Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Uncharacterized protein [173-650]'
TargetUncharacterized protein [173-650](Dog)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50: 105nMAssay Description:Antagonist activity at dog GCGR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 mins prior to...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUncharacterized protein [173-650](Dog)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334481(3-(4-((3-(3,5-dichlorophenyl)-5-(4-(trifluorometho...)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at dog GCGR assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed