Compile Data Set for Download or QSAR
Report error Found 710 Enz. Inhib. hit(s) with Target = 'Sucrase-isomaltase, intestinal'
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024139(1-Hydroxymethyl-5-phenethylamino-cyclohexane-1,2,3...)
Affinity DataIC50: 2.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024120(1-Hydroxymethyl-5-[(thiophen-2-ylmethyl)-amino]-cy...)
Affinity DataIC50: 3.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50156360(2-Hydroxymethyl-6-nonyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50373983(CHEMBL268675)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50226273(CHEMBL3349431)
Affinity DataIC50: 4.60nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50373982(CHEMBL402196)
Affinity DataIC50: 5nMAssay Description:Inhibition of rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024119(5-(2-Hydroxy-cyclohexylamino)-1-hydroxymethyl-cycl...)
Affinity DataIC50: 5.20nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024137(1-Hydroxymethyl-5-(2-hydroxy-2-phenyl-ethylamino)-...)
Affinity DataIC50: 5.80nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024136(5-(3,5-Di-tert-butyl-4-hydroxy-benzylamino)-1-hydr...)
Affinity DataIC50: 6.80nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405395(CHEMBL2051761)
Affinity DataIC50: 7.5nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50373981(CHEMBL403239)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024114(5-(Cyclohexylmethyl-amino)-1-hydroxymethyl-cyclohe...)
Affinity DataIC50: 9.30nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405397(CHEMBL2051983)
Affinity DataIC50: 10nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024118(5-(3,7-Dimethyl-octa-2,6-dienylamino)-1-hydroxymet...)
Affinity DataIC50: 11nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024124(1-Hydroxymethyl-5-(2-hydroxy-1-phenyl-ethylamino)-...)
Affinity DataIC50: 13nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024133(1-Hydroxymethyl-5-(3-phenyl-allylamino)-cyclohexan...)
Affinity DataIC50: 14nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024117(5-Cyclohexylamino-1-hydroxymethyl-cyclohexane-1,2,...)
Affinity DataIC50: 15nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024126(1-Hydroxymethyl-5-[(pyridin-3-ylmethyl)-amino]-cyc...)
Affinity DataIC50: 15nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024128(5-(4-Bromo-benzylamino)-1-hydroxymethyl-cyclohexan...)
Affinity DataIC50: 15nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50048090(CHEMBL3311519)
Affinity DataIC50: 26nMAssay Description:Inhibition of Wistar rat intestinal sucrase assessed as inhibition of D-glucose release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50333455((2S,3S,4S,5S)-2-butyl-5-(hydroxymethyl)pyrrolidine...)
Affinity DataIC50: 32nMAssay Description:Inhibition of Wistar rat intestinal sucrase assessed as inhibition of D-glucose release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50333455((2S,3S,4S,5S)-2-butyl-5-(hydroxymethyl)pyrrolidine...)
Affinity DataIC50: 32nMAssay Description:Inhibition of Wistar rat small intestine sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50333455((2S,3S,4S,5S)-2-butyl-5-(hydroxymethyl)pyrrolidine...)
Affinity DataIC50: 32nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405389(CHEMBL2051982)
Affinity DataIC50: 35nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405396(CHEMBL2051762)
Affinity DataIC50: 36nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Sucrase in rat intestinal brush border membranes by D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Sucrase in rat intestinal brush border membranes by D-glucose oxidase-peroxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50375510(CHEMBL405957)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50180584(CHEMBL3814496)
Affinity DataIC50: 42nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50048086(CHEMBL3311515)
Affinity DataIC50: 45nMAssay Description:Inhibition of Wistar rat intestinal sucrase assessed as inhibition of D-glucose release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024129(Valiolamine | CHEMBL9216 | Valinolamine | 5-Amino-...)
Affinity DataIC50: 49nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50263044(Voglibose | CHEMBL476960)
Affinity DataIC50: 70nMAssay Description:Inhibition of rat intestinal brush border membrane sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50375511(CHEMBL406973)
Affinity DataIC50: 80nMAssay Description:Inhibition of rat isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50405393(CHEMBL2051981)
Affinity DataIC50: 80nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50180582(CHEMBL3814988)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50180583(CHEMBL3815109)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50156356(2-Hydroxymethyl-6-octyl-piperidine-3,4,5-triol | C...)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat intestinal isomaltase using disaccharideMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50242818(1-Oxo-1lambda-4-thia-cyclotridecan-3,4,5,6,8,10,11...)
Affinity DataIC50: 99nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50375510(CHEMBL405957)
Affinity DataIC50: 100nMAssay Description:Inhibition of rat sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50573735(CHEMBL4860203)
Affinity DataIC50: 100nMAssay Description:Inhibition of rat intestinal sucrase using p-nitrophenyl glycoside as substrate assessed as release of p-nitrophenol measured by spectrometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50612995(CHEMBL5276586)
Affinity DataIC50: 100nMAssay Description:Inhibition of sucrase in rat small intestinal brush border membrane vesicles using sucrose as substrate incubated for 30 mins by glucose-oxidase meth...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50048088(CHEMBL3311517)
Affinity DataIC50: 110nMAssay Description:Inhibition of Wistar rat intestinal sucrase assessed as inhibition of D-glucose release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50333457((2S,3S,4S,5S)-2-hexyl-5-(hydroxymethyl)pyrrolidine...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Wistar rat small intestine sucrase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50242271(Glyset | N-Hydroxyethyl-1-deoxynojirimycin | CHEMB...)
Affinity DataIC50: 110nMAssay Description:Inhibition of rat intestinal brush border membrane sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50333457((2S,3S,4S,5S)-2-hexyl-5-(hydroxymethyl)pyrrolidine...)
Affinity DataIC50: 110nMAssay Description:Inhibition of rat intestinal sucrase using sucrose as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50180520(CHEMBL3814838)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat small intestinal sucrase using sucrose as substrate incubated for 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50342937((1S,2R,3S,4S)-1-((2S,3S)-3-ethoxy-2,4-dihydroxybut...)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM18363((2R,3R,4R,5S,6R)-2-(hydroxymethyl)-6-octylpiperidi...)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat intestinal isomaltase using isomaltase as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50573741(CHEMBL4873807)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat intestinal sucrase using p-nitrophenyl glycoside as substrate assessed as release of p-nitrophenol measured by spectrometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Orleans University

Curated by ChEMBL
LigandPNGBDBM50048087(CHEMBL3311516)
Affinity DataIC50: 130nMAssay Description:Inhibition of Wistar rat intestinal sucrase assessed as inhibition of D-glucose release after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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