Compile Data Set for Download or QSAR
Report error Found 227 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase catalytic subunit alpha/beta/gamma'
LigandPNGBDBM50215107(CHEMBL3143638)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of cAMP dependent protein kinase (PKA)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50215105(CHEMBL3143641)
Affinity DataEC50:  150nMAssay Description:Activation of cAMP dependent protein kinase (PKA)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50215106(CHEMBL230552 | CHEBI:84612 | 8-pCPT-cAMP)
Affinity DataEC50:  2.00E+4nMAssay Description:Activation of cAMP dependent protein kinase (PKA)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50188913(N-((S)-1-amino-3-(2,4-dichlorophenyl)propan-2-yl)-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117503(CHEMBL3613621)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117504(CHEMBL3613620)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50044004(CHEMBL3356433)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117489(CHEMBL3613598)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117631(CHEMBL3613610)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117632(CHEMBL3613609)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117370(CHEMBL3613599)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117299(CHEMBL3613605)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117629(CHEMBL3613612)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117630(CHEMBL3613611)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117301(CHEMBL3613603)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117635(CHEMBL3613606)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117300(CHEMBL3613604)
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117634(CHEMBL3613607)
Affinity DataIC50: 22nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117633(CHEMBL3613608)
Affinity DataIC50: 24nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117315(CHEMBL3613600)
Affinity DataIC50: 24nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 30nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285250(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 60nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50117627(CHEMBL3613614)
Affinity DataIC50: 69nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM3152(2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...)
Affinity DataIC50: 70nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285251(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 70nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 80nMAssay Description:Inhibition of protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 80nMAssay Description:Inhibition of cAMP-dependent protein kinase (Protein kinase A)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50117303(CHEMBL3613601)
Affinity DataIC50: 81nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117302(CHEMBL3613602)
Affinity DataIC50: 150nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117502(CHEMBL3613622)
Affinity DataIC50: 332nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 790nMAssay Description:Inhibition of cAMP-dependent protein kinase (Protein kinase A)More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50192071((13R,15S)-13-methyl-16-oxa-8,9,12,22,24-pentaazahe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117626(CHEMBL3613615)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117505(CHEMBL3613619)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117581(CHEMBL3613618)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117598(CHEMBL3613617)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117625(CHEMBL3613616)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117501(CHEMBL3613623)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117500(CHEMBL3613624)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117628(CHEMBL3613613)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of PKA (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM3154(2-({2,6-dihydroxy-4-[({3-[(4-hydroxybenzene)amido]...)
Affinity DataIC50: 1.90E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM2672(6,7,12,13-Tetrahydro-5,7-dioxo-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50213033(CHEMBL329274)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of c-AMP dependent kinase (PKA) using histone II A proteinMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Protein kinase AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50290416({4-[1-(3-Amino-propyl)-1H-indol-4-yl]-pyrimidin-2-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of protein kinase A.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM3158(2-{[2,6-dihydroxy-4-({[(4S)-3-[(4-hydroxybenzene)a...)
Affinity DataIC50: 2.00E+3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article

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