Compile Data Set for Download or QSAR
Report error Found 2453 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 4'
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  4.68E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  4.17E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  2.63E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  8.91E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst4) expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  574nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  353nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  321nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  182nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50081059(CHEMBL3421845 | US10166214, Example 138 | US978908...)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human somatostatin 4 receptor expressed in H4 cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50081060(CHEMBL3421844 | US10166214, Example 101 | US978908...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human somatostatin 4 receptor expressed in H4 cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50081055(CHEMBL3421843 | US10166214, Example 49 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human somatostatin 4 receptor expressed in H4 cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50081058(CHEMBL3421842 | US10166214, Example 22 | US9789082...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human somatostatin 4 receptor expressed in H4 cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation i...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50261729(6-chloro-3-(4-(3-(2-chloro-4-fluorophenyl)-1,2,4-o...)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423297(Obelin | CHEMBL251541)
Affinity DataKd:  1.51E+4nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  8.13E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423465(ERGOLINE)
Affinity DataKd:  4.90E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423458(CHEMBL252232)
Affinity DataKd:  5.62E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  3.63E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275985(US10071974, Example 96 | US10577336, Example 96)
Affinity DataEC50:  13nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275986(US10071974, Example 97 | US10577336, Example 97)
Affinity DataEC50:  40.8nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275987(US10071974, Example 98)
Affinity DataEC50:  85.3nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275988(US10071974, Example 99 | US10577336, Example 99)
Affinity DataEC50:  43.4nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275989(US10071974, Example 100 | US10577336, Example 100)
Affinity DataEC50:  103nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275990(US10071974, Example 103 | US10071974, Example 101 ...)
Affinity DataEC50:  6.5nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275991(US10071974, Example 102 | US10577336, Example 102)
Affinity DataEC50:  31nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275990(US10071974, Example 103 | US10071974, Example 101 ...)
Affinity DataEC50:  60.7nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275993(US10071974, Example 104 | US10577336, Example 104)
Affinity DataEC50:  73.5nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275994(US10071974, Example 105 | US10577336, Example 105)
Affinity DataEC50:  596nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275995(US10071974, Example 106 | US10577336, Example 106)
Affinity DataEC50:  230nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275996(US10071974, Example 107 | US10577336, Example 107)
Affinity DataEC50:  51.1nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275997(US10071974, Example 108 | US10577336, Example 108)
Affinity DataEC50:  58.1nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275998(US10071974, Example 109 | US10577336, Example 109)
Affinity DataEC50:  3.70nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275999(US10071974, Example 111 | US10071974, Example 110 ...)
Affinity DataEC50:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM275999(US10071974, Example 111 | US10071974, Example 110 ...)
Affinity DataEC50:  290nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276001(US10071974, Example 113 | US10071974, Example 112 ...)
Affinity DataEC50:  5.50E+3nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276001(US10071974, Example 113 | US10071974, Example 112 ...)
Affinity DataEC50:  380nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276003(US10071974, Example 115 | US10071974, Example 114 ...)
Affinity DataEC50:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276003(US10071974, Example 115 | US10071974, Example 114 ...)
Affinity DataEC50:  294nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276005(US10071974, Example 117 | US10071974, Example 118 ...)
Affinity DataEC50:  9.30nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276005(US10071974, Example 117 | US10071974, Example 118 ...)
Affinity DataEC50:  2.60nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276005(US10071974, Example 117 | US10071974, Example 118 ...)
Affinity DataEC50:  86.8nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSomatostatin receptor type 4(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM276008(US10071974, Example 120 | US10071974, Example 119 ...)
Affinity DataEC50:  73.9nMpH: 7.4 T: 2°CAssay Description:Compounds are dissolved and diluted in DMSO. The final test solution contains 1% DMSO. The cAMP standard (Lance cAMP 384 Kit; PerkinElmer, Cat# AD026...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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