3167 SMILES Strings for GTPase KRas [G12D]

Compound Name
SMILES String
O=C(CCc1c[nH]c2ccccc12)Nc1nnc([nH]1)-c1ccccn1
CC(Oc1cccc(c1)C#N)C(=O)Nc1nnc([nH]1)-c1ccccn1
Cc1cccc(OCC(=O)Nc2nnc([nH]2)-c2ccccn2)c1
O=c1nc([nH]c2c3ccccc3sc12)-c1ccccn1
COc1ccc(COCC(=O)N2CCCc3c(O)nc(nc23)-c2ccccn2)cc1
CS(=O)(=O)c1cccc(c1)C(=O)N1CCCc2c(O)nc(nc12)-c1ccccn1
Oc1nc(nc2c(csc12)C(=O)N1CCN(CC1)c1ccccc1)-c1ccccn1
Oc1nc(nc2sccc12)-c1ccccn1
OCc1ccnc(c1)-c1nc(O)c2ccsc2n1
Oc1cccc(CN2CCN(CC2)C(=O)c2csc3c(O)nc(nc23)-c2ccccn2)c1
Oc1nc(nc2c(csc12)C(=O)N1CCOC(C1)c1nccs1)-c1ccccn1
CC1CN(CCN1C(=O)c1csc2c(O)nc(nc12)-c1ccccn1)c1ccccc1
COc1ccccc1C1CN(CCO1)C(=O)c1csc2c(O)nc(nc12)-c1ccccn1
Oc1nc(nc2c(csc12)C(=O)N1CCOC(C1)c1ccccc1Cl)-c1ccccn1
COc1cccc(c1)C1CN(CCN1)C(=O)c1csc2c(O)nc(nc12)-c1ccccn1
O=C(COCc1ccc(cc1)C#N)Nc1nc(nc2sccc12)-c1ccccn1
OCc1ccnc(c1)-c1nc(O)c2c(Cl)csc2n1
Oc1ccc(cc1Cl)N1CCN(CC1)C(=O)c1csc2c(O)nc(nc12)-c1ccccn1
CC(N1CCN(CC1)C(=O)c1csc2c(O)nc(nc12)-c1ccccn1)c1ccccc1
Oc1ccc(cc1)C1CN(CCN1)C(=O)c1csc2c(O)nc(nc12)-c1ccccn1
CN1CCN(CC1)c1nc(nc2scc(C(=O)NCCc3cnc(O)nc3)c12)-c1ccccn1
Oc1nc(nc2c(csc12)-c1cc(F)cc(F)c1)-c1ccccn1
CN(C)Cc1ccc(F)c(c1)-c1csc2c(O)nc(nc12)-c1ccccn1
CCn1nc(C)cc1-c1csc2c(O)nc(nc12)-c1ccccn1
COC(=O)c1cc2nc(nc(O)c2s1)-c1ccccn1
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(cc2n1)-c1cc(O)cc2ccccc12 |r|
COc1ccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)cn1
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Cc1cccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)n1
Cn1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Cc1ccc2[nH]ncc2c1-c1ncc2c(nc(OCCc3nccn3C)nc2c1F)N1CC2CCC(C1)N2 |(-3.95,-5,;-5.28,-4.23,;-6.61,-5,;-7.95,-4.23,;-7.95,-2.69,;-9.09,-1.66,;-8.47,-.26,;-6.93,-.42,;-6.61,-1.93,;-5.28,-2.69,;-3.95,-1.93,;-3.95,-.38,;-2.61,.38,;-1.28,-.38,;.05,.38,;1.39,-.38,;1.39,-1.93,;2.72,-2.69,;4.06,-1.93,;5.39,-2.69,;6.72,-1.93,;8.19,-2.4,;9.09,-1.15,;8.19,.09,;6.72,-.38,;5.3,.2,;.05,-2.69,;-1.28,-1.93,;-2.61,-2.69,;-2.61,-4.23,;.05,1.93,;-1.28,2.69,;-1.28,4.23,;-.6,3.39,;.78,3.39,;1.39,4.23,;1.39,2.69,;.05,5,)|
Oc1cc(-c2ncc3c(nc(OCCc4ccccn4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OCc4ccccn4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Cn1nccc1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Fc1ccc2cccc(-c3ncc4c(nc(OCCc5cccnc5)nc4c3F)N3CC4CCC(C3)N4)c2c1
Cc1cccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CC(C)n1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Oc1cc(-c2ncc3c(nc(OCCc4ncccn4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Fc1c(ncc2c(nc(OCCc3cn4ccccc4n3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Cn1ccc(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)n1
Cn1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccccc12
Cn1cnc(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)c1
Cn1cncc1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CN1CCC[C@H]1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Oc1cc(-c2ncc3c(nc(OCCc4ccccc4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CCN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Fc1c(ncc2c(nc(OC[C@@H]3CCCN3Cc3ccccc3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@H]4CCCN4Cc4ccccc4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OCc4cccnc4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN(C)C(=O)CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Cc1cccc2cccc(-c3ncc4c(nc(OCCc5nccn5C)nc4c3F)N3CC4CCC(C3)N4)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)c(Br)c2ccccc12 |r|
Cc1cccc2cccc(-c3ncc4c(nc(OCCc5cccnc5)nc4c3F)N3CC4CCC(C3)N4)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C)c12 |r|
Oc1cc(-c2ncc3c(nc(OCCc4ccc(F)cn4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN1C[C@H](F)C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Clc1cccc2cccc(-c3ccc4c(nc(OCCCN5C[C@@H]6C[C@H]5CO6)nc4c3)N3CC4CCC(C3)N4)c12 |r|
C[C@H](CN(C)C)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Cn1ccnc1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CN(C)CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccc(F)cc12 |r|
Oc1cc(-c2ncc3c(nc(OCCc4cccnc4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccccc12 |r|
CN(C)CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2CCCCc12 |r|
Fc1c(ncc2c(nc(OC[C@@H]3CCCN3Cc3ccccc3)nc12)N1CC2CCC(C1)N2)-c1cccc2ccccc12 |r|
Oc1cc(-c2ncc3c(nc(OCCCN4CCOCC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2CCCc12 |r|
Cn1cncc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Oc1cc(-c2ncc3c(nc(OCCCN4C[C@@H]5CC4CO5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Cn1cncc1CCNc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Oc1cc(-c2ncc3c(nc(OCCN4CCOCC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Cn1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccc(F)cc12
Oc1cc(-c2ncc3c(nc(OCCN4C[C@@H]5CC4CO5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Fc1c(ncc2c(nc(OCCc3cccnc3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CC(Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12)C1CCCN1C
Cn1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12)C(F)(F)F |r|
CN1C[C@H](F)C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CC(C)N1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(cc2n1)-c1cccc2cccc(C)c12 |r|
CC1C(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)=Nc2ccccc12 |c:41|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(cc2n1)-c1cccc2cccc(CCC#N)c12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Oc1cc(-c2ncc3c(nc(nc3c2F)N2CCCC2)N2CC3CCC(C2)N3)c2ccccc2c1
CO[C@@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
Oc1cc(-c2ncc3c(nc(nc3c2F)N2CCC2)N2CC3CCC(C2)N3)c2ccccc2c1
OCC(CO)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN(C)C1CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
OC1CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
OC[C@@H]1CCN1c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Oc1cc(-c2ncc3c(nc(OCCCC(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN(C)C1CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
COCCN1CCC(CC1)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccccc12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(cc2n1)-c1cccc2cccc(Cl)c12 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@H]4CC5CCN4C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r,THB:12:13:19:17.16|
CC1(N)CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
COCCCN1CCC(CC1)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CCC1(N)CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CO[C@@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)N(C)C1 |r|
CN(C)C1(C)CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CCO[C@@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
CN1CC(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)CC1=O
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccc(F)c(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CC1CCCc2cccc(-c3ncc4c(nc(OC[C@@H]5CCCN5C)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Oc1cc(-c2ncc3c(nc(OCC4(CCCC4)C(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Nc1cccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)n1
Oc1cc(-c2ncc3c(nc(OCC(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
COc1cccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
O[C@@H]1CC2CN(C[C@H]1N2)c1nc(OCC23CCCN2CCC3)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OC3CCc4[nH]ncc4C3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Oc1cc(-c2ncc3c(nc(OC[C@@H]4CCCN4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Fc1c(ncc2c(nc(OC3CCc4cn[nH]c4C3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Oc1cc(-c2ncc3c(nc(OCC4(CC4)C(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Fc1c(ncc2c(nc(OCCn3cccn3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Oc1cc(-c2ncc3c(nc(OCC(F)(F)C(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN1CCCC1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cncc2cccc(Cl)c12
Fc1c(ncc2c(nc(OCC3COC3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CC(C)N1CCC[C@H]1COc1nc(N2C[C@H]3C[C@@H](O)C(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C)(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
OC[C@H](O)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(CCC#N)(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
OC[C@@H](O)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
OCC(O)CCOc1nc(C2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(Cl)(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
OCC[C@@H](CO)Oc1nc(C2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2CCC(C)(C)c12 |r|
OCC(COc1nc(C2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)c1cccnc1
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2CCC3(CC3)c12 |r|
[O-][N+]12CCCC1(COc1nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n1)-c1cccc3cccc(Cl)c13)CCC2 |(8,-3.08,;6.67,-2.31,;6.35,-3.82,;4.82,-3.98,;4.19,-2.57,;5.33,-1.54,;4,-.77,;2.67,-1.54,;1.33,-.77,;1.33,.77,;,1.54,;,3.08,;-1.33,3.85,;-1.33,5.39,;-.74,4.48,;.74,4.48,;1.33,5.39,;1.33,3.85,;,6.16,;-1.33,.77,;-2.67,1.54,;-4,.77,;-4,-.77,;-2.67,-1.54,;-2.67,-3.08,;-1.33,-.77,;,-1.54,;-5.33,-1.54,;-6.67,-.77,;-8,-1.54,;-8,-3.08,;-6.67,-3.85,;-6.67,-5.39,;-5.33,-6.16,;-4,-5.39,;-4,-3.85,;-2.67,-4.62,;-5.33,-3.08,;5.65,-.03,;7.19,.13,;7.81,-1.28,)|
Cn1ccnc1CCOc1nc(N2C[C@H]3C[C@@H](O)[C@@H](C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
OC(=O)CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CC1CCc2cccc(c12)-c1ncc2c(nc(OC[C@@H]3CCCN3C)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1cc(-c2ncc3c(nc(OCCc4ccccc4F)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(C#C)c12
COCCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(cccc2c1)C#C
OCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(C)c2n1)-c1cc(O)cc2ccccc12 |r|
COCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)(N3)C=O)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Oc1cc(-c2ncc3c(nc(OC4CCS(=O)(=O)CC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN1CCC[C@H]1COc1nc(N2CC3CCC(CO)(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Oc1cc(-c2ncc3c(nc(OC4CCOCC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OCC4CCCC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OCc4ccccc4F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(nc3c2F)N2CC3(C2)CCOCC3)N2CC3CCC(C2)N3)c2ccccc2c1
CO[C@@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
OCCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Cc1cccc(F)c1-c1ncc2c(nc(OCCc3nccn3C)nc2c1F)N1CC2CCC(C1)N2 |(-4.55,-5,;-5.89,-4.23,;-7.22,-5,;-8.55,-4.23,;-8.55,-2.69,;-7.22,-1.93,;-7.22,-.38,;-5.89,-2.69,;-4.55,-1.93,;-4.55,-.38,;-3.22,.38,;-1.89,-.38,;-.55,.38,;.78,-.38,;.78,-1.93,;2.12,-2.69,;3.45,-1.93,;4.78,-2.69,;6.12,-1.93,;7.52,-2.55,;8.55,-1.41,;7.78,-.07,;6.28,-.39,;5.13,.64,;-.55,-2.69,;-1.89,-1.93,;-3.22,-2.69,;-3.22,-4.23,;-.55,1.93,;-1.89,2.69,;-1.89,4.23,;-1.12,3.26,;.01,3.26,;.78,4.23,;.78,2.69,;-.55,5,)|
Oc1cc(-c2ncc3c(nc(nc3c2F)N2CC3(C2)CCOC3)N2CC3CCC(C2)N3)c2ccccc2c1
COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C)c12
OC[C@@H]1CCCN1c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2C(O)CCc12 |r|
CC(=O)N1CCC(CC1)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CCOC(=O)CCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
Oc1cc(-c2ncc3c(nc(OC4CCSCC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1ccc(CCCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)cc1C=O
Oc1cc(-c2ncc3c(nc(OC4CCC(F)(F)CC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2C[C@H]3C[C@@H](CC#N)[C@@H](C2)N3)c2ccccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OCCC(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OC[C@@]23CCCN2C[C@H](F)C3)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
Oc1cc(-c2ncc3c(nc(OC4CCS(=O)CC4)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CC(F)C(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
Cc1nccn1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CO[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OC[C@@]23CCCN2C[C@H](F)C3)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
CC(C)Cn1ccnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Br)c12
COc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Oc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
OCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
OCCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
NC(=O)Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
NCC#Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
CCC#Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(cccc2c1)C#C |r|
Oc1cc(-c2ncc3c(ncnc3c2F)N2CC3CCC(C2)N3)c2c(cccc2c1)C#C
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)c(F)ccc2c1
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(F)c(F)ccc2c1 |r|
FC(F)Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
FCCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Cc1cc2[nH]ncc2c(c1C)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-6,-5.77,;-6,-4.24,;-7.34,-3.47,;-7.34,-1.93,;-8.48,-.89,;-7.85,.51,;-6.32,.35,;-6,-1.16,;-4.67,-1.93,;-4.67,-3.47,;-3.33,-4.24,;-3.33,-1.16,;-3.33,.38,;-2,1.15,;-.67,.38,;.67,1.15,;2,.38,;2,-1.16,;3.33,-1.93,;4.67,-1.16,;6,-1.93,;6.32,-.42,;7.85,-.26,;8.48,-1.66,;7.34,-2.7,;7.02,-4.2,;5.48,-4.36,;4.86,-2.96,;.67,-1.93,;-.67,-1.16,;-2,-1.93,;-2,-3.47,;.67,2.69,;-.67,3.46,;-.67,5,;-.02,4.08,;1.33,4.08,;2,5,;2,3.46,;.67,5.77,)|
Cc1cc2[nH]ccc2c(c1C)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-8.57,-1.09,;-7.24,-1.86,;-7.24,-3.4,;-5.91,-4.17,;-5.59,-5.68,;-4.06,-5.84,;-3.43,-4.43,;-4.57,-3.4,;-4.57,-1.86,;-5.91,-1.09,;-5.91,.45,;-3.24,-1.09,;-3.24,.45,;-1.91,1.22,;-.57,.45,;.76,1.22,;2.1,.45,;2.1,-1.09,;3.43,-1.86,;4.76,-1.09,;6.1,-1.86,;6.42,-.36,;7.95,-.19,;8.57,-1.6,;7.43,-2.63,;7.11,-4.14,;5.58,-4.3,;4.95,-2.89,;.76,-1.86,;-.57,-1.09,;-1.91,-1.86,;-1.91,-3.4,;.76,2.76,;-.57,3.53,;-.57,5.07,;.08,4.14,;1.42,4.14,;2.1,5.07,;2.1,3.53,;.76,5.84,)|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CCCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
FCCCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Cc1ccc(O)cc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1c2cn[nH]c2cc2ccccc12 |(-2,-3.08,;-2,-1.54,;-3.33,-.77,;-3.33,.77,;-2,1.54,;-.67,.77,;.67,1.54,;2,.77,;2,-.77,;3.33,-1.54,;4.67,-.77,;6,-1.54,;4.86,-2.57,;5.48,-3.98,;7.02,-3.82,;7.34,-2.31,;8.48,-1.28,;7.85,.13,;6.32,-.03,;.67,-1.54,;-.67,-.77,;.67,3.08,;-.67,3.85,;-.67,5.39,;-.02,4.34,;1.36,4.34,;2,5.39,;2,3.85,;.67,6.16,;-4.67,-1.54,;-6,-.77,;-6.32,.74,;-7.85,.9,;-8.48,-.51,;-7.34,-1.54,;-7.34,-3.08,;-6,-3.85,;-6,-5.39,;-4.67,-6.16,;-3.33,-5.39,;-3.33,-3.85,;-4.67,-3.08,)|
CN1CCC[C@H]1COc1nc(N2CC3C[C@@H](O)C(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1c(OC(F)(F)F)ccc2[nH]ncc12 |(-2,-2.69,;-2,-1.15,;-3.33,-.38,;-3.33,1.15,;-2,1.93,;-.67,1.15,;.67,1.93,;2,1.15,;2,-.38,;3.33,-1.15,;4.67,-.38,;6,-1.15,;4.86,-2.19,;5.48,-3.59,;7.02,-3.43,;7.34,-1.93,;8.48,-.89,;7.85,.51,;6.32,.35,;.67,-1.15,;-.67,-.38,;.67,3.47,;-.67,4.23,;-.67,5.78,;-.02,4.72,;1.36,4.72,;2,5.78,;2,4.23,;.67,6.54,;-4.67,-1.15,;-4.67,-2.69,;-3.33,-3.47,;-3.33,-5,;-2,-5.78,;-4.67,-5.78,;-3.33,-6.54,;-6,-3.47,;-7.34,-2.69,;-7.34,-1.15,;-8.48,-.12,;-7.85,1.28,;-6.32,1.12,;-6,-.38,)|
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCc2ccc(F)cn2)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
CCc1cccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)OC(=O)NCCOCc1ccc(O)cc1 |r|
NCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
NC1(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)CCCCC1
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1
CCc1ccc(O)cc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Nc1cccc(F)c1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-6.57,-.32,;-6.57,-1.86,;-7.91,-2.63,;-7.91,-4.17,;-6.57,-4.94,;-5.24,-4.17,;-3.91,-4.94,;-5.24,-2.63,;-3.91,-1.86,;-3.91,-.32,;-2.57,.45,;-1.24,-.32,;.09,.45,;1.43,-.32,;1.43,-1.86,;2.76,-2.63,;4.1,-1.86,;5.43,-2.63,;4.28,-3.66,;4.91,-5.07,;6.44,-4.91,;6.76,-3.4,;7.91,-2.37,;7.28,-.96,;5.75,-1.13,;.09,-2.63,;-1.24,-1.86,;-2.57,-2.63,;-2.57,-4.17,;.09,1.99,;-1.24,2.76,;-1.24,4.3,;-.6,3.24,;.79,3.24,;1.43,4.3,;1.43,2.76,;.09,5.07,)|
Nc1c(Cl)cc(Cl)c(F)c1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-5.91,.38,;-5.91,-1.15,;-7.24,-1.93,;-8.57,-1.16,;-7.24,-3.47,;-5.91,-4.23,;-5.91,-5.78,;-4.57,-3.47,;-3.24,-4.23,;-4.57,-1.93,;-3.24,-1.15,;-3.24,.38,;-1.91,1.15,;-.57,.38,;.76,1.15,;2.1,.38,;2.1,-1.15,;3.43,-1.93,;4.76,-1.15,;6.1,-1.93,;4.95,-2.96,;5.58,-4.36,;7.11,-4.2,;7.43,-2.69,;8.57,-1.66,;7.95,-.26,;6.42,-.42,;.76,-1.93,;-.57,-1.15,;-1.91,-1.93,;-1.91,-3.47,;.76,2.69,;-.57,3.47,;-.57,5,;.07,3.95,;1.45,3.95,;2.1,5,;2.1,3.47,;.76,5.78,)|
Oc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CNc1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CCNc1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Nc1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Oc1cccc(c1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Cc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
COc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Cc1c(Cl)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Cc1cccc(c1C)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Cc1cccc(c1Cl)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc(Cl)c1Cl
Oc1ccc(CC#C)c(c1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
COCCNC(=O)O[C@@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(F)cccc2c1 |r|
Oc1cc(Cl)c(C2CC2)c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1cc(Cl)c(c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2)C(F)(F)F |r|
F[C@@H]1C[C@H]1c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |r|
C[C@@H]1C[C@@H]1c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |r|
C[C@H]1C[C@H]1c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |r|
C[C@@H]1C[C@H]1c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1ccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)cc1C=O
C[C@H]1C[C@@H]1c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2cccc(Cl)c12 |r|
CC(C)c1c(F)cc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CC(C)(C)[Si](C)(C)OCC1CCC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12
CC(C)c1c(Cl)cc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3C(CCl)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Fc1cccc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c1C(F)(F)F
Fc1c(ncc2c(nc(OC[C@@]34CCCN3C(CCl)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
FC(F)c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Cc1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CCc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CN(C)c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1ccccc1C1CC1
CC(C)c1c(Cl)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CC(C)c1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CCC(C)c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CC(C)c1c(C)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
FC(F)Oc1c(F)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
FC(F)Oc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1cccc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c1C1CC1
CC1(CC1)c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CC(C)c1ccncc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CC(C)c1ncccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CN(C)Cc1ccc(COCCNC(=O)O[C@@H]2C[C@@H](COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)N(C)C2)cc1 |r|
CC(C)c1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3C(=O)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1ccccc1Cl
COc1c(Cl)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CCc1c(Cl)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
COc1c(C)cccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
OCCc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3CC(F)(F)C4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccc(C)cc12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc(Cl)c1C1CC1
CN1CCCC1(CO)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2ccccc12
CCc1cccc2cncc(-c3ncc4c(nc(OCC56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Fc1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c2c1Cl
CC1(C)CN2C[C@H](F)CC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
Oc1cc(-c2ncc3c(nc(OC[C@]45CCCN4C[C@@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc(Cl)c1C(F)(F)F
CSc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Oc1cc(-c2ncc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1 |r|
Cc1ccc2[nH]ncc2c1-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wD:25.28,(-3.33,-4.27,;-4.67,-3.5,;-6,-4.27,;-7.34,-3.5,;-7.34,-1.96,;-8.48,-.93,;-7.85,.47,;-6.32,.31,;-6,-1.19,;-4.67,-1.96,;-3.33,-1.19,;-3.33,.35,;-2,1.12,;-.67,.35,;.67,1.12,;2,.35,;2,-1.19,;3.33,-1.96,;4.67,-1.19,;6,-1.96,;6.32,-.46,;7.85,-.3,;8.48,-1.7,;7.34,-2.73,;7.02,-4.24,;5.48,-4.4,;4.71,-5.74,;4.86,-2.99,;.67,-1.96,;-.67,-1.19,;-2,-1.96,;-2,-3.5,;.67,2.66,;-.67,3.43,;-.67,4.97,;-.03,4.12,;1.3,4.12,;2,4.97,;2,3.43,;.67,5.74,)|
Cc1ccc2[nH]ncc2c1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-3.33,-4.94,;-4.67,-4.17,;-6,-4.94,;-7.34,-4.17,;-7.34,-2.63,;-8.48,-1.6,;-7.85,-.19,;-6.32,-.36,;-6,-1.86,;-4.67,-2.63,;-3.33,-1.86,;-3.33,-.32,;-2,.45,;-.67,-.32,;.67,.45,;2,-.32,;2,-1.86,;3.33,-2.63,;4.67,-1.86,;6,-2.63,;4.86,-3.66,;5.48,-5.07,;7.02,-4.91,;7.34,-3.4,;8.48,-2.37,;7.85,-.96,;6.32,-1.13,;.67,-2.63,;-.67,-1.86,;-2,-2.63,;-2,-4.17,;.67,1.99,;-.67,2.76,;-.67,4.3,;-.03,3.45,;1.3,3.45,;2,4.3,;2,2.76,;.67,5.07,)|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3C[C@H](C(C2)N3)n2cncn2)c2ccccc2c1 |r|
Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(C3CC3)c12
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3ccc(F)c(Cl)c23)C1 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1c(Cl)c(O)cc2ccccc12 |r,wD:5.6,(5.13,-4.1,;6.28,-3.07,;7.78,-3.39,;8.55,-2.06,;7.52,-.91,;6.12,-1.54,;4.78,-.77,;3.45,-1.54,;2.12,-.77,;2.12,.77,;.78,1.54,;.78,3.08,;-.55,3.85,;-.55,5.39,;.09,4.54,;1.41,4.54,;2.12,5.39,;2.12,3.85,;.78,6.16,;-.55,.77,;-1.89,1.54,;-3.22,.77,;-3.22,-.77,;-1.89,-1.54,;-1.89,-3.08,;-.55,-.77,;.78,-1.54,;-4.55,-1.54,;-5.89,-.77,;-5.89,.77,;-7.22,-1.54,;-8.55,-.77,;-7.22,-3.08,;-5.89,-3.85,;-5.89,-5.39,;-4.55,-6.16,;-3.22,-5.39,;-3.22,-3.85,;-4.55,-3.08,)|
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2C[C@H]3C[C@@H](CC#N)[C@@H](C2)N3)c2ccccc2c1 |r|
Oc1ccc(OC(F)(F)F)c(c1)-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1ccc(OC(F)(F)F)c(c1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
F[C@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc(Cl)c2C2CC2)C1 |r|
F[C@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2c(ccc3[nH]ncc23)C(F)(F)F)C1 |r,wD:1.0,(4.71,-5.74,;5.48,-4.4,;7.02,-4.24,;7.34,-2.73,;8.48,-1.7,;7.85,-.3,;6.32,-.46,;6,-1.96,;4.67,-1.19,;3.33,-1.96,;2,-1.19,;2,.35,;.67,1.12,;.67,2.66,;-.67,3.43,;-.67,4.97,;-.02,4.2,;1.32,4.2,;2,4.97,;2,3.43,;.67,5.74,;-.67,.35,;-2,1.12,;-3.33,.35,;-3.33,-1.19,;-2,-1.96,;-2,-3.5,;-.67,-1.19,;.67,-1.96,;-4.67,-1.96,;-4.67,-3.5,;-6,-4.27,;-7.34,-3.5,;-7.34,-1.96,;-8.48,-.93,;-7.85,.47,;-6.32,.31,;-6,-1.19,;-3.33,-4.27,;-2,-5.04,;-2.56,-2.94,;-4.1,-5.61,;4.86,-2.99,)|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1c(ccc2[nH]ncc12)C(F)(F)F |(-2,-3.57,;-2,-2.03,;-3.33,-1.26,;-3.33,.28,;-2,1.05,;-.67,.28,;.67,1.05,;2,.28,;2,-1.26,;3.33,-2.03,;4.67,-1.26,;6,-2.03,;4.86,-3.06,;5.48,-4.47,;7.02,-4.3,;7.34,-2.8,;8.48,-1.77,;7.85,-.36,;6.32,-.52,;.67,-2.03,;-.67,-1.26,;.67,2.59,;-.67,3.36,;-.67,4.9,;-.02,4.14,;1.32,4.14,;2,4.9,;2,3.36,;.67,5.67,;-4.67,-2.03,;-4.67,-3.57,;-6,-4.34,;-7.34,-3.57,;-7.34,-2.03,;-8.48,-1,;-7.85,.41,;-6.32,.25,;-6,-1.26,;-3.33,-4.34,;-2,-5.11,;-2.56,-3,;-4.1,-5.67,)|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(OC(F)(F)F)c12
FC(F)Oc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
FCC1CCC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4ccccc34)CCCN12
CC(C)c1ccccc1-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1c(Cl)ccc2ccccc12 |(-2.57,-3.08,;-2.57,-1.54,;-3.91,-.77,;-3.91,.77,;-2.57,1.54,;-1.24,.77,;.09,1.54,;1.43,.77,;1.43,-.77,;2.76,-1.54,;4.1,-.77,;5.43,-1.54,;4.28,-2.57,;4.91,-3.98,;6.44,-3.82,;6.76,-2.31,;7.91,-1.28,;7.28,.13,;5.75,-.03,;.09,-1.54,;-1.24,-.77,;.09,3.08,;-1.24,3.85,;-1.24,5.39,;-.6,4.15,;.72,4.15,;1.43,5.39,;1.43,3.85,;.09,6.16,;-5.24,-1.54,;-6.57,-.77,;-6.57,.77,;-7.91,-1.54,;-7.91,-3.08,;-6.57,-3.85,;-6.57,-5.39,;-5.24,-6.16,;-3.91,-5.39,;-3.91,-3.85,;-5.24,-3.08,)|
Oc1c(F)cc(F)c(c1F)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-8.57,-1.86,;-7.24,-2.63,;-7.24,-4.17,;-8.57,-4.94,;-5.91,-4.94,;-4.57,-4.17,;-3.24,-4.94,;-4.57,-2.63,;-5.91,-1.86,;-5.91,-.32,;-3.24,-1.86,;-3.24,-.32,;-1.91,.45,;-.57,-.32,;.76,.45,;2.1,-.32,;2.1,-1.86,;3.43,-2.63,;4.76,-1.86,;6.1,-2.63,;4.95,-3.66,;5.58,-5.07,;7.11,-4.91,;7.43,-3.4,;8.57,-2.37,;7.95,-.96,;6.42,-1.13,;.76,-2.63,;-.57,-1.86,;-1.91,-2.63,;-1.91,-4.17,;.76,1.99,;-.57,2.76,;-.57,4.3,;.19,2.93,;1.27,2.93,;2.1,4.3,;2.1,2.76,;.76,5.07,)|
CO[C@H]1CN[C@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CC1(N)CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
Fc1c(ncc2c(nc(OC[C@@H]3CC(F)(F)CN3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)NC(=O)c1ccc(C=O)cc1 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)NC(=O)c1cccc(C=O)c1 |r|
CCC1(N)CN(C1)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)NC(=O)c1ccccc1C=O |r|
Fc1c(ncc2c(nc(OCCC3CC(F)(F)C3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CN1CC[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
Fc1c(ncc2c(nc(nc12)N1CC2(CCN2)C1)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CN1CC[C@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CN1CC[C@H](C1)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CN1CC[C@@H](C1)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2cccc(Cl)c12
COc1ccc(OC(F)(F)F)c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
OCC1CCC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12
CC(C)(C)c1ccccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1c(ncc2c(nc(OC[C@@H]3CCCO3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
CNC(C)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
Fc1c(ncc2c(nc(OC[C@H]3CCCO3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
CC(C)c1cccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CO[C@H](C)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
Cc1ccc(O)cc1-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(F)cccc2c1
Nc1ccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)cn1
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2ccccc2C2CC2)C1 |r|
Oc1cccc(F)c1-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wD:23.25,(-6.57,.35,;-6.57,-1.19,;-7.91,-1.96,;-7.91,-3.5,;-6.57,-4.27,;-5.24,-3.5,;-3.91,-4.27,;-5.24,-1.96,;-3.91,-1.19,;-3.91,.35,;-2.57,1.12,;-1.24,.35,;.09,1.12,;1.43,.35,;1.43,-1.19,;2.76,-1.96,;4.1,-1.19,;5.43,-1.96,;5.75,-.46,;7.28,-.3,;7.91,-1.7,;6.76,-2.73,;6.44,-4.24,;4.91,-4.4,;4.14,-5.74,;4.28,-2.99,;.09,-1.96,;-1.24,-1.19,;-2.57,-1.96,;-2.57,-3.5,;.09,2.66,;-1.24,3.43,;-1.24,4.97,;-.59,4.2,;.75,4.2,;1.43,4.97,;1.43,3.43,;.09,5.74,)|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1ccccc1C(F)(F)F
Cn1nccc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
F[C@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2ccccc2C2CCC2)C1 |r|
Cn1ccc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)n1
CSc1cccc2cc(O)cc(-c3ncc4c(nc(OCC56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Cn1cc(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)cn1
Oc1ccc(c(c1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2)C(F)(F)F
C[C@H](N)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
Cn1cnc2ccc(Oc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)cc12
Oc1ccc(c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2)C(F)(F)F |r|
CO[C@H]1CC(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
Cc1cc2[nH]ncc2c(c1Cl)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:20.21,wD:26.29,(-6,-5.78,;-6,-4.23,;-7.34,-3.47,;-7.34,-1.93,;-8.48,-.89,;-7.85,.51,;-6.32,.35,;-6,-1.15,;-4.67,-1.93,;-4.67,-3.47,;-3.33,-4.23,;-3.33,-1.15,;-3.33,.38,;-2,1.16,;-.67,.38,;.67,1.15,;2,.38,;2,-1.15,;3.33,-1.93,;4.67,-1.15,;6,-1.93,;6.32,-.42,;7.85,-.26,;8.48,-1.66,;7.34,-2.69,;7.02,-4.2,;5.48,-4.36,;4.71,-5.7,;4.86,-2.96,;.67,-1.93,;-.67,-1.15,;-2,-1.93,;-2,-3.47,;.67,2.69,;-.67,3.47,;-.67,5,;.1,3.67,;1.23,3.67,;2,5,;2,3.47,;.67,5.78,)|
Fc1c(ncc2c(nc(OCc3cccn4ccnc34)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Cc1cccc(O)c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:17.17,wD:23.25,(-3.91,-4.27,;-5.24,-3.5,;-6.57,-4.27,;-7.91,-3.5,;-7.91,-1.96,;-6.57,-1.19,;-6.57,.35,;-5.24,-1.96,;-3.91,-1.19,;-3.91,.35,;-2.57,1.12,;-1.24,.35,;.09,1.12,;1.43,.35,;1.43,-1.19,;2.76,-1.96,;4.1,-1.19,;5.43,-1.96,;5.75,-.46,;7.28,-.3,;7.91,-1.7,;6.76,-2.73,;6.44,-4.24,;4.91,-4.4,;4.14,-5.74,;4.28,-2.99,;.09,-1.96,;-1.24,-1.19,;-2.57,-1.96,;-2.57,-3.5,;.09,2.66,;-1.24,3.43,;-1.24,4.97,;-.6,4.06,;.78,4.06,;1.43,4.97,;1.43,3.43,;.09,5.74,)|
CN1CCc2cccc(Oc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)c2C1
O[C@@H]1C[C@@H]2CN(CC1N2)c1nc(nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12)N1CCC1 |r|
Fc1c(ncc2c(nc(OC[C@@]34CCCN3CC[C@@H]4C#N)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Nc1ccc(Cl)c(F)c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:18.18,wD:24.26,(-6.57,.38,;-6.57,-1.15,;-7.91,-1.93,;-7.91,-3.47,;-6.57,-4.23,;-6.57,-5.78,;-5.24,-3.47,;-3.91,-4.23,;-5.24,-1.93,;-3.91,-1.15,;-3.91,.38,;-2.57,1.16,;-1.24,.38,;.09,1.15,;1.43,.38,;1.43,-1.15,;2.76,-1.93,;4.1,-1.15,;5.43,-1.93,;5.75,-.42,;7.28,-.26,;7.91,-1.66,;6.76,-2.69,;6.44,-4.2,;4.91,-4.36,;4.14,-5.7,;4.28,-2.96,;.09,-1.93,;-1.24,-1.15,;-2.57,-1.93,;-2.57,-3.47,;.09,2.69,;-1.24,3.47,;-1.24,5,;-.47,3.67,;.66,3.67,;1.43,5,;1.43,3.47,;.09,5.78,)|
Cn1cnnc1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CCc1c(F)ccc2cccc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
O[C@@H]1C[C@@H]2CN(CC1N2)c1nc(OCCC(F)(F)F)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OC[C@@]34CCCN3C[C@H](C4)C(F)(F)F)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2ccccc2CC(F)(F)F)C1 |r|
Oc1cc(-c2ncc3c(nc(OCC45CCCN4C(CF)CC5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
COc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)(N3)C(N)=O)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
Oc1ccc(SC(F)(F)F)c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CC(C)(N)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
COC1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3cccc(F)c23)C1
COC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cc(O)cc4ccccc34)CCCN12 |r|
Fc1c(ncc2c(nc(OC3CCN(CC3)C(=O)CCl)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
COC(c1ccc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2)C(F)(F)F |r|
Fc1c(ncc2c(nc(OCCNC(=O)c3ccc(cc3)S(F)(=O)=O)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
Cc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2cn[nH]c2c1 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)NC(=O)c1ccc(cc1)S(F)(=O)=O |r|
Oc1cccc(OC(F)(F)F)c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:21.21,wD:27.29,(-6.57,1.15,;-6.57,-.39,;-7.91,-1.16,;-7.91,-2.7,;-6.57,-3.47,;-5.24,-2.7,;-3.91,-3.46,;-3.91,-5,;-2.57,-5.77,;-5.24,-5.77,;-3.91,-6.54,;-5.24,-1.16,;-3.91,-.39,;-3.91,1.15,;-2.57,1.93,;-1.24,1.15,;.09,1.92,;1.43,1.15,;1.43,-.39,;2.76,-1.16,;4.1,-.39,;5.43,-1.16,;5.75,.35,;7.28,.51,;7.91,-.89,;6.76,-1.93,;6.44,-3.43,;4.91,-3.59,;4.14,-4.93,;4.28,-2.19,;.09,-1.16,;-1.24,-.39,;-2.57,-1.16,;-2.57,-2.7,;.09,3.46,;-1.24,4.23,;-1.24,5.77,;-.47,4.44,;.66,4.44,;1.43,5.77,;1.43,4.23,;.09,6.54,)|
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCc2nccn2C(F)F)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
Oc1cc(-c2ncc3c(nc(OCCC(F)(F)F)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1
Cc1nccn1CCOc1nc(N2C[C@H]3C[C@@H](O)[C@@H](C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
CC(C)c1cccc(C(C)C)c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:21.21,wD:27.29,(-2.57,-5.03,;-3.91,-4.26,;-4.3,-5.75,;-5.24,-3.49,;-6.57,-4.26,;-7.91,-3.49,;-7.91,-1.95,;-6.57,-1.18,;-6.57,.36,;-7.91,1.13,;-5.24,1.13,;-5.24,-1.95,;-3.91,-1.18,;-3.91,.36,;-2.57,1.13,;-1.24,.36,;.09,1.13,;1.43,.36,;1.43,-1.18,;2.76,-1.95,;4.1,-1.18,;5.43,-1.95,;5.75,-.44,;7.28,-.28,;7.91,-1.69,;6.76,-2.72,;6.44,-4.23,;4.91,-4.39,;4.14,-5.72,;4.28,-2.98,;.09,-1.95,;-1.24,-1.18,;-2.57,-1.95,;-2.57,-3.49,;.09,2.67,;-1.24,3.44,;-1.24,4.98,;-.47,3.65,;.66,3.65,;1.43,4.98,;1.43,3.44,;.09,5.75,)|
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCn2ccnc2CF)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCn2ccnc2C(F)(F)F)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCc2nccn2CF)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
OCc1nccn1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN1CCC(F)(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)CC1
O[C@@H]1C[C@@H]2CN(C[C@H]1N2)c1nc(OCCn2ccnc2C(F)F)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
CC(C)c1ccc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Oc1cc(-c2ncc3c(nc(OCC45CCCN4C(CF)CC5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1
Cc1c(Cl)cc2[nH]ncc2c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:20.21,wD:26.29,(-3.33,-4.23,;-4.67,-3.47,;-6,-4.23,;-6,-5.78,;-7.34,-3.47,;-7.34,-1.93,;-8.48,-.89,;-7.85,.51,;-6.32,.35,;-6,-1.15,;-4.67,-1.93,;-3.33,-1.15,;-3.33,.38,;-2,1.16,;-.67,.38,;.67,1.15,;2,.38,;2,-1.15,;3.33,-1.93,;4.67,-1.15,;6,-1.93,;6.32,-.42,;7.85,-.26,;8.48,-1.66,;7.34,-2.69,;7.02,-4.2,;5.48,-4.36,;4.71,-5.7,;4.86,-2.96,;.67,-1.93,;-.67,-1.15,;-2,-1.93,;-2,-3.47,;.67,2.69,;-.67,3.47,;-.67,5,;.1,3.67,;1.23,3.67,;2,5,;2,3.47,;.67,5.78,)|
Cc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(Cl)cccc2c1
CC(C)(O)c1ccccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
NC(=N)NCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CC(C)c1ccc(O)cc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
NC(=N)NCCCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
COC1(CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1)OC
Nc1nccn1CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
CN(C)C(=O)OC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
CO[C@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3cccc(F)c23)C1 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(-c3c[nH]nn3)c12
CC(C)(F)c1ccccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,TLB:14:32:39:35.36|
Oc1cc(-c2ncc3c(ncnc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CNC(=O)OC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
Nc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2ccccc2C#N)C1 |r|
CNc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
CO[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3cccc(C#C)c23)C1 |r|
CN(C)c1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
COC(=O)NC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
CN(C)C(=O)NC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2ccccc12
CC(=O)NC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
CCc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2ccccc2Cl)C1 |r|
Fc1c(ncc2c(ncnc12)N1CC2CCC(C1)N2)-c1cccc2cccc(C#C)c12
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cnccc2C(F)(F)F)C1 |r|
Fc1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c2c1C#C
CC(C)Oc1ccccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CC(C)Cc1ccccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(Cl)c2n1)-c1cc(O)cc2ccccc12 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](Cn3cccn3)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C#N)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(c23)C(F)(F)F)C1 |r|
OCC#Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
CS(=O)(=O)NC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C#CCO)c12 |r|
CC(C)c1ncccc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CC#Cc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2CCC=C(c12)C(F)(F)F |c:42|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2OC(F)(F)Oc12
COCc1cccc2cccc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc(c1C(F)(F)F)C(F)(F)F
Oc1ccc(CC(F)(F)F)c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(C#N)c12
FC1CN2CC(F)CC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1
CSc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
CCc1c(F)ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Fc1c(ncc2c(nc(OCC34CCCN3CCOC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12
CCn1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C=C)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3CCCc23)C1 |r|
COCCO[C@@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
CC1CCc2cccc(c12)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
F[C@@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cncc3cccc(Cl)c23)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3ccc(F)c(F)c23)C1 |r|
F[C@@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cncc3cccc(C#C)c23)C1 |r|
CCc1cccc2cccc(-c3ncc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCOCC5)CC6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
F[C@@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(C#C)c23)C1 |r|
CCc1cccc2cccc(-c3ncc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)NC)CC6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(C#C)c12 |r|
CCc1cccc2cc(O)cc(-c3ncc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)NC)CC6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cc(C)ccc12 |r|
CCc1cccc2cc(O)cc(-c3ncc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)N(C)C)CC6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)Oc1cccc(c1)S(F)(=O)=O |r|
CNC(=O)O[C@@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)Oc1ccc(cc1)S(F)(=O)=O |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3C[C@H](C4)OC(=O)N3CCOCC3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
CN1CC[C@H](Oc2cccc(c2)S(F)(=O)=O)[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3CCC(C4CC4)c23)C1 |r|
CN1C[C@@H](C[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)NC(=O)c1cccc(c1)S(F)(=O)=O |r|
F[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3C4CC4Cc23)C1 |r|
Oc1cc(-c2ncc3c(nc(OCCNC(=O)c4ccc(cc4)S(F)(=O)=O)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN(C)C(=O)OC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4ccc(F)c(C#C)c34)CCCN12 |r|
Oc1cc(-c2ncc3c(nc(OCCNC(=O)c4cccc(c4)S(F)(=O)=O)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
CN(C)C(=O)OC[C@H]1CC[C@@]2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cc(O)cc4ccc(F)c(C#C)c34)CCCN12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)N(C)C)CC6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Fc1cccc2cccc(-c3ncc4c(nc(CCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](CN3CCOC3=O)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](COC(=O)N3CCCC3)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Cn1cc(cn1)[C@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](COC(=O)N3CCCCC3)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3C[C@@H](C4)c3ccccc3)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](COC(=O)N3CCOCC3)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
OCC12CCCN1CC(C2)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
Cn1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
O[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CCCc1ccccc1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
O[C@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CO[C@H]1CN2CCC[C@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CCc1cccc2cc(O)cc(-c3ncc4c(ncnc4c3F)N3CC4CCC(C3)N4)c12
F[C@H]1CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CC(Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(F)c12)C12CCCN1CCC2
C[C@H]1CN2CCC[C@@]2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1 |r|
CC1(C)CN2CCCC2(COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)C1
C[C@@H]1C[C@H]1c1c(Cl)cc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1ccccc1OC(F)(F)F
Nc1nc2c(cccc2s1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc(Cl)c1OC(F)(F)F
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2scnc12
COc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(cccc2c1)C#C
Nc1nc2c(ccc(F)c2s1)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2
Oc1cc(-c2ncc3c(nc(OCC45CCCN4CCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1
Cc1cc2sc(N)nc2c(c1C)-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-5.93,-5.78,;-5.93,-4.23,;-7.26,-3.47,;-7.26,-1.93,;-8.41,-.89,;-7.78,.51,;-8.55,1.85,;-6.25,.35,;-5.93,-1.15,;-4.6,-1.93,;-4.6,-3.47,;-3.26,-4.24,;-3.26,-1.15,;-3.26,.38,;-1.93,1.15,;-.6,.38,;.74,1.15,;2.07,.38,;2.07,-1.15,;3.41,-1.93,;4.74,-1.15,;6.07,-1.93,;4.93,-2.96,;5.56,-4.36,;7.09,-4.2,;7.41,-2.69,;8.55,-1.66,;7.93,-.26,;6.39,-.42,;.74,-1.93,;-.6,-1.15,;-1.93,-1.93,;-1.93,-3.47,;.74,2.69,;-.6,3.47,;-.6,5,;.17,3.67,;1.3,3.67,;2.07,5,;2.07,3.47,;.74,5.78,)|
C(Oc1nc(N2CC3CCC(C2)N3)c2cnc(cc2n1)-c1cccc2ccccc12)C12CCCN1CCC2
Cc1cc2sc(N)nc2c(c1C)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:27.30,wD:21.22,(-6,-5.78,;-6,-4.23,;-7.34,-3.47,;-7.34,-1.93,;-8.48,-.89,;-7.85,.51,;-8.62,1.85,;-6.32,.35,;-6,-1.15,;-4.67,-1.93,;-4.67,-3.47,;-3.33,-4.24,;-3.33,-1.15,;-3.33,.38,;-2,1.15,;-.67,.38,;.67,1.15,;2,.38,;2,-1.15,;3.33,-1.93,;4.67,-1.15,;6,-1.93,;4.86,-2.96,;5.48,-4.36,;7.02,-4.2,;7.34,-2.69,;8.48,-1.66,;7.85,-.26,;8.62,1.08,;6.32,-.42,;.67,-1.93,;-.67,-1.15,;-2,-1.93,;-2,-3.47,;.67,2.69,;-.67,3.47,;-.67,5,;.1,3.67,;1.23,3.67,;2,5,;2,3.47,;.67,5.78,)|
Fc1cccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c12
Cc1ccc2sc(N)nc2c1-c1ncc2c(nc(OCC34CCCN3CCC4)nc2c1F)N1CC2CCC(C1)N2 |(-3.26,-4.94,;-4.6,-4.17,;-5.93,-4.94,;-7.26,-4.17,;-7.26,-2.63,;-8.41,-1.6,;-7.78,-.19,;-8.55,1.14,;-6.25,-.36,;-5.93,-1.86,;-4.6,-2.63,;-3.26,-1.86,;-3.26,-.32,;-1.93,.45,;-.6,-.32,;.74,.45,;2.07,-.32,;2.07,-1.86,;3.41,-2.63,;4.74,-1.86,;6.07,-2.63,;4.93,-3.66,;5.56,-5.07,;7.09,-4.91,;7.41,-3.4,;8.55,-2.37,;7.93,-.96,;6.39,-1.13,;.74,-2.63,;-.6,-1.86,;-1.93,-2.63,;-1.93,-4.17,;.74,1.99,;-.6,2.76,;-.6,4.3,;.17,2.97,;1.3,2.97,;2.07,4.3,;2.07,2.76,;.74,5.07,)|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(O)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccc(CN2CC[C@@H](O)C2)cc1 |r|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(N)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccccc1CCOC |r,wU:21.40,39.47,wD:13.18,47.51,(-7.19,-7.73,;-7.96,-6.4,;-7.19,-5.06,;-8.09,-3.82,;-7.19,-2.57,;-7.19,-1.03,;-5.85,-.26,;-4.37,.14,;-4.76,-1.35,;-5.71,1.57,;-4.37,2.34,;-4.37,3.88,;-5.71,4.65,;-3.04,4.65,;-3.04,6.19,;-1.71,6.96,;-.37,6.19,;-.37,4.65,;-1.71,3.88,;.96,3.88,;2.29,4.65,;.96,2.34,;-.37,1.57,;-.37,.03,;.96,-.74,;.96,-2.28,;2.29,-3.05,;-.37,-3.05,;-1.71,-2.28,;-1.71,-.74,;-3.05,-3.05,;-3.05,-4.59,;-4.39,-5.36,;-5.72,-4.59,;-5.72,-3.05,;-4.39,-2.28,;2.29,1.57,;3.63,2.34,;3.63,3.88,;4.96,1.57,;4.96,.03,;6.29,-.74,;3.63,-.74,;6.29,2.34,;6.29,3.88,;7.63,1.57,;7.63,.03,;8.96,2.34,;10.43,1.86,;11.33,3.11,;10.43,4.36,;8.96,3.88,;10.83,5.84,;9.74,6.93,;12.31,6.24,;12.71,7.73,;-9.63,-3.82,;-10.4,-5.15,;-11.94,-5.15,;-12.71,-3.82,;-11.94,-2.48,;-10.4,-2.48,;-9.63,-1.15,;-10.4,.19,;-9.63,1.52,;-10.4,2.85,)|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(O)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccc(CN(C)C)cc1 |r|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(O)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccccc1CO |r,wU:21.40,39.47,wD:13.18,47.51,(-7.19,-7.73,;-7.96,-6.4,;-7.19,-5.06,;-8.09,-3.82,;-7.19,-2.57,;-7.19,-1.03,;-5.85,-.26,;-4.37,.14,;-4.76,-1.35,;-5.71,1.57,;-4.37,2.34,;-4.37,3.88,;-5.71,4.65,;-3.04,4.65,;-3.04,6.19,;-1.71,6.96,;-.37,6.19,;-.37,4.65,;-1.71,3.88,;.96,3.88,;2.29,4.65,;.96,2.34,;-.37,1.57,;-.37,.03,;.96,-.74,;.96,-2.28,;2.29,-3.05,;-.37,-3.05,;-1.71,-2.28,;-1.71,-.74,;-3.05,-3.05,;-3.05,-4.59,;-4.39,-5.36,;-5.72,-4.59,;-5.72,-3.05,;-4.39,-2.28,;2.29,1.57,;3.63,2.34,;3.63,3.88,;4.96,1.57,;4.96,.03,;6.29,-.74,;3.63,-.74,;6.29,2.34,;6.29,3.88,;7.63,1.57,;7.63,.03,;8.96,2.34,;10.43,1.86,;11.33,3.11,;10.43,4.36,;8.96,3.88,;10.83,5.84,;9.74,6.93,;12.31,6.24,;12.71,7.73,;-9.63,-3.82,;-10.4,-5.15,;-11.94,-5.15,;-12.71,-3.82,;-11.94,-2.48,;-10.4,-2.48,;-9.63,-1.15,;-10.4,.19,)|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(O)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccccc1CN(C)C |r,wU:21.40,39.47,wD:13.18,47.51,(-7.19,-7.73,;-7.96,-6.4,;-7.19,-5.06,;-8.09,-3.82,;-7.19,-2.57,;-7.19,-1.03,;-5.85,-.26,;-4.37,.14,;-4.76,-1.35,;-5.71,1.57,;-4.37,2.34,;-4.37,3.88,;-5.71,4.65,;-3.04,4.65,;-3.04,6.19,;-1.71,6.96,;-.37,6.19,;-.37,4.65,;-1.71,3.88,;.96,3.88,;2.29,4.65,;.96,2.34,;-.37,1.57,;-.37,.03,;.96,-.74,;.96,-2.28,;2.29,-3.05,;-.37,-3.05,;-1.71,-2.28,;-1.71,-.74,;-3.05,-3.05,;-3.05,-4.59,;-4.39,-5.36,;-5.72,-4.59,;-5.72,-3.05,;-4.39,-2.28,;2.29,1.57,;3.63,2.34,;3.63,3.88,;4.96,1.57,;4.96,.03,;6.29,-.74,;3.63,-.74,;6.29,2.34,;6.29,3.88,;7.63,1.57,;7.63,.03,;8.96,2.34,;10.43,1.86,;11.33,3.11,;10.43,4.36,;8.96,3.88,;10.83,5.84,;9.74,6.93,;12.31,6.24,;12.71,7.73,;-9.63,-3.82,;-10.4,-5.15,;-11.94,-5.15,;-12.71,-3.82,;-11.94,-2.48,;-10.4,-2.48,;-9.63,-1.15,;-10.4,.19,;-11.94,.19,;-9.63,1.52,)|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(O)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C1CCOCC1)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccccc1CCOC |r,wU:21.40,39.51,wD:13.18,50.55,(-7.19,-7.73,;-7.96,-6.4,;-7.19,-5.06,;-8.09,-3.82,;-7.19,-2.57,;-7.19,-1.03,;-5.85,-.26,;-4.37,.14,;-4.76,-1.35,;-5.71,1.57,;-4.37,2.34,;-4.37,3.88,;-5.71,4.65,;-3.04,4.65,;-3.04,6.19,;-1.71,6.96,;-.37,6.19,;-.37,4.65,;-1.71,3.88,;.96,3.88,;2.29,4.65,;.96,2.34,;-.37,1.57,;-.37,.03,;.96,-.74,;.96,-2.28,;2.29,-3.05,;-.37,-3.05,;-1.71,-2.28,;-1.71,-.74,;-3.05,-3.05,;-3.05,-4.59,;-4.39,-5.36,;-5.72,-4.59,;-5.72,-3.05,;-4.39,-2.28,;2.29,1.57,;3.63,2.34,;3.63,3.88,;4.96,1.57,;4.96,.03,;3.87,-1.06,;4.27,-2.55,;5.76,-2.95,;6.85,-1.86,;6.45,-.37,;6.29,2.34,;6.29,3.88,;7.63,1.57,;7.63,.03,;8.96,2.34,;10.43,1.86,;11.33,3.11,;10.43,4.36,;8.96,3.88,;10.83,5.84,;9.74,6.93,;12.31,6.24,;12.71,7.73,;-9.63,-3.82,;-10.4,-5.15,;-11.94,-5.15,;-12.71,-3.82,;-11.94,-2.48,;-10.4,-2.48,;-9.63,-1.15,;-10.4,.19,;-9.63,1.52,;-10.4,2.85,)|
CCn1c(c2CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C(=O)[C@H](Cc3cc(OC(=O)CCN4CCN(C)CC4)cc(c3)-c3ccc1c2c3)NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C1)C(=O)C=C)-c1ccccc1CCOC |r,wU:21.52,50.59,wD:13.18,58.63,(-7.19,-7.73,;-7.96,-6.4,;-7.19,-5.06,;-8.09,-3.82,;-7.19,-2.57,;-7.19,-1.03,;-5.85,-.26,;-4.37,.14,;-4.76,-1.35,;-5.71,1.57,;-4.37,2.34,;-4.37,3.88,;-5.71,4.65,;-3.04,4.65,;-3.04,6.19,;-1.71,6.96,;-.37,6.19,;-.37,4.65,;-1.71,3.88,;.96,3.88,;2.29,4.65,;.96,2.34,;-.37,1.57,;-.37,.03,;.96,-.74,;.96,-2.28,;2.29,-3.05,;2.29,-4.59,;.96,-5.36,;3.63,-5.36,;4.96,-4.59,;6.29,-5.36,;6.29,-6.9,;7.63,-7.67,;8.96,-6.9,;10.3,-7.67,;8.96,-5.36,;7.63,-4.59,;-.37,-3.05,;-1.71,-2.28,;-1.71,-.74,;-3.05,-3.05,;-3.05,-4.59,;-4.39,-5.36,;-5.72,-4.59,;-5.72,-3.05,;-4.39,-2.28,;2.29,1.57,;3.63,2.34,;3.63,3.88,;4.96,1.57,;4.96,.03,;6.29,-.74,;3.63,-.74,;6.29,2.34,;6.29,3.88,;7.63,1.57,;7.63,.03,;8.96,2.34,;10.43,1.86,;11.33,3.11,;10.43,4.36,;8.96,3.88,;10.83,5.84,;9.74,6.93,;12.31,6.24,;12.71,7.73,;-9.63,-3.82,;-10.4,-5.15,;-11.94,-5.15,;-12.71,-3.82,;-11.94,-2.48,;-10.4,-2.48,;-9.63,-1.15,;-10.4,.19,;-9.63,1.52,;-10.4,2.85,)|
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Fc1c(ncc2c(nc(OCCCN3C[C@@H]4C[C@H]3CO4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Oc1cc(-c2ncc3c(nc(OCCCN4C[C@@H]5C[C@H]4CO5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Cn1ccnc1CCNc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cc(O)cc2ccccc12
Oc1cc(-c2ncc3c(nc(OCCN4C[C@@H]5C[C@H]4CO5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Cn1c(CCOc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cc(O)cc3ccccc23)nc2ccccc12
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(CCC#N)c12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cncc2cccc(Cl)c12
O[C@@H]1C[C@@H]2CN(CC1N2)c1nc(OCC23CCCN2CCC3)nc2c(F)c(ncc12)-c1cccc2cccc(Cl)c12 |r|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cncc2cccc(Cl)c12 |r|
CC(C)N1CCC[C@H]1COc1nc(N2C[C@H]3CC(O)C(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
C[C@H](CO)COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
OCC(O)CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
OCC[C@@H](CO)Oc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12 |r|
OCC(COc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12)c1cccnc1
O[N+]12CCCC1(COc1nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n1)-c1cccc3cccc(Cl)c13)CCC2 |(7.96,-3.22,;6.62,-2.45,;6.15,-3.91,;4.61,-3.91,;4.13,-2.45,;5.38,-1.54,;4.04,-.77,;2.71,-1.54,;1.38,-.77,;1.38,.77,;.04,1.54,;.04,3.08,;-1.29,3.85,;-1.29,5.39,;-.52,4.06,;.61,4.06,;1.38,5.39,;1.38,3.85,;.04,6.16,;-1.29,.77,;-2.62,1.54,;-3.96,.77,;-3.96,-.77,;-2.62,-1.54,;-2.62,-3.08,;-1.29,-.77,;.04,-1.54,;-5.29,-1.54,;-6.62,-.77,;-7.96,-1.54,;-7.96,-3.08,;-6.62,-3.85,;-6.62,-5.39,;-5.29,-6.16,;-3.96,-5.39,;-3.96,-3.85,;-2.62,-4.62,;-5.29,-3.08,;5.85,-.08,;7.39,-.08,;7.87,-1.54,)|
Oc1cc(-c2ncc3c(nc(OCCc4ccccc4F)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
FCC1CCC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(c(F)c4n3)-c3cccc4cccc(Cl)c34)CCCN12
Cc1ccc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
CCOc1nc(N2CC3CCC(C2)N3)c2cnc(c(F)c2n1)-c1cccc2cccc(Cl)c12
Oc1ccc(c(c1)-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2)C(F)(F)F |r|
Cc1cc2[nH]ncc2c(-c2ncc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c1C(F)(F)F |r,wD:24.26,(-6.01,-5.77,;-6.01,-4.24,;-7.34,-3.47,;-7.34,-1.93,;-8.49,-.89,;-7.86,.51,;-6.33,.35,;-6.01,-1.16,;-4.67,-1.92,;-3.34,-1.16,;-3.34,.38,;-2.01,1.15,;-.67,.38,;.66,1.15,;1.99,.38,;1.99,-1.16,;3.33,-1.93,;4.66,-1.16,;5.99,-1.93,;6.47,-.46,;8.01,-.46,;8.49,-1.93,;7.24,-2.83,;6.76,-4.29,;5.22,-4.29,;4.45,-5.63,;4.75,-2.83,;.66,-1.93,;-.67,-1.16,;-2.01,-1.93,;-2.01,-3.47,;.66,2.69,;-.67,3.46,;-.67,5,;.1,3.67,;1.22,3.67,;1.99,5,;1.99,3.46,;.66,5.77,;-4.67,-3.46,;-3.34,-4.23,;-2.01,-5,;-2.57,-2.9,;-4.11,-5.57,)|
Cc1cccc(O)c1-c1ncc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wD:23.25,(-3.91,-4.31,;-5.25,-3.54,;-6.58,-4.31,;-7.91,-3.54,;-7.91,-2,;-6.58,-1.23,;-6.58,.31,;-5.25,-2,;-3.91,-1.23,;-3.91,.31,;-2.58,1.08,;-1.25,.31,;.09,1.08,;1.42,.31,;1.42,-1.23,;2.76,-2,;4.09,-1.23,;5.42,-2,;5.9,-.53,;7.44,-.53,;7.91,-2,;6.67,-2.9,;6.19,-4.37,;4.65,-4.37,;3.88,-5.7,;4.18,-2.9,;.09,-2,;-1.25,-1.23,;-2.58,-2,;-2.58,-3.54,;.09,2.62,;-1.25,3.39,;-1.25,4.93,;-.48,3.6,;.65,3.6,;1.42,4.93,;1.42,3.39,;.09,5.7,)|
CO[C@H]1C[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(c(F)c3n2)-c2cccc3cccc(Cl)c23)N(C)C1 |r|
CC(C)c1cccc(c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2)C(C)(C)C |r,wU:18.18,wD:24.26,(-7.91,1.13,;-6.58,.36,;-5.25,1.13,;-6.58,-1.18,;-7.91,-1.95,;-7.91,-3.49,;-6.58,-4.26,;-5.25,-3.49,;-5.25,-1.95,;-3.91,-1.18,;-3.91,.36,;-2.58,1.13,;-1.25,.36,;.09,1.13,;1.42,.36,;1.42,-1.18,;2.76,-1.95,;4.09,-1.18,;5.42,-1.95,;5.9,-.49,;7.44,-.49,;7.91,-1.95,;6.67,-2.86,;6.19,-4.32,;4.65,-4.32,;3.88,-5.65,;4.18,-2.86,;.09,-1.95,;-1.25,-1.18,;-2.58,-1.95,;-2.58,-3.49,;.09,2.67,;-1.25,3.44,;-1.25,4.98,;-.48,3.65,;.65,3.65,;1.42,4.98,;1.42,3.44,;.09,5.75,;-3.91,-4.26,;-4.31,-5.75,;-2.37,-4.26,;-2.58,-5.03,)|
Fc1c(ncc2c(nc(OC[C@]34CCCN3[C@@H](CNC=O)CC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(Cl)c12 |r|
Fc1c(ncc2c(nc(OCC34CCCN3CCC4)nc12)N1CC2CCC(C1)N2)-c1cccc2cccc(c12)C(F)(F)F
C[C@H]1C[C@@H]1c1c(Cl)cc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
C[C@@H]1CC1c1c(Cl)cc(O)cc1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r|
Fc1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c2c1
Oc1cc(-c2ncc3c(nc(OCC45CCCN4C(=O)CC5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Oc1cc(-c2ncc3c(nc(OCC4CCCN5CCCC45)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1
Fc1ccc2cccc(-c3ncc4c(nc(OCC56CCCN5CCC6)nc4c3F)N3CC4CCC(C3)N4)c2c1F
CCc1cccc2cccc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CCc1cccc2cccc(-c3ncc4c(nc(OC[C@]56C[C@@H](O)CN5C[C@@H](O)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
CCc1cccc2cc(O)cc(-c3ncc4c(nc(OC[C@]56CCCN5C[C@@H](F)C6)nc4c3F)N3CC4CCC(C3)N4)c12 |r|
Oc1cc(-c2ncc3c(nc(OC[C@]45C[C@@H](F)CN4CCCC5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2ncc3c(nc(OC[C@]45CCCN4C[C@@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(OC(F)(F)F)cccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)cccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(Cl)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(OC(F)(F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2cc(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(Cl)c(F)ccc2c1 |r|
[#8]-c1cc(-c2nc3-[#8]-[#6]-[#6@@H]-4-[#6@@H]-5-[#6]-[#6]-[#6@H](-[#6]-[#7]-4-c4nc(-[#8]-[#6][C@@]67[#6]-[#6]-[#6]-[#7]6-[#6]-[#6@H](F)-[#6]7)nc(c2F)c34)-[#7]-5)c2c(\[#6]=[#6](/F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(F)c(F)cc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(F)c(F)c(F)c2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67C[C@@H](F)CN6CC(=C)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(CC3CC3)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(Cl)cccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@H]5CC[C@@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2ccccc2c1 |r|
Oc1cc(-c2nc3OC[C@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2ccccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2ccccc2c1 |r|
Oc1cc(-c2nc3OC[C@H]4[C@H]5CC[C@@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2ccccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2ccccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCOCC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[Si](C)(COc1nc2N3C[C@H]4CC[C@H](N4)[C@H]3COc3nc(c(F)c(n1)c23)-c1cc(O)cc2ccc(F)c(C#C)c12)CN1CCOCC1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)c(F)cc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3c(F)cccc23)C1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(F)CC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC[C@H](F)C7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC[C@@H](F)C7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCCOCC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](CN=[N+]=[N-])CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(OC3CC3)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COC(=O)N6CCCCCC6)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
CN(C)C(=O)OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5COc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CCCN12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(F)c(Cl)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(OC(F)(F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(OC3CC3)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC[C@H](C7)C(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC[C@@H](C7)C(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
CN(C(=O)OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5COc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CCCN12)C(F)(F)F |r,TLB:14:15:19.18:21,THB:23:22:19.18:21|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3ccccc23)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cc(F)cc3ccccc23)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2c(F)ccc3ccccc23)C1 |r,wU:7.8,18.19,15.20,wD:1.0,20.22,(4.8,-5.61,;5.54,-4.23,;7.08,-4.07,;7.38,-2.61,;8.54,-1.51,;7.93,-.11,;6.42,-.25,;6.06,-1.76,;4.72,-1.02,;3.42,-1.81,;2.05,-.99,;2.08,.52,;.76,1.35,;1.28,2.58,;2.82,2.7,;3.51,4.07,;2.49,3.71,;1.47,4.1,;1.17,5.31,;2.68,5.61,;.45,3.88,;-1.06,4.04,;-2.13,2.83,;-1.94,1.35,;-3.23,.52,;-3.26,-.99,;-1.88,-1.76,;-1.88,-3.38,;-.59,-.99,;.76,-1.81,;-.56,.55,;-4.55,-1.79,;-4.58,-3.3,;-3.23,-4.18,;-5.87,-4.1,;-7.22,-3.33,;-7.22,-1.79,;-8.54,-.99,;-8.54,.55,;-7.22,1.32,;-5.9,.55,;-5.9,-.99,;4.94,-2.81,)|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](Cn6ccnn6)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(CC(F)(F)F)c(F)ccc2c1 |r|
CN(C(=O)OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5COc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CCCN12)c1cccc(c1)S(F)(F)(F)(F)F |r|
Oc1cc(-c2cc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(SC(F)(F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@@H](CC7)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2cc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3cc(F)c(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(OC(F)(F)F)c23)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3cc(F)ccc23)C1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC[C@@H](F)C7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@]12CC[C@H](N1)[C@H]1CCc3nc(c(F)c4nc(OCC5(CN6CCC(F)CC6)CC5)nc(N1C2)c34)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC7)C(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC[C@H](C7)C(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3O[C@@H](C4CC4)[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2ccc(F)c3ccccc23)C1 |r|
Cc1ccc2cc(O)cc(-c3nc4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C(Cl)=C |r|
Oc1cc(-c2nc3CCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3OCC[C@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[Si]1(C)CCCN(CC2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CC2)CC1 |r|
C[C@@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3O[C@H](C(F)F)[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cc(O)cc2ccc(F)c(F)c12)N3 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@@]4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@@H]1[C@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c-5nc([C@@H]1C#Cc1c(F)ccc6cccc-5c16)c24)N3 |r|
C[C@@H]1[C@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c-5nc([C@@H]1C#Cc1c(F)ccc6cc(O)cc-5c16)c24)N3 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CCC(CC5)OC(F)(F)F)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CC[C@@H](C5)OC(F)(F)F)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
CC[C@@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
CC[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
CC[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
C[C@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
C[C@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cc(O)cc2ccc(F)c(C#C)c12)N3 |r|
C[C@@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
C[C@@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cc(O)cc2ccc(F)c(C#C)c12)N3 |r|
Oc1cc(-c2nc3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](N4)[C@H]2CC3(F)F)c2c(C#C)c(F)ccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CC(F)(F)c4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@@]6(CC6(F)F)C7)nc(c2F)c34)N5)c2c(OC(F)(F)F)c(F)ccc2c1 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CCC[Si](C)(C)CC5)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CCN(CC(F)(F)F)CC5)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC7)OC(F)(F)F)CC6)nc(c2F)c34)N5)c2c(OC(F)(F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC[C@@H](C7)OC(F)(F)F)CC6)nc(c2F)c34)N5)c2c(OC(F)(F)F)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COc6cccc(c6)S(F)(F)(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4[C@H](COc4cccc(c4)S(F)(F)(F)(F)F)CC5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC7)OC(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CCC(CC8)OC(F)(F)F)CC7)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cccc(c7)S(F)(F)(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
CC(OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CCCN12)(C(F)(F)F)C(F)(F)F |r,TLB:12:13:17.16:19,THB:21:20:17.16:19|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COC(C6CC6)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r,TLB:16:15:11.12:44,THB:8:9:11.12:44|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COC(C7CC7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:49,THB:13:14:16.17:49|
CC(OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12)(C(F)(F)F)C(F)(F)F |r,TLB:12:13:17.16:19,THB:21:20:17.16:19|
F[C@H]1CN2CC3(CC3)C[C@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@]78CCCN7CC(C8)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:53,THB:13:14:16.17:53|
CC(OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12)(C(F)(F)F)C(F)(F)F |r,TLB:12:13:17.16:19,THB:21:20:17.16:19|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COC(C7CC7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r,TLB:22:21:17.18:50,THB:14:15:17.18:50|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cccc(c7)S(F)(F)(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
CC(C)(C)OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CCC(CC8)OC(F)(F)F)CC7)nc(c3F)c45)N6)c2c1OC(F)(F)F |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@@]7(CC7(F)F)C8)nc(c3F)c45)N6)c2c1C#C |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@@]6(CC6(F)F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3OCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCOc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CC[C@@H](C8)OC(F)(F)F)CC7)nc(c3F)c45)N6)c2c1OC(F)(F)F |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CC[C@@H](C8)OC(F)(F)F)CC7)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CCC(CC8)OC(F)(F)F)CC7)nc(c3F)c45)N6)c2c1C#C |r|
CCC[C@@H]1NCCN2[C@@H]1CCc1cc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc2c13)-c1cc(O)cc2ccc(F)c(CC)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@@H](C7)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@@H](C8)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r|
CCc1c(F)ccc2cccc(-c3nc4C[C@H](C)[C@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c12 |r|
Oc1cc(-c2nc3CCC[C@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](C7)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r,TLB:16:15:11.12:48,THB:8:9:11.12:48|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](C8)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:53,THB:13:14:16.17:53|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CCC6(CC6(F)F)CC5)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC78CCCN7C[C@@H](C8)OC(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC67CCCN6C[C@@H](C7)OC(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6CC(C7)OC(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r,TLB:16:15:11.12:39,THB:8:9:11.12:39|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](C8)OC(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:44,THB:13:14:16.17:44|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@]67CCCN6C[C@H](C7)OC(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r,TLB:16:15:11.12:39,THB:8:9:11.12:39|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@]78CCCN7C[C@H](C8)OC(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:44,THB:13:14:16.17:44|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@]67CCCN6C[C@@H](C7)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@]78CCCN7C[C@@H](C8)OC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)nc(c3F)c45)N6)c2c1C#C |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC4(CN5CCC(CC5)C(F)(F)F)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COc6ccnc(n6)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COc6cc(ncn6)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COC(C(F)(F)F)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7ccnc(n7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cc(ncn7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cc(ncn7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COc6cnc(cn6)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@H]1CCc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC45CCCN4CCC5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@H]1Cc2nc(c(F)c3nc(OCC45CC6(CC6)CN4CC4(CC4)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@@H]1CCc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COc6ncccc6OC(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC7)OC(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC[C@@H](C7)OC(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COCC(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COCC(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](CF)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
FC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC(F)(F)F)CC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
COC1(CCN(CC2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc5nc(c(F)c(n3)c45)-c3cc(O)cc4ccc(F)c(C#C)c34)CC2)CC1)C(F)(F)F |r|
CC[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@@H]4CCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
C[C@@H]1CC[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4C[C@H](F)c4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4C[C@@H](F)c4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
C[C@H]1CC[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
CC[C@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC8CC8C7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC8(CC8)CC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC7(CN8CCC9(CC9)CC8)CC7)nc(c3F)c45)N6)c2c1C#C |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CC8CC(C8)C7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r,wU:10.44,13.43,wD:9.15,(-7.51,-5.83,;-7.48,-4.21,;-6.13,-3.44,;-6.13,-1.87,;-4.78,-1.1,;-4.78,.41,;-3.41,1.24,;-4.18,2.53,;-3.41,3.93,;-2.03,3.55,;-2.01,5.11,;-1.24,4.04,;-.08,4.07,;.69,5.09,;.69,3.55,;-.69,2.72,;-.69,1.21,;.69,.41,;.69,-1.13,;2.03,-1.92,;3.41,-1.1,;4.76,-1.9,;6.08,-1.07,;7.48,-1.87,;7.51,-3.38,;8.88,-4.07,;8.83,-2.53,;10.12,-1.81,;10.2,-3.33,;8.8,-1.04,;4.01,-3.19,;5.53,-3.16,;-.69,-1.95,;-2.03,-1.13,;-3.38,-1.87,;-3.38,-3.49,;-2.01,.44,;-.69,5.83,;-7.51,-1.1,;-7.48,.44,;-6.63,1.68,;-5.75,3.05,;-8.85,1.21,;-8.85,2.72,;-10.2,.44,;-10.2,-1.1,;-8.83,-1.87,;-8.83,-3.44,)|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC(CC7)Oc7ccnc(n7)C(F)(F)F)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
Oc1cc(-c2nc3CCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
CC[C@@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
Oc1cc(-c2nc3CC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OCC6(CN7CCC8(CC8(F)F)CC7)CC6)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
O[C@@H]1C[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
Fc1ccc2cccc(-c3nc4CC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r,TLB:21:20:16.17:54,THB:13:14:16.17:54|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCCCc4nc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
Oc1cc(-c2nc3CCCC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(C#C)c(F)ccc2c1 |r|
C[C@]12CC[C@H](N1)[C@H]1CCc3nc(c(F)c4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(N1C2)c34)-c1cc(O)cc2ccc(F)c(C#C)c12 |r|
C[C@]12CC[C@H](N1)[C@H]1CCc3nc(c(F)c4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(N1C2)c34)-c1cccc2ccc(F)c(C#C)c12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCCc4cc(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r|
C[C@H]1Cc2cc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(N)cc2ccc(F)c(C#C)c12 |r|
C[C@@H]1CC[C@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4c(F)c(nc1c24)-c1cc(N)cc2ccc(F)c(C#C)c12)N3 |r|
C[C@@H]1CC[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4[C@H](CF)CC5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
C[C@H]1Cc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@H]14)c23)-c1cc(N)cc2ccc(F)c(C#C)c12 |r|
CCC[C@@H]1NCCN2[C@@H]1CCCc1nc(c(F)c3nc(OC[C@@]45CCCN4[C@H](COc4cnc(cn4)C(F)(F)F)CC5)nc2c13)-c1cccc2ccc(F)c(C#C)c12 |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cc(cnn7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](COc7cnnc(c7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
FC(F)c1cnc(OC[C@@H]2CC[C@]3(COc4nc5N6C[C@H]7CC[C@H](N7)[C@H]6CCCc6nc(c(F)c(n4)c56)-c4cccc5ccc(F)c(C#C)c45)CCCN23)cn1 |r|
Fc1ccc2cccc(-c3nc4CCC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7[C@H](CSc7cc(ncn7)C(F)(F)F)CC8)nc(c3F)c45)N6)c2c1C#C |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4CCc4c(Cl)c(c(F)c(n2)c34)-c2cccc3ccc(F)c(C#C)c23)C1 |r,wU:7.8,18.19,15.20,wD:1.0,20.22,(4.97,-6.12,;5.72,-4.93,;7.27,-4.77,;7.61,-3.3,;8.77,-2.22,;8.13,-.83,;6.61,-.97,;6.25,-2.47,;4.92,-1.72,;3.56,-2.52,;2.26,-1.88,;2.26,-.39,;.9,.42,;.87,3.02,;2.26,3.77,;2.31,5.32,;1.54,4.35,;.29,4.3,;-.35,5.43,;.98,6.12,;-.43,3.85,;-1.93,3.49,;-2.7,1.86,;-1.79,.42,;-3.12,-.33,;-3.53,1.11,;-3.12,-1.88,;-1.76,-2.63,;-1.79,-4.24,;-.46,-1.86,;.87,-2.69,;-.43,-.36,;-4.75,-2.77,;-4.75,-4.35,;-6.08,-5.1,;-7.44,-4.32,;-7.41,-2.77,;-8.77,-2.02,;-8.77,-.5,;-7.44,.3,;-7.44,1.8,;-6.11,-.47,;-5.31,.83,;-4.56,2.24,;-6.11,-2,;5.14,-3.52,)|
C[C@@H]1CC[C@@H]2[C@@H]3CC[C@H](CN2c2nc(OC[C@@]45CCCN4[C@H](COc4cc(ncn4)C(F)(F)F)CC5)nc4c(F)c(nc1c24)-c1cccc2ccc(F)c(C#C)c12)N3 |r|
Oc1cc(-c2c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCc(c2Cl)c34)c2c(C#C)c(F)ccc2c1 |r,wU:12.11,28.30,25.31,wD:18.19,30.33,(-6.07,-6.4,;-6.04,-4.8,;-4.72,-4,;-4.69,-2.49,;-3.1,-1.58,;-1.78,-2.33,;-1.75,-3.95,;-.43,-1.56,;.92,-2.41,;2.24,-1.58,;3.54,-2.22,;4.86,-1.42,;6.21,-2.16,;6.56,-.67,;8.11,-.54,;8.71,-1.91,;7.56,-3.01,;7.25,-4.47,;5.71,-4.64,;4.94,-6.01,;5.11,-3.26,;2.24,-.1,;.92,.73,;.87,3.32,;2.24,4.09,;2.33,5.63,;1.56,4.64,;.32,4.58,;-.34,5.74,;1,6.4,;-.43,4.14,;-1.91,3.78,;-2.68,2.16,;-1.75,.73,;-3.1,-.01,;-3.51,1.42,;-.43,-.04,;-6.07,-1.69,;-6.07,-.18,;-5.24,1.14,;-4.5,2.55,;-7.39,.59,;-7.36,2.11,;-8.71,-.18,;-8.71,-1.72,;-7.36,-2.46,;-7.36,-4.03,)|
FC(F)c1cc(OC[C@@H]2CC[C@]3(COc4nc5N6C[C@H]7CC[C@H](N7)[C@H]6CCCc6nc(c(F)c(n4)c56)-c4cccc5ccc(F)c(C#C)c45)CCCN23)ncn1 |r|
FC(F)c1cncnc1OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12 |r|
FC(F)c1nccnc1OC[C@@H]1CC[C@]2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5CCCc5nc(c(F)c(n3)c45)-c3cccc4ccc(F)c(C#C)c34)CCCN12 |r|
FC(F)c1nccc(OC[C@@H]2CC[C@]3(COc4nc5N6C[C@H]7CC[C@H](N7)[C@H]6CCCc6nc(c(F)c(n4)c56)-c4cccc5ccc(F)c(C#C)c45)CCCN23)n1 |r|
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(Br)c23)CC1
Oc1cc(N2CCc3c(C2)nc(OCC2(CN4CC[C@@H](F)C4)CC2)nc3N2CC3CCC(C2)N3)c2c(Br)cccc2c1 |r|
Oc1cc(N2CCc3c(C2)nc(OCC2(CN4CCOCC4)CC2)nc3N2CC3CCC(C2)N3)c2c(Br)cccc2c1
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(C)c23)CC1
Cc1cccc2cc(O)cc(N3CCc4c(C3)nc(OCC3(CN5CC[C@@H](F)C5)CC3)nc4N3CC4CCC(C3)N4)c12 |r|
Cc1cccc2cc(O)cc(N3CCc4c(C3)nc(OCC3(CN5CCOCC5)CC3)nc4N3CC4CCC(C3)N4)c12
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(I)c23)CC1
Oc1cc(N2CCc3c(C2)nc(OCC2(CN4CC[C@@H](F)C4)CC2)nc3N2CC3CCC(C2)N3)c2c(I)cccc2c1 |r|
Oc1cc(N2CCc3c(C2)nc(OCC2(CN4CCOCC4)CC2)nc3N2CC3CCC(C2)N3)c2c(I)cccc2c1
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CCOCC5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(cccc2c1)C#C
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CC[C@@H](F)C5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(cccc2c1)C#C |r|
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CC[C@@H](F)C5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(I)cccc2c1 |r|
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CCOCC5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(I)cccc2c1
CN(C)CC1(COc2nc(N3CC4CCC(C3)N4)c3cc(Cl)c(c(F)c3n2)-c2cc(O)cc3ccccc23)CC1 |TLB:9:10:13.14:17,(6.54,-6.48,;6.94,-4.99,;8.42,-4.59,;5.85,-3.9,;6.25,-2.42,;4.91,-1.65,;3.58,-2.42,;2.25,-1.65,;2.25,-.11,;.91,.66,;.91,2.2,;.51,3.69,;-.82,4.46,;-2.36,4.46,;-1.27,5.55,;.27,5.55,;1.6,4.78,;-.13,7.04,;-.42,-.11,;-1.76,.66,;-3.09,-.11,;-4.42,.66,;-3.09,-1.65,;-1.76,-2.42,;-1.76,-3.96,;-.42,-1.65,;.91,-2.42,;-4.42,-2.42,;-5.76,-1.65,;-7.09,-2.42,;-8.42,-1.65,;-7.09,-3.96,;-5.76,-4.73,;-5.76,-6.27,;-4.42,-7.04,;-3.09,-6.27,;-3.09,-4.73,;-4.42,-3.96,;7.79,-2.42,;7.02,-1.08,)|
CN(C)CC1(COc2nc(N3CC4CCC(C3)N4)c3ccc(c(F)c3n2)-c2cc(O)cc3ccccc23)CC1 |TLB:9:10:13.14:17|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)N3)c2ccc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r,TLB:10:11:14.15:18|
CN(C)[C@@H]1CC[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2ccc(c(F)c2n1)-c1cc(O)cc2ccccc12 |r|
CN(C)CC1(COc2nc(N3CC4CCC(C3)N4)c3cc(F)c(c(F)c3n2)-c2cc(O)cc3ccccc23)CC1 |(73.89,-11.38,;75.22,-12.15,;75.23,-13.69,;76.55,-11.38,;76.54,-9.83,;75.21,-9.07,;73.88,-9.84,;72.54,-9.07,;72.54,-7.52,;71.2,-6.76,;71.2,-5.22,;69.86,-4.46,;69.86,-2.92,;70.33,-4.08,;71.91,-4.02,;72.53,-2.92,;72.53,-4.45,;71.2,-2.15,;69.88,-7.53,;68.55,-6.76,;67.21,-7.52,;65.88,-6.74,;67.2,-9.06,;68.54,-9.85,;68.53,-11.39,;69.87,-9.08,;71.2,-9.85,;65.87,-9.82,;64.54,-9.04,;63.2,-9.8,;61.87,-9.02,;63.19,-11.34,;64.53,-12.12,;64.53,-13.64,;65.85,-14.41,;67.18,-13.65,;67.18,-12.12,;65.86,-11.36,;77.3,-8.5,;78.08,-9.82,)|
CCc1cc2c(nc(OCC3(CN(C)C)CC3)nc2c(F)c1-c1cc(O)cc2ccccc12)N1CC2CCC(C1)N2 |TLB:5:33:36.37:40,(-5.76,-.11,;-4.42,.66,;-3.09,-.11,;-1.76,.66,;-.42,-.11,;.91,.66,;2.25,-.11,;2.25,-1.65,;3.58,-2.42,;4.91,-1.65,;6.25,-2.42,;5.85,-3.9,;6.94,-4.99,;6.54,-6.48,;8.42,-4.59,;7.73,-2.81,;7.34,-1.33,;.91,-2.42,;-.42,-1.65,;-1.76,-2.42,;-1.76,-3.96,;-3.09,-1.65,;-4.42,-2.42,;-5.76,-1.65,;-7.09,-2.42,;-8.42,-1.65,;-7.09,-3.96,;-5.76,-4.73,;-5.76,-6.27,;-4.42,-7.04,;-3.09,-6.27,;-3.09,-4.73,;-4.42,-3.96,;.91,2.2,;.51,3.69,;-.82,4.46,;-2.36,4.46,;-1.27,5.55,;.27,5.55,;1.6,4.78,;-.13,7.04,)|
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2C[C@@H]3CC[C@H]2CN3)c2cc(O)cc3cccc(Br)c23)CC1 |r|
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(Br)c23)CC1(F)F
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2nc(N)cc3cccc(Br)c23)CC1
CN(C)CC1(COc2nc3CC(OCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(C#C)c23)CC1
CN(C)CC1(COc2nc3CC(CCc3c(n2)N2CC3CCC(C2)N3)c2cccc3cccc(C#C)c23)CC1
Ic1cccc2cccc(N3CCc4c(C3)nc(OCC3(CN5CCOCC5)CC3)nc4N3CC4CCC(C3)N4)c12
CN1CCC[C@@H]1COc1nc2CN(CCc2c(n1)N1CC2CCC(C1)N2)c1cc(O)cc2cccc(Br)c12 |r|
CN1C[C@H](F)C[C@H]1COc1nc2CN(CCc2c(n1)N1CC2CCC(C1)N2)c1cc(O)cc2cccc(Br)c12 |r|
Oc1cc(N2CCc3c(C2)nc(OCC2(CN4CCOCC4)CC2)nc3N2C[C@@H]3CC[C@H]2CN3)c2c(Br)cccc2c1 |r|
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cccc3cccc(Br)c23)CC1(F)F
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(Br)c23)CC1(C)C
CN1CCC[C@H]1COc1nc2CN(CCc2c(n1)N1CC2CCC(C1)N2)c1cc(O)cc2cccc(Br)c12 |r|
CO[C@@H]1C[C@@H](COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(Br)c23)N(C)C1 |r|
Oc1cc(C2Cc3nc(OCC4(CN5CCOCC5)CC4)nc(N4CC5CCC(C4)N5)c3CO2)c2c(cccc2c1)C#C
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CC[C@@H](F)C5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(C=C)cccc2c1 |r|
Oc1cc(C(=O)N2Cc3nc(OCC4(CN5CCOCC5)CC4)nc(N4CC5CCC(C4)N5)c3C2)c2c(C=C)cccc2c1
CN(C)CC1(COc2nc3CN(CCc3c(n2)N2CC3CCC(C2)N3)c2nc(N)cc3cccc(C#C)c23)CC1
CN(C)CC1(COc2nc3CC(OCc3c(n2)N2CC3CCC(C2)N3)c2cc(O)cc3cccc(Br)c23)CC1
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc4nc(c(F)c(n2)c34)-c2cccc3cccc(Cl)c23)C1 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(cccc2c1)C#C |r|
Cn1ncc2ccc(F)c(-c3nc4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c12 |r,wU:19.46,16.47,33.35,wD:15.21,27.27,(-5.28,1.03,;-6.31,-.12,;-7.84,.05,;-8.47,-1.36,;-7.33,-2.39,;-7.33,-3.93,;-5.99,-4.7,;-4.66,-3.93,;-3.33,-4.7,;-4.66,-2.39,;-3.33,-1.62,;-3.33,-.08,;-1.99,.69,;-2.38,2.21,;-1.34,3.36,;.16,3.35,;.74,4.68,;.94,3.25,;1.75,2.88,;3.08,3.65,;2.47,2.36,;1.03,2.19,;.68,.69,;2.01,-.08,;2.01,-1.62,;3.34,-2.39,;4.68,-1.62,;6.01,-2.39,;4.92,-3.48,;5.62,-4.85,;7.14,-4.61,;7.38,-3.09,;8.47,-2,;7.77,-.63,;8.47,.74,;6.25,-.87,;.68,-2.39,;-.66,-1.62,;-1.99,-2.39,;-1.99,-3.93,;-.66,-.08,;2.18,4.85,;-5.99,-1.62,)|
CCc1cccc2cc(O)cc(-c3nc4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2cccc(Cl)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2cccc(Cl)c12 |r|
CCc1cccc2cc(O)cc(-c3nc4O[C@@H](C)[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2cccc(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc(N)c1F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(C)c(F)c(N)c1 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(F)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(F)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(C)c(F)c(N)c1F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2cccc(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2cccc(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OCC45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2cccc(Cl)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OCC45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OCC45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(C)cc(N)c1F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2ccccc12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4C[C@@H](F)CN4C)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2cccc(Cl)c12 |r|
CCc1cccc2cc(O)cc(-c3nc4O[C@@H](C)[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OCC78CC(C7)OC8)nc(c3F)c45)N6)c12 |r,wU:22.46,19.47,16.16,wD:18.24,(-4.55,2.92,;-4.55,1.38,;-5.89,.61,;-7.22,1.38,;-8.55,.61,;-8.55,-.93,;-7.22,-1.7,;-7.22,-3.24,;-5.89,-4.01,;-5.89,-5.55,;-4.55,-3.24,;-4.55,-1.7,;-3.22,-.93,;-3.22,.61,;-1.89,1.38,;-2.28,2.91,;-1.23,4.05,;-2,5.39,;.27,4.05,;.84,5.38,;1.04,3.95,;1.86,3.58,;3.19,4.35,;2.58,3.05,;1.14,2.88,;.78,1.38,;2.12,.61,;2.12,-.93,;3.45,-1.7,;4.78,-.93,;6.12,-1.7,;7.52,-1.07,;8.55,-2.22,;7.21,-2.79,;7.78,-3.55,;6.28,-3.23,;.78,-1.7,;-.55,-.93,;-1.89,-1.7,;-1.89,-3.24,;-.55,.61,;2.29,5.55,;-5.89,-.93,)|
C[C@@H]1Oc2nc(c(F)c3nc(OCC45CCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cncc2ccccc12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@@H](C5)OCc4ccc(cc4)-c4ccccc4C#N)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)cc(C)c1C(F)(F)F |r,wU:13.12,1.0,29.31,26.32,wD:31.35,(-2.53,5.47,;-1.76,4.13,;-2.81,2.82,;-2.42,1.46,;-3.75,.69,;-3.75,-.85,;-2.42,-1.62,;-2.42,-3.16,;-1.09,-.85,;.25,-1.62,;1.58,-.85,;2.92,-1.62,;4.25,-.85,;5.58,-1.62,;4.68,-2.86,;5.92,-3.77,;6.83,-2.52,;8.08,-1.62,;7.6,-.15,;8,1.34,;9.09,.25,;6.06,-.15,;1.58,.69,;.25,1.46,;.6,2.8,;2.05,2.79,;2.82,4.13,;1.48,3.36,;.51,3.92,;.51,5.46,;2.05,5.46,;-.26,4.13,;-1.09,.69,;-5.09,-1.62,;-5.09,-3.16,;-3.75,-3.93,;-6.42,-3.93,;-6.42,-5.47,;-7.75,-3.16,;-7.75,-1.62,;-9.09,-.85,;-6.42,-.85,;-6.42,.69,;-7.75,1.46,;-5.09,1.46,;-6.42,2.23,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)cc(C)c1C(F)(F)F |r,wU:1.0,29.31,26.32,19.20,wD:31.35,13.12,(-2.17,5.47,;-1.4,4.13,;-2.45,2.82,;-2.06,1.46,;-3.39,.69,;-3.39,-.85,;-2.06,-1.62,;-2.06,-3.16,;-.73,-.85,;.61,-1.62,;1.94,-.85,;3.27,-1.62,;4.61,-.85,;5.94,-1.62,;4.7,-2.52,;5.17,-3.99,;6.71,-3.99,;7.19,-2.52,;8.43,-1.62,;7.96,-.15,;8.73,1.18,;6.42,-.15,;1.94,.69,;.61,1.46,;.96,2.8,;2.41,2.79,;3.18,4.13,;1.84,3.36,;.87,3.92,;.87,5.46,;2.41,5.46,;.1,4.13,;-.73,.69,;-4.73,-1.62,;-4.73,-3.16,;-3.39,-3.93,;-6.06,-3.93,;-6.06,-5.47,;-7.39,-3.16,;-7.39,-1.62,;-8.73,-.85,;-6.06,-.85,;-6.06,.69,;-7.39,1.46,;-4.73,1.46,;-6.06,2.23,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)ccc1C(F)(F)F |r,wU:1.0,29.31,26.32,19.20,wD:31.35,13.12,(-2.84,5.47,;-2.07,4.13,;-3.12,2.82,;-2.73,1.46,;-4.06,.69,;-4.06,-.85,;-2.73,-1.62,;-2.73,-3.16,;-1.39,-.85,;-.06,-1.62,;1.27,-.85,;2.61,-1.62,;3.94,-.85,;5.28,-1.62,;4.03,-2.52,;4.5,-3.99,;6.04,-3.99,;6.52,-2.52,;7.77,-1.62,;7.29,-.15,;8.06,1.18,;5.75,-.15,;1.27,.69,;-.06,1.46,;.3,2.8,;1.74,2.79,;2.51,4.13,;1.17,3.36,;.2,3.92,;.2,5.46,;1.74,5.46,;-.57,4.13,;-1.39,.69,;-5.39,-1.62,;-5.39,-3.16,;-4.06,-3.93,;-6.73,-3.93,;-6.73,-5.47,;-8.06,-3.16,;-8.06,-1.62,;-6.73,-.85,;-6.73,.69,;-8.06,1.46,;-5.39,1.46,;-6.73,2.23,)|
Cc1cc(N)c(F)c(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c1C(F)(F)F |r,wU:14.45,17.44,31.33,wD:13.19,25.25,(-6.59,-5.75,;-6.59,-4.21,;-7.92,-3.44,;-7.92,-1.9,;-9.25,-1.13,;-6.59,-1.13,;-6.59,.41,;-5.25,-1.9,;-2.56,-.56,;-2.56,.98,;-1.22,1.75,;-1.62,3.11,;-.57,4.42,;.93,4.42,;1.7,5.75,;1.7,4.21,;2.68,3.65,;4.01,4.42,;3.24,3.08,;1.8,3.09,;1.44,1.75,;2.78,.98,;2.78,-.56,;4.11,-1.33,;5.44,-.56,;6.78,-1.33,;5.64,-2.37,;6.28,-3.77,;7.81,-3.6,;8.12,-2.09,;9.25,-1.05,;8.62,.35,;9.24,1.76,;7.09,.18,;1.44,-1.33,;.11,-.56,;-1.22,-1.33,;-1.22,-2.87,;.11,.98,;3.24,5.75,;-5.25,-3.44,;-3.92,-4.21,;-2.59,-3.44,;-3.92,-5.75,;-2.59,-4.98,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cncc2cccc(Cl)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cncc2cccc(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cncc2cccc(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)cc2ccccc12 |r|
Cc1cc(N)nc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6CC6(CC6(F)F)C7)nc(c2F)c34)N5)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)cc(C)c1C(F)(F)F |r|
Cc1cc(N)nc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)C14)c23)-c1nc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC(=C)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)cc(C)c1C(F)(F)F |r|
CN1CCC2COc3nc(c(F)c4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(N2CC1)c34)-c1cc(O)cc2cccc(F)c12 |r|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N(CCCF)C5)c2c(cccc2c1)C#C |r,THB:36:35:15.9.14:11.12|
Oc1cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N(CC2COC2)C5)c2c(cccc2c1)C#C |r,THB:36:35:15.9.14:11.12|
Cc1cc(N)nc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4ncnc(c2F)c34)N5)c1C(F)(F)F |r|
Fc1c(nc2OC[C@@H]3[C@@H]4CC[C@H](CN3c3ncnc1c23)N4)-c1cccc2cccc(Cl)c12 |r|
C[C@@H]1Oc2nc(c(F)c3ncnc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2cccc(C#C)c12 |r|
Nc1nc2c(ccc(F)c2s1)-c1nc2OC[C@@H]3[C@@H]4CC[C@H](CN3c3ncnc(c1F)c23)N4 |r|
C[C@@H]1Oc2nc(c(F)c3ncnc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2ccc(F)c(C#C)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC(=C)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C=O |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1C(F)(F)F |r|
Cc1c(F)c(N)cc(-c2nc3OC[C@@H]4[C@@H]5CC[C@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C\C(C5)=C/F)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC(F)(F)CN4C)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@H]4CC(F)(F)CN4C)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)ccc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)cc1C(C)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(C)c1Cl |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1CC(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)c(F)c(C)c1Cl |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc(F)c1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cnccc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cccc2nc(N)ccc12 |r|
CCc1cccc2cc(O)cc(-c3nc4O[C@@H](C)[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7CC(=C)C8)nc(c3F)c45)N6)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(O)cc2ccc(F)c(F)c12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)cc2CCCc12 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)ccc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4CC4(CC4(F)F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nc(N)c(F)cc1C(F)(F)F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1nccc(C)c1C(F)(F)F |r|
COc1cc2ccccc2c(n1)-c1nc2O[C@@H](C)[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@]56CCN5CC(F)(F)C6)nc(c1F)c23)N4 |r|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)c(F)cc1C(F)(F)F |r,wU:26.32,29.31,1.0,19.20,wD:13.12,31.35,(-2.06,5.23,;-1.29,3.9,;-2.23,2.68,;-1.85,1.19,;-3.19,.42,;-3.19,-1.12,;-1.85,-1.89,;-1.85,-3.43,;-.52,-1.12,;.82,-1.89,;2.15,-1.12,;3.48,-1.89,;4.82,-1.12,;6.15,-1.89,;5.25,-3.14,;6.15,-4.38,;7.61,-3.91,;7.61,-2.37,;8.52,-1.12,;7.61,.13,;8.38,1.46,;6.15,-.35,;2.15,.42,;.82,1.19,;1.2,2.68,;2.72,2.89,;3.3,4.32,;2.29,3.84,;1.24,4.28,;.83,5.32,;2.36,5.53,;.25,3.9,;-.52,.42,;-4.52,-1.89,;-5.85,-1.12,;-5.85,.42,;-7.19,-1.89,;-8.52,-1.12,;-7.19,-3.43,;-8.52,-4.2,;-5.85,-4.2,;-4.47,-3.5,;-3.14,-4.28,;-1.82,-5.07,;-3.93,-5.61,;-2.36,-2.96,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)c(F)c(C)c1C(F)(F)F |r,wU:1.0,29.31,26.32,19.20,wD:13.12,31.35,(-2.06,5.44,;-1.29,4.11,;-2.23,2.89,;-1.85,1.4,;-3.19,.63,;-3.19,-.91,;-1.85,-1.68,;-1.85,-3.22,;-.52,-.91,;.82,-1.68,;2.15,-.91,;3.48,-1.68,;4.82,-.91,;6.15,-1.68,;5.25,-2.93,;6.15,-4.17,;7.61,-3.7,;7.61,-2.16,;8.52,-.91,;7.61,.33,;8.38,1.67,;6.15,-.14,;2.15,.63,;.82,1.4,;1.2,2.89,;2.72,2.9,;3.55,4.53,;2.41,4.09,;1.41,4.49,;1.08,5.53,;2.62,5.53,;.25,4.11,;-.52,.63,;-4.52,-1.68,;-5.85,-.91,;-5.85,.63,;-7.19,-1.68,;-8.52,-.91,;-7.19,-3.22,;-8.52,-3.99,;-5.85,-3.99,;-5.85,-5.53,;-4.44,-3.31,;-3.12,-4.09,;-1.8,-4.88,;-2.33,-2.77,;-3.91,-5.42,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@]45CCN4CC(F)(F)C5)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)cc(C)c1C(F)(F)F |r,wU:1.0,29.31,26.32,wD:13.12,31.35,(-2.62,5.44,;-1.85,4.11,;-2.8,2.89,;-2.42,1.4,;-3.75,.63,;-3.75,-.91,;-2.42,-1.68,;-2.42,-3.22,;-1.08,-.91,;.25,-1.68,;1.58,-.91,;2.92,-1.68,;4.25,-.91,;5.58,-1.68,;4.68,-2.93,;5.92,-3.83,;6.83,-2.59,;8.08,-1.68,;7.6,-.22,;8,1.27,;9.09,.18,;6.06,-.22,;1.58,.63,;.25,1.4,;.63,2.89,;2.16,2.9,;2.98,4.53,;1.84,4.09,;.84,4.49,;.51,5.53,;2.05,5.53,;-.31,4.11,;-1.08,.63,;-5.09,-1.68,;-6.42,-.91,;-6.42,.63,;-7.75,-1.68,;-9.09,-.91,;-7.75,-3.22,;-6.42,-3.99,;-6.42,-5.53,;-5.01,-3.31,;-3.69,-4.09,;-2.36,-4.88,;-2.9,-2.77,;-4.47,-5.42,)|
C[C@@H]1Oc2nc(c(Cl)c3ncnc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)cc(C)c1C(F)(F)F |r,wU:1.0,18.18,15.19,wD:20.22,(.43,5.44,;1.2,4.11,;.25,2.89,;.64,1.4,;-.7,.63,;-.7,-.91,;.64,-1.68,;.64,-3.22,;1.97,-.91,;3.3,-1.68,;4.64,-.91,;4.64,.63,;3.3,1.4,;3.68,2.89,;5.21,2.9,;6.03,4.53,;4.89,4.09,;3.89,4.49,;3.56,5.53,;5.1,5.53,;2.74,4.11,;1.97,.63,;-2.03,-1.68,;-3.37,-.91,;-3.37,.63,;-4.7,-1.68,;-6.03,-.91,;-4.7,-3.22,;-3.37,-3.99,;-3.37,-5.53,;-1.92,-3.24,;-.58,-4,;.77,-4.75,;.17,-2.65,;-1.33,-5.34,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)c(F)c(C)c1C(F)(F)F |r,wU:1.0,29.31,26.32,16.22,wD:13.12,31.35,(-2.06,5.79,;-1.29,4.46,;-2.23,3.24,;-1.85,1.75,;-3.19,.98,;-3.19,-.56,;-1.85,-1.33,;-1.85,-2.87,;-.52,-.56,;.82,-1.33,;2.15,-.56,;3.48,-1.33,;4.82,-.56,;6.15,-1.33,;7.61,-.86,;8.52,-2.1,;7.61,-3.35,;7.94,-4.85,;6.79,-5.88,;5.33,-5.41,;5.01,-3.9,;6.15,-2.87,;2.15,.98,;.82,1.75,;1.2,3.24,;2.72,3.25,;3.55,4.88,;2.41,4.44,;1.41,4.84,;1.08,5.88,;2.62,5.88,;.25,4.46,;-.52,.98,;-4.52,-1.33,;-5.85,-.56,;-5.85,.98,;-7.19,-1.33,;-8.52,-.56,;-7.19,-2.87,;-8.52,-3.64,;-5.85,-3.64,;-5.85,-5.18,;-4.44,-2.96,;-3.12,-3.74,;-1.8,-4.53,;-2.33,-2.42,;-3.91,-5.07,)|
C[C@@H]1Oc2nc(c(F)c3nc(OC[C@@H]4CC[C@H]5COCCN45)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1c(F)c(N)cc(C)c1C(F)(F)F |r,wU:1.0,29.31,26.32,16.22,wD:13.12,31.35,(-2.06,5.79,;-1.29,4.46,;-2.23,3.24,;-1.85,1.75,;-3.19,.98,;-3.19,-.56,;-1.85,-1.33,;-1.85,-2.87,;-.52,-.56,;.82,-1.33,;2.15,-.56,;3.48,-1.33,;4.82,-.56,;6.15,-1.33,;7.61,-.86,;8.52,-2.1,;7.61,-3.35,;7.94,-4.85,;6.79,-5.88,;5.33,-5.41,;5.01,-3.9,;6.15,-2.87,;2.15,.98,;.82,1.75,;1.2,3.24,;2.72,3.25,;3.55,4.88,;2.41,4.44,;1.41,4.84,;1.08,5.88,;2.62,5.88,;.25,4.46,;-.52,.98,;-4.52,-1.33,;-5.85,-.56,;-5.85,.98,;-7.19,-1.33,;-8.52,-.56,;-7.19,-2.87,;-5.85,-3.64,;-5.85,-5.18,;-4.44,-2.96,;-3.12,-3.74,;-1.8,-4.53,;-2.33,-2.42,;-3.91,-5.07,)|
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C[C@@H]1Oc2nc(c(F)c3nc(OCC4(CN5CC(C5)C(F)F)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)nc(C)c1C(F)(F)F |r|
CO[C@@H]1CCN(CC2(COc3nc4N5C[C@H]6CC[C@H](N6)[C@H]5[C@H](C)Oc5nc(c(F)c(n3)c45)-c3cc(N)nc(C)c3C(F)(F)F)CC2)C[C@@H]1F |r|
C[C@@H]1Oc2nc(c(F)c3nc(OCC4(CN5CCC(C5)C(F)F)CC4)nc(N4C[C@H]5CC[C@H](N5)[C@@H]14)c23)-c1cc(N)nc(C)c1C(F)(F)F |r|
Oc1cc(-c2c(Cl)cc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r,wU:20.21,(-9.09,-.65,;-7.75,-1.42,;-6.42,-.65,;-5.08,-1.42,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,;-5.08,-2.96,;-3.75,-3.73,;-3.75,-5.27,;-5.08,-6.04,;-6.42,-5.27,;-6.42,-3.73,;-7.75,-2.96,)|
Nc1nc2c(ccc(F)c2s1)-c1c(Cl)cc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:27.30,(-8.09,3.65,;-7.77,2.15,;-6.36,1.52,;-6.52,-.01,;-5.49,-1.16,;-5.97,-2.62,;-7.47,-2.94,;-8.51,-1.8,;-10.01,-2.12,;-8.03,-.33,;-8.8,1,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,)|
Oc1cc(-c2ccc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r|
Nc1nc2c(ccc(F)c2s1)-c1c(F)cc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1Cl)N1CC2CCC(C1)N2 |r,wU:27.30,(-8.58,3.35,;-8.1,1.89,;-6.64,1.41,;-6.64,-.13,;-5.49,-1.16,;-5.81,-2.66,;-7.28,-3.14,;-8.42,-2.11,;-9.89,-2.58,;-8.1,-.6,;-9.01,.64,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,)|
Oc1cc(-c2c(F)cc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2Cl)N2CC3CCC(C2)N3)c2ccccc2c1 |r,wU:20.21,(-7.6,-4.65,;-7.28,-3.14,;-5.81,-2.66,;-5.49,-1.16,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,;-6.64,-.13,;-6.32,1.38,;-7.46,2.41,;-8.93,1.93,;-9.25,.43,;-8.1,-.6,;-8.42,-2.11,)|
Nc1nc2c(ccc(F)c2s1)-c1c(F)cc2c(nc(OCC34CCCN3C[C@H](F)C4)nc2c1F)N1CC2CCC(C1)N2 |r,wU:27.30,(-8.58,3.35,;-8.1,1.89,;-6.64,1.41,;-6.64,-.13,;-5.49,-1.16,;-5.81,-2.66,;-7.28,-3.14,;-8.42,-2.11,;-9.83,-2.74,;-8.1,-.6,;-9.01,.64,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,)|
Oc1cc(-c2c(Cl)cc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2ccccc2c1 |r,wU:20.21,(-7.6,-4.65,;-7.28,-3.14,;-5.81,-2.66,;-5.49,-1.16,;-3.75,-.65,;-3.75,.9,;-5.08,1.67,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,;-6.64,-.13,;-6.32,1.38,;-7.46,2.41,;-8.93,1.93,;-9.25,.43,;-8.1,-.6,;-8.42,-2.11,)|
Nc1cc(-c2ccc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r|
Nc1cc(-c2c(Cl)cc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r,wU:20.21,(-7.6,-4.65,;-7.28,-3.14,;-5.81,-2.66,;-5.49,-1.16,;-3.75,-.65,;-3.75,.9,;-5.16,.27,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,;-6.64,-.13,;-6.32,1.38,;-4.85,1.86,;-3.39,2.33,;-7.46,2.41,;-7.14,3.92,;-8.93,1.93,;-9.25,.43,;-8.1,-.6,;-8.42,-2.11,)|
Nc1cc(-c2c(F)cc3c(nc(OCC45CCCN4C[C@H](F)C5)nc3c2F)N2CC3CCC(C2)N3)c2c(C#C)c(F)ccc2c1 |r,wU:20.21,(-7.6,-4.65,;-7.28,-3.14,;-5.81,-2.66,;-5.49,-1.16,;-3.75,-.65,;-3.75,.9,;-5.16,.27,;-2.42,1.67,;-1.08,.9,;.25,1.66,;1.58,.89,;1.58,-.65,;2.92,-1.42,;2.92,-2.96,;4.16,-3.86,;3.02,-4.89,;3.65,-6.3,;5.18,-6.14,;5.5,-4.63,;6.64,-3.6,;6.02,-2.19,;6.79,-.86,;4.48,-2.35,;.25,-1.42,;-1.08,-.65,;-2.42,-1.42,;-2.42,-2.96,;.25,3.2,;-1.08,3.97,;-1.08,5.52,;-.18,4.27,;1.06,4.18,;1.58,5.52,;1.58,3.97,;.25,6.28,;-6.64,-.13,;-6.32,1.38,;-4.85,1.86,;-3.39,2.33,;-7.46,2.41,;-7.14,3.92,;-8.93,1.93,;-9.25,.43,;-8.1,-.6,;-8.42,-2.11,)|
CN1CCC[C@H]1COc1nc(N2C3CCC2CNCC3)c2cc(Cl)c(c(F)c2n1)-c1cc(O)cc2ccccc12 |r,wD:5.6,(5.1,-4.28,;6.25,-3.25,;7.78,-3.54,;8.55,-2.2,;7.52,-1.06,;6.12,-1.69,;4.78,-.92,;3.45,-1.69,;2.12,-.92,;2.12,.62,;.78,1.39,;.78,2.93,;-.61,3.6,;.06,4.77,;1.6,4.77,;2.17,3.6,;2.51,5.1,;1.55,6.31,;.01,6.31,;-.95,5.1,;-.55,.62,;-1.89,1.39,;-3.22,.62,;-4.55,1.39,;-3.22,-.92,;-1.89,-1.69,;-1.89,-3.23,;-.55,-.92,;.78,-1.69,;-4.55,-1.69,;-5.89,-.92,;-7.22,-1.69,;-8.55,-.92,;-7.22,-3.23,;-5.89,-4,;-5.89,-5.54,;-4.55,-6.31,;-3.22,-5.54,;-3.22,-4,;-4.55,-3.23,)|
CN1CCC[C@H]1COc1nc(N2CCN3CCC2CC3)c2cc(Cl)c(c(F)c2n1)-c1cc(O)cc2ccccc12 |r,wD:5.6,(5.23,-4.71,;6.32,-3.62,;7.87,-3.83,;8.57,-2.46,;7.48,-1.37,;6.1,-2.07,;4.77,-1.3,;3.44,-2.07,;2.1,-1.3,;2.1,.24,;.77,1.01,;.77,2.55,;-.62,3.22,;-.96,4.72,;,5.92,;1.54,5.92,;2.5,4.72,;2.16,3.22,;1.54,4.38,;,4.38,;-.56,.24,;-1.9,1.01,;-3.23,.24,;-4.56,1.01,;-3.23,-1.3,;-1.9,-2.07,;-1.9,-3.61,;-.56,-1.3,;.77,-2.07,;-4.56,-2.07,;-4.56,-3.61,;-5.9,-4.38,;-5.9,-5.92,;-7.23,-3.61,;-7.23,-2.07,;-8.57,-1.3,;-8.57,.24,;-7.23,1.01,;-5.9,.24,;-5.9,-1.3,)|
CN1CCC[C@H]1COc1nc(N2CCC3CCC(C2)N3)c2cc(Cl)c(c(F)c2n1)-c1nc(N)cc(C)c1C(F)(F)F |r,wD:5.6,(5.1,-4.66,;6.25,-3.63,;7.78,-3.92,;8.55,-2.59,;7.52,-1.45,;6.12,-2.07,;4.78,-1.3,;3.45,-2.07,;2.12,-1.3,;2.12,.24,;.78,1.01,;.78,2.55,;-.61,3.22,;-.95,4.72,;.01,5.92,;-.01,4.68,;1.32,3.91,;2.51,4.72,;2.17,3.22,;1.55,5.92,;-.55,.24,;-1.89,1.01,;-3.22,.24,;-4.55,1.01,;-3.22,-1.3,;-1.89,-2.07,;-1.89,-3.61,;-.55,-1.3,;.78,-2.07,;-4.55,-2.07,;-5.89,-1.3,;-7.22,-2.07,;-8.55,-1.3,;-7.22,-3.61,;-5.88,-4.43,;-5.89,-5.97,;-4.52,-3.64,;-3.18,-4.4,;-1.83,-5.15,;-2.42,-3.05,;-3.93,-5.74,)|
CN1CCC[C@H]1COc1nc(N2CC3CCC(C2)NC3)c2cc(Cl)c(c(F)c2n1)-c1nc(N)cc(C)c1C(F)(F)F |r,wD:5.6,(5.23,-4.71,;6.32,-3.62,;7.87,-3.83,;8.57,-2.46,;7.48,-1.37,;6.1,-2.07,;4.77,-1.3,;3.44,-2.07,;2.1,-1.3,;2.1,.24,;.77,1.01,;.77,2.55,;-.62,3.22,;-.96,4.72,;.53,5.12,;1.86,4.35,;2.5,4.72,;2.16,3.22,;1.54,5.92,;,5.92,;-.56,.24,;-1.9,1.01,;-3.23,.24,;-4.56,1.01,;-3.23,-1.3,;-1.9,-2.07,;-1.9,-3.61,;-.56,-1.3,;.77,-2.07,;-4.56,-2.07,;-5.9,-1.3,;-7.23,-2.07,;-8.57,-1.3,;-7.23,-3.61,;-5.91,-4.43,;-5.96,-5.97,;-4.52,-3.7,;-3.19,-4.48,;-1.86,-5.26,;-2.41,-3.15,;-3.97,-5.81,)|
CN1CCC[C@@]2(COc3nc(N4CC[C@H]5CC[C@@H](C4)N5)c4cc(Cl)c(c(F)c4n3)-c3nc(N)cc(C)c3C(F)(F)F)CCC[C@@H]12 |r,wU:5.5,wD:44.48,17.19,14.20,(9.34,-2.66,;8,-1.89,;8,-.35,;6.67,.42,;5.33,-.35,;5.33,-1.89,;4,-1.12,;2.67,-1.89,;1.33,-1.12,;1.33,.42,;,1.19,;,2.73,;-1.39,3.4,;-1.73,4.9,;-.77,6.1,;-.77,4.56,;.74,3.99,;1.73,4.9,;1.39,3.4,;.77,6.1,;-1.33,.42,;-2.67,1.19,;-4,.42,;-5.33,1.19,;-4,-1.12,;-2.67,-1.89,;-2.67,-3.43,;-1.33,-1.12,;,-1.89,;-5.33,-1.89,;-6.67,-1.12,;-8,-1.89,;-9.34,-1.12,;-8,-3.43,;-6.67,-4.2,;-6.67,-5.74,;-5.33,-3.43,;-4.56,-4.77,;-3.02,-4.77,;-5.33,-6.1,;-3.79,-6.1,;4.19,-2.92,;4.82,-4.33,;6.35,-4.17,;6.67,-2.66,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wU:23.24,wD:36.42,33.43,17.16,(-5.37,-5.52,;-5.32,-3.98,;-6.65,-3.16,;-6.65,-1.62,;-7.98,-.85,;-5.31,-.85,;-3.98,-1.62,;-2.64,-.85,;-2.64,.69,;-3.98,1.46,;-1.31,1.46,;.02,.69,;1.36,1.46,;2.69,.69,;2.69,-.85,;4.02,-1.62,;4.02,-3.16,;5.36,-3.93,;4.21,-4.96,;4.84,-6.37,;6.37,-6.21,;6.69,-4.7,;7.84,-3.67,;7.21,-2.27,;7.98,-.93,;5.68,-2.43,;1.36,-1.62,;.02,-.85,;-1.31,-1.62,;-1.31,-3.16,;1.36,3,;-.03,3.67,;-.37,5.17,;.59,6.37,;.59,4.83,;2.09,4.26,;3.09,5.17,;2.74,3.67,;2.13,6.37,;-3.93,-3.25,;-2.6,-4.03,;-1.27,-4.81,;-1.83,-2.7,;-3.38,-5.36,)|
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Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OC[C@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wU:17.16,23.24,wD:33.43,36.42,(-5.37,-5.52,;-5.32,-3.98,;-6.65,-3.16,;-6.65,-1.62,;-7.98,-.85,;-5.31,-.85,;-3.98,-1.62,;-2.64,-.85,;-2.64,.69,;-3.98,1.46,;-1.31,1.46,;.02,.69,;1.36,1.46,;2.69,.69,;2.69,-.85,;4.02,-1.62,;4.02,-3.16,;5.36,-3.93,;4.21,-4.96,;4.84,-6.37,;6.37,-6.21,;6.69,-4.7,;7.84,-3.67,;7.21,-2.27,;7.98,-.93,;5.68,-2.43,;1.36,-1.62,;.02,-.85,;-1.31,-1.62,;-1.31,-3.16,;1.36,3,;-.03,3.67,;-.37,5.17,;.59,6.37,;.59,4.83,;2.07,4.43,;3.09,5.17,;2.74,3.67,;2.13,6.37,;-3.93,-3.25,;-2.6,-4.03,;-1.27,-4.81,;-1.83,-2.7,;-3.38,-5.36,)|
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CN1CCC[C@H]1COc1nc(N2CC[C@H]3CC[C@@H](C2)N3)c2cc(Cl)c(c(F)c2n1)-c1cc(O)cc2ccccc12 |r,wD:17.20,14.21,5.6,(5.03,-4.26,;6.19,-3.25,;7.78,-3.54,;8.55,-2.21,;7.52,-1.06,;6.12,-1.69,;4.78,-.92,;3.45,-1.69,;2.12,-.92,;2.12,.62,;.78,1.39,;.78,2.93,;-.58,3.68,;-.86,5.2,;.07,6.31,;.04,4.83,;1.47,4.33,;2.53,5.09,;2.18,3.62,;1.64,6.31,;-.55,.62,;-1.89,1.39,;-3.22,.62,;-4.55,1.39,;-3.22,-.92,;-1.89,-1.69,;-1.89,-3.23,;-.55,-.92,;.78,-1.69,;-4.55,-1.69,;-5.89,-.92,;-7.22,-1.69,;-8.55,-.92,;-7.22,-3.23,;-5.89,-4,;-5.89,-5.54,;-4.55,-6.31,;-3.22,-5.54,;-3.22,-4,;-4.55,-3.23,)|
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CCc1cccc2cc(O)cc(-c3c(Cl)cc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@H]4CC[C@@H](C3)N4)c12 |r,wU:28.29,wD:22.21,41.47,38.48,(-1.74,-5.94,;-1.74,-4.4,;-3.23,-4,;-3.23,-5.54,;-4.56,-6.31,;-5.9,-5.54,;-5.9,-4,;-7.23,-3.23,;-7.23,-1.69,;-8.57,-.92,;-5.9,-.92,;-4.56,-1.69,;-3.23,-.92,;-3.23,.62,;-4.56,1.39,;-1.9,1.39,;-.56,.62,;.77,1.39,;2.1,.62,;2.1,-.92,;3.44,-1.69,;4.77,-.92,;6.1,-1.69,;5.02,-2.78,;5.71,-4.15,;7.24,-3.91,;7.48,-2.39,;8.57,-1.3,;7.87,.08,;8.57,1.45,;6.35,-.17,;.77,-1.69,;-.56,-.92,;-1.9,-1.69,;-1.9,-3.23,;.77,2.93,;-.62,3.6,;-.96,5.1,;,6.31,;,4.77,;1.44,4.13,;2.5,5.1,;2.16,3.6,;1.54,6.31,;-4.56,-3.23,)|
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Oc1cc(-c2c(Cl)cc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2c(F)cccc2c1 |r,wU:20.21,wD:14.13,33.39,30.40,(-8.65,-.92,;-7.31,-1.69,;-5.98,-.92,;-4.65,-1.69,;-3.31,-.92,;-3.31,.62,;-4.65,1.39,;-1.98,1.39,;-.64,.62,;.69,1.39,;2.02,.62,;2.02,-.92,;3.36,-1.69,;4.69,-.92,;6.02,-1.69,;4.88,-2.72,;5.51,-4.12,;7.04,-3.96,;7.36,-2.46,;8.5,-1.43,;7.88,-.02,;8.65,1.31,;6.34,-.18,;.69,-1.69,;-.64,-.92,;-1.98,-1.69,;-1.98,-3.23,;.69,2.93,;-.7,3.6,;-1.04,5.1,;-.08,6.31,;-.08,4.77,;1.33,4.01,;2.42,5.1,;2.08,3.6,;1.46,6.31,;-4.65,-3.23,;-3.31,-4,;-1.98,-4.77,;-3.31,-5.54,;-4.65,-6.31,;-5.98,-5.54,;-5.98,-4,;-7.31,-3.23,)|
Oc1cc(-c2c(Cl)cc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2ccccc2c1 |r,wU:20.21,wD:14.13,33.39,30.40,(-8.65,-.92,;-7.31,-1.69,;-5.98,-.92,;-4.65,-1.69,;-3.31,-.92,;-3.31,.62,;-4.65,1.39,;-1.98,1.39,;-.64,.62,;.69,1.39,;2.02,.62,;2.02,-.92,;3.36,-1.69,;4.69,-.92,;6.02,-1.69,;4.88,-2.72,;5.51,-4.12,;7.04,-3.96,;7.36,-2.46,;8.5,-1.43,;7.88,-.02,;8.65,1.31,;6.34,-.18,;.69,-1.69,;-.64,-.92,;-1.98,-1.69,;-1.98,-3.23,;.69,2.93,;-.7,3.6,;-1.04,5.1,;-.08,6.31,;-.08,4.77,;1.33,4.01,;2.42,5.1,;2.08,3.6,;1.46,6.31,;-4.65,-3.23,;-3.31,-4,;-3.31,-5.54,;-4.65,-6.31,;-5.98,-5.54,;-5.98,-4,;-7.31,-3.23,)|
Oc1cc(-c2c(Cl)cc3c(nc(OC[C@]45CCCN4C[C@@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2ccccc2c1 |r,wU:14.13,wD:33.39,30.40,20.21,(-8.65,-.92,;-7.31,-1.69,;-5.98,-.92,;-4.65,-1.69,;-3.31,-.92,;-3.31,.62,;-4.65,1.39,;-1.98,1.39,;-.64,.62,;.69,1.39,;2.02,.62,;2.02,-.92,;3.36,-1.69,;4.69,-.92,;6.02,-1.69,;4.88,-2.72,;5.51,-4.12,;7.04,-3.96,;7.36,-2.46,;8.5,-1.43,;7.88,-.02,;8.65,1.31,;6.34,-.18,;.69,-1.69,;-.64,-.92,;-1.98,-1.69,;-1.98,-3.23,;.69,2.93,;-.7,3.6,;-1.04,5.1,;-.08,6.31,;-.08,4.77,;1.33,4.01,;2.42,5.1,;2.08,3.6,;1.46,6.31,;-4.65,-3.23,;-3.31,-4,;-3.31,-5.54,;-4.65,-6.31,;-5.98,-5.54,;-5.98,-4,;-7.31,-3.23,)|
CN1CCC[C@@]2(COc3nc(N4CC[C@H]5CC[C@@H](C4)N5)c4ccc(c(F)c4n3)-c3cc(O)cc4ccccc34)CCC[C@@H]12 |r|
CN1CCC[C@@]2(COc3nc(N4CC[C@H]5CC[C@@H](C4)N5)c4ccc(c(F)c4n3)-c3cc(O)cc4cccc(F)c34)CCC[C@@H]12 |r|
CCc1cccc2cc(O)cc(-c3ccc4c(nc(OC[C@]56CCC[C@H]5N(C)CCC6)nc4c3F)N3CC[C@H]4CC[C@@H](C3)N4)c12 |r|
CN1CCC[C@@]2(COc3nc(N4CC[C@H]5CC[C@@H](C4)N5)c4ccc(c(F)c4n3)-c3cc(O)cc4ccc(F)c(C#C)c34)CCC[C@@H]12 |r|
CN(C)CC1(COc2nc(N3CC[C@H]4CC[C@@H](C3)N4)c3cc(Cl)c(c(F)c3n2)-c2nc(N)cc(C)c2C(F)(F)F)CC1 |r,wD:13.19,16.18,(9.43,-.13,;8.34,-1.22,;8.74,-2.71,;6.85,-.82,;5.76,-1.91,;4.43,-1.14,;3.1,-1.91,;1.76,-1.14,;1.76,.4,;.43,1.17,;.43,2.71,;-.96,3.38,;-1.3,4.88,;-.34,6.08,;-.34,4.54,;1.15,4.14,;2.16,4.88,;1.82,3.38,;1.2,6.08,;-.91,.4,;-2.24,1.17,;-3.57,.4,;-4.91,1.17,;-3.57,-1.14,;-2.24,-1.91,;-2.24,-3.45,;-.91,-1.14,;.43,-1.91,;-5.43,-2.23,;-6.76,-1.46,;-8.1,-2.23,;-9.43,-1.46,;-8.1,-3.77,;-6.76,-4.54,;-6.76,-6.08,;-5.43,-3.77,;-4.09,-4.54,;-2.76,-5.31,;-4.09,-6.08,;-2.76,-3.77,;4.99,-3.25,;6.53,-3.25,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5C6CCC5COC6)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:39.46,36.47,(-5.67,-5.54,;-5.67,-4,;-7,-3.23,;-7,-1.69,;-8.33,-.92,;-5.67,-.93,;-4.33,-1.69,;-2.34,-.53,;-2.34,1.01,;-3.67,1.78,;-1,1.78,;.33,1.01,;1.67,1.78,;3,1.01,;3,-.53,;4.33,-1.3,;5.67,-.53,;7,-1.3,;5.67,-2.07,;5.67,-3.61,;4.33,-4.38,;4.92,-5.17,;6.41,-5.17,;7,-4.38,;7,-5.92,;5.67,-6.69,;4.33,-5.92,;8.33,-2.07,;8.33,-.53,;1.67,-1.3,;.33,-.53,;-1,-1.3,;-1,-2.84,;1.67,3.32,;.28,3.99,;-.06,5.49,;.9,6.69,;.9,5.15,;2.31,4.4,;3.4,5.49,;3.05,3.99,;2.44,6.69,;-4.33,-3.23,;-3,-4.01,;-1.67,-3.24,;-3.01,-5.55,;-1.67,-4.78,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5CCCC(F)C5)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,w:23.23,wD:38.44,35.45,(-5.67,-5.54,;-5.67,-4,;-7,-3.23,;-7,-1.69,;-8.33,-.92,;-5.67,-.93,;-4.33,-1.69,;-2.34,-.53,;-2.34,1.01,;-3.67,1.78,;-1,1.78,;.33,1.01,;1.67,1.78,;3,1.01,;3,-.53,;4.33,-1.3,;5.67,-.53,;7,-1.3,;5.67,-2.07,;5.67,-3.61,;4.33,-4.38,;4.33,-5.92,;5.67,-6.69,;7,-5.92,;8.33,-6.69,;7,-4.38,;8.33,-2.07,;8.33,-.53,;1.67,-1.3,;.33,-.53,;-1,-1.3,;-1,-2.84,;1.67,3.32,;.28,3.99,;-.06,5.49,;.9,6.69,;.9,5.15,;2.31,4.4,;3.4,5.49,;3.05,3.99,;2.44,6.69,;-4.33,-3.23,;-3,-4.01,;-1.67,-3.24,;-3.01,-5.55,;-1.67,-4.78,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5CC[C@@H](F)C5)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:37.43,34.44,22.22,(-5.67,-5.22,;-5.67,-3.68,;-7,-2.92,;-7,-1.38,;-8.33,-.61,;-5.67,-.62,;-4.33,-1.38,;-2.34,-.22,;-2.34,1.32,;-3.67,2.09,;-1,2.09,;.33,1.32,;1.67,2.09,;3,1.32,;3,-.22,;4.33,-.99,;5.67,-.22,;7,-.99,;5.67,-1.76,;5.67,-3.3,;4.42,-4.21,;4.9,-5.67,;6.44,-5.67,;7.21,-7,;6.91,-4.21,;8.33,-1.76,;8.33,-.22,;1.67,-.99,;.33,-.22,;-1,-.99,;-1,-2.53,;1.67,3.63,;.28,4.3,;-.06,5.8,;.9,7,;.9,5.46,;2.31,4.71,;3.4,5.8,;3.05,4.3,;2.44,7,;-4.33,-2.92,;-3,-3.69,;-1.67,-2.93,;-3.01,-5.23,;-1.67,-4.46,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OC[C@@]45CCCN4C[C@H](C5)OC(F)F)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:39.45,36.46,17.16,23.26,(-6.32,-6.11,;-6.32,-4.57,;-7.65,-3.81,;-7.65,-2.27,;-8.98,-1.49,;-6.32,-1.5,;-4.98,-2.27,;-2.98,-1.1,;-2.98,.44,;-4.31,1.21,;-1.65,1.21,;-.31,.44,;1.02,1.21,;2.36,.44,;2.36,-1.1,;3.69,-1.87,;5.02,-1.1,;6.36,-1.87,;5.21,-2.9,;5.84,-4.31,;7.37,-4.15,;7.69,-2.64,;8.83,-1.61,;8.21,-.21,;6.68,-.37,;8.98,1.13,;10.52,1.13,;11.29,2.46,;11.29,-.21,;1.02,-1.87,;-.31,-1.1,;-1.65,-1.87,;-1.65,-3.41,;1.02,2.75,;-.37,3.41,;-.71,4.92,;.25,6.12,;.25,4.58,;1.66,3.83,;2.75,4.92,;2.41,3.41,;1.79,6.12,;-4.98,-3.81,;-3.65,-4.58,;-2.31,-3.81,;-3.65,-6.12,;-2.31,-5.35,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5CCOCC5)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:37.43,34.44,(-5.67,-5.54,;-5.67,-4,;-7,-3.23,;-7,-1.69,;-8.33,-.92,;-5.67,-.93,;-4.33,-1.69,;-2.34,-.53,;-2.34,1.01,;-3.67,1.78,;-1,1.78,;.33,1.01,;1.67,1.78,;3,1.01,;3,-.53,;4.33,-1.3,;5.67,-.53,;7,-1.3,;5.67,-2.07,;5.67,-3.61,;4.33,-4.38,;4.33,-5.92,;5.67,-6.69,;7,-5.92,;7,-4.38,;8.33,-2.07,;8.33,-.53,;1.67,-1.3,;.33,-.53,;-1,-1.3,;-1,-2.84,;1.67,3.32,;.28,3.99,;-.06,5.49,;.9,6.69,;.9,5.15,;2.31,4.4,;3.4,5.49,;3.05,3.99,;2.44,6.69,;-4.33,-3.23,;-3,-4.01,;-1.67,-3.24,;-3.01,-5.55,;-1.67,-4.78,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5CCCCC5)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:37.43,34.44,(-5.67,-5.54,;-5.67,-4,;-7,-3.23,;-7,-1.69,;-8.33,-.92,;-5.67,-.93,;-4.33,-1.69,;-2.34,-.53,;-2.34,1.01,;-3.67,1.78,;-1,1.78,;.33,1.01,;1.67,1.78,;3,1.01,;3,-.53,;4.33,-1.3,;5.67,-.53,;7,-1.3,;5.67,-2.07,;5.67,-3.61,;4.33,-4.38,;4.33,-5.92,;5.67,-6.69,;7,-5.92,;7,-4.38,;8.33,-2.07,;8.33,-.53,;1.67,-1.3,;.33,-.53,;-1,-1.3,;-1,-2.84,;1.67,3.32,;.28,3.99,;-.06,5.49,;.9,6.69,;.9,5.15,;2.31,4.4,;3.4,5.49,;3.05,3.99,;2.44,6.69,;-4.33,-3.23,;-3,-4.01,;-1.67,-3.24,;-3.01,-5.55,;-1.67,-4.78,)|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OCC4(CN5CCCC(F)C5)CC4)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wD:38.44,35.45,(-5.67,-5.54,;-5.67,-4,;-7,-3.23,;-7,-1.69,;-8.33,-.92,;-5.67,-.93,;-4.33,-1.69,;-2.34,-.53,;-2.34,1.01,;-3.67,1.78,;-1,1.78,;.33,1.01,;1.67,1.78,;3,1.01,;3,-.53,;4.33,-1.3,;5.67,-.53,;7,-1.3,;5.67,-2.07,;5.67,-3.61,;4.33,-4.38,;4.33,-5.92,;5.67,-6.69,;7,-5.92,;8.33,-6.69,;7,-4.38,;8.33,-2.07,;8.33,-.53,;1.67,-1.3,;.33,-.53,;-1,-1.3,;-1,-2.84,;1.67,3.32,;.28,3.99,;-.06,5.49,;.9,6.69,;.9,5.15,;2.31,4.4,;3.4,5.49,;3.05,3.99,;2.44,6.69,;-4.33,-3.23,;-3,-4.01,;-1.67,-3.24,;-3.01,-5.55,;-1.67,-4.78,)|
CN(C)CC1(COc2nc(N3CC[C@H]4CC[C@@H](C3)N4)c3ccc(c(F)c3n2)-c2cc(O)cc3ccc(F)c(C#C)c23)CC1 |r|
Nc1cc(-c2ccc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2c(F)cccc2c1 |r|
C[C@H]1CN2CCC[C@@]2(COc2nc(N3CC[C@@H]4CC[C@H](C3)N4)c3ccc(c(F)c3n2)-c2cc(N)cc3cccc(F)c23)C1 |r|
Nc1cc2cccc(F)c2c(n1)-c1ccc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CC[C@H]2CC[C@@H](C1)N2 |r|
CCc1cccc2cc(N)cc(-c3ccc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@H]4CC[C@@H](C3)N4)c12 |r|
Nc1cc(-c2ccc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2c(C#C)c(F)ccc2c1 |r|
Nc1cc(-c2ccc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c2ccccc2c1 |r|
CCc1cccc2cccc(-c3ccc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@H]4CC[C@@H](C3)N4)c12 |r|
Cc1cc(N)nc(-c2ccc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r|
Cc1cc(N)nc(-c2ccc3c(nc(OC[C@]45CCCN4C[C@H](F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r|
Cc1cc(N)nc(-c2ccc3c(nc(OCC45CCCN4CC(F)(F)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,w:15.15|
Cc1cc(N)nc(-c2c(Cl)cc3c(nc(OC[C@@]45C[C@@H](F)CN4CC4(CC4)C5)nc3c2F)N2CC[C@H]3CC[C@@H](C2)N3)c1C(F)(F)F |r,wU:17.16,19.19,wD:38.45,35.46,(-5.32,-4.76,;-5.3,-3.22,;-6.65,-2.41,;-6.65,-.87,;-7.98,-.1,;-5.31,-.1,;-3.98,-.87,;-2.64,-.1,;-2.64,1.44,;-3.98,2.21,;-1.31,2.21,;.02,1.44,;1.36,2.21,;2.69,1.44,;2.69,-.1,;4.02,-.87,;4.02,-2.41,;5.36,-3.18,;5.68,-1.67,;7.21,-1.51,;7.98,-.18,;7.84,-2.92,;6.69,-3.95,;6.37,-5.46,;4.84,-5.62,;3.51,-6.39,;4.84,-7.16,;4.21,-4.21,;1.36,-.87,;.02,-.1,;-1.31,-.87,;-1.31,-2.41,;1.36,3.75,;-.06,4.35,;-.48,5.83,;.42,7.08,;.42,5.57,;1.91,5.11,;2.98,6,;2.71,4.49,;1.96,7.16,;-3.94,-2.44,;-2.6,-3.2,;-1.26,-3.95,;-1.85,-1.85,;-3.36,-4.54,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@@H](O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H](O)C[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ccc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H](O)C[C@H]3C(=O)OC)c12 |r|
Cc1ccc2[nH]ncc2c1-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CCCC2(CCO2)C1 |r,wU:25.28,wD:19.20,(-3.41,-5.3,;-4.74,-4.53,;-6.07,-5.3,;-7.41,-4.53,;-7.41,-2.99,;-8.55,-1.96,;-7.93,-.55,;-6.39,-.71,;-6.07,-2.22,;-4.74,-2.99,;-3.41,-2.22,;-3.41,-.68,;-2.07,.09,;-.74,-.68,;.6,.09,;1.93,-.68,;1.93,-2.22,;3.26,-2.99,;4.6,-2.22,;5.93,-2.99,;4.79,-4.02,;5.41,-5.43,;6.94,-5.27,;7.26,-3.76,;8.41,-2.73,;7.78,-1.32,;8.55,.01,;6.25,-1.48,;.6,-2.99,;-.74,-2.22,;-2.07,-2.99,;-2.07,-4.53,;.6,1.63,;-.74,2.4,;-.74,3.94,;.6,4.71,;1.93,3.94,;2.33,5.43,;3.81,5.03,;3.42,3.54,;1.93,2.4,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3C(N)=O)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCC4(CCO4)C3)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3C(=O)OC)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3c(Cl)cc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCO4)C3)c12 |r,wU:29.30,wD:23.22,(-.95,-4.43,;-2.29,-3.66,;-3.62,-4.43,;-3.62,-5.97,;-2.29,-6.74,;-4.95,-6.74,;-6.29,-5.97,;-6.29,-4.43,;-7.62,-3.66,;-7.62,-2.12,;-8.95,-1.35,;-6.29,-1.35,;-4.95,-2.12,;-3,-.91,;-3,.63,;-4.34,1.4,;-1.67,1.4,;-.34,.63,;1,1.4,;2.33,.63,;2.33,-.91,;3.67,-1.68,;5,-.91,;6.33,-1.68,;5.19,-2.71,;5.81,-4.12,;7.35,-3.96,;7.67,-2.45,;8.81,-1.42,;8.18,-.01,;8.95,1.32,;6.65,-.17,;1,-1.68,;-.34,-.91,;-1.67,-1.68,;-1.67,-3.22,;1,2.94,;-.34,3.71,;-.34,5.25,;1,6.02,;2.33,5.25,;2.73,6.74,;4.22,6.34,;3.82,4.85,;2.33,3.71,;-4.95,-3.66,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3C(O)=O)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCO4)C3)c12 |r,wU:29.30,wD:23.22,(-.95,-4.43,;-2.29,-3.66,;-3.62,-4.43,;-3.62,-5.97,;-2.29,-6.74,;-4.95,-6.74,;-6.29,-5.97,;-6.29,-4.43,;-7.62,-3.66,;-7.62,-2.12,;-8.95,-1.35,;-6.29,-1.35,;-4.95,-2.12,;-3,-.91,;-3,.63,;-4.34,1.4,;-1.67,1.4,;-.34,.63,;1,1.4,;2.33,.63,;2.33,-.91,;3.67,-1.68,;5,-.91,;6.33,-1.68,;5.19,-2.71,;5.81,-4.12,;7.35,-3.96,;7.67,-2.45,;8.81,-1.42,;8.18,-.01,;8.95,1.32,;6.65,-.17,;1,-1.68,;-.34,-.91,;-1.67,-1.68,;-1.67,-3.22,;1,2.94,;-.34,3.71,;-.34,5.25,;1,6.02,;2.33,5.25,;2.73,6.74,;4.22,6.34,;3.82,4.85,;2.33,3.71,;-4.95,-3.66,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3[C@H]4CC[C@@H]3C[C@H](O)C4)c12 |r,THB:17:35:40.41.43:37.38|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(CCC4O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3[C@H]4CC[C@@H]3C[C@@H](O)C4)c12 |r,THB:17:35:40.41.43:37.38|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(CCC4=O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C4CCC3COC4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)C3CCCC4(C3)OCCO4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CCC(C3)O4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CCOC4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC33COC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCOCC6)CC5)nc4c3F)N3CCCC4(CCO4)C3)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C4CCC3CC4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@H]5C[C@@H](F)CN5C)nc4c3F)N3CCCC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC(C)(O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCN4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C4CCC3CCC4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H](C3)OC)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC(C)(O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC3c3ccccc3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4CC(CO)(C4)C3)c12 |r,wU:28.29,wD:22.21,(-4.65,2.7,;-4.65,1.16,;-5.98,.39,;-7.31,1.16,;-7.31,2.7,;-8.65,.39,;-8.65,-1.15,;-7.31,-1.92,;-7.31,-3.46,;-5.98,-4.23,;-5.98,-5.78,;-4.65,-3.46,;-4.65,-1.92,;-3.31,-1.15,;-3.31,.38,;-1.98,1.15,;-.64,.38,;.69,1.15,;2.02,.38,;2.02,-1.15,;3.36,-1.93,;4.69,-1.15,;6.02,-1.93,;4.88,-2.96,;5.51,-4.36,;7.04,-4.2,;7.36,-2.69,;8.5,-1.66,;7.88,-.26,;8.65,1.08,;6.34,-.42,;.69,-1.93,;-.64,-1.15,;-1.98,-1.93,;-1.98,-3.47,;.69,2.69,;-.64,3.47,;-.64,5,;.69,5.78,;2.02,5,;3.36,5.78,;4.69,5.01,;.69,4.23,;2.02,3.47,;-5.98,-1.15,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC(C3)c3ccccc3)c12 |r|
Oc1cc(-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCCC3(CCO3)C2)c2ccccc2c1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC(F)(F)C[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCCCC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@@]3(C)CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCCC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3CN)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@H](C)OC)nc4c3F)N3CCCC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC3c3cccnc3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCN(C)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC(Cl)(CCO)C3)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3ccc(c(F)c3n2)-c2c(C)ccc3[nH]ncc23)CC1 |r,wD:14.17,(7.91,-4.59,;7.91,-3.05,;9.24,-2.28,;6.57,-2.28,;5.24,-3.05,;3.91,-2.28,;2.57,-3.05,;1.24,-2.28,;1.24,-.74,;-.09,.03,;-.09,1.57,;1.24,2.34,;1.24,3.88,;-.09,4.65,;-1.43,3.88,;-2.92,3.48,;-3.31,4.97,;-1.83,5.36,;-1.43,2.34,;-1.43,-.74,;-2.76,.03,;-4.1,-.74,;-4.1,-2.28,;-2.76,-3.05,;-2.76,-4.59,;-1.43,-2.28,;-.09,-3.05,;-5.43,-3.05,;-5.43,-4.59,;-4.1,-5.36,;-6.76,-5.36,;-8.1,-4.59,;-8.1,-3.05,;-9.24,-2.02,;-8.61,-.62,;-7.08,-.78,;-6.76,-2.28,;4.47,-4.39,;6.01,-4.39,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@@H]4C[C@@H](O)[C@H]3C4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ccc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(NC5CC6(CCC6)C5)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@](C)(O)C3)c3cnc(c(F)c3n2)-c2cc(N)cc(Cl)c2C(F)(F)F)CC1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@H](C3)C(C)(C)O)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3cnc(c(F)c3n2)-c2cc(N)ccc2-c2cccs2)CC1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3CN3CCCC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC7(COC7)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCN([C@H](C)C3)C(C)=O)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC7(CC(C7)N7CCC(CC7)c7ccc8cnn(C)c8c7)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@@H](CO)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC7(CC(C7)N7CCOCC7)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@@H](N)C[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC7(CC(C7)N7CCCCC7)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCN[C@H](C)C3)c12 |r|
CCc1c(F)ccc2cc(OC(=O)C(C)C)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@@H]4C[C@H]3CO4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC7(CCC7)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(CC(O)C4)C3)c12 |r|
CCc1c(F)ccc2cc(OC(=O)N(C)C)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@@H]4C[C@H](O)[C@H]3C4)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3cnc(c(F)c3n2)-c2cc(O)ccc2-c2cccs2)CC1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC[C@@H](N)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC(C)(C)CN(C)C)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H](F)C[C@H]3CO)c12 |r|
CCN(CC)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3cnc(c(F)c3n2)-c2cc(O)cc3ccc(F)c(CC)c23)CC1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(C3)CCCCC4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CC(F)(F)C6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC(O)(CO)CC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC(F)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC(F)(F)CC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CNC(=O)O4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CC(N)=O)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(C3)CC(=O)C4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N(C)CC(C)(C)O)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H]3C(C)(C)O)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC(CC6)C(O)=O)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H]4C[C@@H]3C(=O)N4)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(OC[C@@]56CCCN5C[C@H](F)C6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3cnc(c(F)c3n2)-c2ccc(F)c3sc(N)c(C#N)c23)CC1 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC[C@H](CO)C3)c12 |r|
CN(C)CC1(COc2nc(N3CCC=CC3)c3cnc(c(F)c3n2)-c2cc(O)cc3ccc(F)c(C#C)c23)CC1 |c:13|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC(CC3)C(C)=O)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CC5)N(C)C)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(COC4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CC4CC(C4)C3)c12 |(-5.33,2.7,;-5.33,1.16,;-6.67,.39,;-8,1.16,;-8,2.7,;-9.34,.39,;-9.34,-1.15,;-8,-1.92,;-8,-3.46,;-6.67,-4.23,;-6.67,-5.78,;-5.33,-3.46,;-5.33,-1.92,;-4,-1.15,;-4,.38,;-2.67,1.15,;-1.33,.38,;,1.15,;1.33,.38,;1.33,-1.15,;2.67,-1.93,;4,-1.15,;5.33,-1.92,;6.67,-1.15,;8,-1.92,;8,-3.46,;9.34,-1.15,;4.56,-3.26,;6.1,-3.26,;,-1.93,;-1.33,-1.15,;-2.67,-1.93,;-2.67,-3.47,;,2.69,;1.33,3.47,;1.33,5,;,5.78,;-1.33,5,;,4.23,;-1.33,3.47,;-6.67,-1.15,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H](O)[C@@H](O)[C@H](O)[C@H]3CO)c12 |r|
CN(C)CC1(COc2nc(N3CCC[C@]4(CCO4)C3)c3cc(Cl)c(c(F)c3n2)-c2ccc(F)c3sc(N)c(C#N)c23)CC1 |r,wU:14.17,(8.24,-4.48,;8.24,-2.94,;9.58,-2.17,;6.91,-2.17,;5.58,-2.94,;4.24,-2.17,;2.91,-2.94,;1.58,-2.17,;1.58,-.63,;.24,.14,;.24,1.68,;-1.09,2.45,;-1.09,3.99,;.24,4.76,;1.58,3.99,;3.06,3.59,;3.46,5.08,;1.97,5.47,;1.58,2.45,;-1.09,-.63,;-2.43,.14,;-3.76,-.63,;-5.09,.14,;-3.76,-2.17,;-2.43,-2.94,;-2.43,-4.48,;-1.09,-2.17,;.24,-2.94,;-5.58,-3.16,;-5.58,-4.7,;-6.91,-5.47,;-8.24,-4.7,;-9.58,-5.47,;-8.24,-3.16,;-9.39,-2.13,;-8.76,-.73,;-9.53,.61,;-7.23,-.89,;-6.2,.26,;-5.17,1.4,;-6.91,-2.39,;4.81,-4.28,;6.35,-4.28,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4CC4(O)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCC(CC3)OC)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(COC4)CC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN6CCC(F)C6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r,w:27.27|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CC4(COC4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCC(CC3)C#N)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3C[C@H](N)C[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCCCC3)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC(C)(CO)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCC(O)CC3)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3[C@@H]4C[C@@H]4C[C@H]3CO)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCCC(C3)OC)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CCCC4=O)CC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCCCC(O)C3)c12
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CCC4=O)CC3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)C)CC5)nc4c3F)N3CCC=CCC3)c12 |c:39|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CCO4)CC3)c12 |r|
Nc1sc2c(F)ccc(-c3c(Cl)cc4c(nc(OCC5(CN6CCCCC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c2c1C#N |r,wD:37.44,(-10.2,.61,;-9.43,-.73,;-10.06,-2.13,;-8.91,-3.16,;-8.91,-4.7,;-10.24,-5.47,;-7.58,-5.47,;-6.24,-4.7,;-6.24,-3.16,;-4.43,-2.17,;-4.43,-.63,;-4.82,.85,;-3.09,.14,;-1.76,-.63,;-.43,.14,;.91,-.63,;.91,-2.17,;2.24,-2.94,;3.58,-2.17,;4.91,-2.94,;6.24,-2.17,;7.58,-2.94,;7.58,-4.48,;8.91,-5.25,;10.24,-4.48,;10.24,-2.94,;8.91,-2.17,;4.14,-4.28,;5.68,-4.28,;-.43,-2.94,;-1.76,-2.17,;-3.09,-2.94,;-3.09,-4.48,;-.43,1.68,;.91,2.45,;.91,3.99,;-.43,4.76,;-1.76,3.99,;-3.25,3.59,;-3.64,5.08,;-2.16,5.47,;-1.76,2.45,;-7.58,-2.39,;-7.9,-.89,;-6.87,.26,;-5.84,1.4,)|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(COC4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)CC6COC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC4(CCO4)C3)c12 |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OCC5(CN(C)CC6CCOC6)CC5)nc4c3F)N3CCC[C@]4(CCO4)C3)c12 |r|
Nc1cc(Cl)c(c(c1)-c1ncc2c(nc(OC[C@@]34CCCN3C[C@H](F)C4)nc2c1F)N1CCCC2(COC2)C1)C(F)(F)F |r|
CCc1c(F)ccc2cc(O)cc(-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCC4(CCOC4)C3)c12 |r|
Oc1cc2-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@H](C3)NC(=O)CCCc3cccc(c1)c23 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CC[C@@H](F)C(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3cccc(CCCC(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3ccc(F)c(CCCC(=O)N2)c13 |r|
CN1C[C@H](F)C[C@H]1COc1nc2N3CCC[C@](C)(C3)NC(=O)CCCc3c(F)ccc4cc(O)cc(-c5ncc2c(n1)c5F)c34 |r|
COc1nc2N3CCC[C@](C)(C3)NC(=O)CCCc3c(F)ccc4cc(O)cc(-c5ncc2c(n1)c5F)c34 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCCC(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3cccc(CCCCC(=O)N2)c13 |r|
Oc1cc2-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCCN(CC3)C(=O)CCCCc3cccc(c1)c23 |r|
C[C@@]12CCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3ccc(F)c(CCCC(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCC(F)C(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CC[C@H](F)C(=O)N2)c13 |r|
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C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ccc13)-c1cc(O)cc3ccc(F)c(CCCC(=O)N2)c13 |r|
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Cc1c-2ncc3c(nc(OCC(C)(C)O)nc13)N1CCC[C@](C)(C1)NC(=O)CCCc1c(F)ccc3cc(O)cc-2c13 |r|
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C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3CCC[C@@H](CCCC(=O)N2)c13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)CCCc4cccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)CC\C=C/c4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r,c:26|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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Cc1cc2[nH]ncc2c-2c1CCCOC(=O)O[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)CC1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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Oc1cc2-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCC[C@](CF)(C3)OC(=O)CCCc3c(F)ccc(c1)c23 |r|
C[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@](C)(C4)OC(=O)CCCc4c(F)ccc5cc(O)cc(-c6ncc3c(n2)c6F)c45)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCCCCC1(O)CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)OC[C@@H]4C[C@@H]4c4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)OC[C@H]4C[C@H]4c4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cc(O)cc3ccc(F)c(CCCCC(=O)N2)c13 |r|
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Cc1cc2[nH]ncc2c-2c1CCC[C@H](F)C(=O)N[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCCC1=O)c(C)cc1[nH]ncc21 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCC[C@H](F)C1=O)c(C)cc1[nH]ncc21 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCC[C@@H](F)C1=O)c(C)cc1[nH]ncc21 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCCC1=O)c(Cl)cc1[nH]ncc21 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N[C@@H]1CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCC(F)C(=O)N[C@@H]1COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N1CC3(C1)CCCN(C3)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r,wU:30.33,wD:36.41,(8.72,-1.45,;7.39,-2.22,;7.39,-3.76,;6.06,-4.53,;5.74,-6.04,;4.2,-6.2,;3.58,-4.79,;4.72,-3.76,;4.72,-2.22,;6.06,-1.45,;6.06,.09,;4.72,.86,;4.72,2.4,;3.39,3.17,;3.39,4.71,;4.72,5.48,;2.61,5.8,;2.21,4.31,;.72,4.71,;1.12,6.2,;-.61,5.48,;-1.95,4.71,;-1.95,3.17,;-.61,2.4,;.72,3.17,;-.61,.86,;-1.95,.09,;-1.95,-1.45,;-3.28,-2.22,;-4.61,-1.45,;-5.95,-2.22,;-4.75,-3.19,;-5.3,-4.63,;-6.84,-4.55,;-7.24,-3.06,;-8.44,-2.09,;-7.88,-.65,;-8.72,.64,;-6.35,-.73,;-.61,-2.22,;.72,-1.45,;2.05,-2.22,;2.05,-3.76,;3.39,-1.45,;3.39,.09,;2.05,.86,;.72,.09,)|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N1CC3CCN(CC3C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N1C[C@@H]3CCN(CC3C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)NC(=O)CCCCc4c(Cl)cccc4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC5CCN([C@H]5C4)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@@H]5CCN([C@@H]5C4)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@H]5CCN([C@H]5C4)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N1CC[C@@H]3CCN(C[C@H]13)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
CN1C2COCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCCC1=O)c(Cl)cc1[nH]ncc21 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N[C@@H]1COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N[C@]1(C)COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)NC(=O)CCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)CCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@@H]5CCN([C@@H]5C4)C(=O)CCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@H]5CCN([C@H]5C4)C(=O)CCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3cc(nnc23)-c2c(CCCCC1=O)c(Cl)cc1[nH]ncc21 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCOC1=O)c(Cl)cc1[nH]ncc21 |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)N1CC[C@@H]3CCN(C[C@H]13)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
CC12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCOC(=O)N2)c13 |r|
C[C@@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCOC(=O)N2)c13 |r|
C[C@]12CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCOC(=O)N2)c13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)NC(=O)OCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)OC1CN(CC3(CC3)C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)OC1CN(CC(F)(F)C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)OC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)O[C@@H]1COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CN1C[C@H](F)C[C@H]1COc1nc2N3CCCC[C@H](C3)OC(=O)CCCCc3c(Cl)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)OC1CC[C@@H]3CC[C@H]1N3c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r,THB:25:24:19.18.17:21.22|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)CCCCc4c(cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C(F)(F)F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC(C4)CC(=O)OCCc4cccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
CC1CCCc2c(Cl)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCC[C@H](C2)OC1=O |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)OC(=O)COCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CC1COC(=O)O[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(Cl)cc1[nH]ncc21 |r|
CN1C[C@H](F)C[C@H]1COc1nc2N3CCCC[C@H](C3)OC(=O)OCCCc3c(C)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)O[C@H]1CN(CC[C@H]1F)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
C[C@@H]1CCN2C[C@@H]1OC(=O)OCCCc1c(C)cc3[nH]ncc3c1-c1ncc3c2nc(OC[C@@]24CCCN2C[C@H](F)C4)nc3c1F |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)O[C@@H]1C[C@H](F)CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)OC1CC[C@@H]3CC[C@H]1N3c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r,THB:25:24:17.18.19:21.22|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)O[C@@H]1COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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CN1CCO[C@@H](COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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Cc1cc2[nH]ncc2c-2c1CCCCOC[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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Cc1cc2[nH]ncc2c-2c1CCCCCO[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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Cc1cc2[nH]ncc2c-2c1CC\C=C\CO[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r,t:14|
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Cc1cc2[nH]ncc2c-2c1CCCn1ccc(n1)C1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)Cn4ncc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
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Cc1cc2[nH]ncc2c-2c1CCCC(F)C(=O)N[C@@H]1CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N[C@H]1CN(C[C@H]3C[C@@H]13)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5C[C@H]5[C@H](C4)NC(=O)[C@H](F)CCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@H]5CCN([C@H]5C4)C(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CN1[C@@H]2COCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCOC1=O)c(Cl)cc1[nH]ncc21 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4C[C@H]5C[C@H]5[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CN1CCC[C@H]1COc1nc2N3CCOC[C@@](C)(C3)OC(=O)OCCCc3c(Cl)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
CN1CCC[C@H]1COc1nc2N3CCOC[C@](C)(C3)OC(=O)OCCCc3c(Cl)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
CN1CCC[C@H]1COc1nc2N3CCOC[C@@](C)(C3)OC(=O)OCCCc3c(C)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
CN1CCC[C@H]1COc1nc2N3CCOC[C@](C)(C3)OC(=O)OCCCc3c(C)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@H]3[C@@H](F)CN4CCCC34)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(F)cc2[nH]ncc12 |r|
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F[C@H]1CN2CCCC2[C@@H]1COc1nc2N3CCOC[C@H](C3)OC(=O)OCCCc3c(Cl)cccc3-c3ncc2c(n1)c3F |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4c(F)cc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ccc3c(n2)c4F)C1 |r|
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C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=S)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc(Cl)c1CCCOC(=O)O2 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCc4cccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
CN1CCC[C@H]1COc1nc2N3CCCC[C@H](C3)OC(=O)OCCCc3c(Cl)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
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CN1CCC[C@H]1COc1nc2N3CCCC4(CC(C4)OC(=O)OCCc4c(C)cc5[nH]ncc5c4-c4ncc2c(n1)c4F)C3 |r,wU:5.6,(-5.13,-4.78,;-6.28,-3.75,;-7.78,-4.07,;-8.55,-2.74,;-7.52,-1.59,;-6.12,-2.22,;-4.78,-1.45,;-3.45,-2.22,;-2.12,-1.45,;-2.12,.09,;-.78,.86,;-.78,2.4,;-2.12,3.17,;-2.12,4.71,;-.78,5.48,;.55,4.71,;2.04,4.31,;2.44,5.8,;.95,6.2,;3.53,4.71,;3.22,3.17,;1.89,2.4,;4.55,2.4,;4.55,.86,;5.89,.09,;5.89,-1.45,;7.22,-2.22,;6.32,-3.47,;7.22,-3.76,;5.89,-4.53,;5.57,-6.04,;4.03,-6.2,;3.41,-4.79,;4.55,-3.76,;4.55,-2.22,;3.22,-1.45,;3.22,.09,;1.89,.86,;.55,.09,;.55,-1.45,;-.78,-2.22,;1.89,-2.22,;1.89,-3.76,;.55,3.17,)|
CN1CCC[C@H]1COc1nc2N3CCCC[C@H](C3)OC(=O)OCCCc3c(C)cc4[nH]ncc4c3-c3ncc2c(n1)c3F |r|
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C[C@@]12COCCN(C1)c1nc(OCC34CCCN3CCC4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
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CC(=O)n1ncc2c-3c(CCCOC(=O)O[C@@H]4COCCN(C4)c4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc5c(F)c-3ncc45)c(Cl)cc12 |r|
C[C@H]1COC(=O)O[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(C)cc1[nH]ncc21 |r|
C[C@@H]1COC(=O)O[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(C)cc1[nH]ncc21 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc(cc4-c4ncc3c(n2)c4F)C#N)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)COC(=O)OCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCOC(=O)OC[C@H]1CN(CCO1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOCC(C4)COC(=O)OCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)CCOCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c2-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCO[C@H](C3)COCC[C@H]3C[C@H]3c12 |r|
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Cc1cc2[nH]ncc2c-2c1CCCCOCC1CN(CCC1(F)F)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC(CC5(CC5)C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOCC(C4)CC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)Cc4ncc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC(C4)Cc4ncn(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
O[C@H]1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCc3cnc1o3)c(Cl)cc1[nH]ncc21 |r|
O[C@@H]1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCc3cnc1o3)c(Cl)cc1[nH]ncc21 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC(C4)CCC(=O)CCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCC[C@H](O)CC[C@@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCC[C@H](O)CC[C@H]1CCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)COCCCCc4c(F)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@@H](C4)COCCCCc4c(F)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
C[C@H]1OCCCCc2c(C)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCO[C@@H]1C2 |r|
C[C@@H]1OCCCCc2c(C)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCO[C@@H]1C2 |r|
C[C@H]1OCCCCc2c(C)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCO[C@H]1C2 |r|
C[C@@H]1OCCCCc2c(C)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCO[C@H]1C2 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@]5(C[C@@H](C5)OC(=O)OCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,17.21,19.20,wD:1.0,(-8.01,1.28,;-7.61,-.2,;-8.52,-1.45,;-7.61,-2.7,;-7.61,-4.24,;-6.15,-4.71,;-5.25,-3.47,;-6.15,-2.22,;-4.82,-1.45,;-3.48,-2.22,;-2.15,-1.45,;-2.15,.09,;-.82,.86,;-.82,2.4,;-2.15,3.17,;-2.15,4.71,;-.82,5.48,;.52,4.71,;.92,6.2,;2.4,5.8,;2.01,4.31,;3.19,4.71,;3.19,3.17,;1.85,2.4,;4.52,2.4,;4.52,.86,;5.85,.09,;5.85,-1.45,;7.19,-2.22,;8.52,-1.45,;7.19,-3.76,;5.85,-4.53,;5.53,-6.04,;4,-6.2,;3.37,-4.79,;4.52,-3.76,;4.52,-2.22,;3.19,-1.45,;3.19,.09,;1.85,.86,;.52,.09,;.52,-1.45,;-.82,-2.22,;1.85,-2.22,;1.85,-3.76,;.52,3.17,;-6.15,-.68,)|
C[C@H]1CCOC[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(C)cc1[nH]ncc21 |r|
C[C@@H]1CCOC[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(C)cc1[nH]ncc21 |r|
C[C@H]1CCOC[C@H]2CN(CCO2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(Cl)cc1[nH]ncc21 |r|
C[C@@H]1CCOC[C@H]2CN(CCO2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(C1)c(Cl)cc1[nH]ncc21 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@H](C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC(C4)c4cnc(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)Oc4nccc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOCC(C4)Cn4ncc(\C=C/c5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r,c:27|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,17.17,wD:1.0,17.50,19.22,(.09,-7.54,;.86,-8.87,;.23,-10.28,;1.38,-11.31,;1.7,-12.81,;3.23,-12.97,;3.85,-11.57,;2.71,-10.54,;4.04,-9.77,;5.38,-10.54,;6.71,-9.77,;6.71,-8.23,;8.04,-7.46,;8.04,-5.92,;6.71,-5.15,;6.71,-3.61,;8.04,-2.84,;9.38,-3.61,;9.78,-2.12,;11.26,-2.52,;10.87,-4,;12.05,-3.61,;12.05,-5.15,;13.38,-5.92,;13.38,-7.46,;14.71,-8.23,;14.71,-9.77,;16.05,-10.54,;17.38,-9.77,;16.05,-12.08,;14.71,-12.85,;14.39,-14.35,;12.86,-14.51,;12.23,-13.11,;13.38,-12.08,;13.38,-10.54,;12.05,-9.77,;12.05,-8.23,;10.71,-7.46,;9.38,-8.23,;9.38,-9.77,;8.04,-10.54,;10.71,-10.54,;10.71,-12.08,;9.38,-5.15,;2.39,-9.03,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,19.20,wD:1.0,17.21,(-8.01,1.28,;-7.61,-.2,;-8.52,-1.45,;-7.61,-2.7,;-7.61,-4.24,;-6.15,-4.71,;-5.25,-3.47,;-6.15,-2.22,;-4.82,-1.45,;-3.48,-2.22,;-2.15,-1.45,;-2.15,.09,;-.82,.86,;-.82,2.4,;-2.15,3.17,;-2.15,4.71,;-.82,5.48,;.52,4.71,;.92,6.2,;2.4,5.8,;2.01,4.31,;3.58,4.66,;3.58,3.12,;4.92,2.35,;4.52,.86,;5.85,.09,;5.85,-1.45,;7.19,-2.22,;8.52,-1.45,;7.19,-3.76,;5.85,-4.53,;5.53,-6.04,;4,-6.2,;3.37,-4.79,;4.52,-3.76,;4.52,-2.22,;3.19,-1.45,;3.19,.09,;1.85,.86,;.52,.09,;.52,-1.45,;-.82,-2.22,;1.85,-2.22,;1.85,-3.76,;.52,3.17,;-6.15,-.68,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,wD:1.0,17.18,19.19,(-8.01,1.28,;-7.61,-.2,;-8.52,-1.45,;-7.61,-2.7,;-7.61,-4.24,;-6.15,-4.71,;-5.25,-3.47,;-6.15,-2.22,;-4.82,-1.45,;-3.48,-2.22,;-2.15,-1.45,;-2.15,.09,;-.82,.86,;-.82,2.4,;-2.15,3.17,;-2.15,4.71,;-.82,5.48,;.52,4.71,;2.01,4.31,;2.4,5.8,;.92,6.2,;3.58,4.66,;3.58,3.12,;4.92,2.35,;4.52,.86,;5.85,.09,;5.85,-1.45,;7.19,-2.22,;8.52,-1.45,;7.19,-3.76,;5.85,-4.53,;5.53,-6.04,;4,-6.2,;3.37,-4.79,;4.52,-3.76,;4.52,-2.22,;3.19,-1.45,;3.19,.09,;1.85,.86,;.52,.09,;.52,-1.45,;-.82,-2.22,;1.85,-2.22,;1.85,-3.76,;.52,3.17,;-6.15,-.68,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,20.21,wD:1.0,18.22,(-8.01,1.21,;-7.61,-.28,;-8.52,-1.53,;-7.61,-2.77,;-7.61,-4.31,;-6.15,-4.79,;-5.25,-3.54,;-6.15,-2.3,;-4.82,-1.53,;-3.48,-2.3,;-2.15,-1.53,;-2.15,.01,;-.82,.78,;-.82,2.32,;-2.32,2.66,;-2.99,4.05,;-2.32,5.44,;-.82,5.78,;.39,4.82,;.9,6.28,;2.35,5.77,;1.84,4.31,;3.58,4.58,;3.58,3.04,;4.92,2.27,;4.52,.78,;5.85,.01,;5.85,-1.53,;7.19,-2.3,;8.52,-1.53,;7.19,-3.84,;5.85,-4.61,;5.53,-6.11,;4,-6.28,;3.37,-4.87,;4.52,-3.84,;4.52,-2.3,;3.19,-1.53,;3.19,.01,;1.85,.78,;.52,.01,;.52,-1.53,;-.82,-2.3,;1.85,-2.3,;1.85,-3.84,;.39,3.28,;-6.15,-.76,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,wD:1.0,18.19,20.20,(-8.01,1.21,;-7.61,-.28,;-8.52,-1.53,;-7.61,-2.77,;-7.61,-4.31,;-6.15,-4.79,;-5.25,-3.54,;-6.15,-2.3,;-4.82,-1.53,;-3.48,-2.3,;-2.15,-1.53,;-2.15,.01,;-.82,.78,;-.82,2.32,;-2.32,2.66,;-2.99,4.05,;-2.32,5.44,;-.82,5.78,;.39,4.82,;1.84,4.31,;2.35,5.77,;.9,6.28,;3.58,4.58,;3.58,3.04,;4.92,2.27,;4.52,.78,;5.85,.01,;5.85,-1.53,;7.19,-2.3,;8.52,-1.53,;7.19,-3.84,;5.85,-4.61,;5.53,-6.11,;4,-6.28,;3.37,-4.87,;4.52,-3.84,;4.52,-2.3,;3.19,-1.53,;3.19,.01,;1.85,.78,;.52,.01,;.52,-1.53,;-.82,-2.3,;1.85,-2.3,;1.85,-3.84,;.39,3.28,;-6.15,-.76,)|
O[C@H]1C[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCCOC2)c(Cl)cc2[nH]ncc12 |r|
[H][C@]12CCB(COc3nc4N5CCC[C@H](C5)COCCCCc5c(C)cc6[nH]ncc6c5-c5ncc4c(n3)c5F)N1CCOC2 |r|
CN1CCC[C@H]1COc1nc2N3CC[C@H]4CCN([C@H]4C3)C(=O)COCCCc3c(Cl)cc4[nH]ncc4c3-c3ncc2c(n1)c3F
CN(C)CC1(COc2nc3N4CC[C@H]5CCN([C@H]5C4)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)CC1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC5CCN(C(C5)C4)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)COCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)COCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@]5(C[C@@H](C5)NC(=O)CCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,19.19,wD:1.0,17.18,(-8.47,.76,;-7.72,-.55,;-8.32,-2.01,;-7.23,-3.1,;-6.89,-4.6,;-5.43,-4.75,;-4.79,-3.32,;-5.92,-2.23,;-4.64,-1.49,;-3.31,-2.26,;-1.98,-1.49,;-1.98,.05,;-.64,.82,;-.64,2.36,;-1.98,3.13,;-1.98,4.67,;-.64,5.44,;.69,4.67,;2.18,4.27,;2.58,5.76,;1.09,6.16,;4.07,6.16,;5.54,4.83,;7.08,4.83,;4.55,3.43,;5.64,2.34,;4.55,1.25,;5.88,.48,;5.88,-1.54,;7.15,-2.32,;8.47,-1.57,;7.15,-3.9,;5.84,-4.65,;5.48,-6.07,;4.02,-6.16,;3.48,-4.8,;4.61,-3.86,;4.61,-2.32,;3.36,-1.49,;3.36,.05,;2.03,.82,;.69,.05,;.69,-1.49,;-.64,-2.26,;2.03,-2.26,;2.03,-3.8,;.69,3.13,;-6.22,-.74,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC5(CC(C5)NC(=O)CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,wD:1.0,(-8.47,.76,;-7.72,-.55,;-8.32,-2.01,;-7.23,-3.1,;-6.89,-4.6,;-5.43,-4.75,;-4.79,-3.32,;-5.92,-2.23,;-4.64,-1.49,;-3.31,-2.26,;-1.98,-1.49,;-1.98,.05,;-.64,.82,;-.64,2.36,;-1.98,3.13,;-1.98,4.67,;-.64,5.44,;.69,4.67,;2.18,4.27,;2.58,5.76,;1.09,6.16,;4.07,6.16,;4.85,4.83,;6.39,4.83,;4.45,3.34,;5.93,2.46,;5.26,.62,;5.88,-1.54,;7.15,-2.32,;8.47,-1.57,;7.15,-3.9,;5.84,-4.65,;5.48,-6.07,;4.02,-6.16,;3.48,-4.8,;4.61,-3.86,;4.61,-2.32,;3.36,-1.49,;3.36,.05,;2.03,.82,;.69,.05,;.69,-1.49,;-.64,-2.26,;2.03,-2.26,;2.03,-3.8,;.69,3.13,;-6.22,-.74,)|
O[C@H]1C[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCCC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
O[C@@H]1C[C@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCCC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
Cc1cc2[nH]ncc2c-2c1CCCOCC(=O)N1CC[C@@H]3CCN(C[C@H]13)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c3[C@H](CCc3cc3[nH]ncc23)CCOCC1=O |r|
CN1[C@@H]2CCCN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c3[C@@H](CCc3cc3[nH]ncc23)CCOCC1=O |r|
Cc1cc2[nH]ncc2c-2c1CCCCC(=O)N[C@]1(C)CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
C[C@@]12CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCC[C@H](F)C(=O)N2)c(Cl)cc2[nH]ncc12 |r|
O[C@H]1CC[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
O[C@@H]1CC[C@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
O[C@H]1CC2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
O[C@@H]1C[C@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
CN1[C@@H]2C[C@H](O)CN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCOC1=O)c(Cl)cc1[nH]ncc21 |r|
CN1C2C[C@@H](O)CN(C2)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc23)-c2c(CCCOC1=O)c(Cl)cc1[nH]ncc21 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)OC(=O)NCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@@]5(C[C@@H](C5)NC(=O)OCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,17.18,wD:1.0,19.19,(-8.65,.8,;-7.88,-.53,;-8.5,-1.94,;-7.36,-2.97,;-7.04,-4.47,;-5.51,-4.63,;-4.88,-3.23,;-6.02,-2.2,;-4.69,-1.43,;-3.36,-2.2,;-2.02,-1.43,;-2.02,.11,;-.69,.88,;-.69,2.42,;-2.02,3.19,;-2.02,4.73,;-.69,5.5,;.64,4.73,;1.18,6.17,;2.63,5.63,;2.09,4.19,;4.3,4.92,;5.36,3.8,;6.86,4.16,;4.63,2.45,;4.63,.91,;5.97,.14,;5.98,-1.43,;7.31,-2.2,;8.65,-1.43,;7.31,-3.74,;5.98,-4.51,;5.66,-6.01,;4.13,-6.17,;3.5,-4.77,;4.65,-3.74,;4.65,-2.2,;3.31,-1.43,;3.31,.11,;1.98,.88,;.64,.11,;.64,-1.43,;-.69,-2.2,;1.98,-2.2,;1.98,-3.74,;.64,3.19,;-6.34,-.69,)|
C[C@@]12CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)N2)c(Cl)cc2[nH]ncc12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)OCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)N[C@]1(C)CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
Cc1cc2[nH]ncc2c-2c1CCCOC(=O)N[C@@]1(C)CCCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c-2ncc13 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC(C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@@H](C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@@H](C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)c4cnn(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
O[C@@H]1C[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCn3ncc2n3)c(Cl)cc2[nH]ncc12 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)OCC[C@@H]4CCc5cc6[nH]ncc6c(c45)-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@H](C4)NC(=O)OCC[C@H]4CCc5cc6[nH]ncc6c(c45)-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4cc(n2)c3cn4)C1 |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1cccc3ccc(F)c(CCOC(=O)O2)c13 |r|
CN(C)CC1(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4c(F)cc3c(n2)c4F)CC1 |r|
CO[C@@H]1C[C@@H](COc2nc3N4CCCC5(C[C@@H](C5)OC(=O)OCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)N(C)C1 |r,wU:4.4,16.16,wD:2.1,(-9.85,-1.29,;-9.32,-2.74,;-7.78,-2.74,;-6.75,-1.59,;-5.35,-2.22,;-4.01,-1.45,;-2.68,-2.22,;-1.35,-1.45,;-1.35,.09,;-.01,.86,;-.01,2.4,;-1.35,3.17,;-1.35,4.71,;-.01,5.48,;1.32,4.71,;1.72,6.2,;3.21,5.8,;2.81,4.31,;4.3,4.71,;3.99,3.17,;2.66,2.4,;5.32,2.4,;5.32,.86,;6.66,.09,;6.66,-1.45,;7.99,-2.22,;9.32,-1.45,;7.99,-3.76,;6.66,-4.53,;6.34,-6.04,;4.8,-6.2,;4.18,-4.79,;5.32,-3.76,;5.32,-2.22,;3.99,-1.45,;3.99,.09,;2.66,.86,;1.32,.09,;1.32,-1.45,;-.01,-2.22,;2.66,-2.22,;2.66,-3.76,;1.32,3.17,;-5.51,-3.75,;-4.36,-4.78,;-7.01,-4.07,)|
C[C@@]12COCCN(C1)c1nc(OC[C@H]3CC[C@@H]4COCCN34)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@H]3CC[C@H]4COCCN34)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
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F[C@@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@]5(C[C@@H](C5)OC(=O)OCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)C1 |r,wU:7.8,1.0,17.21,19.20,(-8.65,.78,;-7.88,-.55,;-8.5,-1.96,;-7.36,-2.99,;-7.04,-4.5,;-5.51,-4.66,;-4.88,-3.25,;-6.02,-2.22,;-4.69,-1.45,;-3.36,-2.22,;-2.02,-1.45,;-2.02,.09,;-.69,.86,;-.69,2.4,;-2.02,3.17,;-2.02,4.71,;-.69,5.48,;.64,4.71,;1.04,6.2,;2.53,5.8,;2.13,4.31,;3.86,5.03,;3.47,3.54,;1.98,3.14,;4.65,2.4,;4.65,.86,;5.98,.09,;5.98,-1.45,;7.31,-2.22,;8.65,-1.45,;7.31,-3.76,;5.98,-4.53,;5.66,-6.04,;4.13,-6.2,;3.5,-4.79,;4.65,-3.76,;4.65,-2.22,;3.31,-1.45,;3.31,.09,;1.98,.86,;.64,.09,;.64,-1.45,;-.69,-2.22,;1.98,-2.22,;1.98,-3.76,;.64,3.17,;-6.34,-.71,)|
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C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
F[C@@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
Oc1cc2-c3ncc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)N3CCOC[C@H](C3)OC(=O)OCCc3c(F)ccc(c1)c23 |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3cc(nnc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
C[C@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3cc(nnc13)-c1c(CCCOC(=O)O2)c(Cl)cc2[nH]ncc12 |r|
C[C@@]12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c3[C@@H](CCc3cc3[nH]ncc13)CCOC(=O)O2 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCC[C@@H]4CCc5cc6[nH]ncc6c(c45)-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)OC(=O)OCCc4c(F)ccc5cccc(-c6ncc3c(n2)c6F)c45)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)CC(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)Cc4ncc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@@H](C4)Cc4ncc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCOC[C@H](C4)Cc4ncc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
O[C@H]1C[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCc3nc2no3)c(Cl)cc2[nH]ncc12 |r|
CC12COCCN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCc3nc2no3)c(Cl)cc2[nH]ncc12 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCCC(C4)c4noc(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)Cn4ncc(n4)[C@@H]4C[C@@H]4c4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@@H](C4)c4coc(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)c4coc(CCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)n4)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCC[C@H](C4)Cc4nnc(CCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)o4)C1 |r|
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F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCO[C@H](C4)COCC[C@H]4C[C@H]4c4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CN1CCC[C@H]1COc1nc2N3CCC[C@H](C3)[C@H](O)c3ncc(CCc4c(Cl)cc5[nH]ncc5c4-c4ncc2c(n1)c4F)o3 |r|
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O[C@@]12C[C@]3(C1)CCCN(C3)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCOCC2)c(Cl)cc2[nH]ncc12 |r,wU:15.16,3.2,1.0,wD:21.24,(3.17,6.66,;2.4,5.33,;2.01,3.84,;.52,4.24,;.92,5.73,;-.82,5.01,;-2.15,4.24,;-2.15,2.7,;-.82,1.93,;.52,2.7,;-.82,.39,;-2.15,-.38,;-2.15,-1.92,;-3.48,-2.69,;-4.82,-1.92,;-6.15,-2.69,;-5.25,-3.93,;-6.15,-5.18,;-7.61,-4.7,;-7.61,-3.16,;-8.52,-1.92,;-7.61,-.67,;-8.01,.82,;-6.15,-1.15,;-.82,-2.69,;.52,-1.92,;1.85,-2.69,;1.85,-4.23,;3.19,-1.92,;3.19,-.38,;1.85,.39,;.52,-.38,;4.52,-2.69,;5.85,-1.92,;5.85,-.38,;4.52,.39,;5.07,2.25,;3.74,3.02,;3.74,4.56,;7.19,-2.69,;8.52,-1.92,;7.19,-4.23,;5.85,-5,;5.53,-6.5,;4,-6.66,;3.37,-5.26,;4.52,-4.23,)|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@@](F)(C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CCCC[C@](F)(C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
CN(C)CC1(COc2nc3N4CCCC[C@](F)(C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)CC1 |r|
CN(C)CC1(COc2nc3N4CCCC[C@@](F)(C4)COCCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)CC1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@H]5[C@@H](C4)N(CC5(F)F)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
F[C@H]1CN2CCC[C@@]2(COc2nc3N4CC[C@@H]5[C@H](C4)N(CC5(F)F)C(=O)CCCCc4c(Cl)cc5[nH]ncc5c4-c4ncc3c(n2)c4F)C1 |r|
O[C@@H]1CCOCCc2c(Cl)cc3[nH]ncc3c2-c2ncc3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)N2CCC[C@@H]1C2 |r|
CN(C)CC1(COc2nc3N4CCC[C@]5(C[C@@H](C5)OCCCCc5c(Cl)cc6[nH]ncc6c5-c5ncc3c(n2)c5F)C4)CC1 |r,wU:14.17,16.16,(-9.34,-1.45,;-8,-2.22,;-8,-3.76,;-6.67,-1.45,;-5.33,-2.22,;-4,-1.45,;-2.67,-2.22,;-1.33,-1.45,;-1.33,.09,;,.86,;,2.4,;-1.33,3.17,;-1.33,4.71,;,5.48,;1.33,4.71,;1.73,6.2,;3.22,5.8,;2.82,4.31,;4.4,4.66,;4,3.17,;5.33,2.4,;5.33,.86,;6.67,.09,;6.67,-1.45,;8,-2.22,;9.34,-1.45,;8,-3.76,;6.67,-4.53,;6.35,-6.04,;4.82,-6.2,;4.19,-4.79,;5.33,-3.76,;5.33,-2.22,;4,-1.45,;4,.09,;2.67,.86,;1.33,.09,;1.33,-1.45,;,-2.22,;2.67,-2.22,;2.67,-3.76,;1.33,3.17,;-6.1,-3.55,;-4.56,-3.55,)|
O[C@@H]1C[C@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCCOC2)c(Cl)cc2[nH]ncc12 |r|
O[C@@H]1C[C@@H]2CN(C1)c1nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3c(F)c(ncc13)-c1c(CCCCOC2)c(Cl)cc2[nH]ncc12 |r|
Oc1cc(-c2nc3OC[C@H]4[C@H]5CC[C@@H](CN4c4nc(OC[C@@]67CCCN6C[C@H](F)C7)nc(c2F)c34)N5)c2c(cccc2c1)C#C |r|
Nc1sc2cccc(-c3c(Cl)c4OCC5C6CCC(CN5c5ncnc(c3F)c45)N6)c2c1C#N |(.08,-40.94,;-.69,-39.61,;-2.22,-39.45,;-2.54,-37.94,;-3.88,-37.17,;-3.88,-35.63,;-2.54,-34.86,;-1.21,-35.63,;.12,-34.86,;.12,-33.32,;-1.21,-32.55,;1.46,-32.55,;1.23,-31.03,;2.28,-29.9,;3.81,-30.01,;4.27,-28.54,;5.7,-27.98,;7.03,-28.75,;7.26,-30.27,;6.21,-31.4,;4.68,-31.29,;4.13,-32.55,;5.46,-33.32,;5.46,-34.86,;4.13,-35.63,;2.79,-34.86,;1.46,-35.63,;1.46,-37.17,;2.79,-33.32,;5.27,-30.01,;-1.21,-37.17,;-.06,-38.2,;1.44,-37.88,;2.95,-37.56,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-1.56,-15.02,;-2.33,-13.68,;-3.86,-13.52,;-4.18,-12.01,;-5.51,-11.24,;-5.51,-9.7,;-4.18,-8.93,;-2.85,-9.7,;-1.51,-8.93,;-1.51,-7.39,;-2.85,-6.62,;-.18,-6.62,;-.41,-5.1,;.64,-3.97,;2.17,-4.09,;2.63,-2.62,;4.06,-2.05,;5.4,-2.82,;5.62,-4.35,;4.58,-5.48,;3.04,-5.36,;2.49,-6.62,;3.82,-7.39,;3.82,-8.93,;5.15,-9.7,;6.49,-8.93,;7.82,-9.7,;8.14,-8.2,;9.67,-8.04,;10.3,-9.44,;9.16,-10.47,;8.84,-11.98,;7.3,-12.14,;6.53,-13.48,;6.68,-10.74,;2.49,-9.7,;1.15,-8.93,;-.18,-9.7,;-.18,-11.24,;1.15,-7.39,;3.81,-4.02,;-2.85,-11.24,;-1.7,-12.28,;-.2,-11.96,;1.31,-11.63,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-3.95,-6.8,;-4.72,-5.47,;-6.25,-5.31,;-6.57,-3.8,;-7.91,-3.03,;-7.91,-1.49,;-6.57,-.72,;-5.24,-1.49,;-3.91,-.72,;-3.91,.82,;-5.24,1.59,;-2.57,1.59,;-2.8,3.11,;-1.75,4.24,;-.22,4.13,;.23,5.6,;1.67,6.16,;3,5.39,;3.23,3.87,;2.18,2.74,;.65,2.85,;.09,1.59,;1.43,.82,;1.43,-.72,;2.76,-1.49,;4.1,-.72,;5.43,-1.49,;5.75,.02,;7.28,.18,;7.91,-1.23,;6.76,-2.26,;6.44,-3.77,;4.91,-3.93,;4.14,-5.26,;4.28,-2.52,;.09,-1.49,;-1.24,-.72,;-2.57,-1.49,;-2.57,-3.03,;-1.24,.82,;1.42,4.19,;-5.24,-3.03,;-4.1,-4.06,;-2.59,-3.74,;-1.08,-3.42,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,32.34,wD:14.20,(-1.55,-22.68,;-2.32,-21.35,;-3.86,-21.19,;-4.18,-19.68,;-5.51,-18.91,;-5.51,-17.37,;-4.18,-16.6,;-2.84,-17.37,;-1.51,-16.6,;-1.51,-15.06,;-2.84,-14.29,;-.17,-14.29,;-.4,-12.77,;.64,-11.64,;2.18,-11.76,;2.63,-10.28,;4.07,-9.72,;5.4,-10.49,;5.63,-12.01,;4.58,-13.14,;3.05,-13.03,;2.49,-14.29,;3.83,-15.06,;3.83,-16.6,;5.16,-17.37,;6.49,-16.6,;7.83,-17.37,;8.15,-15.87,;9.68,-15.7,;10.31,-17.11,;9.16,-18.14,;8.84,-19.65,;7.31,-19.81,;6.54,-21.14,;6.68,-18.4,;2.49,-17.37,;1.16,-16.6,;-.17,-17.37,;-.17,-18.91,;1.16,-15.06,;3.82,-11.69,;-2.84,-18.91,;-1.7,-19.94,;-.19,-19.62,;1.32,-19.3,)|
Nc1sc2c(F)ccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5ncnc(c3F)c45)N6)c2c1C#N |r,wU:16.34,19.33,wD:15.21,(-1.02,-16.96,;-1.72,-15.53,;-3.26,-15.41,;-3.61,-13.91,;-4.98,-13.14,;-6.32,-13.91,;-4.95,-11.59,;-3.64,-10.87,;-2.3,-11.59,;-.55,-10.59,;-.52,-9.04,;-1.89,-8.28,;.79,-8.28,;.59,-6.74,;1.67,-5.63,;3.18,-5.72,;3.68,-4.26,;5.02,-3.68,;6.41,-4.44,;6.56,-5.95,;5.6,-7.09,;4.05,-7,;3.47,-8.26,;4.84,-9.04,;4.81,-10.59,;3.5,-11.37,;2.13,-10.56,;.82,-11.34,;.82,-12.89,;2.16,-9.04,;4.58,-5.66,;-2.3,-13.11,;-1.13,-14.11,;.37,-13.76,;1.87,-13.4,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5ncnc(c3F)c45)N6)c2c1C#N |r,wU:15.33,18.32,wD:14.20,(-1.7,-16.96,;-2.39,-15.54,;-3.93,-15.41,;-4.28,-13.92,;-5.65,-13.14,;-5.62,-11.6,;-4.31,-10.88,;-2.97,-11.6,;-1.22,-10.59,;-1.19,-9.05,;-2.56,-8.29,;.12,-8.29,;-.08,-6.74,;.99,-5.64,;2.51,-5.72,;3,-4.27,;4.34,-3.69,;5.74,-4.44,;5.89,-5.96,;4.93,-7.09,;3.38,-7.01,;2.8,-8.26,;4.17,-9.05,;4.14,-10.59,;2.83,-11.38,;1.46,-10.56,;.15,-11.35,;.15,-12.9,;1.49,-9.05,;3.91,-5.67,;-2.97,-13.11,;-1.8,-14.12,;-.3,-13.76,;1.2,-13.4,)|
Nc1sc2c(F)ccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:27.27,16.47,19.46,wD:15.21,33.35,(-3.3,-6.63,;-4.07,-5.26,;-5.6,-5.13,;-5.95,-3.63,;-7.32,-2.86,;-8.65,-3.62,;-7.26,-1.3,;-5.96,-.58,;-4.6,-1.3,;-3.27,-.52,;-3.24,1.01,;-4.6,1.76,;-1.91,1.76,;-2.31,3.27,;-1.3,4.48,;.23,4.46,;.61,5.96,;2,6.63,;3.38,5.93,;3.65,4.43,;2.75,3.27,;1.16,3.27,;.78,1.76,;2.11,.98,;2.11,-.55,;3.47,-1.3,;4.8,-.55,;6.13,-1.3,;6.48,.17,;8.01,.35,;8.65,-1.07,;7.49,-2.08,;7.17,-3.59,;5.61,-3.73,;4.83,-5.07,;5.01,-2.37,;.78,-1.3,;-.61,-.52,;-1.91,-1.3,;-1.94,-2.86,;-.55,1.01,;1.79,4.54,;-4.63,-2.84,;-3.47,-3.85,;-1.97,-3.5,;-.47,-3.16,)|
Nc1sc2c(F)ccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@]78CCCN7C[C@@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:16.47,19.46,33.35,wD:27.27,15.21,(-3.3,-6.63,;-4.07,-5.26,;-5.6,-5.13,;-5.95,-3.63,;-7.32,-2.86,;-8.65,-3.62,;-7.26,-1.3,;-5.96,-.58,;-4.6,-1.3,;-3.27,-.52,;-3.24,1.01,;-4.6,1.76,;-1.91,1.76,;-2.31,3.27,;-1.3,4.48,;.23,4.46,;.61,5.96,;2,6.63,;3.38,5.93,;3.65,4.43,;2.75,3.27,;1.16,3.27,;.78,1.76,;2.11,.98,;2.11,-.55,;3.47,-1.3,;4.8,-.55,;6.13,-1.3,;6.48,.17,;8.01,.35,;8.65,-1.07,;7.49,-2.08,;7.17,-3.59,;5.61,-3.73,;4.83,-5.07,;5.01,-2.37,;.78,-1.3,;-.61,-.52,;-1.91,-1.3,;-1.94,-2.86,;-.55,1.01,;1.79,4.54,;-4.63,-2.84,;-3.47,-3.85,;-1.97,-3.5,;-.47,-3.16,)|
CC(C)(C)OC(=O)Nc1nc2c(cccc2s1)-c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r,wU:24.57,27.56,35.37,wD:23.31,41.45,(-7.35,-17.29,;-5.81,-17.29,;-5.04,-18.62,;-4.27,-17.29,;-5.04,-15.95,;-5.81,-14.62,;-7.35,-14.62,;-5.04,-13.29,;-5.81,-11.95,;-5.19,-10.55,;-6.33,-9.52,;-6.33,-7.97,;-7.66,-7.2,;-9,-7.97,;-9,-9.52,;-7.66,-10.29,;-7.34,-11.79,;-5,-7.2,;-5,-5.66,;-6.33,-4.89,;-3.66,-4.89,;-3.89,-3.37,;-2.84,-2.24,;-1.31,-2.36,;-.86,-.89,;.58,-.32,;1.91,-1.09,;2.14,-2.62,;1.09,-3.75,;-.44,-3.63,;-1,-4.89,;.34,-5.66,;.34,-7.2,;1.67,-7.97,;3.01,-7.2,;4.34,-7.97,;4.66,-6.47,;6.19,-6.31,;6.82,-7.71,;5.67,-8.75,;5.35,-10.25,;3.82,-10.41,;3.05,-11.75,;3.2,-9.01,;-1,-7.97,;-2.33,-7.2,;-3.66,-7.97,;-3.66,-9.52,;-2.33,-5.66,;.17,-2.37,)|
Nc1nc2c(cccc2s1)-c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r,wU:17.50,20.49,28.30,wD:16.24,34.38,(-2.64,-29.27,;-3.41,-27.94,;-2.79,-26.53,;-3.93,-25.5,;-3.93,-23.96,;-5.27,-23.19,;-6.6,-23.96,;-6.6,-25.5,;-5.27,-26.27,;-4.95,-27.78,;-2.6,-23.19,;-2.6,-21.65,;-3.93,-20.88,;-1.26,-20.88,;-1.49,-19.36,;-.45,-18.23,;1.09,-18.35,;1.54,-16.88,;2.98,-16.31,;4.31,-17.08,;4.54,-18.61,;3.49,-19.73,;1.96,-19.62,;1.4,-20.88,;2.74,-21.65,;2.74,-23.19,;4.07,-23.96,;5.4,-23.19,;6.74,-23.96,;7.06,-22.46,;8.59,-22.3,;9.22,-23.7,;8.07,-24.73,;7.75,-26.24,;6.22,-26.4,;5.45,-27.73,;5.59,-24.99,;1.4,-23.96,;.07,-23.19,;-1.26,-23.96,;-1.26,-25.5,;.07,-21.65,;2.57,-18.36,)|
Nc1nn2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-1.04,-20.79,;-1.81,-19.46,;-3.34,-19.3,;-3.66,-17.79,;-5,-17.02,;-5,-15.48,;-3.66,-14.71,;-2.33,-15.48,;-1,-14.71,;-1,-13.17,;-2.33,-12.4,;.34,-12.4,;.11,-10.88,;1.16,-9.75,;2.69,-9.86,;3.14,-8.39,;4.58,-7.83,;5.91,-8.6,;6.14,-10.12,;5.09,-11.25,;3.56,-11.14,;3,-12.4,;4.34,-13.17,;4.34,-14.71,;5.67,-15.48,;7.01,-14.71,;8.34,-15.48,;8.66,-13.97,;10.19,-13.81,;10.82,-15.22,;9.67,-16.25,;9.35,-17.76,;7.82,-17.92,;7.08,-18.99,;7.19,-16.51,;3,-15.48,;1.67,-14.71,;.34,-15.48,;.34,-17.02,;1.67,-13.17,;4.19,-9.66,;-2.33,-17.02,;-1.19,-18.05,;.32,-17.73,;1.83,-17.41,)|
Nc1sc2ccc(F)c(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:16.47,19.46,27.27,wD:15.21,33.35,(-7.84,-6.25,;-8.61,-4.91,;-10.14,-4.75,;-10.47,-3.24,;-11.8,-2.47,;-11.8,-.93,;-10.47,-.16,;-10.47,1.38,;-9.13,-.93,;-7.8,-.16,;-7.8,1.38,;-8.95,2.13,;-6.46,2.15,;-6.69,3.67,;-5.65,4.8,;-4.11,4.68,;-3.66,6.15,;-2.22,6.72,;-.89,5.95,;-.66,4.42,;-1.71,3.29,;-3.24,3.41,;-3.8,2.15,;-2.46,1.38,;-2.46,-.16,;-1.13,-.93,;.2,-.16,;1.54,-.93,;1.86,.57,;3.39,.73,;4.02,-.67,;2.87,-1.7,;2.55,-3.21,;1.02,-3.37,;.25,-4.71,;.39,-1.97,;-3.8,-.93,;-5.13,-.16,;-6.46,-.93,;-6.45,-2.38,;-5.13,1.38,;-2.17,5.75,;-9.13,-2.47,;-7.99,-3.5,;-6.48,-3.18,;-4.97,-2.86,)|
Nc1cc2c(c(Cl)ccc2s1)-c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r,wU:29.31,18.51,21.50,wD:17.25,35.39,(-3.99,-6.66,;-4.77,-5.31,;-4.14,-3.89,;-5.31,-2.82,;-5.28,-1.31,;-6.63,-.52,;-6.63,.8,;-7.96,-1.31,;-7.96,-2.85,;-6.6,-3.61,;-6.32,-5.15,;-3.92,-.52,;-3.92,1.02,;-5.28,1.78,;-2.6,1.78,;-2.98,3.29,;-2.06,4.52,;-.46,4.49,;-.08,6,;1.31,6.66,;2.69,5.97,;2.95,4.46,;2.03,3.26,;.49,3.29,;.05,1.81,;1.43,1.02,;1.43,-.52,;2.76,-1.31,;4.11,-.55,;5.43,-1.28,;5.81,.2,;7.32,.36,;7.96,-1.06,;6.82,-2.1,;6.47,-3.61,;4.96,-3.73,;4.18,-5.08,;4.33,-2.38,;.11,-1.31,;-1.28,-.49,;-2.6,-1.28,;-2.6,-2.85,;-1.24,1.02,;1.12,4.58,)|
Nc1cc2cc(ccc2s1)-c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r|
CC(Oc1nc2N3C[C@H]4CC[C@H](N4)[C@H]3COc3c(Cl)c(c(F)c(n1)c23)-c1cccc2sc(N)c(C#N)c12)[C@@]12CCCN1C[C@H](F)C2 |r,wU:11.11,8.12,37.43,wD:13.14,43.51,(-.57,1.61,;-.57,-.46,;-1.9,-1.23,;-3.24,-.46,;-3.24,1.08,;-4.57,1.85,;-4.02,3.12,;-2.48,3,;-1.43,4.13,;-1.66,5.65,;-3,6.42,;-4.43,5.86,;-2.94,5.46,;-4.88,4.39,;-6.42,4.5,;-7.47,3.38,;-7.24,1.85,;-8.57,1.08,;-9.82,1.73,;-8.57,-.46,;-7.24,-1.23,;-7.25,-2.62,;-5.9,-.46,;-4.57,-1.23,;-5.9,1.08,;-9.9,-1.23,;-11.24,-.46,;-12.57,-1.23,;-12.57,-2.77,;-11.24,-3.54,;-10.92,-5.04,;-9.39,-5.21,;-8.62,-6.54,;-8.76,-3.8,;-7.25,-3.48,;-5.75,-3.16,;-9.91,-2.77,;.76,-1.23,;1.09,.28,;2.62,.44,;3.24,-.97,;2.1,-2,;1.78,-3.5,;.25,-3.67,;-.52,-5,;-.38,-2.26,)|
CC(Oc1nc2N3C[C@H]4CC[C@H](N4)[C@@H]3COc3c(Cl)c(c(F)c(n1)c23)-c1cccc2sc(N)c(C#N)c12)[C@@]12CCCN1C[C@@H](F)C2 |r,wU:13.14,11.11,8.12,37.43,43.51,(-.57,1.61,;-.57,-.46,;-1.9,-1.23,;-3.24,-.46,;-3.24,1.08,;-4.57,1.85,;-4.02,3.12,;-2.48,3,;-1.43,4.13,;-1.66,5.65,;-3,6.42,;-4.43,5.86,;-2.94,5.46,;-4.88,4.39,;-6.42,4.5,;-7.47,3.38,;-7.24,1.85,;-8.57,1.08,;-9.82,1.73,;-8.57,-.46,;-7.24,-1.23,;-7.25,-2.62,;-5.9,-.46,;-4.57,-1.23,;-5.9,1.08,;-9.9,-1.23,;-11.24,-.46,;-12.57,-1.23,;-12.57,-2.77,;-11.24,-3.54,;-10.92,-5.04,;-9.39,-5.21,;-8.62,-6.54,;-8.76,-3.8,;-7.25,-3.48,;-5.75,-3.16,;-9.91,-2.77,;.76,-1.23,;1.09,.28,;2.62,.44,;3.24,-.97,;2.1,-2,;1.78,-3.5,;.25,-3.67,;-.52,-5,;-.38,-2.26,)|
CC(Oc1nc2N3C[C@H]4CC[C@H](N4)[C@H]3COc3c(Cl)c(c(F)c(n1)c23)-c1c(F)ccc2sc(N)c(C#N)c12)[C@@]12CCCN1C[C@H](F)C2 |r,wU:38.44,11.11,8.12,wD:13.14,44.52,(4.08,1.04,;4.08,-.51,;2.77,-1.33,;1.39,-.51,;1.42,1.01,;.07,1.8,;.45,3.29,;2,3.26,;2.91,4.46,;2.68,5.98,;1.27,6.69,;-.07,6.01,;1.1,4.58,;-.45,4.52,;-2,4.55,;-2.94,3.29,;-2.59,1.8,;-3.88,1.04,;-5.25,1.77,;-3.94,-.51,;-2.59,-1.27,;-2.59,-2.85,;-1.27,-.51,;.07,-1.3,;-1.24,1.04,;-5.22,-1.3,;-6.57,-.54,;-6.57,1.04,;-7.89,-1.3,;-7.89,-2.88,;-6.57,-3.63,;-6.2,-5.13,;-4.67,-5.25,;-3.96,-6.69,;-4.08,-3.82,;-2.58,-3.46,;-1.09,-3.1,;-5.25,-2.82,;5.43,-1.24,;5.75,.19,;7.27,.37,;7.89,-1.04,;6.74,-2.09,;6.42,-3.61,;4.9,-3.73,;4.12,-5.08,;4.26,-2.38,)|
Nc1nc2c(ccc(F)c2s1)-c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r,wU:18.51,21.50,29.31,wD:17.25,35.39,(-3.55,3.51,;-4.32,4.85,;-3.68,6.26,;-4.81,7.28,;-4.78,8.81,;-6.13,9.54,;-7.41,8.84,;-7.47,7.31,;-8.81,6.53,;-6.11,6.52,;-5.79,4.99,;-3.04,9.81,;-3.02,11.35,;-4.35,12.12,;-1.67,12.08,;-1.88,13.58,;-.85,14.72,;.74,14.55,;1.23,16.02,;2.63,16.58,;3.97,15.77,;4.09,14.27,;3.12,13.15,;1.59,13.29,;.96,12.06,;2.33,11.26,;2.31,9.84,;3.65,9.07,;4.98,9.84,;6.32,9.07,;6.64,10.58,;8.18,10.74,;8.81,9.33,;7.66,8.29,;7.34,6.78,;5.8,6.62,;5.03,5.28,;5.17,8.03,;.97,8.97,;-.41,9.77,;-1.72,9.04,;-1.72,7.49,;-.35,11.3,;2.13,14.62,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-8.81,3.66,;-9.74,5.27,;-11.59,5.46,;-11.98,7.29,;-13.31,8.06,;-13.31,9.6,;-11.98,10.37,;-10.65,9.6,;-9.31,10.37,;-9.31,11.91,;-10.56,12.56,;-7.98,12.68,;-8.21,14.2,;-7.16,15.33,;-5.62,15.21,;-5.17,16.68,;-3.74,17.25,;-2.4,16.48,;-2.17,14.95,;-3.22,13.83,;-4.76,13.94,;-5.31,12.68,;-3.98,11.91,;-3.98,10.37,;-2.64,9.6,;-1.31,10.37,;.02,9.6,;.34,11.1,;1.88,11.26,;2.5,9.86,;1.36,8.83,;1.04,7.32,;-.49,7.16,;-1.26,5.83,;-1.12,8.57,;-5.31,9.6,;-6.64,10.37,;-7.98,9.6,;-7.99,8.2,;-6.64,11.91,;-3.68,16.29,;-10.37,8.22,;-8.98,6.97,;-7.16,7.36,;-5.34,7.75,)|
Cc1ccc2sc(N)c(C#N)c2c1-c1c(F)c2nc(OC[C@@]34CCCN3C[C@H](F)C4)nc3N4C[C@H]5CC[C@H](N5)[C@H]4COc(c1Cl)c23 |r,wU:21.22,37.41,34.42,wD:39.44,27.30,(-6.58,1.01,;-6.58,-.54,;-7.93,-1.32,;-7.93,-2.84,;-6.61,-3.61,;-6.26,-5.11,;-4.73,-5.24,;-3.95,-6.61,;-4.13,-3.82,;-2.63,-3.47,;-1.13,-3.12,;-5.3,-2.81,;-5.27,-1.29,;-3.92,-.51,;-2.57,-1.26,;-2.57,-2.84,;-1.26,-.51,;.09,-1.29,;1.41,-.54,;2.78,-1.32,;4.1,-.54,;5.45,-1.26,;5.77,.21,;7.3,.36,;7.93,-1.05,;6.79,-2.06,;6.46,-3.59,;4.91,-3.71,;4.11,-5.04,;4.28,-2.3,;1.44,1.02,;.06,1.8,;.48,3.29,;2,3.26,;2.93,4.43,;2.69,5.92,;1.26,6.61,;-.06,5.95,;1.11,4.58,;-.45,4.46,;-1.97,4.49,;-2.96,3.26,;-2.6,1.77,;-3.92,1.02,;-5.27,1.77,;-1.23,1.02,)|
Nc1nc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2n1C(F)F |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-4.15,-23.26,;-4.92,-21.92,;-6.45,-21.76,;-6.77,-20.26,;-8.1,-19.49,;-8.1,-17.95,;-6.77,-17.18,;-5.44,-17.95,;-4.1,-17.18,;-4.1,-15.64,;-5.44,-14.87,;-2.77,-14.87,;-3,-13.34,;-1.95,-12.22,;-.42,-12.33,;.04,-10.86,;1.47,-10.3,;2.81,-11.07,;3.04,-12.59,;1.99,-13.72,;.45,-13.6,;-.1,-14.87,;1.23,-15.64,;1.23,-17.18,;2.57,-17.95,;3.9,-17.18,;5.23,-17.95,;5.55,-16.44,;7.08,-16.28,;7.71,-17.69,;6.57,-18.72,;6.25,-20.22,;4.72,-20.38,;3.98,-21.46,;4.09,-18.98,;-.1,-17.95,;-1.44,-17.18,;-2.77,-17.95,;-2.77,-19.49,;-1.44,-15.64,;1.18,-12.09,;-5.44,-19.49,;-4.29,-20.52,;-2.75,-20.52,;-1.26,-20.12,;-2.55,-22.04,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,26.26,wD:14.20,32.34,(-4.92,-13.3,;-5.69,-11.97,;-7.22,-11.81,;-7.54,-10.3,;-8.87,-9.53,;-8.87,-7.99,;-7.54,-7.22,;-6.2,-7.99,;-4.87,-7.22,;-4.87,-5.68,;-6.2,-4.91,;-3.54,-4.91,;-3.77,-3.39,;-2.72,-2.26,;-1.18,-2.37,;-.73,-.9,;.7,-.34,;2.04,-1.11,;2.27,-2.63,;1.22,-3.76,;-.32,-3.64,;-.87,-4.91,;.46,-5.68,;.46,-7.22,;1.8,-7.99,;3.13,-7.22,;4.46,-7.99,;4.79,-6.48,;6.32,-6.32,;6.94,-7.73,;5.8,-8.76,;5.48,-10.27,;3.95,-10.43,;3.21,-11.5,;3.32,-9.02,;-.87,-7.99,;-2.2,-7.22,;-3.54,-7.99,;-3.54,-9.53,;-2.2,-5.68,;.53,-2,;-6.2,-9.53,;-5.06,-10.56,;-3.55,-10.24,;-2.05,-9.92,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@]78CCCN7C[C@@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:15.46,18.45,32.34,wD:14.20,26.26,(-4.92,-13.3,;-5.69,-11.97,;-7.22,-11.81,;-7.54,-10.3,;-8.87,-9.53,;-8.87,-7.99,;-7.54,-7.22,;-6.2,-7.99,;-4.87,-7.22,;-4.87,-5.68,;-6.2,-4.91,;-3.54,-4.91,;-3.77,-3.39,;-2.72,-2.26,;-1.18,-2.37,;-.73,-.9,;.7,-.34,;2.04,-1.11,;2.27,-2.63,;1.22,-3.76,;-.32,-3.64,;-.87,-4.91,;.46,-5.68,;.46,-7.22,;1.8,-7.99,;3.13,-7.22,;4.46,-7.99,;4.79,-6.48,;6.32,-6.32,;6.94,-7.73,;5.8,-8.76,;5.48,-10.27,;3.95,-10.43,;3.21,-11.5,;3.32,-9.02,;-.87,-7.99,;-2.2,-7.22,;-3.54,-7.99,;-3.54,-9.53,;-2.2,-5.68,;.53,-2,;-6.2,-9.53,;-5.06,-10.56,;-3.55,-10.24,;-2.05,-9.92,)|
Nc1sc2CCC=C(c2c1C#N)c1c(Cl)c2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r,c:6|
Nc1n[nH]c2sc3cccc(-c4c(Cl)c5OC[C@@H]6[C@@H]7CC[C@H](CN6c6nc(OC[C@@]89CCCN8C[C@H](F)C9)nc(c4F)c56)N7)c3c12 |r,wU:18.49,21.48,29.29,wD:17.23,35.37,(1.47,-35.88,;.14,-36.65,;.46,-38.16,;-.88,-38.93,;-2.02,-37.9,;-3.55,-37.74,;-3.87,-36.23,;-5.21,-35.46,;-5.21,-33.92,;-3.87,-33.15,;-2.54,-33.92,;-1.21,-33.15,;-1.21,-31.61,;-2.54,-30.84,;.13,-30.84,;-.1,-29.32,;.95,-28.19,;2.48,-28.31,;2.94,-26.83,;4.37,-26.27,;5.7,-27.04,;5.93,-28.56,;4.88,-29.69,;3.35,-29.58,;2.8,-30.84,;4.13,-31.61,;4.13,-33.15,;5.46,-33.92,;6.8,-33.15,;8.13,-33.92,;8.45,-32.42,;9.98,-32.26,;10.61,-33.66,;9.46,-34.69,;9.14,-36.2,;7.61,-36.36,;6.84,-37.69,;6.99,-34.95,;2.8,-33.92,;1.46,-33.15,;.13,-33.92,;.13,-35.46,;1.46,-31.61,;4.13,-28.02,;-2.54,-35.46,;-1.39,-36.49,)|
CC(C)(C)OC(=O)Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:33.33,22.53,25.52,wD:39.41,21.27,(-10.26,-4.23,;-9.37,-2.56,;-7.7,-3.46,;-11.03,-1.66,;-8.46,-.88,;-9.79,.65,;-11.74,.17,;-9.2,2.6,;-9.77,4.54,;-11.65,4.74,;-12.04,6.59,;-13.38,7.36,;-13.38,8.9,;-12.04,9.67,;-10.71,8.9,;-9.38,9.67,;-9.38,11.21,;-10.71,11.98,;-8.04,11.98,;-8.27,13.5,;-7.23,14.63,;-5.69,14.52,;-5.24,15.99,;-3.8,16.55,;-2.47,15.78,;-2.24,14.26,;-3.29,13.13,;-4.82,13.24,;-5.38,11.98,;-4.04,11.21,;-4.04,9.67,;-2.71,8.9,;-1.38,9.67,;-.04,8.9,;.28,10.41,;1.81,10.57,;2.44,9.16,;1.29,8.13,;.97,6.62,;-.56,6.46,;-1.33,5.13,;-1.19,7.87,;-5.38,8.9,;-6.71,9.67,;-8.04,8.9,;-8.04,7.36,;-6.71,11.21,;-3.88,14.87,;-10.41,7.54,;-9,6.27,;-6.9,5.62,;-5.39,4.26,)|
Nc1sc2cccc(-c3c(Cl)c4OC[C@@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c2c1C#N |r,wU:26.26,15.46,18.45,wD:32.34,14.20,(-9.21,2.6,;-9.77,4.54,;-11.65,4.74,;-12.04,6.59,;-13.38,7.36,;-13.38,8.9,;-12.04,9.67,;-10.71,8.9,;-9.38,9.67,;-9.38,11.21,;-10.71,11.98,;-8.04,11.98,;-8.27,13.5,;-7.23,14.63,;-5.69,14.52,;-5.24,15.99,;-3.8,16.55,;-2.47,15.78,;-2.24,14.26,;-3.29,13.13,;-4.82,13.24,;-5.38,11.98,;-4.04,11.21,;-4.04,9.67,;-2.71,8.9,;-1.38,9.67,;-.04,8.9,;.28,10.41,;1.81,10.57,;2.44,9.16,;1.29,8.13,;.97,6.62,;-.56,6.46,;-1.33,5.13,;-1.19,7.87,;-5.38,8.9,;-6.71,9.67,;-8.04,8.9,;-8.04,7.36,;-6.71,11.21,;-3.88,14.87,;-10.41,7.54,;-9,6.27,;-6.9,5.62,;-5.39,4.26,)|
CN1CCC[C@@H]1COc1nc2N3C[C@H]4CC[C@H](N4)[C@H]3COc3c(Cl)c(c(F)c(n1)c23)-c1cccc2sc(N)c(C#N)c12 |r,wU:5.6,16.17,13.18,wD:18.20,(-.12,-1.59,;1.02,-.56,;2.53,-.88,;3.3,.45,;2.27,1.59,;.86,.97,;-.47,1.74,;-1.8,.97,;-3.14,1.74,;-3.14,3.28,;-4.47,4.05,;-3.92,5.31,;-2.38,5.2,;-1.34,6.33,;-1.56,7.85,;-2.9,8.62,;-4.33,8.06,;-2.92,7.09,;-4.79,6.58,;-6.32,6.7,;-7.37,5.57,;-7.14,4.05,;-8.47,3.28,;-9.81,4.05,;-8.47,1.74,;-7.14,.97,;-7.14,-.57,;-5.81,1.74,;-4.47,.97,;-5.81,3.28,;-9.81,.97,;-11.14,1.74,;-12.47,.97,;-12.47,-.57,;-11.14,-1.34,;-10.82,-2.85,;-9.29,-3.01,;-8.68,-4.53,;-8.66,-1.6,;-7.08,-1.58,;-5.49,-2.1,;-9.81,-.57,)|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4CC5CCC(C4)N5)c3CO2)c1C(F)(F)F |r,w:8.7|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4CC5CC(C4)N5)c3CO2)c1C(F)(F)F |r,w:8.7|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@@H]5NCC[C@H]45)c3CO2)c1C(F)(F)F |r,w:8.7|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C5CCC4CNC5)c3CO2)c1C(F)(F)F |r,w:8.7|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4C[C@@H]5CC[C@H]4CN5)c3CO2)c1C(F)(F)F |r,w:8.7|
Cc1cc(N)c(F)c(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4CC5NC(C4)C=C5)c3CO2)c1C(F)(F)F |r,w:8.7,c:35|
Oc1cc(C2Cc3nc(OC[C@@]45CCCN4C[C@H](F)C5)nc(N4CC5CCC(C4)N5)c3CO2)c2ccccc2c1 |r|
COc1ccc(CN(Cc2ccc(OC)cc2)c2cc(C)c(c(C3OCc4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4N4CC5CCC(C4)N5)C3C)c2F)C(F)(F)F)cc1 |r,TLB:42:43:50:46.47|
COc1ccc(CN(Cc2ccc(OC)cc2)c2cc(C)c(c(C3Cc4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(N5CC6CCC(C5)N6)c4C(C)O3)c2F)C(F)(F)F)cc1 |r,TLB:40:41:48:44.45|
CCc1cccc2cc(O)cc(-c3cc4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc5N6C[C@H]7CC[C@H](N7)[C@H]6COc(n3)c45)c12 |r|
Oc1cc(Cl)c(C2CC2)c(c1)-c1nc2OC[C@@H]3[C@@H]4CC[C@H](CN3c3nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(c1F)c23)N4 |r|
[H][C@]12CC[C@]([H])(N1)[C@@]1([H])COc3nc(c(F)c4nc(OC[C@@]56CCCN5C[C@H](F)C6)nc(N1C2)c34)-c1cc(O)cc2ccc(F)c(CC)c12 |r|
CCc1cccc2cc(O)cc(-c3nc4OC[C@H]5[C@@H]6CC[C@H](CN5c5nc(OC[C@@]78CCCN7C[C@H](F)C8)nc(c3F)c45)N6)c12 |r|
Cc4cc(N)nc(c3cc1ncnc2c1c(OCCN2CCN(C)C)c3Cl)c4C(F)(F)F
Cc4cc(N)nc(c3cc1ncnc2c1c(OCCN2CCN(C)CCO)c3Cl)c4C(F)(F)F
CNCCN2CCOc3c(Cl)c(c1nc(N)cc(C)c1C(F)(F)F)cc4ncnc2c34
Cc5cc(N)nc(c4cc1ncnc2c1c(OCCN2CCN3CCOCC3)c4Cl)c5C(F)(F)F
Cc5cc(N)nc(c4cc1ncnc2c1c(OCCN2[C@@H]3CCNC3)c4Cl)c5C(F)(F)F
Cc5cc(N)nc(c4cc1ncnc2c1c(OCCN2[C@H]3CCNC3)c4Cl)c5C(F)(F)F
Cc5cc(N)nc(c4cc1ncnc2c1c(OC[C@H](CC#N)N2[C@@H]3CCNC3)c4Cl)c5C(F)(F)F
Cc5cc(N)nc(c4cc1ncnc2c1c(OC[C@H](CC#N)N2[C@H]3CCNC3)c4Cl)c5C(F)(F)F
Cc5cc(N)nc(c4cc2nc(OC[C@@H]1C[C@@H](F)CN1C)nc3c2c(OCCN3CCN(C)C)c4Cl)c5C(F)(F)F
Cc6cc(N)nc(c5cc3nc(OCC12CCCN1CCC2)nc4c3c(OCCN4CCN(C)C)c5Cl)c6C(F)(F)F
C=C6CN1CCC[C@@]1(COc5nc2c4c(OCCN2CCN(C)C)c(Cl)c(c3nc(N)cc(C)c3C(F)(F)F)cc4n5)C6
C=C7CN1CCC[C@@]1(COc6nc2c5c(OCCN2CCN(C)C)c(Cl)c(c3c(F)ccc4cnn(C)c34)cc5n6)C7
C=C6CN1CCC[C@@]1(COc5nc2c4c(OCCN2CCN(C)C)c(Cl)c(c3nc(N)cc(C)c3C(F)(F)F)c(F)c4n5)C6
C=C6CN1CCC[C@@]1(COc5nc2c4c(OCCN2CCN(C)C)c(Cl)c(c3nc(N)cc(C)c3C(F)(F)F)c(F)c4n5)C6
C=C7CN1CCC[C@@]1(COc6nc2c5c(OCCN2C3CCNC3)c(Cl)c(c4nc(N)cc(C)c4C(F)(F)F)c(F)c5n6)C7
C=C7CN1CCC[C@@]1(COc6nc2c5c(OCCN2[C@@H]3CCNC3)c(Cl)c(c4nc(N)cc(C)c4C(F)(F)F)c(F)c5n6)C7
C=C7CN1CCC[C@@]1(COc6nc2c5c(OCCN2[C@H]3CCNC3)c(Cl)c(c4nc(N)cc(C)c4C(F)(F)F)c(F)c5n6)C7
C=C7CN1CCC[C@@]1(COc6nc2c5c(OCCN2C3CCNC3)c(Cl)c(c4nc(N)cc(C)c4C(F)(F)F)c(F)c5n6)C7
C=C6CN1CCC[C@]1(COc5nc2c4c(OCCN2CCN(C)C)c(F)c(c3nc(N)cc(C)c3C(F)(F)F)c(F)c4n5)C6
C=C6CN1CCC[C@@]1(COc5nc2c4c(OCCN2CCN(C)C)c(F)c(c3nc(N)cc(C)c3C(F)(F)F)c(F)c4n5)C6
C#Cc1c(F)ccc2cc(O)cc(-c3cc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOCC3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3cc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3cc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3cc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
Oc1cc(-c2nc3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2CCCOC[C@H]2CC3)c2c(F)c(F)ccc2c1
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCOCCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOCC3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OCC67CCCN6CCC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OCC67CCCN6CCC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)ncn6)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCOCCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6nccnc6C(F)C(C)F)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)ncn6)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CC5(COCC3CC4)OCCO5)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CC(F)(F)COCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C=C4C)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C=C4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCCCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3c(F)c4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3c(F)c4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C/C(=CF)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C[C@@H]4F)c12
C#Cc1c(F)ccc2cc(O)cc(C3=C(F)C4N=C(OC[C@@]56CCCN5C[C@H](F)C6)N=C5C4C(=C3F)C(C)=C[C@H]3COCCCN53)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)ncn6)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)cnn6)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6nccnc6C(F)F)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C=C4C)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@H]3C=C4C)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C[C@H]4C)c12
C#Cc1c(F)ccc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3C[C@@H]4C)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(F)c4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
CCc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCOCC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCOCC[C@H]3CCC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCOCC[C@@H]3CCC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCCC3CCn3nncc3-4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OCC6(CN7CCCCC7)CC6)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OCC6(CN7CCCCC7)CC6)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COC(=O)N(CC)CC)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COC(=O)N6CCCCC6)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cccc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COC(=O)NCC)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CC(F)(F)COC[C@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CC(F)(F)COC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)ncn6)CC7)nc5c3F)N3CCCOC[C@@H]3C=C4C)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COc6cc(C(F)(F)F)cnn6)CC7)nc5c3F)N3CCCOC[C@@H]3C=C4C)c12
Oc1cc(-c2nc3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2CCCOC[C@@H]2CC3)c2c(Cl)cccc2c1
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCCC[C@@H]3CC4)c12
Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2CCCOCC2CC3)c1C(F)(F)F
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6CC(=C)C7)nc5c3F)N3CCCOCC3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@@]6(CC6(F)F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6[C@H](COC(C(F)(F)F)(C(F)(F)F)C(F)(F)F)CC7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOCC3C[C@@H]4O)c12
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOCC3C[C@H]4F)c12
C#Cc7c(F)ccc8cc(O)cc(c4nc5CCC1COCCCN1c6nc(OCC23CCCN2[C@H](COC(C(F)(F)F)C(F)(F)F)CC3)nc(c4F)c56)c78
C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OCC67CCCN6[C@H](COCC(F)(F)F)CC7)nc5c3F)N3CCCOCC3CC4)c12
C#Cc1c(F)c(F)cc2cc(N)cc(-c3nc4c5c(nc(OC[C@@]67CCCN6C[C@H](F)C7)nc5c3F)N3CCCOC[C@@H]3CC4)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(Cl)cc4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(F)cc4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(F)cc4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3ccc4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3cc(OC)c4c(N5CC6C=CC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(F)cc4c(N5CC6C=CC(C5)N6)nc(OC[C@]56CCCN5CC(=C)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(F)cc4c(N5CC6C=CC(C5)N6)nc(OC[C@]56CCCN5C/C(=CF)C6)nc4c3F)c12
C#Cc1c(F)ccc2cc(N)cc(-c3c(Cl)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)c12
Nc1nc2c(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c3F)ccc(F)c2s1
Oc1cc(-c2c(Cl)cc3c(N4C5CCC4CNC5)nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)c2ccccc2c1
Fc1c(-c2c(C3CC3)c(Cl)cc3[nH]ncc23)nc2c3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc13)N1CCCOC[C@H]1CO2
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C6CC6)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
Fc1c(-c2cccc3[nH]ncc23)nc2c3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc13)N1CCCOC[C@H]1CO2
Fc1c(-c2c(Cl)c(Cl)cc3[nH]ncc23)nc2c3c(nc(OC[C@@]45CCCN4C[C@H](F)C5)nc13)N1CCCC[C@H]1CO2
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C)ccc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(Cl)ccc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C(F)F)ccc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(Cl)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C(F)(F)F)ccc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C(F)(F)F)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(Cl)c(C)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(Cl)c(C)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
C=C1CN2CC(F)C[C@@]2(COc2nc3c4c(nc(-c5c(C6CC6)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
F/C=C1/CN2CCC[C@@]2(COc2nc3c4c(nc(-c5c(C6CC6)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
F/C=C\9CN1CCC[C@@]1(COc6nc7c5c(nc(c3c(C2CC2)c(Cl)cc4[nH]ncc34)c(F)c5n6)OC[C@@H]8COCCCN78)C9
C=C1CN2C[C@@H](O)C[C@@]2(COc2nc3c4c(nc(-c5c(C6CC6)c(Cl)cc6[nH]ncc56)c(F)c4n2)OC[C@@H]2COCCCN32)C1
Fc1c(-c2c(C3CC3)c(Cl)cc3[nH]ncc23)nc2c3c(nc(OC[C@@]45CCCN4CC4(CC4)C5)nc13)N1CCCOC[C@H]1CO2
Fc1c(-c2c(C3CC3)c(Cl)cc3[nH]ncc23)nc2c3c(nc(OC[C@]45CCCN4CC4(CC4)C5)nc13)N1CCCOC[C@H]1CO2
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Cc1cc(N)nc(-c2c(Cl)c3c4c(ncnc4c2F)N2C[C@H]4CC[C@H](N4)[C@H]2[C@H](C)O3)c1C(F)(F)F
Cc1cc(N)nc(-c2c(Cl)c3c4c(ncnc4c2F)N2C[C@H]4CC[C@H](N4)[C@H]2[C@H](C)O3)c1C(F)(F)F
COn9ncc8ccc(F)c(c7c(F)c3nc(OC[C@@]12CCCN1C[C@H](F)C2)nc4c3c(O[C@@H](C)[C@@H]5[C@@H]6CC[C@H](CN45)N6)c7Cl)c89
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Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](CN4CCCF)[C@H]2CO3)c1C(F)(F)F
Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](CN4CCCF)[C@H]2CO3)c1C(F)(F)F
Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](CN4C)[C@H]2CO3)c1C(F)(F)F
Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](CN4CC4COC4)[C@H]2CO3)c1C(F)(F)F
Cc1cc(N)nc(-c2c(Cl)c3c4c(nc(OC[C@@]56CCCN5C[C@H](F)C6)nc4c2F)N2C[C@H]4CC[C@H](CN4CCCC#N)[C@H]2CO3)c1C(F)(F)F
Cc8cc(N)nc(c7c(F)c3nc(OC[C@@]12CCCN1C/C(=C/F)C2)nc4c3c(OC[C@@H]5[C@@H]6CC[C@H](CN45)NC6)c7Cl)c8C(F)(F)F
Cc8cc(N)nc(c7c(F)c3nc(OC[C@@]12CCCN1C/C(=C/F)C2)nc4c3c(OC[C@@H]5[C@@H]6CC[C@H](CN45)N(CCCF)C6)c7Cl)c8C(F)(F)F
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCN(C(=O)C#CCN3CCOCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CN(C(=O)CCl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CC(C)[C@@H](C(=O)N[C@H]1Cc2cc(O)cc(c2)-c2ccc3c(C(C)(C)C#N)cn(c3c2)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)N1CCCC2(CCN(C(=O)CCl)C2)C1=O
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(F)Cl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC(C=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)/C=C/n3cncn3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H](F)Cl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCCC3(CCN(C(=O)[C@H](F)Cl)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncc(N2CCN(C)CC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(F)CCN(C(=O)[C@H](F)Cl)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncc(N2CCN(C)CC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H](F)Cl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncc(N2CCN(C)CC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CC[C@]3(CCN(C(=O)[C@H](F)Cl)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncc(N2CCN(C)CC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CC[C@]3(CCN(C(=O)[C@H](F)Cl)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncc(N2CCOCC2)cc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H](F)Cl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(CC(F)(F)F)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H](F)Cl)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC1CN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N1COCC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncccc1-c1c2c3cc(ccc3n1C)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncccc1-c1c2c3cc(ccc3n1C)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(CCO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(CCO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(CCO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCc1ncccc1-c1c2c3cc(ccc3n1CC)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CNC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@@H](O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCNCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCN3CCOCC13)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)Cc1cc[nH]n1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CNC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(S(=O)(=O)CC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC3CCCCN3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCC[C@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(O)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC3CC1CN3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCN[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@@]3(C)CCCN3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)NC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(CN)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN3CC(O)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC13CNC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(=C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1[C@H](C)CCN1C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(cc(NC(C)=O)c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC13CCNC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
C=C[C@@H]1C[C@]1(N)C(=O)N(C)[C@H](C(=O)N[C@H]1Cc2cc(O)cc(c2)-c2ccc3c(c2)c(c(-c2cccnc2[C@H](C)OC)n3CC)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)C(C)C
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(C(=O)O)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC13CCNCC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1nc(cs1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(cc3nc[nH]c13)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(cc(S(C)(=O)=O)c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C13CNCC1C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC13CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CC1(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CC1(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(C#N)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN1C[C@@H](C(=O)N(C)[C@H](C(=O)N[C@H]2Cc3cc(O)cc(c3)-c3ccc4c(c3)c(c(-c3cnccc3COC)n4CC)CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C2=O)C(C)C)CC1=O
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1C[C@@H]1F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@@H]1F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@H]1F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1[C@@H]3CNC[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1[C@@H]3CNC[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn5c(c1cccnc1[C@@H](C)OC)c6CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C3(F)CC3)Cc4cc(O)cc(c4)c7ccc5c6c7
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CC1(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CC1(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(N)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](NC(C)=O)C(C)(C)OC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C3CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1CCCCCN1C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)CCc1ccncc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)CC(C)c1ccncc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(C)Cc1ccncc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C13CCCC1C3(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C1CCC3C1C3(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H]1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(C1CC1)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OCc1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)CC#N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)CC1OCCC13CNC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)CC1CCC3(CNC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)N1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)CCN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)C1CS(=O)(=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)c1cnc[nH]1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)N1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)c1ccc(O)cc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)c1cn(C)c(C)n1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)c1ccc(OC)cc1OC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN3CC[C@H](O)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NS(=O)(=O)CC1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CCc3ccccc3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC3CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2ccccc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN(C3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1[C@H]3C[C@H]3CN1C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1[C@@H](C)CCN1C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCOC(=O)N1CC[C@H](C(=O)N(C)[C@H](C(=O)N[C@H]2Cc3cc(O)cc(c3)-c3ccc4c(c3)c(c(-c3cccnc3[C@H](C)OC)n4CC)CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C2=O)C(C)C)C1
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCCC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CCN(C)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](NC(C)=O)C(C)(C)O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CN(C(C)=O)C[C@H]1C(F)(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CNC[C@H]1C(F)(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1NC[C@@H]3C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CCN(S(C)(=O)=O)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CCN(C(=O)OC)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CN(C)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C1CCC1C#N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCc3ccccc3N1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1NCCC1C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1NCCC13CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CNCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(CCO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCC(=O)N1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CN[C@@H]3CCO[C@H]13)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(CO)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC(C)(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CN(S(C)(=O)=O)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(CN(C(=O)OC)C3)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(C)C1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(S(C)(=O)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(S(C)(=O)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@H](O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn5c(c1cccnc1[C@H](C)OC)c6CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]3CCN(C(C)=O)C3)Cc4nc(cs4)c7ccc5c6c7
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCc3ncccc3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN1CC(C(=O)N(C)[C@H](C(=O)N[C@H]2Cc3cc(O)cc(c3)-c3ccc4c(c3)c(c(-c3cccnc3[C@H](C)OC)n4CC)CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C2=O)C(C)C)CC1=O
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1Cc3nccn3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)cc2cc(-c3cc(O)cc(C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N4CCC[C@@H](C(=O)OCC(C)C)N4)c3)ccc21
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1Cc3cccnc3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CNC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC(=O)N(C3CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C1[C@H]3COC[C@@H]13)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C1CCCC1C(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCNCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(C)C1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C1CCCC1C(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN1C[C@@H](C(=O)N(C)[C@H](C(=O)N[C@H]2Cc3cc(O)cc(c3)-c3ccc4c(c3)c(c(-c3cnccc3COC)n4CC)CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C2=O)C(C)C)CC1=O
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CC[C@@H]1COC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCC[C@@H]1COC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC1C(=O)O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1[C@H](C)CN(C)C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13CCN(C)CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn6c(c1cccnc1[C@H](C)OC)c7CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N3CCC34CN(C)C4)Cc5nc(cs5)c8ccc6c7c8
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1[C@H](C)COC[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1[C@H](C)COC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](C)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](C)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N(C)C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H]1C(=O)NC)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H]1C(=O)NC)C(=O)N1CC(C)C[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H](C)N(C)C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3CC(C1)N3C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C3CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H]1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N3CCN(C)CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C(C)(C)O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)CN(C)C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(C)=O)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H](C)N(C)C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H](C)N(C)C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC3(CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N3CCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN3CCOCC3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(n3nc(C)cc3C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C)(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H](C)N(C)C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3CC(C1)O3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC(F)F)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncccc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)CO)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)CC13CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3CCC1CN3C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@@H](C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C[C@@H](C)O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@H](C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)C3(CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3COC[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3CN(C)C[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3C[C@H]1CN3C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncccc1-c1c2c3cc(ccc3n1CC(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCCN(C)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN(CC)C1CN(C(=O)N(C)[C@H](C(=O)N[C@H]2Cc3nc(cs3)-c3ccc4c(c3)c(c(-c3cccnc3[C@H](C)OC)n4CC)CC(C)(C)COC(=O)[C@@H]3CCCN(N3)C2=O)C(C)C)C1
CCn1c(-c2cccnc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)C1(F)COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)S(=O)(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@@H]1O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H]1[C@@H](C)CCCN1C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CN(C(=O)OC)C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2C2CCCC2)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CC(Br)C[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2C2CCCC2)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CO[C@@H](C)c1ncccc1-c1c2c3cc(ccc3n1CC(F)(F)F)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N3CCCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2ccccc2CCOC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC(F)(F)F)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)CC(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN(C(=O)N(C)[C@H](C(=O)N[C@H]1Cc2nc(cs2)-c2ccc3c(c2)c(c(-c2cccnc2[C@H](C)OC)n3CC)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)C(C)C)C(C)C
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN(C)C(=O)N(C)[C@H](C(=O)N[C@H]1Cc2nc(cs2)-c2ccc3c(c2)c(c(-c2cccnc2[C@H](C)OC)n3CC)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)C(C)C
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N3CCOCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)N(C)CC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN(C(=O)[C@]3(C)CCCN3C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C(=O)O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N1CNCC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@@H]1O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1C[C@H]1O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)OC3CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(S(=O)(=O)N3CC(N)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCN(CC)C(=O)N(C)[C@H](C(=O)N[C@H]1Cc2nc(cs2)-c2ccc3c(c2)c(c(-c2cccnc2[C@H](C)OC)n3CC)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)C(C)C
CCN(C(=O)N(C)[C@H](C(=O)N[C@H]1Cc2nc(cs2)-c2ccc3c(c2)c(c(-c2cccnc2[C@H](C)OC)n3CC)CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C1=O)C(C)C)C1CC1
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(CO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCS(=O)(=O)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@@H]1CCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2ccccc2CCOC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CCCN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H]1CCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)C1(F)CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)C1(F)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)c1ccccn1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)N1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(S(=O)(=O)N3CC(O)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@@H]3CCCN3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H]3CCCN3C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCNCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H](O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@H]3CCCN3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@@]3(C)CCCN3C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)c1ncco1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@]3(C)CCCN3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C#N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(S(C)(=O)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@@H]3CCCN3C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)[C@@H](C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(COC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(c3cn[nH]c3c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCN(C)C1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC1COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CC[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CC[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCNC13CCC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCC[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCCC[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCC(C3CCCO3)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CC[C@@H](CN(C)C)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)C(C)=C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N1CCCC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H](O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CN3CCCN1CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCC(=O)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C13CC(CO1)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OC[C@@H]3CCC[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCC(C(F)(F)F)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCC3(CCOC3)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C13CCC(CO1)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C13CCC(CO1)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C13CCC(CC1)O3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CC3(CCOCC3)CO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CC[C@@H](C(N)=O)O1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(C(F)F)CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1[C@H]3CC[C@H](C3)[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1COC[C@@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCC[C@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1OCC[C@H]1N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1[C@@H](N)[C@@H]3CC[C@H]1O3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC(C(=O)C(F)(F)F)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)[C@H]1OCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)N1CCS(=N)(=O)CC1)C(=O)N1CCC[C@H](N1)C(=O)CCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1OCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)N1CCS(=O)(=NC)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC(C(=O)C(F)(F)F)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1OCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1OCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CO)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(C#N)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)NCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CNCCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC3(CC1)CN(C)CCO3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@]13CCCNC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@]13CCCNC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@@]3(CCN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)[C@H](c3ccccc3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13CCNCC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCS1(=O)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N1CCCCC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCCS1(=O)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@]3(CCN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@]13CCCN(C)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)C3(N(C)C)CC3)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3OCCN(C)[C@@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3OCCN(C)[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3CN(C)C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1[C@@H]3CN(C)C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1[C@@H]3CNC[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCNC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C3CCOCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccncc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3OCCN(C)[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C#N)(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CCCN(C)C3=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1(COC)COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N)(C#N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N4CC(F)C4)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)CCN(C)C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C3CCC1CN(C)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@]3(CCN(C)C3=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3CN(C)CC[C@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H]1CN)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)[C@@H]1CCN(C)[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N(C)CCO)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@]13CCCN(C)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C[C@H]1CCN1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C[C@H](C)O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H]3CN(C)C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H]3CN(C)C[C@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3[C@@H](C1)OCCN3C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C[C@H]1CCCN1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC13COC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC3(COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H](C)N(C)C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](C)CO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@]3(CCNC3=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H](N)CCCNC(=N)N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@]3(CCNC3=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3CN(C)CC[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(C1)CS(=O)(=O)CCN3C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13CCN(C)CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(C3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N(C)C(C)C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N4CCOCC4)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](C)CO)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](C)NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)[C@@H](O)[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(C)COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1cccnc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC[C@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC[C@@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@H](N(C)C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@@H](N(C)C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@]3(CCN(C)C3=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C3CC1CS(=O)(=O)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3CN(C)C[C@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC13CCN(C)CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CN(C)CCO3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn6c(c1cccnc1[C@H](C)OC)c7CC(C)(C)COC(=O)[C@@H]2CCCN(N2)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N4CC(Cc3cnn(C)c3)C4)Cc5nc(cs5)c8ccc6c7c8
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN(C(=O)OC)[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H]1CN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC3(CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C[C@@H]1CCCN1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(C3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H](F)[C@H](NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN(C(=O)CN(C)C)[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H]1CN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(CF)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(O)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N(C)C4COC4)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(NCCOC)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CCN(C)CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](CO)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](CO)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@@H]3CCN(C)C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3CCN(C)C[C@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@@H]1CN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@H]1CN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)c1ncco1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC13CCOCC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CCOCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CCCO3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)[C@@H](c3ccccc3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)N1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1(C)COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC13COC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C1CCCC1)N(C)C(=O)N1CCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](OC(=O)N(C)C)C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13CCS(=O)(=O)CC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CC(N(C)CCOC)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](C)COC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@@H](C)COC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](C)NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN3C(=O)CN(C)C[C@@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN3C(=O)CN(C)C[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC([C@H](C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3CCN(C)CC31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C3COCC1C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C3CC1CN(C)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C(=O)N3CCOCC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1C[C@@H](c3ccccc3)CC1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC13CN(C)C3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1cccnc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN3CCOC[C@@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN3CCOC[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(S(=O)(=O)NC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(N(C)S(C)(=O)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(S(=O)(=O)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(NS(C)(=O)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(O)(COC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1C[C@H]1O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(CCc1ccncc1)C1CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)CCc1ccncc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H]1CN)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H](F)[C@H](N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](NC(=O)c1ncco1)C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13COC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N1CCC3(COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)[C@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)[C@@H]1CCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC3(CCN(C)CC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H](N)[C@@H](F)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H]3CCN(C)[C@H]3C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)S(C)(=O)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC(N(C)C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC[C@@H]1CN(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@H](CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@@H](CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(CN(C)C)(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(C3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](CC1CC1)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CC[C@H](C)[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H](OC)[C@@H](N)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1C[C@H](N)[C@@H](O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@H](c3ccccc3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)[C@@H]1CCCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)[C@H]1CCCN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCCC3(CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@@H](OC(=O)N1CCCC1)C(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@H](CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@@H](CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(cc(C(F)F)c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cc(N3CCN(C)CC3)cnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1OCC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)[C@H]3CCCN3C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)[C@@H]3CCCN3C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(O)(CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)[C@@H](OC)[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC[C@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN3CC[C@@H](O)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCO[C@@H](c3ccccc3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCC13CCOCC3)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC3(CCN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC[C@H](N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCOC[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCN[C@@H]1c1ccccc1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)C3COC3)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CCN(C(=O)C3CC3)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C3CN(C)C3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1[C@@H](C)CN(C)C[C@@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1[C@H](C)CN(C)C[C@H]1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N(C)C1CN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2C(C)C)c2c3cc(cnc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2C(C)C)c2c3nc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)N1CC(C(C)(C)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@]1(F)CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@]1(F)CCN(C(=O)OC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CN/C(N)=N/C#N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)c1cnc(N)[nH]c1=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)c1ncc[nH]1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CN1CCOCC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CCCCN)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CCN)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CNC(=N)N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2ccccc2CCOC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CNC(=N)N)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(C)=O)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2ccccc2CCOC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)CCN)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H]([C@H](C)OC)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H]([C@@H](C)OC)N(C)C(C)=O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)CC(F)(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1NC[C@@H]3C[C@@H]31)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CNC[C@@H]1C(F)(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C(C)(C)N(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CN(C(C)=O)C[C@@H]1C(F)(F)F)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)OC1CNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)O[C@@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCN1C)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CCN(C)CC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)c1nccs1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CNC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1CN(C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)C1(O)COC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)C3COC3)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCCO1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H](C)O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H](C)O)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cnccc2COC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@@H]1CCOC1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cc(O)cc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CN(C)C)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1cccc(c1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CNC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2
CCn1c(-c2cccnc2[C@H](C)OC)c2c3cc(ccc31)-c1csc(n1)C[C@H](NC(=O)[C@H](C(C)C)N(C)C(=O)[C@H]1CCN(C(=O)CNC)C1)C(=O)N1CCC[C@H](N1)C(=O)OCC(C)(C)C2