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Report error Found 7763 Enz. Inhib. hit(s) with Target = 'Toll-like receptor 9' Sort by
TargetToll-like receptor 9(Mouse)
Princ

Curated by ChEMBL
LigandPNGBDBM50543465(CHEMBL4636498)
Affinity DataEC50:  25nMAssay Description:Invivo antagonist activity at TLR9 in po dosed C57BL/6 mouse assessed as reduction of CpG-ODN-1585-induced IL-6 production pretreated for 30 mins fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50239681(CHEMBL4074408)
Affinity DataEC50:  5.66E+3nMAssay Description:Agonist activity at human TLR9More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50239681(CHEMBL4074408)
Affinity DataEC50:  5.66E+3nMAssay Description:Agonist activity at human TLR9 expressed in HEK293 cells assessed as induction of NF-kB activation-mediated SEAP production after 24 hrs by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2019
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033123(CHEMBL3356618)
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033119(CHEMBL3357062)
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033101(CHEMBL2144205)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50587873(CHEMBL5169681)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at TLR9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50581965(CHEMBL5094930)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue-HTLR7 cells assessed as inhibition of CpGB-induced NFkappaB activation measured after overnig...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033108(CHEMBL3357064)
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033124(CHEMBL3356617)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50252308(CHEMBL4065452)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human TLR9 expressed in HEK293 cells coexpressing firefly luciferase assessed as inhibition of CpGB-induced NFkappaB activatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033107(CHEMBL3357065)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033102(CHEMBL3357070)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595527(CHEMBL5176310)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue hTLR9 cells assessed as inhibition of CpGB-induced NFkappaB activation preincubated with comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50252308(CHEMBL4065452)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human TLR9 expressed in HEK293 cells assessed as inhibition of CpGB-induced NF-kappaB activation after 24 hrs by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM444287(US10660877, Example 877)
Affinity DataIC50: 16nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2021
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033126(CHEMBL3356616)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595519(CHEMBL5177422)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue hTLR9 cells assessed as inhibition of CpGB-induced NFkappaB activation preincubated with comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM444220(US10660877, Example 810)
Affinity DataIC50: 19nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2021
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595498(CHEMBL5193639)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue hTLR9 cells assessed as inhibition of CpGB-induced NFkappaB activation preincubated with comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50274714(2-(4-(4-methylpiperazin-1-yl)phenyl)-N-(2-morpholi...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK293 cells assessed as blockade of CpG oligonucleotide-induced immune response by NF-kappaB lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467773(CHEMBL4282131)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50274714(2-(4-(4-methylpiperazin-1-yl)phenyl)-N-(2-morpholi...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue hTLR9 cells assessed as activation of NFkappaB incubated for 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467784(CHEMBL4278635)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467770(CHEMBL4279467)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467766(CHEMBL4276673)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033132(CHEMBL3356615)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033132(CHEMBL3356615)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue hTLR9 cells assessed as activation of NFkappaB incubated for 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM444221(US10660877, Example 811)
Affinity DataIC50: 23nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2021
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM235724(US9359361, 67 | US10117875, Example 67)
Affinity DataIC50: 25nMT: 2°CAssay Description:Day 1: A cell suspension of HEK-Blue™-hTLR9 cells at ~450,000 cells per ml in test medium which contained 5% (v/v) heat inactivated FBS was pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM235724(US9359361, 67 | US10117875, Example 67)
Affinity DataIC50: 25nMAssay Description:HEK-Blue-hTLR9 cells were obtained from InvivoGen Inc. and used to determine test compound antagonism of human TLR9 (hTLR9) driven responses. HEK-Blu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM655054(US11912703, Example 9)
Affinity DataIC50: 26nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033140(CHEMBL3356611)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50033103(CHEMBL3357069)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human TLR9 transfected in HEK293 cells after 6 hrs by NF-kappaB luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595508(CHEMBL5183377)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at TLR9 in human pDCs inhibition of CpGB-induced NFkappaB activation by measuring IFN-alpha levels preincubated with compound for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595518(CHEMBL5187807)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue hTLR9 cells assessed as inhibition of CpGB-induced NFkappaB activation preincubated with comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467786(CHEMBL4281194)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467794(CHEMBL4290314)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467774(CHEMBL4286933)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50274715(N-(2-(dimethylamino)ethyl)-2-(4-(4-methylpiperazin...)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK293 cells assessed as blockade of CpG oligonucleotide-induced immune response by NF-kappaB lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467782(CHEMBL4279648)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50467775(CHEMBL4278682)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-Blue cells assessed as reduction in CpGB-induced NF-kappaB levels after 24 hrs by spectrophotometr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM443949(US10660877, Example 537)
Affinity DataIC50: 32nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2021
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50582802(CHEMBL5092293)
Affinity DataIC50: 32nMAssay Description:Inhibition of human TLR9 expressed in HEK-Blue hTLR9 cells assessed as inhibition of TLR9 by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50587877(CHEMBL5207784)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at R848 stimulated TRL9 in HEK-Blue hTLR9 cells assessed as inhibition of NF kappa B/Ap-1 activation measured after 20 hrs by SEA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50582805(CHEMBL5075053)
Affinity DataIC50: 32nMAssay Description:Inhibition of human TLR9 expressed in HEK-Blue hTLR9 cells assessed as inhibition of TLR9 by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50587876(CHEMBL5208108)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at R848 stimulated TRL9 in HEK-Blue hTLR9 cells assessed as inhibition of NF kappa B/Ap-1 activation measured after 20 hrs by SEA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM655201(US11912703, Example 342 | US11912703, Example 317)
Affinity DataIC50: 34nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2024
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM444222(US10660877, Example 812)
Affinity DataIC50: 35nMAssay Description:HEK-Blue-cells (Invivogen) overexpressing human TLR7, TLR8 or TLR9 receptors were used for screening inhibitors of these receptors using an inducible...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2021
Entry Details
Go to US Patent

TargetToll-like receptor 9(Human)
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50595516(CHEMBL5197857)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human TLR9 expressed in HEK-blue hTLR9 cells assessed as inhibition of CpGB-induced NFkappaB activation preincubated with comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
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