Compile Data Set for Download or QSAR
Report error Found 122 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 5'
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <5.01E+4nMAssay Description:Induction of human TRPM5 opening expressed in HEK293 cells by FLIPR membrane potential/summary (Abse5) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571574(CHEMBL4873144)
Affinity DataEC50:  4.68E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571570(CHEMBL4876211)
Affinity DataEC50:  331nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571575(CHEMBL4858947)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571576(CHEMBL4877096)
Affinity DataEC50:  2.29E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571577(CHEMBL4853398)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571578(CHEMBL4870747)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571579(CHEMBL4873490)
Affinity DataEC50:  5.13E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571580(CHEMBL1440011)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571581(CHEMBL4855094)
Affinity DataEC50:  3.02E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571582(CHEMBL4876435)
Affinity DataEC50:  6.03E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571583(CHEMBL4852732)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571584(CHEMBL4868164)
Affinity DataEC50:  1.35E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571585(CHEMBL4847994)
Affinity DataEC50:  1.62E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571586(CHEMBL4846618)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571587(CHEMBL4858831)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571588(CHEMBL4847928)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571589(CHEMBL4849590)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571590(CHEMBL4851802)
Affinity DataEC50:  5.13E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571591(CHEMBL4859679)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571592(CHEMBL4855887)
Affinity DataEC50:  457nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571593(CHEMBL4877090)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571594(CHEMBL4850328)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571595(CHEMBL4876532)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571596(CHEMBL4855627)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571571(CHEMBL4849726)
Affinity DataEC50:  89nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571597(CHEMBL4871574)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571598(CHEMBL4874619)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571599(CHEMBL4866780)
Affinity DataEC50:  575nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571600(CHEMBL4849306)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571601(CHEMBL4867233)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571602(CHEMBL4853883)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571603(CHEMBL4857099)
Affinity DataEC50:  4.68E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571604(CHEMBL4872851)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571605(CHEMBL4869736)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571606(CHEMBL4863555)
Affinity DataEC50:  447nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571607(CHEMBL4863223)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571608(CHEMBL4873210)
Affinity DataEC50:  5.13E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571609(CHEMBL4856537)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571610(CHEMBL4865623)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571611(CHEMBL4849797)
Affinity DataEC50:  468nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571612(CHEMBL4875178)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571613(CHEMBL4869125)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571614(CHEMBL4861541)
Affinity DataEC50:  7.59E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571615(CHEMBL4850518)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571616(CHEMBL4867011)
Affinity DataEC50:  832nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571617(CHEMBL4860824)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571618(CHEMBL4869759)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571619(CHEMBL4873593)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571620(CHEMBL4858854)
Affinity DataEC50:  468nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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