Compile Data Set for Download or QSAR
Report error Found 1552 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A'
LigandPNGBDBM50213779(CHEMBL313598)
Affinity DataIC50: 0.0200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213551(CHEMBL90618)
Affinity DataIC50: 0.0300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213592(CHEMBL315236)
Affinity DataIC50: 0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213695(CHEMBL89032)
Affinity DataIC50: 0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213685(CHEMBL431853)
Affinity DataIC50: 0.0600nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213561(CHEMBL312937)
Affinity DataIC50: 0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213505(CHEMBL314975)
Affinity DataIC50: 0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213687(CHEMBL87244)
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213697(CHEMBL84908)
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213687(CHEMBL87244)
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213593(CHEMBL91046)
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213688(CHEMBL86538)
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213782(CHEMBL264304)
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50470233(CHEMBL80177)
Affinity DataIC50: 0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50213680(CHEMBL87091)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213681(CHEMBL433010)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50470229(CHEMBL76870)
Affinity DataIC50: 0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50213504(CHEMBL89369)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213457(CHEMBL84686)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213500(CHEMBL86337)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213456(CHEMBL315000)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213552(CHEMBL328302)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213567(CHEMBL315983)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213460(CHEMBL85081)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213591(CHEMBL84795)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213458(CHEMBL90672)
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213591(CHEMBL84795)
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213783(CHEMBL328985)
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50470236(CHEMBL309313)
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50470239(CHEMBL311312)
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50283305(3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propy...)
Affinity DataIC50: 0.110nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283317(2-Propyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonyla...)
Affinity DataIC50: 0.130nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283300(2-Butyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonylam...)
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283312(4'-[2-Ethyl-6-(3-isopropyl-ureido)-4-oxo-4H-quinaz...)
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283310(4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-...)
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50213499(CHEMBL88653)
Affinity DataIC50: 0.150nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50230790(CHEMBL292892)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50283316(3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propy...)
Affinity DataIC50: 0.170nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50067536(5-Hydroxy-2,4-dimethyl-8-[2'-(2H-tetrazol-5-yl)-bi...)
Affinity DataIC50: 0.170nMAssay Description:Compound was evaluated for the in vitro inhibition of specific binding of [125I]-A II to Angiotensin II receptor, type 1 from rat adrenal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50213550(CHEMBL87847)
Affinity DataIC50: 0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213557(CHEMBL309602)
Affinity DataIC50: 0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213554(CHEMBL314527)
Affinity DataIC50: 0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213564(CHEMBL316234)
Affinity DataIC50: 0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213569(CHEMBL78866)
Affinity DataIC50: 0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50285769(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285761(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50285760(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50213679(CHEMBL327297 | 5-Beta-Ketosulfoxide Imidazolyl Bip...)
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

LigandPNGBDBM50213781(CHEMBL327927)
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
In DepthDetails

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