BindingDB PrimarySearch

Report error Found 2958 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor'

Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75537(5-amino-N-(2,3-dimethylphenyl)-1-(2-methylbenzyl)-...)

EC50: >2.99E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75538((Z)-but-2-enedioic acid;1-(3-chloro-5,6-dihydroben...)

EC50: 2.13E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM47719(MLS000539990 | 4-chloro-N-(4-chloro-2-methylphenyl...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75539(cid_2865612 | 2-[(4-chlorophenyl)thio]-N-[4-(4-mor...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

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BDBM75540(SMR000131950 | cid_6280515 | 5-[2-[(E)-(5-methoxy-...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75541(cid_2368087 | SMR000154872 | MLS000569286 | 2-[[5-...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM42052(2-N,3-N-dimethyl-6,7-dinitroquinoxaline-2,3-diamin...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75542(SMR000198437 | cid_2940387 | N-[4-[(4-fluorophenyl...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75543(2-(4-Methoxy-phenyl)-thiazolidine-3-carbothioic ac...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75544(SMR000253424 | 5-(2,4-dichlorophenyl)-5-methyl-3-[...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM74897(1-[3-[(4-fluoranylphenoxy)methyl]-4-methoxy-phenyl...)

EC50: 2.08E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75545(MLS000662389 | cid_2944534 | N-(1,3-benzodioxol-5-...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75546(SMR000280908 | 1-(5-bromo-2-thiophenyl)-2-[2-imino...)

EC50: 1.51E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75547(SMR000282370 | MLS000712603 | 1-carbazol-9-yl-3-[2...)

EC50: 1.27E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75548(3-[2-(4-acetyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-oxoe...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75549((4-Methoxy-benzyl)-(5H-pyrimido[5,4-b]indol-4-yl)-...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75550(cid_24979260 | N-[2-(2-furanyl)-2-(1-piperidinyl)e...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM58926(Ethylhexadecyldimethylammonium bromide | MLS001335...)

EC50: >3.32E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75551(SMR001307039 | 4-chloranyl-2-[[(4-fluorophenyl)met...)

EC50: 1.10E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75552(2-(4-fluorophenoxy)-N-[4-(3,4,5,6-tetrahydro-2H-az...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75553(4-chloro-2-[[(6-chloropyridin-3-yl)methylamino]met...)

EC50: 1.75E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75554((4aR,5R,6aS,6bR,10S,12aR)-2,2,6a,6b,9,9,12a-heptam...)

EC50: 2.33E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM50247213(CHEMBL473106 | cid_2369069 | 3-ethyl-4-(1-(furan-2...)

EC50: 1.05E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM52365(SMR000176434 | 2-(2-hydroxyethyl)-6-piperidin-1-yl...)

EC50: 4.75E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM47577(cid_2584707 | (5Z)-3-ethyl-2-sulfanylidene-5-[(1,2...)

EC50: >9.98E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75711(cid_3484134 | 1-(3,4-dichlorophenyl)-3-[1-(4-morph...)

EC50: 6.23E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75712(SMR000280693 | (4Z)-4-[(2Z)-2-(3-ethyl-1,3-benzoxa...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75713(N-[[3-aminocarbonyl-7-(diethylamino)chromen-2-ylid...)

EC50: 1.86E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75714(MLS001018457 | 1-[1-(4-morpholinyl)-1-phenylpropan...)

EC50: 4.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75715(SMR000549804 | cid_1471100 | MLS001165292 | 6-brom...)

EC50: 6.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM4810(cid_5329098 | CHEMBL276711 | SU5146 | (3Z)-3-[(3,5...)

EC50: 1.21E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75716(SMR000710903 | [1-[methyl-(phenylmethyl)amino]-1-o...)

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM66022(KE-IK | MLS002153668 | SMR001231046 | cid_25163004)

EC50: 8.37E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay

BDBM75717(7-[(4-ethylphenyl)hydrazo]-4-benzimidazolone | cid...)

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)

Kd: 0.640nMAssay Description:Binding potency against V1 receptor in rat liver cellsMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50406623(CHEMBL2115369)

Kd: 0.182nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008092(CHEMBL2372415 | cyclo(Ppa-Phe(NO2)-Phe-Val-Asn-Cys...)

Kd: 3.20nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50406622(CHEMBL2115364)

Kd: 0.479nMAssay Description:Negative log of Kd.More data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008096(CHEMBL2372414 | cyclo(Ppa-Phe(N3)-Phe-Val-Asn-Cys)...)

Kd: 35nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008084(1-[13-Benzyl-7-carbamoylmethyl-10-isopropyl-16-(4-...)

Kd: 41nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008088(CHEMBL2372416 | cyclo(Depa-Phe(N3)-Phe-Val-Asn-Cys...)

Kd: 2.60nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008083([2-({1-[19-Amino-10-(2-carbamoyl-ethyl)-7-carbamoy...)

Kd: 54nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50008085([2-({1-[19-Amino-13-(4-azido-benzyl)-10-(2-carbamo...)

Kd: 76nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50453152(CHEMBL2115365)

Kd: 2.63nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50453150(CHEMBL2372420)

Kd: 27nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50453151(CHEMBL2372421)

Kd: 33nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50453148(CHEMBL2372422)

Kd: 16nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50038603(3-N3-C6H4CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Ar...)

Kd: 0.0540nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50038599(4-N3-C6H4CH2CH2CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro...)

Kd: 0.0400nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair

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Vasopressin V1a receptor(Rat)
University of Sherbrooke

Curated by ChEMBL

BDBM50038602(4-N3-C6H4CH2CO-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-T...)

Kd: 0.150nMAssay Description:Tested for dissociation constant at V1a receptor of rat liver membraneMore data for this Ligand-Target Pair

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Displayed 1 to 50 (of 2958 total ) | Next | Last >>

Filter my 2958 hits

Targets 1▿
- Vasopressin V1a receptor 2958
Publications 50▿
- US Patent US11186577 (2021) 259
- US Patent US10092551 (2018) 173
- Bioorg Med Chem Lett 27: 2331-2335 (2017) 137
- J Med Chem 57: 5306-17 (2014) 132
- J Med Chem 54: 4388-98 (2011) 89
- Bioorg Med Chem Lett 30: (2020) 84
- Bioorg Med Chem 15: 2054-80 (2007) 79
- US Patent US11578077 (2023) 72
- US Patent US11149023 (2021) 70
- J Med Chem 39: 3547-55 (1996) 67
- Bioorg Med Chem Lett 20: 3742-5 (2010) 59
- J Med Chem 36: 2011-7 (1993) 57
- Bioorg Med Chem Lett 21: 4622-8 (2011) 53
- Bioorg Med Chem Lett 21: 3163-7 (2011) 52
- J Med Chem 61: 8670-8692 (2018) 50
- Eur J Med Chem 143: 1644-1656 (2018) 48
- Bioorg Med Chem Lett 30: (2020) 48
- J Med Chem 58: 2275-89 (2015) 45
- US Patent US9617226 (2017) 45
- J Med Chem 35: 151-7 (1992) 44
- Bioorg Med Chem Lett 14: 3143-6 (2004) 36
- Bioorg Med Chem Lett 14: 2747-52 (2004) 34
- Bioorg Med Chem Lett 21: 5684-7 (2011) 34
- J Med Chem 48: 7882-905 (2005) 34
- Bioorg Med Chem Lett 17: 6623-8 (2007) 32
- Eur J Med Chem 108: 730-40 (2016) 31
- US Patent US9687476 (2017) 30
- Bioorg Med Chem Lett 19: 6018-22 (2009) 30
- J Med Chem 45: 2589-98 (2002) 30
- US Patent US10889569 (2021) 30
- J Med Chem 64: 10445-10468 (2021) 30
- US Patent US9187466 (2015) 30
- Bioorg Med Chem Lett 13: 2195-8 (2003) 28
- J Med Chem 41: 2442-4 (1998) 27
- J Med Chem 35: 3905-18 (1992) 24
- J Med Chem 47: 2375-88 (2004) 24
- J Med Chem 53: 6525-38 (2010) 24
- Bioorg Med Chem 17: 3130-41 (2009) 23
- Bioorg Med Chem Lett 5: 119-122 (1995) 22
- PubChem Bioassay (2010) 22
- J Med Chem 50: 835-47 (2007) 22
- Bioorg Med Chem Lett 10: 695-8 (2000) 21
- Bioorg Med Chem Lett 20: 516-20 (2010) 21
- J Med Chem 61: 10173-10184 (2018) 20
- US Patent US9180120 (2015) 19
- J Med Chem 37: 1841-9 (1994) 17
- J Med Chem 38: 1762-9 (1995) 17
- Bioorg Med Chem Lett 14: 2987-9 (2004) 17
- Bioorg Med Chem Lett 12: 3081-4 (2002) 17
- Bioorg Med Chem 7: 1743-54 (1999) 16
- ...
Institutions 32▿
- Blackthorn Therapeutics 259
- Hoffmann-La Roche 245
- Ferring Research Institute 221
- Gedeon Richter 162
- Otsuka Pharmaceutical 140
- Takeda Pharmaceutical 137
- Pfizer 114
- Msd 105
- The University of Sydney 79
- Bayer Intellectual Property 79
- Lehigh University 79
- Johnson and Johnson Pharmaceutical Research and Development 70
- Bayer Pharma Aktiengesellschaft 70
- Johnson & Johnson Pharmaceutical Research & Development 66
- Umr7200 Cnrs/Universit£ 50
- Wyeth-Ayerst Research 48
- F. Hoffmann-La Roche 45
- Abbvie Deutschland 45
- University of Sherbrooke 44
- University of Montpellier 42
- Medical College of Ohio 41
- Serono Pharmaceutical Research Institute 34
- Yamanouchi Pharmaceutical 30
- Jiangsu Hengrui Medicine 30
- Schering-Plough Research Institute 30
- Wyeth Research 28
- Merck Research Laboratories 24
- Drugmoldesign 24
- Astellas Pharma 23
- TBA 22
- The Scripps Research Institute Molecular Screening Center 22
- Upr 9023 Cnrs 17
- ...
Affinity: 0.0040 to 5.4E+5 nM▿
- Ki 1319
- IC50 1160
- Kd 73
- EC50 406
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 111