Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'Toll-like receptor 5'
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50239681(CHEMBL4074408)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human TLR5 expressed in HEK293 cells assessed as induction of NF-kB activation-mediated SEAP production after 24 hrs by HTS assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50552136(CHEMBL4795753)
Affinity DataIC50: 850nMAssay Description:Inhibition of Flagellin-BS binding to human TLR5 expressed in HEK293 cells harboring SEAP reporter gene preincubated for 24 hrs followed by compound ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50552136(CHEMBL4795753)
Affinity DataIC50: 850nMAssay Description:Antagonist activity at TLR5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50563780(CHEMBL4795714)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human TLR5 stably expressed in HEK293 cells cotransfected with secreted alkaline phosphatase assessed as assessed as inhibition of flag...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50622095(CHEMBL5423509)
Affinity DataIC50: 3.13E+3nMAssay Description:Antagonist activity at TLR5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50622094(CHEMBL5436800)
Affinity DataIC50: 3.38E+3nMAssay Description:Antagonist activity at TLR5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50543142(CHEMBL4641633)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at TLR5 in human PBMC assessed as inhibition of flagellin-induced TNFalpha production preincubated for 30 mins followed by flagel...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetToll-like receptor 5(Human)
University of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50622093(CHEMBL5435694)
Affinity DataIC50: 5.05E+4nMAssay Description:Antagonist activity at TLR5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed