Compile Data Set for Download or QSAR
Report error Found 4314 Enz. Inhib. hit(s) with Target = 'Substance-P receptor'
TargetSubstance-P receptor(Rat)
University of Arizona Tucson

LigandPNGBDBM21010(H-Tyr-D-Ala-Gly-Phe-Pro-Leu-Trp-NH-Bzl | (2S)-2-{[...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Rat)
University of Arizona Tucson

LigandPNGBDBM21011(H-Tyr-D-Ala-Gly-Phe-Pro-Leu-Trp-NMe-Bzl | (2S)-2-{...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007962(CHEMBL81919 | pGlu6-Phe-NMePhe-Gly-Leu-Met-NH2)
Affinity DataEC50:  600nMAssay Description:Effective dose was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007824(CHEMBL293747 | 2-(2-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50: >3.57E+3nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007823(CHEMBL2372953 | 1-{2-[2-(4-Amino-butyrylamino)-3-p...)
Affinity DataEC50:  188nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007825(CHEMBL291903 | 2-(2-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50:  130nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007828(CHEMBL292435 | 2-(1-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007830(CHEMBL301477 | 1-{2-[2-(4-Amino-butyrylamino)-3-ph...)
Affinity DataEC50:  400nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007822(CHEMBL2372954 | 2-(2-{2-[2-(4-Amino-butyrylamino)-...)
Affinity DataEC50:  892nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataEC50:  1nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007831(CHEMBL54622 | 2-(2-{2-[2-(4-Amino-butyrylamino)-3-...)
Affinity DataEC50:  6.90nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007826(CHEMBL2372949 | 2-(2-{2-[2-(4-Amino-butyrylamino)-...)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007832(CHEMBL299503 | 2-(3-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007827(CHEMBL301841 | 2-(3-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50:  15nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007829(CHEMBL280020 | 2-(1-{2-[2-(4-Amino-butyrylamino)-3...)
Affinity DataEC50:  63nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50452295(CHEMBL2371799)
Affinity DataEC50:  2.20nMAssay Description:Compound was evaluated for effective dose against muscular receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50016358(CHEMBL428532 | 4-Amino-4-{1-[1-({[1-(1-carbamoyl-3...)
Affinity DataEC50:  4nMAssay Description:Compound was evaluated for effective dose against Neuronal receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007822(CHEMBL2372954 | 2-(2-{2-[2-(4-Amino-butyrylamino)-...)
Affinity DataEC50: >100nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataEC50:  4.90nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Rat)
University of Arizona Tucson

LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  0.970nMAssay Description:Scatchard analysis at concentration of the 1 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Rat)
University of Arizona Tucson

LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  1.5nMAssay Description:Scatchard analysis at concentration of the 10 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Rat)
University of Arizona Tucson

LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataKd:  0.180nMAssay Description:Scatchard analysis at concentration of the 3 uM :Apparent affinity constant (Kd) against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007972(CHEMBL311917 | pGlu6-Phe-Phe8(psi)CH2O-Gly-Leu-Met...)
Affinity DataEC50:  40nMAssay Description:Effective dose was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007963(CHEMBL441061 | pGlu6-Phe-Phe-Gly-Leu-Met-NH2)
Affinity DataEC50:  2.20nMAssay Description:Effective dose was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030212((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  180nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030211((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  5nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030213((S)-2-{2-[(2R,5S,8R)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  11nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50030214((S)-2-{2-[(6R,9S,12R)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001603(CHEMBL133362 | 2-(1-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  307nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001593(N-{1-[1-(1-{1-[1-(1-Carbamoyl-3-methylsulfanyl-pro...)
Affinity DataEC50:  4.24E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001594(N-(1-{1-[1-({[1-(1-Carbamoyl-3-methylsulfanyl-prop...)
Affinity DataEC50:  61nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001602(CHEMBL339391 | 2-(1-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  3.73E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001606(CHEMBL335248 | 2-(2-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001595(CHEMBL407511 | 1-{2-[2-(5-Amino-pentanoylamino)-3-...)
Affinity DataEC50:  13nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001607(CHEMBL262048 | 1-{2-[2-(5-Amino-pentanoylamino)-3-...)
Affinity DataEC50:  830nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001604(CHEMBL262049 | 2-(2-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  38nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001600(N-{1-[1-(1-Benzyl-2-{5-[1-(1-carbamoyl-3-methylsul...)
Affinity DataEC50:  1.03E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001447(His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu-Met-NH2(Neurok...)
Affinity DataEC50:  14nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001596(3-(2-Acetylamino-6-amino-hexanoylamino)-N-{1-[1-(1...)
Affinity DataEC50:  44nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001598(CHEMBL337037 | 2-(1-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  5.23E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001592(N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-methylsulfanyl-pro...)
Affinity DataEC50:  1.13E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001599(CHEMBL134012 | 2-(1-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  545nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataEC50:  68nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataEC50:  5.60nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001601(CHEMBL135186 | 2-(3-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001605(CHEMBL337465 | 2-(1-{2-[2-(5-Amino-pentanoylamino)...)
Affinity DataEC50:  3.77E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50001597(N-(1-{1-[1-({[1-(1-Carbamoyl-3-methylsulfanyl-prop...)
Affinity DataEC50:  45nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052515((S)-2-{2-[(2S,5R,8S)-5,8-Dibenzyl-2-(3-guanidino-p...)
Affinity DataEC50:  11nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052516((S)-2-{2-[(3S,6R,9S)-3,6-Dibenzyl-9-(3-guanidino-p...)
Affinity DataEC50:  60nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSubstance-P receptor(Guinea pig)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50052517((S)-2-{2-[(6S,9R,12S)-6,9-Dibenzyl-12-(3-guanidino...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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