10:14.13.12,THB:8:9:12:16.7.15,8:7:10.9.14:12,15:7:10:14.13.12,15:13:10:16.8.7,6:7:10.9.14:12|
N#C\N=C(\NCCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:14:15:18:22.21.20,THB:16:17:20:24.15.23,16:15:18.17.22:20,23:15:18:22.21.20,23:21:18:24.16.15|
N#C\N=C(\Nc1ccccc1)NC12CC3CC(CC(C3)C1)C2 |TLB:11:12:15:19.18.17,THB:13:14:17:21.12.20,13:12:15.14.19:17,20:12:15:19.18.17,20:18:15:21.13.12,11:12:15.14.19:17|
N#C\N=C(\NCc1ccccc1)NC12CC3CC(CC(C3)C1)C2 |TLB:12:13:16:20.19.18,THB:14:15:18:22.13.21,14:13:16.15.20:18,21:13:16:20.19.18,21:19:16:22.14.13,12:13:16.15.20:18|
N#C\N=C(\NCc1cccnc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:13:14:17:21.20.19,THB:22:20:17:15.23.14,22:14:17:21.20.19,19:20:15:17.18.23,19:18:15:21.22.20|
N#C\N=C(\NCc1ccccc1)NCC12CC3CC(CC(C3)C1)C2 |TLB:13:14:17:21.20.19,THB:15:16:19:23.14.22,15:14:17.16.21:19,22:14:17:21.20.19,22:20:17:23.15.14|
Fc1cccc(CN\C(NCC23CC4CC(CC(C4)C2)C3)=N\C#N)c1 |TLB:10:11:14:18.17.16,THB:19:17:14:12.20.11,19:11:14:18.17.16,16:17:12:14.15.20,16:15:12:18.19.17|
N#C\N=C(/NCC12CC3CC(CC(C3)C1)C2)Nc1cccc2ncccc12 |TLB:5:6:9.8.13:11,THB:7:8:11:15.6.14,7:6:9.8.13:11,14:6:9:13.12.11,14:12:9:15.7.6|
Fc1ccccc1CN\C(NCC12CC3CC(CC(C3)C1)C2)=N\C#N |TLB:11:12:15:19.18.17,THB:20:18:15:13.21.12,20:12:15:19.18.17,17:18:13:15.16.21,17:16:13:19.20.18|
N#C\N=C(/NCC12CC3CC(CC(C3)C1)C2)Nc1ccccn1 |TLB:5:6:9.8.13:11,THB:7:8:11:15.6.14,7:6:9.8.13:11,14:6:9:13.12.11,14:12:9:15.7.6|