Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with Target = 'Telomeric repeat-binding factor 2' Sort by
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136331(CHEMBL3752722)
Affinity DataKd:  11nMAssay Description:Binding affinity to RAP1 (unknown origin) incubated for 1 to 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136337(CHEMBL3752164)
Affinity DataKd:  11nMAssay Description:Binding affinity to RAP1 (unknown origin) incubated for 1 to 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136326(CHEMBL3752569)
Affinity DataKd:  300nMAssay Description:Binding affinity to RAP1 (unknown origin) incubated for 1 to 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136330(CHEMBL3753350)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to RAP1 (unknown origin) incubated for 1 to 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546766(CHEMBL4745325)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to biotinylated TRF2 (unknown origin) by biolayer interferometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136318(CHEMBL3752561)
Affinity DataIC50: 65nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136317(CHEMBL3752190)
Affinity DataIC50: 100nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136315(CHEMBL3751889)
Affinity DataIC50: 120nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136319(CHEMBL3752814)
Affinity DataIC50: 120nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136320(CHEMBL3752958)
Affinity DataIC50: 130nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136311(CHEMBL3752264)
Affinity DataIC50: 180nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136310(CHEMBL3754578)
Affinity DataIC50: 280nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136316(CHEMBL3752170)
Affinity DataIC50: 610nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136305(CHEMBL3752828)
Affinity DataIC50: 700nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136300(CHEMBL3752803)
Affinity DataIC50: 7.10E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136313(CHEMBL3752883)
Affinity DataIC50: 8.30E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136314(CHEMBL3752069)
Affinity DataIC50: 9.30E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136309(CHEMBL3754122)
Affinity DataIC50: 9.70E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136301(CHEMBL3753586)
Affinity DataIC50: 1.38E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136308(CHEMBL3754737)
Affinity DataIC50: 1.50E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136312(CHEMBL3753717)
Affinity DataIC50: 2.70E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136305(CHEMBL3752828)
Affinity DataIC50: 2.85E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136306(CHEMBL3754019)
Affinity DataIC50: 3.65E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136307(CHEMBL3754707)
Affinity DataIC50: 3.78E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136298(CHEMBL3752820)
Affinity DataIC50: 4.33E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136302(CHEMBL3752348)
Affinity DataIC50: 6.44E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136304(CHEMBL3751917)
Affinity DataIC50: 9.03E+4nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136299(CHEMBL3752992)
Affinity DataIC50: 1.37E+5nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136303(CHEMBL3752934)
Affinity DataIC50: 1.82E+5nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136340(CHEMBL3752470)
Affinity DataIC50: 2.00E+5nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136318(CHEMBL3752561)
Affinity DataKi:  7nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136317(CHEMBL3752190)
Affinity DataKi:  16nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136315(CHEMBL3751889)
Affinity DataKi:  19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136319(CHEMBL3752814)
Affinity DataKi:  19nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136320(CHEMBL3752958)
Affinity DataKi:  22nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136311(CHEMBL3752264)
Affinity DataKi:  32nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136310(CHEMBL3754578)
Affinity DataKi:  53nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338579(CHEMBL4166000)
Affinity DataKi:  90nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338579(CHEMBL4166000)
Affinity DataKi:  90nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136316(CHEMBL3752170)
Affinity DataKi:  130nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136305(CHEMBL3752828)
Affinity DataKi:  140nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338573(CHEMBL4163499)
Affinity DataKi:  210nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338561(CHEMBL4172926)
Affinity DataKi:  240nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546773(CHEMBL4782698)
Affinity DataKi:  330nMAssay Description:Binding affinity to TRFH domain of TRF2 (residues 42 to 245) (unknown origin) by FP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338565(CHEMBL4176290)
Affinity DataKi:  340nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338580(CHEMBL4163072)
Affinity DataKi:  380nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338572(CHEMBL4161391)
Affinity DataKi:  510nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338555(CHEMBL4161856)
Affinity DataKi:  720nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50338574(CHEMBL4159482)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of 5-((2R,6S,9S,12S,15S,18S,21S,24S)-3-((S)-2-((S)-1-amino-3-methyl-1-oxobutan-2-ylcarbamoyl)pyrrolidine-1-carbonyl)-15-(4-aminobutyl)-2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTelomeric repeat-binding factor 2-interacting protein 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50136300(CHEMBL3752803)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive binding to RAP1 (unknown origin) incubated for 1 hr by fluorescence polarization-based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2017
Entry Details Article
PubMed
Displayed 1 to 50 (of 116 total ) | Next | Last >>
Jump to: