Compile Data Set for Download or QSAR
Report error Found 149 Enz. Inhib. hit(s) with Target = 'Small conductance calcium-activated potassium channel protein 1/2/3'
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.0120nMAssay Description:Displacement of [125I]apamin from rat brain SkCa channel after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50155248(CHEMBL3774478)
Affinity DataIC50: 0.0160nMAssay Description:Displacement of [125I]apamin from rat cerebral cortex small conductance calcium-activated potassium channelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50092131(CHEMBL612120 | UCL-1848 | CHEMBL420873 | 1,7-diazo...)
Affinity DataIC50: 2nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50061977(CHEMBL117908 | 17,25-diazonia-2,9-diazaheptacyclo[...)
Affinity DataIC50: 3nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50061977(CHEMBL117908 | 17,25-diazonia-2,9-diazaheptacyclo[...)
Affinity DataIC50: 3nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474856(CHEMBL184300)
Affinity DataIC50: 9nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474870(CHEMBL185146)
Affinity DataIC50: 10nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474869(CHEMBL181911)
Affinity DataIC50: 12nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474865(CHEMBL183644)
Affinity DataIC50: 15nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474867(CHEMBL184858)
Affinity DataIC50: 16nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474866(CHEMBL181912)
Affinity DataIC50: 25nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473100(CHEMBL344807)
Affinity DataIC50: 25nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473103(CHEMBL430146)
Affinity DataIC50: 28nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473103(CHEMBL430146)
Affinity DataIC50: 28nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474868(CHEMBL184891)
Affinity DataIC50: 30nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474871(CHEMBL182716)
Affinity DataIC50: 31nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474863(CHEMBL360624)
Affinity DataIC50: 35nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474872(CHEMBL1180184)
Affinity DataIC50: 40nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474858(CHEMBL186139)
Affinity DataIC50: 60nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50150389(17,23-diazonia-2,9-diazahexacyclo[21.6.2.24,7.210,...)
Affinity DataIC50: 60nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473097(CHEMBL136488)
Affinity DataIC50: 60nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474859(CHEMBL185258)
Affinity DataIC50: 65nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473106(CHEMBL137175)
Affinity DataIC50: 70nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473106(CHEMBL137175)
Affinity DataIC50: 70nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084848(BIs-cyclo(4N-pentyl-1-(4-methylbenzyl)-4-quinolini...)
Affinity DataIC50: 80nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473094(CHEMBL137155)
Affinity DataIC50: 90nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473098(CHEMBL342213)
Affinity DataIC50: 100nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084852(4N-[10-(1-methyl-4-quinoliniumylamino)decyl]-1-[3-...)
Affinity DataIC50: 110nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473099(CHEMBL140380)
Affinity DataIC50: 120nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474857(CHEMBL185106)
Affinity DataIC50: 130nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473107(CHEMBL341700)
Affinity DataIC50: 130nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473107(CHEMBL341700)
Affinity DataIC50: 130nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474862(CHEMBL425707)
Affinity DataIC50: 150nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474873(CHEMBL185137)
Affinity DataIC50: 150nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473102(CHEMBL137266)
Affinity DataIC50: 150nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084849(Bis-quinolinium cyclophane analogue | Cyclo(N-deca...)
Affinity DataIC50: 150nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084839(Bis-quinolinium cyclophane analogue | cyclo N-deca...)
Affinity DataIC50: 170nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084851(Bis-quinolinium cyclophane analogue | Cyclo N-deca...)
Affinity DataIC50: 180nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474864(CHEMBL119859)
Affinity DataIC50: 190nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50054105(1-{4-[2-[4-(4-amino-1-quinoliniumylmethyl)phenyl]-...)
Affinity DataIC50: 190nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473108(CHEMBL137116)
Affinity DataIC50: 210nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473111(CHEMBL137256)
Affinity DataIC50: 250nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50474861(CHEMBL185230)
Affinity DataIC50: 260nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473109(CHEMBL136303)
Affinity DataIC50: 260nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473096(CHEMBL434234)
Affinity DataIC50: 280nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50054098(CHEMBL6354 | 1-{3-[3-(4-amino-1-quinoliniumylmethy...)
Affinity DataIC50: 290nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50084846(1-[7-(4-amino-1-quinoliniumylmethyl)-9H-2-fluoreny...)
Affinity DataIC50: 310nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473105(CHEMBL133311)
Affinity DataIC50: 360nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50054103(CHEMBL269729 | CHEMBL370040 | 1-{4-[4-(4-amino-1-q...)
Affinity DataIC50: 380nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50473101(CHEMBL344620)
Affinity DataIC50: 380nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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