Compile Data Set for Download or QSAR
Report error Found 1730 Enz. Inhib. hit(s) with Target = 'Wee1-like protein kinase'
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13216(N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyeth...)
Affinity DataKd:  7.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataKd:  770nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  3.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  1.60E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  1.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13534(VX680 | N-[4-[[4-(4-methylpiperazino)-6-[(5-methyl...)
Affinity DataKd:  3.20E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM36838(cid_647878 | SMR000001049 | MLS000070497 | 1-ethen...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM36923((Z)-3,4-bis(benzenesulfonyl)but-2-en-1-ol | cid_53...)
Affinity DataEC50: >5.53E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43753(MLS000081058 | cid_665867 | N-benzyl-6-methyl-1H-b...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM38931(6-methyl-2-[3-methyl-5-(4-methylanilino)pyrazol-1-...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43754(SMR000031817 | 4-[[2-(4-ethoxyphenyl)-4-quinolinyl...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM38959(4-(1-methyl-2-oxoquinolin-4-yl)oxy-N-(4-methylpyri...)
Affinity DataEC50:  7.87E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM40850(cid_5771404 | 7-(2,3-dimethoxyphenyl)-5-(3-methoxy...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM38993(SMR000020833 | cid_5286934 | MLS000085704 | (1Z,3Z...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43755(cid_690911 | SMR000069284 | 3-oxidanyl-7-phenyl-py...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43756(N-Cyclohexyl-2-[(3-ethoxy-phenyl)-(2-thiophen-2-yl...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM41591(MLS000540304 | (Z)-2,3-bis(chloranyl)-N-(6-methoxy...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM41593(MLS000540302 | cid_1472216 | (Z)-2,3-dichloro-N-(6...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43757(MLS000554170 | Furan-2-yl-(8-methyl-2-thioxo-2H-[1...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43758(cid_2162384 | methyl 1-[(E)-3-(4-methoxyphenyl)pro...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43759(SMR000130859 | N-(thiophen-2-ylmethyl)-3-(3,4,5-tr...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43375(2-[1-Cyano-2,2,2-trifluoro-eth-(E)-ylidene]-5-phen...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43760(N'-(5-bromanyl-2-oxidanylidene-indol-3-yl)-2-pyrro...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43761([2-methoxy-5-[(naphthalene-2-carbonylhydrazinylide...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43762(N-(4-chloro-2-methylphenyl)-N'-2-pyridinylthio...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43763(4,5-Dimethoxy-1H-indole-2-carboxylic acid [1-(2,3-...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43764(cid_760177 | N'-[4-(diethylamino)benzylidene]-...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43765(N-(furan-2-ylmethyl)-6-propyl-benzo[b][1,4]benzoth...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43766(SMR000156275 | 5,7-dihydroxy-2-(1-hydroxy-4-oxocyc...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43767(cid_2564901 | 2-[4-(4-fluorophenyl)carbonylphenoxy...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43768(1-(3,4-Dichloro-phenyl)-3-thiazol-2-yl-urea | cid_...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43769(MLS000715629 | cid_3128426 | 3-[[4-(2-methyl-3-imi...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43728((E)-N-(5-chloro-2-pyridinyl)-3-phenyl-2-propenamid...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43770((3Z)-3-(2-oxo-2-thiophen-2-ylethylidene)-1,4-dihyd...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43771(SMR000280785 | MLS000711018 | N-[[4-(diethylamino)...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43772(cid_7206036 | SMR000323857 | 3-[(2-fluorophenyl)me...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43773(4-(diethylsulfamoyl)-N-[2-(2-pyridinyl)ethyl]benza...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43774(MLS001017252 | SMR000353528 | N-[4-[(1,3-benzothia...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43775(N-[(5-methylthiophen-2-yl)methylideneamino]-2,3-di...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43776(SMR000436531 | MLS000333177 | cid_941925 | 5-[1-(1...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43477(MLS000766145 | 1,4-Pentadien-3-one, 1,5-di-3-pyrid...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43777(5-(4-methoxyanilino)-2-(4-methoxyphenyl)-1,3-oxazo...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25469(2-[(7-nitro-2,1,3-benzoxadiazol-4-yl)sulfanyl]-1-o...)
Affinity DataEC50: >1.84E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM43778(MLS000860689 | N1-benzyl-2-{[4-(3,4-dimethylthieno...)
Affinity DataEC50: >4.98E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetWee1-like protein kinase 2(Human)
Ambit Biosciences

Curated by ChEMBL
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to WEE2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to WEE1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetWee1-like protein kinase 2(Human)
Ambit Biosciences

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to WEE2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to WEE1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | Vargatef | US10981896, Co...)
Affinity DataKd:  2.90E+3nMAssay Description:Binding constant for WEE1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetWee1-like protein kinase(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  1.60E+3nMAssay Description:Binding constant for WEE1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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