Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with Target = 'Ubiquitin-like modifier-activating enzyme 1'
TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50616172(CHEMBL5440318)
Affinity DataKd:  630nMAssay Description:Binding affinity to Uba1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fluorescence polarisati...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50616173(CHEMBL5433769)
Affinity DataKd:  720nMAssay Description:Binding affinity to Uba1 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by fluorescence polarisati...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329794(US9663525, Compound I-002 | US9663525, Compound I-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329795(US9663525, Compound I-003 | (rac)((1R,2R,3S,4R)-4-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329797(US9663525, Compound I-005 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329799(US9663525, Compound I-007 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329802(US9663525, Compound I-010 | US9663525, Compound I-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329807(US9663525, Compound I-015 | US9663525, Compound I-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329808(US9663525, Compound I-016 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329809(US9663525, Compound I-017 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329810(US9663525, Compound I-018 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329811(US9663525, Compound I-019 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329812(US9663525, Compound I-020 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329813(US9663525, Compound I-021 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329814(US9663525, Compound I-022 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329816(US9663525, Compound I-024 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329818(US9663525, Compound I-026 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329819(US9663525, Compound I-027 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329820(US9663525, Compound I-028 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329821(US9663525, Compound I-029 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329822(US9663525, Compound I-030 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329823(US9663525, Compound I-031 | (rac)-[(1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329824(US9663525, Compound I-032 | (rac)-[(1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329825(US9663525, Compound I-033 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329826(US9663525, Compound I-034 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329827(US9663525, Compound I-035 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329828(US9663525, Compound I-036 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329829(US9663525, Compound I-037 | (rac)-[(1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329830(US9663525, Compound I-038 | (rac)-[(1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329831(US9663525, Compound I-039 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329832(US9663525, Compound I-040 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329833(US9663525, Compound I-041 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329834(US9663525, Compound I-042 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329835(US9663525, Compound I-043 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329836(US9663525, Compound I-044 | US9663525, Compound I-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329837(US9663525, Compound I-045 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329838(US9663525, Compound I-046 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329839(US9663525, Compound I-047 | (rac)-(1R,2R,3S,4R)-4-...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329840(US9663525, Compound I-048 | (rac)-[(1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329841(US9663525, Compound I-049 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329842(US9663525, Compound I-050 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329844(US9663525, Compound I-052 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329845(US9663525, Compound I-053 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329846(US9663525, Compound I-054 | (rac)-[(1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329847(US9663525, Compound I-055 | (rac)-[(1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329848(US9663525, Compound I-056 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329849(US9663525, Compound I-057 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329850(US9663525, Compound I-058 | (rac)-((1R,2R,3S,4R)-2...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329853(US9663525, Compound I-061 | (rac)-((1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetUbiquitin-like modifier-activating enzyme 1(Human)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM329854(US9663525, Compound I-062 | (rac)-[(1R,2R,3S,4R)-4...)
Affinity DataIC50: 10nMAssay Description:The UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubi...More data for this Ligand-Target Pair
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US Patent

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