Report error Found 116 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LasR'
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 3.60nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 119nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli BL21 DE3 after 4 to 6 hrs by GFP reporter gene assayMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.30E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 2.10E+4nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa PAO1 MW1 (pUM15) LasR after 8 hrs by beta-galactosidase reporter gene assay relative to OdDHLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.88E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 906nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 256nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 162nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.40E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 139nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 4.20E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: 71nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at Pseudomonas aeruginosa MW1 LasR assessed as inhibition of protein interaction with OdDHL by beta-galactosidase reporter gene a...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in presence of 7.5 nM natural auto-inducer 3-oxo-C12-HSLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in presence of 7.5 nM natural auto-inducer 3-oxo-C12-HSLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli DH5alpha assessed as inhibition of protein interaction with OdDHL af...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in presence of 7.5 nM natural auto-inducer 3-oxo-C12-HSLMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli DH5alpha assessed as inhibition of protein interaction with OdDHL af...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli DH5alpha assessed as inhibition of protein interaction with OdDHL af...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Antagonist activity at LasR in Pseudomonas aeruginosa PAO1 harboring GFP-fused quorum sensing lasB measured every 15 mins for 14 hrs by GFP reporter ...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli DH5alpha assessed as inhibition of protein interaction with OdDHL af...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Rowan University
Curated by ChEMBL
Rowan University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
