Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with Target = 'Solute carrier family 2, facilitated glucose transporter member 4'
LigandPNGBDBM50510641(CHEMBL4435909)
Affinity DataEC50:  230nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510640(CHEMBL4529010)
Affinity DataEC50:  47nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510631(CHEMBL4576794)
Affinity DataEC50:  4.70E+3nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510632(CHEMBL4550275)
Affinity DataEC50:  110nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510633(CHEMBL4439282)
Affinity DataEC50:  650nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510634(CHEMBL4570366)
Affinity DataEC50:  230nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510635(CHEMBL4452486)
Affinity DataEC50:  24nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510636(CHEMBL4539293)
Affinity DataEC50:  120nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510637(CHEMBL4466592)
Affinity DataEC50:  140nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510638(CHEMBL4469586)
Affinity DataEC50:  76nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50510639(CHEMBL4588796)
Affinity DataEC50:  140nMAssay Description:Induction of GLUT4 translocation in rat L6-GLUT4myc differentiated myotube cells after 20 mins by chemiluminescent methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277370(CHEMBL4171968)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277370(CHEMBL4171968)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at rat C-terminal 6His/Myc-tagged GLUT4 assessed as reduction in 2-[3H]deoxyglucose uptake measured after 6 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50565143(CHEMBL4793560)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277369(CHEMBL4160688)
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277373(CHEMBL4165190)
Affinity DataIC50: 1.82E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277387(CHEMBL4164091)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50565142(CHEMBL4776246)
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50565144(CHEMBL4786111)
Affinity DataIC50: 1.52E+5nMAssay Description:Inhibition of transport activity of human GLUT4 expressed in hexose transporter deficient W4000fgy1 erg4 yeast cells assessed as reduction in transpo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50277375(CHEMBL4173323)
Affinity DataKi:  2.60E+4nMAssay Description:Antagonist activity at GLUT4 in rat adipocytes assessed as reduction in insulin-stimulated [3H]2-deoxyglucose uptake preincubated for 1 min followed ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed