Compile Data Set for Download or QSAR
Report error Found 522 Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-3'
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM85507(NSC_4488 | CAS_4394-00-7 | Niflumic acid (Hit 16) ...)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to human His-tagged TEAD4 YBD (217 to 434 residues) expressed in Escherichia coli BL21(DE3) after 30 mins by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to N-terminal His6 tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells incubated for 30 mins by i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataKd:  8.40E+4nMAssay Description:Binding affinity to N-terminal His6 tagged human TEAD4-YBD (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM30815(4-(4-methylphenoxy)aniline;hydrochloride | MLS0000...)
Affinity DataKd:  4.10E+4nMAssay Description:Binding affinity to N-terminal His6 tagged human TEAD4-YBD (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50535722(CHEMBL4468725)
Affinity DataKd:  25nMAssay Description:Binding affinity to Avi-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 (DE3) by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM85507(NSC_4488 | CAS_4394-00-7 | Niflumic acid (Hit 16) ...)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to N-terminal His6-tagged human TEAD4 YAP binding domain (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells by ITC ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to N-terminal His6-tagged human TEAD4 YAP binding domain (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells by ITC ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM85507(NSC_4488 | CAS_4394-00-7 | Niflumic acid (Hit 16) ...)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YPD domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by isothermal titrati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM626316(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)
Affinity DataEC50:  50nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626317(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)
Affinity DataEC50:  90nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50:  30nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626319(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50:  160nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626320(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626321(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50:  1.00E+3nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626322(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50:  430nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626323(methyl 2-[[[4-cyano-7-(4- isopropylphenyl)-2,3- ...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626324(US11787775, Compound 29 | 2-[[[4-cyano-7-(4-isopro...)
Affinity DataEC50:  280nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626325(1-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)
Affinity DataEC50:  2.10E+3nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626326(7-(4-isopropylphenyl)-5-[(2- methylene-3-oxo-buty...)
Affinity DataEC50:  80nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626327(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)
Affinity DataEC50:  750nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626328(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)
Affinity DataEC50:  180nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626329(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)
Affinity DataEC50:  890nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626330(2-[[[4-cyano-7-[4- (trifluoromethyl)phenyl]-2,3- ...)
Affinity DataEC50:  250nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626331(US11787775, Compound 16-C)
Affinity DataEC50:  10nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626332(US11787775, Compound 16-D)
Affinity DataEC50:  100nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626333(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)
Affinity DataEC50:  60nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626334(2-[[[4-cyano-7-[4-(1,1- difluoroethyl)phenyl]-2,3...)
Affinity DataEC50:  230nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626335(2-[[[4-(4-isopropylphenyl)-6,7- dihydrofuro[3,2-d...)
Affinity DataEC50:  40nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626336(2-[[[4-fluoro-7-(4-isopropylphenyl)- 2,3-dihydrob...)
Affinity DataEC50:  30nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626337(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrofu...)
Affinity DataEC50:  100nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626338(2-[[[7-cyano-4-[4-(1,1- difluoroethyl)phenyl]-1,3...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626339(2-[[[6-methoxy-5-[(E)-2-[trans-4- (trifluoromethy...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626341(2-[[[4-cyano-7-(2,6-difluoro-4- isopropyl-phenyl)...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626342(2-[[[4-cyano-7-(2-fluoro-4- isopropyl-phenyl)-2,3...)
Affinity DataEC50:  40nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626343(2-[[[4-carbamoyl-7-(4- isopropylphenyl)-2,3- dih...)
Affinity DataEC50:  700nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626344(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)
Affinity DataEC50: >5.00E+4nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626345(2-[[[4-cyano-7-(5-isopropyl-2- pyridyl)-2,3-dihyd...)
Affinity DataEC50:  3.40E+3nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM626346(2-[[[7-(4-isopropylphenyl)-4- methylsulfonyl-2,3-...)
Affinity DataEC50:  2.00E+3nMAssay Description:Table 4-5: Purified His-tagged TEAD protein (YAP Binding Domain, amino acids 217-447) is pre-incubated with Europium labelled anti-His antibody trace...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50600845(CHEMBL5173440)
Affinity DataKd:  7.60E+3nMAssay Description:Binding affinity to human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50600846(CHEMBL5170406)
Affinity DataKd:  5.40E+3nMAssay Description:Binding affinity to human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21 Star (DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50626272(CHEMBL5408794)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to TEAD 4 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50626273(CHEMBL5406847)
Affinity DataKd:  2.94E+4nMAssay Description:Binding affinity to TEAD 4 (unknown origin) assessed as dissociation constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataKd:  7.30E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50626275(CHEMBL23827)
Affinity DataKd:  2.34E+5nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM85507(NSC_4488 | CAS_4394-00-7 | Niflumic acid (Hit 16) ...)
Affinity DataKd:  2.80E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM69368(SMR000372165 | MLS000760860 | cid_2398458 | 2-[[4-...)
Affinity DataKd:  3.10E+4nMAssay Description:Binding affinity to His-tagged TEAD4 YAP-binding domain (217 to 434 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isot...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50447134(SJ000018297 | CHEMBL602720)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to CM5 chip immobilised N-terminal histidine -tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli (DE3) cells ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50626286(CHEMBL5411056)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to CM5 chip immobilised N-terminal histidine -tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli (DE3) cells ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTranscriptional enhancer factor TEF-3(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50630291(US12110276, Compound 48 | CHEMBL5411200)
Affinity DataIC50: 0.880nMAssay Description:His-tagged TEAD proteins are pre-incubated with TEAD project compounds for 30 minutes or 4 hours at room temperature. Biotinylated lipid pocket probe...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM706074(US20240382600, Example 3)
Ligand InfoPC cidPC sid
In DepthDetails

Displayed 1 to 50 (of 522 total ) | Next | Last >>
Jump to: