Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with Target = 'YEATS domain-containing protein 2'
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566877(CHEMBL4863719)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625612(CHEMBL5416331)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625604(CHEMBL5439680)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625613(CHEMBL5394670)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625614(CHEMBL5427853)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625615(CHEMBL5435042)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625616(CHEMBL5398308)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625617(CHEMBL5421606)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625618(CHEMBL5429859)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50625620(CHEMBL4762606)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of YEATS2 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566867(CHEMBL4855926)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566873(CHEMBL4859531)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50566890(CHEMBL4865432)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetYEATS domain-containing protein 2(Human)
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50616143(CHEMBL5439514)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity to human his-tagged recombinant YEATS2 expressed in Escherichia coli assessed as inhibition constant using biotin tagged lysine 27-c...More data for this Ligand-Target Pair
In DepthDetails
PubMed