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Report error Found 117 Enz. Inhib. hit(s) with Target = 'Tau-tubulin kinase 1'
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM4622(CHEMBL127907 | 3-[(6,7-dimethoxyquinazolin-4-yl)am...)
Affinity DataKd:  240nMAssay Description:Binding affinity to phosphorylated TTBK1 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50506661(CHEMBL4517951)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to phosphorylated TTBK1 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM4622(CHEMBL127907 | 3-[(6,7-dimethoxyquinazolin-4-yl)am...)
Affinity DataKd:  240nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal His6/TEV fused-GST-tagged human TTBK1 (14 to 313 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50506661(CHEMBL4517951)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal His6/TEV fused-GST-tagged human TTBK1 (14 to 313 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602886(CHEMBL5182036)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609143(CHEMBL5268795)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609151(CHEMBL5283456)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609159(CHEMBL5280210)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609138(CHEMBL5272364)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609144(CHEMBL5279863)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609137(CHEMBL5282072)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609160(CHEMBL5268080)
Affinity DataIC50: 10nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609145(CHEMBL5271137)
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609158(CHEMBL5282902)
Affinity DataIC50: 20nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609142(CHEMBL5290581)
Affinity DataIC50: 32nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609157(CHEMBL5274162)
Affinity DataIC50: 37nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609139(CHEMBL5280803)
Affinity DataIC50: 39nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609151(CHEMBL5283456)
Affinity DataIC50: 42nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609141(CHEMBL5288487)
Affinity DataIC50: 57nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609136(CHEMBL5278744)
Affinity DataIC50: 60nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609140(CHEMBL5274528)
Affinity DataIC50: 86nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609143(CHEMBL5268795)
Affinity DataIC50: 98nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609137(CHEMBL5282072)
Affinity DataIC50: 114nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50506660(CHEMBL4528881)
Affinity DataIC50: 120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602885(CHEMBL5193906)
Affinity DataIC50: 120nMAssay Description:Inhibition of TTBK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609156(CHEMBL5290252)
Affinity DataIC50: 124nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609144(CHEMBL5279863)
Affinity DataIC50: 164nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609138(CHEMBL5272364)
Affinity DataIC50: 177nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609161(CHEMBL5279159)
Affinity DataIC50: 185nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50429615(CHEMBL2334586)
Affinity DataIC50: 199nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609158(CHEMBL5282902)
Affinity DataIC50: 224nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609160(CHEMBL5268080)
Affinity DataIC50: 239nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602904(CHEMBL5204869)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609146(CHEMBL5273263)
Affinity DataIC50: 259nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609159(CHEMBL5280210)
Affinity DataIC50: 315nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602917(CHEMBL5200069)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602907(CHEMBL5193488)
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609156(CHEMBL5290252)
Affinity DataIC50: 352nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609162(CHEMBL5275588)
Affinity DataIC50: 352nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602930(CHEMBL5181249)
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602922(CHEMBL5184336)
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609162(CHEMBL5275588)
Affinity DataIC50: 377nMAssay Description:Inhibition of TTBK1 in human HEK293T cells incubated for 1 hrs by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602921(CHEMBL5180098)
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602903(CHEMBL5198544)
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602932(CHEMBL5178965)
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50609152(CHEMBL5272862)
Affinity DataIC50: 414nMAssay Description:Inhibition of GST-tagged TTBK1 (1 to 421) (unknown origin) using DNA Topoisomerase 2-alpha-Thr1342 as substrate incubated for 15 mins followed by ATP...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602910(CHEMBL5209196)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602906(CHEMBL5187459)
Affinity DataIC50: 440nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetTau-tubulin kinase 1(Human)
Technical University of Madrid

Curated by ChEMBL
LigandPNGBDBM50602920(CHEMBL5187125)
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant human TTBK1 using RICDLHDDEEDEAMSITA as substrate incubated for 30 mins in presence of 33P-gamma-ATPMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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